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—— 5-chloro-2-hydroxy-N'-[(1E)-1-(2-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)ethyl]benzohydrazide —— C15H13ClN2O4
5-chloro-2-hydroxy-N'-[(1E)-1-(2-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)ethyl]benzohydrazide
—— (5E)-2-(2,6-dimethylmorpholin-4-yl)-5-[[3-[3-methyl-4-(3-methylbutoxy)phenyl]-1-phenylpyrazol-4-yl]methylidene]-1,3-thiazol-4-one —— C31H36N4O3S
(5E)-2-(2,6-dimethylmorpholin-4-yl)-5-[[3-[3-methyl-4-(3-methylbutoxy)phenyl]-1-phenylpyrazol-4-yl]methylidene]-1,3-thiazol-4-one
—— (5S,7S)-3-(3-nitro-1,2,4-triazol-1-yl)-N-(2-phenylsulfanylphenyl)adamantane-1-carboxamide —— C25H25N5O3S
(5S,7S)-3-(3-nitro-1,2,4-triazol-1-yl)-N-(2-phenylsulfanylphenyl)adamantane-1-carboxamide
—— (5E)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H28FN5O3S2
(5E)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-3-[(2-fluorophenyl)methyl]-5-[[1-(4-fluorophenyl)pyrrol-2-yl]methylidene]imidazolidine-2,4-dione —— C21H15F2N3O2
(5E)-3-[(2-fluorophenyl)methyl]-5-[[1-(4-fluorophenyl)pyrrol-2-yl]methylidene]imidazolidine-2,4-dione
—— (5E)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[7-methyl-2-(octylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C25H32N4O4S3
(5E)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[7-methyl-2-(octylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-(3,4-dimethylphenyl)-5-[(5-ethylthiophen-2-yl)methylidene]-1-methyl-2-sulfanylideneimidazolidin-4-one —— C19H20N2OS2
(5Z)-3-(3,4-dimethylphenyl)-5-[(5-ethylthiophen-2-yl)methylidene]-1-methyl-2-sulfanylideneimidazolidin-4-one
—— (5R,7R)-3-(3-chloro-1,2,4-triazol-1-yl)-N-(1-ethylbenzimidazol-2-yl)adamantane-1-carboxamide —— C22H25ClN6O
(5R,7R)-3-(3-chloro-1,2,4-triazol-1-yl)-N-(1-ethylbenzimidazol-2-yl)adamantane-1-carboxamide
—— (5S,7S)-N-(4-phenylmethoxyphenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C26H28N4O2
(5S,7S)-N-(4-phenylmethoxyphenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5R,7R)-N-[(4-sulfamoylphenyl)methyl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C20H25N5O3S
(5R,7R)-N-[(4-sulfamoylphenyl)methyl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5E)-3-Methyl-5-{[3-(4-methylphenyl)-1-phenyl-1H-pyrazol-4-YL]methylene}-2-thioxo-1,3-thiazolidin-4-one —— C21H17N3OS2
(5E)-3-Methyl-5-{[3-(4-methylphenyl)-1-phenyl-1H-pyrazol-4-YL]methylene}-2-thioxo-1,3-thiazolidin-4-one
—— [(5S,7S)-3-(5-bromo-3-nitro-1,2,4-triazol-1-yl)-1-adamantyl]-(4-methylpiperazin-1-yl)methanone —— C18H25BrN6O3
[(5S,7S)-3-(5-bromo-3-nitro-1,2,4-triazol-1-yl)-1-adamantyl]-(4-methylpiperazin-1-yl)methanone
—— (5,7-dibromoquinolin-8-yl) (1S,4S)-4,7,7-trimethyl-3-oxobicyclo[2.2.1]heptane-1-carboxylate —— C20H19Br2NO3
(5,7-dibromoquinolin-8-yl) (1S,4S)-4,7,7-trimethyl-3-oxobicyclo[2.2.1]heptane-1-carboxylate
—— (5Z)-5-[[2-(4-benzylpiperidin-1-yl)-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(2R)-butan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H32N4O2S2
(5Z)-5-[[2-(4-benzylpiperidin-1-yl)-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(2R)-butan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[2-(4-methoxyphenyl)ethyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H28N4O4S2
(5Z)-5-[[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[2-(4-methoxyphenyl)ethyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-{[5-(2,4-dichloro-5-nitrophenyl)furan-2-yl]methylidene}-3-phenyl-1,3-thiazolidine-2,4-dione —— C20H10Cl2N2O5S
(5Z)-5-{[5-(2,4-dichloro-5-nitrophenyl)furan-2-yl]methylidene}-3-phenyl-1,3-thiazolidine-2,4-dione
—— (5S,7S)-N-(2-methylsulfanylphenyl)-3-(3-nitro-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C20H23N5O3S
(5S,7S)-N-(2-methylsulfanylphenyl)-3-(3-nitro-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5S,7S)-N-(3,5-dimethoxyphenyl)-3-(3-nitro-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C21H25N5O5
(5S,7S)-N-(3,5-dimethoxyphenyl)-3-(3-nitro-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5Z)-5-[[2-(4-benzylpiperidin-1-yl)-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(2S)-butan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H32N4O2S2
(5Z)-5-[[2-(4-benzylpiperidin-1-yl)-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(2S)-butan-2-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[5-(4-acetylphenyl)furan-2-yl]methylidene]-1-[(2S)-2-hydroxypropyl]-4-methyl-2,6-dioxopyridine-3-carbonitrile —— C23H20N2O5
(5E)-5-[[5-(4-acetylphenyl)furan-2-yl]methylidene]-1-[(2S)-2-hydroxypropyl]-4-methyl-2,6-dioxopyridine-3-carbonitrile
—— (5R,7R)-N-(3-chloro-4-methylphenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C20H23ClN4O
(5R,7R)-N-(3-chloro-4-methylphenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5S,7S)-3-(3-nitro-1,2,4-triazol-1-yl)-N-(1,2-oxazol-3-yl)adamantane-1-carboxamide —— C16H18N6O4
(5S,7S)-3-(3-nitro-1,2,4-triazol-1-yl)-N-(1,2-oxazol-3-yl)adamantane-1-carboxamide
—— (5R,7R)-N-(2-methylsulfanylphenyl)-3-(3-nitro-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C20H23N5O3S
(5R,7R)-N-(2-methylsulfanylphenyl)-3-(3-nitro-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5Z)-3-Benzyl-5-{[5-(3-bromophenyl)furan-2-YL]methylidene}-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H14BrNO2S2
(5Z)-3-Benzyl-5-{[5-(3-bromophenyl)furan-2-YL]methylidene}-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R,7R)-N-[4-[acetyl(methyl)amino]phenyl]-3-(3-chloro-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C22H26ClN5O2
(5R,7R)-N-[4-[acetyl(methyl)amino]phenyl]-3-(3-chloro-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5R,7R)-3-(3-nitro-1,2,4-triazol-1-yl)-N-(1,2-oxazol-3-yl)adamantane-1-carboxamide —— C16H18N6O4
(5R,7R)-3-(3-nitro-1,2,4-triazol-1-yl)-N-(1,2-oxazol-3-yl)adamantane-1-carboxamide
—— (5E)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H28FN5O3S2
(5E)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,7S)-N-[4-[acetyl(methyl)amino]phenyl]-3-(3-chloro-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C22H26ClN5O2
(5S,7S)-N-[4-[acetyl(methyl)amino]phenyl]-3-(3-chloro-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— [(5R,7R)-3-(5-bromo-3-nitro-1,2,4-triazol-1-yl)-1-adamantyl]-(4-methylpiperazin-1-yl)methanone —— C18H25BrN6O3
[(5R,7R)-3-(5-bromo-3-nitro-1,2,4-triazol-1-yl)-1-adamantyl]-(4-methylpiperazin-1-yl)methanone
—— (5Z)-5-{[5-(4-Nitrophenyl)furan-2-YL]methylidene}-2-sulfanylidene-3-[3-(trifluoromethyl)phenyl]-1,3-thiazolidin-4-one —— C21H11F3N2O4S2
(5Z)-5-{[5-(4-Nitrophenyl)furan-2-YL]methylidene}-2-sulfanylidene-3-[3-(trifluoromethyl)phenyl]-1,3-thiazolidin-4-one
—— (5Z)-5-[[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[2-(4-methoxyphenyl)ethyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H28N4O4S2
(5Z)-5-[[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[2-(4-methoxyphenyl)ethyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-cyclohexyl-5-{2-[(4-fluorobenzyl)oxy]benzylidene}-2-thioxoimidazolidin-4-one —— C23H23FN2O2S
(5Z)-3-cyclohexyl-5-{2-[(4-fluorobenzyl)oxy]benzylidene}-2-thioxoimidazolidin-4-one
—— (5E)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[9-methyl-2-(octylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C25H32N4O4S3
(5E)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[9-methyl-2-(octylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,7S)-N-(2,5-difluorophenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C19H20F2N4O
(5S,7S)-N-(2,5-difluorophenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5Z)-3-[(dibutylamino)methyl]-5-[4-(diethylamino)benzylidene]-1,3-thiazolidine-2,4-dione —— C23H35N3O2S
(5Z)-3-[(dibutylamino)methyl]-5-[4-(diethylamino)benzylidene]-1,3-thiazolidine-2,4-dione
—— (5R,7R)-N-(3-morpholin-4-ylsulfonylphenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C23H29N5O4S
(5R,7R)-N-(3-morpholin-4-ylsulfonylphenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5E)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[2-[4-(2-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H24FN5O4S3
(5E)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[2-[4-(2-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,7S)-N-(6-methyl-1,3-benzothiazol-2-yl)-3-(3-nitro-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C21H22N6O3S
(5S,7S)-N-(6-methyl-1,3-benzothiazol-2-yl)-3-(3-nitro-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5E)-5-[(4-methoxynaphthalen-1-yl)methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H15NO2S2
(5E)-5-[(4-methoxynaphthalen-1-yl)methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[7-methyl-2-(octylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C25H32N4O4S3
(5E)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[7-methyl-2-(octylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[2-[4-(2-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H24FN5O4S3
(5E)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[2-[4-(2-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H26FN5O3S2
(5E)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H28FN5O3S2
(5E)-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-2-butanoyl-5-[(2S)-2-ethylsulfanylpropyl]-3-(hexylamino)cyclohex-2-en-1-one —— C21H37NO2S
(5S)-2-butanoyl-5-[(2S)-2-ethylsulfanylpropyl]-3-(hexylamino)cyclohex-2-en-1-one
—— (5S,7S)-3-(3-chloro-1,2,4-triazol-1-yl)-N-(1-ethylbenzimidazol-2-yl)adamantane-1-carboxamide —— C22H25ClN6O
(5S,7S)-3-(3-chloro-1,2,4-triazol-1-yl)-N-(1-ethylbenzimidazol-2-yl)adamantane-1-carboxamide
—— (5Z)-5-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methylidene]-3-(4-ethoxyphenyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H20ClN3O2S2
(5Z)-5-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methylidene]-3-(4-ethoxyphenyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-(1,3-benzodioxol-5-ylmethyl)-5-[[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H24N4O5S2
(5Z)-3-(1,3-benzodioxol-5-ylmethyl)-5-[[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-(1,3-benzodioxol-5-ylmethyl)-5-[[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H24N4O5S2
(5Z)-3-(1,3-benzodioxol-5-ylmethyl)-5-[[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H24FN5O4S3
(5E)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[2-[4-(4-fluorophenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-[(3-methylanilino)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C19H16N2O3S2
(5Z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-[(3-methylanilino)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one