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—— (5R,7R)-N-benzyl-3-chloro-5-(4-methylphenyl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H24ClF3N4O
(5R,7R)-N-benzyl-3-chloro-5-(4-methylphenyl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-benzyl-3-chloro-5-(4-methylphenyl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H24ClF3N4O
(5S,7S)-N-benzyl-3-chloro-5-(4-methylphenyl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S)-5-[1-[(2-chloro-6-fluorophenyl)methyl]indol-3-yl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C34H28ClFN2O
(5S)-5-[1-[(2-chloro-6-fluorophenyl)methyl]indol-3-yl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one
—— (5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[3-[(1S)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H24ClF3N4O4
(5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[3-[(1S)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-5-[1-[(2-chloro-6-fluorophenyl)methyl]indol-3-yl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C34H28ClFN2O
(5R)-5-[1-[(2-chloro-6-fluorophenyl)methyl]indol-3-yl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one
—— (5R,7S)-N-[4-chloro-2-[(R)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H22ClF3N4O2
(5R,7S)-N-[4-chloro-2-[(R)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[(2,6-dichlorophenyl)methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C25H26Cl2N4O3S
5-[(2,6-dichlorophenyl)methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S,7S)-N-[4-chloro-2-[(R)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H22ClF3N4O2
(5S,7S)-N-[4-chloro-2-[(R)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[(5-bromothiophen-2-yl)methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C23H25BrN4O4S
5-[(5-bromothiophen-2-yl)methyl]-1,3-dimethyl-5-[[(1R,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— (5R,7S)-N-[(6R)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H21ClF3N5O2S2
(5R,7S)-N-[(6R)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-benzyl-3-chloro-5-(4-methylphenyl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H24ClF3N4O
(5S,7R)-N-benzyl-3-chloro-5-(4-methylphenyl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[3-[(1S)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H24ClF3N4O4
(5R,7S)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[3-[(1S)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[3-[(1R)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H24ClF3N4O4
(5R,7S)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[3-[(1R)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-[(6R)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H21ClF3N5O2S2
(5R,7R)-N-[(6R)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5Z)-2-amino-5-[[3-bromo-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-4,6-dimethylcyclopenta[b]pyridine-3,7-dicarbonitrile —— C26H18BrFN4O
(5Z)-2-amino-5-[[3-bromo-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-4,6-dimethylcyclopenta[b]pyridine-3,7-dicarbonitrile
—— (5S,7R)-3-bromo-N-(2,4-dichlorophenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H12BrCl2F3N4OS
(5S,7R)-3-bromo-N-(2,4-dichlorophenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-[4-chloro-2-[(R)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H22ClF3N4O2
(5S,7R)-N-[4-chloro-2-[(R)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-3-(3-hydroxypropyl)-4-imino-5-phenyl-5H-chromeno[2,3-d]pyrimidin-8-ol —— C20H19N3O3
(5R)-3-(3-hydroxypropyl)-4-imino-5-phenyl-5H-chromeno[2,3-d]pyrimidin-8-ol
—— 5-amino-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-chlorobenzamide —— C16H21ClN2O
5-amino-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-chlorobenzamide
—— 5-[(1R)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-ium-1-yl]-3-(2,4-dimethylphenyl)-6-oxo-2-sulfanylidenepyrimidin-4-olate —— C23H25N3O4S
5-[(1R)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-ium-1-yl]-3-(2,4-dimethylphenyl)-6-oxo-2-sulfanylidenepyrimidin-4-olate
—— 5-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]methyl]-1,3,4-oxadiazol-2-amine —— C10H15N3O
5-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]methyl]-1,3,4-oxadiazol-2-amine
—— (5E)-1-phenyl-5-[[[(2S)-2-pyridin-3-ylpiperidin-1-yl]amino]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C21H21N5O2S
(5E)-1-phenyl-5-[[[(2S)-2-pyridin-3-ylpiperidin-1-yl]amino]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-amino-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-chlorobenzamide —— C16H21ClN2O
5-amino-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-chlorobenzamide
—— (5E)-5-[[3-(dimethylamino)propylamino]methylidene]-1-(2-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H22N4O3S
(5E)-5-[[3-(dimethylamino)propylamino]methylidene]-1-(2-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]-3-methylthiophene-2-carboxylic acid —— C15H19NO3S
5-[[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]-3-methylthiophene-2-carboxylic acid
—— 5-[[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]-3-methylthiophene-2-carboxylic acid —— C15H19NO3S
5-[[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]-3-methylthiophene-2-carboxylic acid
—— (5S)-3-(3-hydroxypropyl)-4-imino-5-phenyl-5H-chromeno[2,3-d]pyrimidin-8-ol —— C20H19N3O3
(5S)-3-(3-hydroxypropyl)-4-imino-5-phenyl-5H-chromeno[2,3-d]pyrimidin-8-ol
—— (5Z)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-ylidene]-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1,3-thiazolidine-2,4-dione —— C22H21N3O4S
(5Z)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-ylidene]-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1,3-thiazolidine-2,4-dione
—— (5R,7R)-N-(4-fluorophenyl)-3-(4-methylphenyl)adamantane-1-carboxamide —— C24H26FNO
(5R,7R)-N-(4-fluorophenyl)-3-(4-methylphenyl)adamantane-1-carboxamide
—— (5S,7S)-N-(4-fluorophenyl)-3-(4-methylphenyl)adamantane-1-carboxamide —— C24H26FNO
(5S,7S)-N-(4-fluorophenyl)-3-(4-methylphenyl)adamantane-1-carboxamide
—— (5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C24H14BrF4NO3
(5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— (5R)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C24H14BrF4NO3
(5R)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— (5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-nitrophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C24H14BrF3N2O5
(5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-nitrophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— (5S,7S)-3-(4-ethoxyphenyl)adamantane-1-carboxylic acid —— C19H24O3
(5S,7S)-3-(4-ethoxyphenyl)adamantane-1-carboxylic acid
—— (5R)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(3-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C24H14BrF4NO3
(5R)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(3-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— (5R)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C24H14BrF4NO3
(5R)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— (5E)-5-[[1-(4-chlorophenyl)pyrrol-2-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one —— C16H14ClN3OS
(5E)-5-[[1-(4-chlorophenyl)pyrrol-2-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
—— (5E)-5-[[[(1R,2R)-2-aminocyclohexyl]amino]methylidene]-1-(4-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H22N4O3S
(5E)-5-[[[(1R,2R)-2-aminocyclohexyl]amino]methylidene]-1-(4-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5E)-5-[(4-hydroxyphenyl)methylidene]-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-4-one —— C13H13NO2S2
(5E)-5-[(4-hydroxyphenyl)methylidene]-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,7S)-3-chloro-N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-methyladamantane-1-carboxamide —— C21H26Cl2N2O3
(5S,7S)-3-chloro-N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-methyladamantane-1-carboxamide
—— (5Z,7S)-5-[(Z)-(4-methoxyphenyl)methylidenehydrazinylidene]-7-phenyl-2,6,7,8-tetrahydrocinnolin-3-one —— C22H20N4O2
(5Z,7S)-5-[(Z)-(4-methoxyphenyl)methylidenehydrazinylidene]-7-phenyl-2,6,7,8-tetrahydrocinnolin-3-one
—— (5Z)-1,3-dimethyl-5-(thiophen-2-ylmethylidene)-2-thioxoimidazolidin-4-one —— C10H10N2OS2
(5Z)-1,3-dimethyl-5-(thiophen-2-ylmethylidene)-2-thioxoimidazolidin-4-one
—— (5E)-5-(4-bromobenzylidene)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1,3-thiazolidine-2,4-dione —— C22H20BrN3O3S
(5E)-5-(4-bromobenzylidene)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1,3-thiazolidine-2,4-dione
—— (5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C24H14BrF4NO3
(5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— (5E)-3-[(2S)-butan-2-yl]-5-[[1-(4-methoxyphenyl)pyrrol-2-yl]methylidene]-1,3-thiazolidine-2,4-dione —— C19H20N2O3S
(5E)-3-[(2S)-butan-2-yl]-5-[[1-(4-methoxyphenyl)pyrrol-2-yl]methylidene]-1,3-thiazolidine-2,4-dione
—— (5Z)-5-[(E)-3-[4-(dimethylamino)phenyl]prop-2-enylidene]-3-(4-methoxyphenyl)-2-sulfanylideneimidazolidin-4-one —— C21H21N3O2S
(5Z)-5-[(E)-3-[4-(dimethylamino)phenyl]prop-2-enylidene]-3-(4-methoxyphenyl)-2-sulfanylideneimidazolidin-4-one
—— (5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(3-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C24H14BrF4NO3
(5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(3-fluorophenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— 5-bromo-N-[(Z)-[3-[(4-bromo-5-methyl-3-nitropyrazol-1-yl)methyl]-4-methoxyphenyl]methylideneamino]-2-hydroxybenzamide —— C20H17Br2N5O5
5-bromo-N-[(Z)-[3-[(4-bromo-5-methyl-3-nitropyrazol-1-yl)methyl]-4-methoxyphenyl]methylideneamino]-2-hydroxybenzamide
—— (5R,7R)-N-(2,3-dimethylphenyl)-3-(4-methylphenyl)adamantane-1-carboxamide —— C26H31NO
(5R,7R)-N-(2,3-dimethylphenyl)-3-(4-methylphenyl)adamantane-1-carboxamide
—— (5E)-3-benzyl-5-[[4-(dimethylamino)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C19H19N3OS
(5E)-3-benzyl-5-[[4-(dimethylamino)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one