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—— 5-[(S)-(2-methoxyphenyl)-piperidin-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22N4O2S
5-[(S)-(2-methoxyphenyl)-piperidin-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O2S
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5R)-3-(4-bromophenyl)-7-(4-methylphenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione —— C19H15BrN2O3
(5R)-3-(4-bromophenyl)-7-(4-methylphenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione
—— 5,7-difluoro-3-[1-(4-methoxyphenyl)-2H-tetrazol-5-ylidene]indole —— C16H11F2N5O
5,7-difluoro-3-[1-(4-methoxyphenyl)-2H-tetrazol-5-ylidene]indole
—— 5-[(S)-(2,4-dimethoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22N4O4S
5-[(S)-(2,4-dimethoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-methoxyphenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H21N4O2S+
5-[(R)-(2-methoxyphenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5R)-5-(2-fluorophenyl)-4-[hydroxy-(3-methoxyphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-2,3-dione —— C22H17FN2O5
(5R)-5-(2-fluorophenyl)-4-[hydroxy-(3-methoxyphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-2,3-dione
—— (5R)-5-[[(1R,2R)-2-aminocyclohexyl]iminomethyl]-1-(2-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H22N4O3S
(5R)-5-[[(1R,2R)-2-aminocyclohexyl]iminomethyl]-1-(2-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-7-naphthalen-2-yl-3-(3-nitrophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione —— C22H15N3O5
(5S)-7-naphthalen-2-yl-3-(3-nitrophenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione
—— (5S)-5-(4-fluorophenyl)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-2,3-dione —— C22H17FN2O4
(5S)-5-(4-fluorophenyl)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-2,3-dione
—— (5R)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-1-(3-methoxypropyl)-5-(5-methylfuran-2-yl)pyrrolidine-2,3-dione —— C22H23NO7
(5R)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-1-(3-methoxypropyl)-5-(5-methylfuran-2-yl)pyrrolidine-2,3-dione
—— (5R)-1-[(2S)-butan-2-yl]-5-(2-morpholin-4-ium-4-ylethyliminomethyl)-6-oxo-2-sulfanylidene-5H-pyrimidin-4-olate —— C15H24N4O3S
(5R)-1-[(2S)-butan-2-yl]-5-(2-morpholin-4-ium-4-ylethyliminomethyl)-6-oxo-2-sulfanylidene-5H-pyrimidin-4-olate
—— (5S)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-5-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C22H20FNO6
(5S)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-5-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— (5S)-4-[(4-ethoxyphenyl)-hydroxymethylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(4-methylphenyl)pyrrolidine-2,3-dione —— C24H22N2O5
(5S)-4-[(4-ethoxyphenyl)-hydroxymethylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(4-methylphenyl)pyrrolidine-2,3-dione
—— (5R)-4-[hydroxy(phenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(3-prop-2-enoxyphenyl)pyrrolidine-2,3-dione —— C24H20N2O5
(5R)-4-[hydroxy(phenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(3-prop-2-enoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-4-[hydroxy(phenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(3-propoxyphenyl)pyrrolidine-2,3-dione —— C24H22N2O5
(5S)-4-[hydroxy(phenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(3-propoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-4-[hydroxy-(4-prop-2-enoxyphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-phenylpyrrolidine-2,3-dione —— C24H20N2O5
(5S)-4-[hydroxy-(4-prop-2-enoxyphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-phenylpyrrolidine-2,3-dione
—— (5S)-4-[hydroxy-(3-methoxyphenyl)methylidene]-5-pyridin-2-yl-1-(pyridin-3-ylmethyl)pyrrolidine-2,3-dione —— C23H19N3O4
(5S)-4-[hydroxy-(3-methoxyphenyl)methylidene]-5-pyridin-2-yl-1-(pyridin-3-ylmethyl)pyrrolidine-2,3-dione
—— (5S)-4-[hydroxy(phenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(4-propoxyphenyl)pyrrolidine-2,3-dione —— C24H22N2O5
(5S)-4-[hydroxy(phenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(4-propoxyphenyl)pyrrolidine-2,3-dione
—— 5-(3-Carboxylatopropanoylamino)-2-chlorobenzoate —— C11H8ClNO5-2
5-(3-Carboxylatopropanoylamino)-2-chlorobenzoate
—— 5-bromo-2-[[(2S)-2-methylbutanoyl]amino]benzoate —— C12H13BrNO3-
5-bromo-2-[[(2S)-2-methylbutanoyl]amino]benzoate
—— (5R)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-thiophen-2-ylpyrrolidine-2,3-dione —— C20H16N2O4S
(5R)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-thiophen-2-ylpyrrolidine-2,3-dione
—— 5-chloro-2-[[(2R)-2-methylbutanoyl]amino]benzoate —— C12H13ClNO3-
5-chloro-2-[[(2R)-2-methylbutanoyl]amino]benzoate
—— (5R)-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-phenylpyrrolidine-2,3-dione —— C22H18N2O5
(5R)-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-phenylpyrrolidine-2,3-dione
—— (5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(3-hydroxyphenyl)-1-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-2,3-dione —— C21H15ClN2O5
(5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(3-hydroxyphenyl)-1-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-2,3-dione
—— (5R)-4-[hydroxy(phenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(4-propoxyphenyl)pyrrolidine-2,3-dione —— C24H22N2O5
(5R)-4-[hydroxy(phenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(4-propoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-4-[hydroxy-(3-methyl-4-propan-2-yloxyphenyl)methylidene]-1-(2-methoxyethyl)-5-pyridin-4-ylpyrrolidine-2,3-dione —— C23H26N2O5
(5R)-4-[hydroxy-(3-methyl-4-propan-2-yloxyphenyl)methylidene]-1-(2-methoxyethyl)-5-pyridin-4-ylpyrrolidine-2,3-dione
—— (5R,7S)-5-(furan-2-yl)-N-propyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C15H17F3N4O2
(5R,7S)-5-(furan-2-yl)-N-propyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-4-[hydroxy-(4-methylphenyl)methylidene]-5-(3-methoxyphenyl)-1-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-2,3-dione —— C23H20N2O5
(5R)-4-[hydroxy-(4-methylphenyl)methylidene]-5-(3-methoxyphenyl)-1-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-2,3-dione
—— (5S,7R)-N-butyl-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C16H19F3N4O2
(5S,7R)-N-butyl-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-5-(furan-2-yl)-N-propyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C15H17F3N4O2
(5S,7R)-5-(furan-2-yl)-N-propyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S)-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(4-methylphenyl)pyrrolidine-2,3-dione —— C23H20N2O5
(5S)-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-(5-methyl-1,2-oxazol-3-yl)-5-(4-methylphenyl)pyrrolidine-2,3-dione
—— (5R,7R)-N-[(2S)-butan-2-yl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C16H19F3N4O2
(5R,7R)-N-[(2S)-butan-2-yl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-chloro-2-[[(2R)-2-phenylbutanoyl]amino]benzoate —— C17H15ClNO3-
5-chloro-2-[[(2R)-2-phenylbutanoyl]amino]benzoate
—— 5,5-Dimethyl-2-[2-[4-(2-methylpropanoyl)piperazin-1-yl]ethyliminomethyl]cyclohexane-1,3-dione —— C19H31N3O3
5,5-Dimethyl-2-[2-[4-(2-methylpropanoyl)piperazin-1-yl]ethyliminomethyl]cyclohexane-1,3-dione
—— (5S,7S)-5-(furan-2-yl)-N-propyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C15H17F3N4O2
(5S,7S)-5-(furan-2-yl)-N-propyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-Hydroxy-7-methyl-6-(piperidin-1-ium-1-ylmethyl)-4-propylchromen-2-one —— C19H26NO3+
5-Hydroxy-7-methyl-6-(piperidin-1-ium-1-ylmethyl)-4-propylchromen-2-one
—— [(5R,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2S)-2-methyl-2,3-dihydroindol-1-yl]methanone —— C21H19F3N4O2
[(5R,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2S)-2-methyl-2,3-dihydroindol-1-yl]methanone
—— 5-[(3S)-3-(2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acid —— C20H20N2O4
5-[(3S)-3-(2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acid
—— (5E)-5-[(4-butoxyphenyl)methylidene]-2-(4-methylpiperazin-4-ium-1-yl)-1,3-thiazol-4-one —— C19H26N3O2S+
(5E)-5-[(4-butoxyphenyl)methylidene]-2-(4-methylpiperazin-4-ium-1-yl)-1,3-thiazol-4-one
—— 5-[(4E)-4-benzylidene-3-methyl-5-oxopyrazol-1-yl]-2-chlorobenzoate —— C18H12ClN2O3-
5-[(4E)-4-benzylidene-3-methyl-5-oxopyrazol-1-yl]-2-chlorobenzoate
—— (5Z)-3-[(2S)-butan-2-yl]-5-[[2-(2-hydroxyethylamino)-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C19H22N4O3S2
(5Z)-3-[(2S)-butan-2-yl]-5-[[2-(2-hydroxyethylamino)-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[(3R)-3-(2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acid —— C20H20N2O4
5-[(3R)-3-(2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acid
—— (5Z)-3-[(2R)-butan-2-yl]-5-[[2-(2-hydroxyethylamino)-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C19H22N4O3S2
(5Z)-3-[(2R)-butan-2-yl]-5-[[2-(2-hydroxyethylamino)-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R)-5-(2-methoxyphenyl)-2-propylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione —— C21H23N3O3S
(5R)-5-(2-methoxyphenyl)-2-propylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione
—— (5R)-5-(4-nitrophenyl)-2-prop-2-enylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione —— C20H18N4O4S
(5R)-5-(4-nitrophenyl)-2-prop-2-enylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione
—— (5Z)-3-[(2R)-butan-2-yl]-5-[[2-(2-hydroxyethylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H20N4O3S2
(5Z)-3-[(2R)-butan-2-yl]-5-[[2-(2-hydroxyethylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-chloro-4-methylsulfanyl-1H-pyridazin-6-one —— C5H5ClN2OS
5-chloro-4-methylsulfanyl-1H-pyridazin-6-one
—— 5-Nitro-1-(2-oxo-2-pyrrolidin-1-ylethyl)pyridin-2-one —— C11H13N3O4
5-Nitro-1-(2-oxo-2-pyrrolidin-1-ylethyl)pyridin-2-one
—— 5-[N-[(4-chlorophenyl)methyl]-C-methylcarbonimidoyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C12H11ClN2OS2
5-[N-[(4-chlorophenyl)methyl]-C-methylcarbonimidoyl]-2-sulfanylidene-1,3-thiazolidin-4-one