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—— (5R)-3-(2-furyl)-3-(imidazol-1-ylmethyl)-5-[(4-methoxyphenoxy)methyl]-2-methyl-isoxazolidine —— C20H23N3O4
(5R)-3-(2-furyl)-3-(imidazol-1-ylmethyl)-5-[(4-methoxyphenoxy)methyl]-2-methyl-isoxazolidine
—— (5R,7R)-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-3-(4-methoxyphenyl)adamantane-1-carboxamide —— C27H31NO3
(5R,7R)-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-3-(4-methoxyphenyl)adamantane-1-carboxamide
—— (5S,7S)-3-(4-methoxyphenyl)-N-(2-thiophen-2-ylethyl)adamantane-1-carboxamide —— C24H29NO2S
(5S,7S)-3-(4-methoxyphenyl)-N-(2-thiophen-2-ylethyl)adamantane-1-carboxamide
—— (5S,7S)-3-(4-methoxyphenyl)-N-[4-(pyrrolidin-1-ylmethyl)-1,3-thiazol-2-yl]adamantane-1-carboxamide —— C26H33N3O2S
(5S,7S)-3-(4-methoxyphenyl)-N-[4-(pyrrolidin-1-ylmethyl)-1,3-thiazol-2-yl]adamantane-1-carboxamide
—— 5-(benzyloxy)-1-methyl-4-oxo-N-phenyl-1,4-dihydropyridine-2-carboxamide —— C20H18N2O3
5-(benzyloxy)-1-methyl-4-oxo-N-phenyl-1,4-dihydropyridine-2-carboxamide
—— (5S,7S)-N-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-(4-methoxyphenyl)adamantane-1-carboxamide —— C28H33NO4
(5S,7S)-N-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-(4-methoxyphenyl)adamantane-1-carboxamide
—— 5-[[3-(phenylmethoxy)-4-(2-phenylethoxy)phenyl]methylene]-4-oxo-2-thioxo-3-thiazolidineacetic acid —— C27H23NO5S2
5-[[3-(phenylmethoxy)-4-(2-phenylethoxy)phenyl]methylene]-4-oxo-2-thioxo-3-thiazolidineacetic acid
—— 5-[(2S)-2-(benzotriazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H17FN6O
5-[(2S)-2-(benzotriazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R,7R)-N-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-(4-methoxyphenyl)adamantane-1-carboxamide —— C28H33NO4
(5R,7R)-N-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-(4-methoxyphenyl)adamantane-1-carboxamide
—— (5Z)-5-[[3-(4-butoxy-3-methylphenyl)-1-phenylpyrazol-4-yl]methylidene]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H31N3O3S2
(5Z)-5-[[3-(4-butoxy-3-methylphenyl)-1-phenylpyrazol-4-yl]methylidene]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[(E)-2-bromoethenyl]-1-[(2R,4R,5S)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidine-2,4-dione —— C11H13BrN2O5
5-[(E)-2-bromoethenyl]-1-[(2R,4R,5S)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidine-2,4-dione
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N6O3
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— {5-[1-{3-Benzyloxy-4-[2-(4-trifluoromethoxy-phenyl)-ethoxy]-phenyl}-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid —— C28H22F3NO6S2
{5-[1-{3-Benzyloxy-4-[2-(4-trifluoromethoxy-phenyl)-ethoxy]-phenyl}-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid
—— 5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N6O
5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-fluoro-1-isopropylsulfonyl-6-[(E)-1-phenylbut-1-en-3-ynyl]benzimidazol-2-amine —— C20H18FN3O2S
5-fluoro-1-isopropylsulfonyl-6-[(E)-1-phenylbut-1-en-3-ynyl]benzimidazol-2-amine
—— 5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19FN6O
5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S,7S)-3-(4-methoxyphenyl)-N-[(3-methoxyphenyl)methyl]-N-methyladamantane-1-carboxamide —— C27H33NO3
(5S,7S)-3-(4-methoxyphenyl)-N-[(3-methoxyphenyl)methyl]-N-methyladamantane-1-carboxamide
—— 5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H20N4O3S
5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H22N4O3
5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5E)-3-amino-5-[(4-fluorophenyl)methylene]-2-thioxo-thiazolidin-4-one —— C10H7FN2OS2
(5E)-3-amino-5-[(4-fluorophenyl)methylene]-2-thioxo-thiazolidin-4-one
—— 5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H20N4O3S
5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S,7S)-3-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]adamantane-1-carboxamide —— C26H31NO3
(5S,7S)-3-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]adamantane-1-carboxamide
—— 5-nitro-2-[(E)-2-(5-nitro-2-furyl)vinyl]thiazole —— C9H5N3O5S
5-nitro-2-[(E)-2-(5-nitro-2-furyl)vinyl]thiazole
—— [(5R,7R)-3-(4-methoxyphenyl)-1-adamantyl]-(4-pyrimidin-2-ylpiperazin-1-yl)methanone —— C26H32N4O2
[(5R,7R)-3-(4-methoxyphenyl)-1-adamantyl]-(4-pyrimidin-2-ylpiperazin-1-yl)methanone
—— (5R,7R)-3-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]adamantane-1-carboxamide —— C26H31NO3
(5R,7R)-3-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]adamantane-1-carboxamide
—— 5-Hydroxy-8-(3-hydroxy-2,5-dimethoxy-phenyl)-2,2-dimethyl-pyrano[3,2-g]chromen-6-one —— C22H20O7
5-Hydroxy-8-(3-hydroxy-2,5-dimethoxy-phenyl)-2,2-dimethyl-pyrano[3,2-g]chromen-6-one
—— 5-Styryl-pyrimidine-2,4-diamine —— C12H12N4
5-Styryl-pyrimidine-2,4-diamine
—— 5-[1,1-Dioxo-2-[4-((E)-styryl)-benzyl]-2,3-dihydro-1H-1λ<sup>6</sup>-benzo[e][1,2]thiazin-(4E)-ylidene]-thiazolidine-2,4-dione —— C26H20N2O4S2
5-[1,1-Dioxo-2-[4-((E)-styryl)-benzyl]-2,3-dihydro-1H-1λ<sup>6</sup>-benzo[e][1,2]thiazin-(4E)-ylidene]-thiazolidine-2,4-dione
—— 5-Allylpyrido[3,4-b][1,4]benzothiazine; fumaric acid —— C18H16N2O4S
5-Allylpyrido[3,4-b][1,4]benzothiazine; fumaric acid
—— 5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-ethyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N6O
5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-ethyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R)-3-amino-5-(5-methylthiophen-2-yl)cyclohex-2-en-1-one —— C11H13NOS
(5R)-3-amino-5-(5-methylthiophen-2-yl)cyclohex-2-en-1-one
—— (5S,7S)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-(4-methoxyphenyl)adamantane-1-carboxamide —— C22H27N3O2S
(5S,7S)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-(4-methoxyphenyl)adamantane-1-carboxamide
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19FN6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H20N6OS
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-ethyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-ethyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[[2-(4-chlorophenyl)benzimidazol-1-yl]methyl]-N-phenyl-1,3,4-thiadiazol-2-amine —— C22H16ClN5S
5-[[2-(4-chlorophenyl)benzimidazol-1-yl]methyl]-N-phenyl-1,3,4-thiadiazol-2-amine
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H20N4O3S
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19ClN4O2
5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H20N4O3
5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H20N4O3
5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N6O3
5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-4-[(E)-prop-1-enyl]-2-(3-pyridylmethylamino)phenol —— C16H18N2O
5-methyl-4-[(E)-prop-1-enyl]-2-(3-pyridylmethylamino)phenol
—— 5-[(1S)-1-(2-methoxyphenoxy)ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H19N3O3
5-[(1S)-1-(2-methoxyphenoxy)ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-((E)-2-Chloro-vinyl)-1-((2S,4S)-2-hydroxymethyl-[1,3]dioxolan-4-yl)-1H-pyrimidine-2,4-dione —— C10H11ClN2O5
5-((E)-2-Chloro-vinyl)-1-((2S,4S)-2-hydroxymethyl-[1,3]dioxolan-4-yl)-1H-pyrimidine-2,4-dione
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H24N4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— {5-[1-[3-Benzyloxy-4-(3-phenyl-propoxy)-phenyl]-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid —— C28H25NO5S2
{5-[1-[3-Benzyloxy-4-(3-phenyl-propoxy)-phenyl]-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid
—— (5S)-3-amino-5-(5-methylthiophen-2-yl)cyclohex-2-en-1-one —— C11H13NOS
(5S)-3-amino-5-(5-methylthiophen-2-yl)cyclohex-2-en-1-one