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—— 5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(4-ethylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H28N4O2S
5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(4-ethylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3,4-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O3S+
5-[(R)-(3,4-dimethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,4-dichlorophenyl)-piperidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H21Cl2N4OS+
5-[(S)-(2,4-dichlorophenyl)-piperidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-ethoxyphenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H31N5O2S+2
5-[(S)-(4-ethoxyphenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-chlorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H22ClN5OS
5-[(R)-(2-chlorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(3,4-difluorophenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H25F2N4OS+
5-[(R)-(3,4-difluorophenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H26ClN5O2S+2
5-[(S)-(3-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(4-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H24FN4O3S+
5-[(R)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(4-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3-chlorophenyl)-morpholin-4-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H19ClN4O2S
5-[(R)-(3-chlorophenyl)-morpholin-4-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-dichlorophenyl)-piperidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H20Cl2N4OS
5-[(S)-(3,4-dichlorophenyl)-piperidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(2-chlorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24ClN4OS+
5-[(S)-(2-chlorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-thiophen-2-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H25N4OS2+
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-thiophen-2-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-methylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4OS+
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-methylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-carbamoylpiperidin-1-ium-1-yl)-(4-methoxyphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H25N5O3S
5-[(R)-(4-carbamoylpiperidin-1-ium-1-yl)-(4-methoxyphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(3,4-difluorophenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25F2N5OS+2
5-[(S)-(3,4-difluorophenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-difluorophenyl)-morpholin-4-ium-4-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H19F2N4O2S+
5-[(S)-(3,4-difluorophenyl)-morpholin-4-ium-4-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-chlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H23ClN4OS
5-[(S)-(4-chlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-[(3R,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-methylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4OS+
5-[(R)-[(3R,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-methylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-thiophen-2-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H25N4OS2+
5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-thiophen-2-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl(phenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H24N4O3S
5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl(phenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(4-methylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O2S
5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(4-methylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-chlorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5OS
5-[(S)-(2-chlorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H26ClN5O2S+2
5-[(S)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-benzylpiperidin-1-ium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C23H27N4O2S+
5-[(R)-(4-benzylpiperidin-1-ium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(2-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H24FN4O3S+
5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(2-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-(4-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H23FN4O2S
5-[(R)-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-(4-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-chlorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H22ClN5OS
5-[(R)-(4-chlorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(3-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H26ClN5O2S+2
5-[(R)-(3-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-benzylpiperidin-1-ium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C23H27N4O2S+
5-[(S)-(4-benzylpiperidin-1-ium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(3R,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H24N4O2S
5-[(R)-[(3R,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-methoxyphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O2S+
5-[(R)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-methoxyphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-chlorophenyl)-[(3R,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H25ClN4OS
5-[(R)-(2-chlorophenyl)-[(3R,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(4-ethylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O2S+
5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(4-ethylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3-chlorophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C17H19ClN4OS
5-[(R)-(3-chlorophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(3-chlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H23ClN4OS
5-[(S)-(3-chlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(4-Nitrophenyl)methoxy]-2-(1,2,3,4-tetrahydroisoquinolin-2-ium-2-ylmethyl)pyran-4-one —— C22H21N2O5+
5-[(4-Nitrophenyl)methoxy]-2-(1,2,3,4-tetrahydroisoquinolin-2-ium-2-ylmethyl)pyran-4-one
—— 5-[(R)-(2-chlorophenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H25ClN4OS
5-[(R)-(2-chlorophenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(3,4-difluorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H23F2N4OS+
5-[(R)-(3,4-difluorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(3-Fluorophenyl)methoxy]-2-[[4-(furan-2-carbonyl)piperazin-1-ium-1-yl]methyl]pyran-4-one —— C22H22FN2O5+
5-[(3-Fluorophenyl)methoxy]-2-[[4-(furan-2-carbonyl)piperazin-1-ium-1-yl]methyl]pyran-4-one
—— 5-[(R)-(4-bromophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H20BrN4OS+
5-[(R)-(4-bromophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3,4-difluorophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C17H18F2N4OS
5-[(R)-(3,4-difluorophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethoxy]-2-(1,2,3,4-tetrahydroisoquinolin-2-ium-2-ylmethyl)pyran-4-one —— C23H29N2O5+
5-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethoxy]-2-(1,2,3,4-tetrahydroisoquinolin-2-ium-2-ylmethyl)pyran-4-one
—— 5-[2-(2,3-Dihydroindol-1-yl)-2-oxoethoxy]-2-(1,2,3,4-tetrahydroisoquinolin-2-ium-2-ylmethyl)pyran-4-one —— C25H25N2O4+
5-[2-(2,3-Dihydroindol-1-yl)-2-oxoethoxy]-2-(1,2,3,4-tetrahydroisoquinolin-2-ium-2-ylmethyl)pyran-4-one
—— 5-(2-Morpholin-4-yl-2-oxoethoxy)-2-(1,2,3,4-tetrahydroisoquinolin-2-ium-2-ylmethyl)pyran-4-one —— C21H25N2O5+
5-(2-Morpholin-4-yl-2-oxoethoxy)-2-(1,2,3,4-tetrahydroisoquinolin-2-ium-2-ylmethyl)pyran-4-one
—— (5-acetyl-2-methoxyphenyl)methyl 3-oxo-4H-1,4-benzothiazine-6-carboxylate —— C19H17NO5S
(5-acetyl-2-methoxyphenyl)methyl 3-oxo-4H-1,4-benzothiazine-6-carboxylate
—— 5,6-Dihydro-1,4-dioxin-2-yl[4-(6-ethyl-1,3-benzothiazol-2-yl)piperazino]methanone —— C18H21N3O3S
5,6-Dihydro-1,4-dioxin-2-yl[4-(6-ethyl-1,3-benzothiazol-2-yl)piperazino]methanone
—— [5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]methyl 5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylate —— C20H20N2O6S
[5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]methyl 5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylate
—— 5-(4-methoxyphenyl)-2-methyl-N-(2-methylpropyl)-1-phenylpyrrole-3-carboxamide —— C23H26N2O2
5-(4-methoxyphenyl)-2-methyl-N-(2-methylpropyl)-1-phenylpyrrole-3-carboxamide
—— 5-methyl-2-[(1R)-1-thiophen-2-ylethyl]pyrazol-3-amine —— C10H13N3S
5-methyl-2-[(1R)-1-thiophen-2-ylethyl]pyrazol-3-amine
—— (5E)-5-(3-bromo-4-methoxybenzylidene)-1-methyl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione —— C13H11BrN2O3S
(5E)-5-(3-bromo-4-methoxybenzylidene)-1-methyl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione