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—— (5E)-3-(butan-2-yl)-5-[4-(morpholin-4-yl)benzylidene]-1,3-thiazolidine-2,4-dione —— C18H22N2O3S
(5E)-3-(butan-2-yl)-5-[4-(morpholin-4-yl)benzylidene]-1,3-thiazolidine-2,4-dione
—— (5Z)-5-{5-bromo-2-[(4-fluorobenzyl)oxy]benzylidene}-2-thioxo-1,3-thiazolidin-4-one —— C17H11BrFNO2S2
(5Z)-5-{5-bromo-2-[(4-fluorobenzyl)oxy]benzylidene}-2-thioxo-1,3-thiazolidin-4-one
—— (5E)-2-(2,6-dimethylmorpholin-4-yl)-5-[[1-phenyl-3-(4-prop-2-enoxyphenyl)pyrazol-4-yl]methylidene]-1,3-thiazol-4-one —— C28H28N4O3S
(5E)-2-(2,6-dimethylmorpholin-4-yl)-5-[[1-phenyl-3-(4-prop-2-enoxyphenyl)pyrazol-4-yl]methylidene]-1,3-thiazol-4-one
—— 5-[(2R)-1-[(3,4-dimethylphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H33N5O2
5-[(2R)-1-[(3,4-dimethylphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(2-methylphenyl)methyl]piperidin-2-yl]-11-prop-2-enoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H29N5O2
5-[(2R)-1-[(2-methylphenyl)methyl]piperidin-2-yl]-11-prop-2-enoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-butanoylpiperidin-2-yl]-11-(cyclobutanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H31N5O3
5-[(2R)-1-butanoylpiperidin-2-yl]-11-(cyclobutanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-fluoro-N-[(Z)-[6-[[(5S)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl]-4,7-dimethoxy-1,3-benzodioxol-5-yl]methylideneamino]-1H-indole-2-carboxamide —— C29H24F2N4O6
5-fluoro-N-[(Z)-[6-[[(5S)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl]-4,7-dimethoxy-1,3-benzodioxol-5-yl]methylideneamino]-1H-indole-2-carboxamide
—— 5-[(2S)-1-butanoylpiperidin-2-yl]-11-(cyclopentanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[(2S)-1-butanoylpiperidin-2-yl]-11-(cyclopentanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-(4-ethoxyphenyl)-3-hydroxy-1-(2-methoxyethyl)-4-{[3-methyl-4-(2-methylpropoxy)phenyl]carbonyl}-1,5-dihydro-2H-pyrrol-2-one —— C27H33NO6
5-(4-ethoxyphenyl)-3-hydroxy-1-(2-methoxyethyl)-4-{[3-methyl-4-(2-methylpropoxy)phenyl]carbonyl}-1,5-dihydro-2H-pyrrol-2-one
—— 5-[(2S)-1-[(3-hydroxyphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O3
5-[(2S)-1-[(3-hydroxyphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(2-Hydroxyacetyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C19H25N5O4
5-[1-(2-Hydroxyacetyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[(2R)-2-hydroxypropanoyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H27N5O4
5-[1-[(2R)-2-hydroxypropanoyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(2-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H33N5O2
5-[(2R)-1-[(2-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(3-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H33N5O2
5-[(2S)-1-[(3-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(3-hydroxyphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O3
5-[(2R)-1-[(3-hydroxyphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-fluoro-N-[(Z)-[6-[[(5R)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl]-4,7-dimethoxy-1,3-benzodioxol-5-yl]methylideneamino]-1H-indole-2-carboxamide —— C29H24F2N4O6
5-fluoro-N-[(Z)-[6-[[(5R)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl]-4,7-dimethoxy-1,3-benzodioxol-5-yl]methylideneamino]-1H-indole-2-carboxamide
—— 5-[(2R)-1-butanoylpiperidin-2-yl]-11-prop-2-enoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C21H27N5O3
5-[(2R)-1-butanoylpiperidin-2-yl]-11-prop-2-enoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-benzylpiperidin-2-yl]-11-(cyclobutanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H31N5O2
5-[(2R)-1-benzylpiperidin-2-yl]-11-(cyclobutanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[(1S)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H31N5O3
5-[1-[(1S)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-(cyclopropanecarbonyl)piperidin-2-yl]-11-(3-methoxypropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H29N5O4
5-[(2S)-1-(cyclopropanecarbonyl)piperidin-2-yl]-11-(3-methoxypropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-butanoylpiperidin-2-yl]-11-(cyclobutanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H31N5O3
5-[(2S)-1-butanoylpiperidin-2-yl]-11-(cyclobutanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(3,4-dimethylphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H33N5O2
5-[(2S)-1-[(3,4-dimethylphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5Z)-5-[(4-ethoxyphenyl)methylidene]-3-phenyl-2-sulfanylideneimidazolidin-4-one —— C18H16N2O2S
(5Z)-5-[(4-ethoxyphenyl)methylidene]-3-phenyl-2-sulfanylideneimidazolidin-4-one
—— 5-[(2R)-1-(cyclopropanecarbonyl)piperidin-2-yl]-11-(3-methoxypropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H29N5O4
5-[(2R)-1-(cyclopropanecarbonyl)piperidin-2-yl]-11-(3-methoxypropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-benzoylpiperidin-2-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H27N5O3
5-[(2S)-1-benzoylpiperidin-2-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-benzylpiperidin-2-yl]-11-(cyclobutanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H31N5O2
5-[(2S)-1-benzylpiperidin-2-yl]-11-(cyclobutanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-cyclohexylpiperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H35N5O2
5-[(2R)-1-cyclohexylpiperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-benzoylpiperidin-2-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H27N5O3
5-[(2R)-1-benzoylpiperidin-2-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(4-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H33N5O2
5-[(2R)-1-[(4-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-acetylpiperidin-2-yl]-11-butanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H27N5O3
5-[(2S)-1-acetylpiperidin-2-yl]-11-butanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-acetylpiperidin-2-yl]-11-butanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H27N5O3
5-[(2R)-1-acetylpiperidin-2-yl]-11-butanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(4-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H33N5O2
5-[(2S)-1-[(4-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(2-Ethylbutanoyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H33N5O3
5-[1-(2-Ethylbutanoyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(2-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H33N5O2
5-[(2S)-1-[(2-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(3-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H33N5O2
5-[(2R)-1-[(3-methylphenyl)methyl]piperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-benzylpiperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O2
5-[(2R)-1-benzylpiperidin-2-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5Z)-5-[(2,5-dimethyl-1-phenylpyrrol-3-yl)methylidene]-3-phenyl-1,3-thiazolidine-2,4-dione —— C22H18N2O2S
(5Z)-5-[(2,5-dimethyl-1-phenylpyrrol-3-yl)methylidene]-3-phenyl-1,3-thiazolidine-2,4-dione
—— 5-[(2S)-1-cyclohexylpiperidin-2-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O2
5-[(2S)-1-cyclohexylpiperidin-2-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-cyclohexylpiperidin-2-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O2
5-[(2R)-1-cyclohexylpiperidin-2-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[(1R)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H31N5O3
5-[1-[(1R)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[(2S)-2-hydroxypropanoyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H27N5O4
5-[1-[(2S)-2-hydroxypropanoyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(2-Methylpropanoyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C21H29N5O3
5-[1-(2-Methylpropanoyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H29N5O4
5-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[2-[(1S)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H31N5O3
5-[1-[2-[(1S)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H31N5O3
5-[1-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H29N5O4
5-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O3
5-[1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-(1-Benzylpiperidin-4-yl)-11-butanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O2
5-(1-Benzylpiperidin-4-yl)-11-butanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(2-Cyclopentylacetyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[1-(2-Cyclopentylacetyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(Cyclopentanecarbonyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H31N5O3
5-[1-(Cyclopentanecarbonyl)piperidin-4-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one