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—— 5-[(1R)-1-[(4-methoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H25N5O2
5-[(1R)-1-[(4-methoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-N-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)cyclohexyl]methyl]pyrazine-2-carboxamide —— C22H26N6O
5-methyl-N-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)cyclohexyl]methyl]pyrazine-2-carboxamide
—— 5-[(1S)-1-[(3-methoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H25N5O2
5-[(1S)-1-[(3-methoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1R)-2-methyl-1-[(4-propan-2-yloxyphenyl)methylamino]propyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H29N5O2
5-[(1R)-2-methyl-1-[(4-propan-2-yloxyphenyl)methylamino]propyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-ethyl-4-methyl-N-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)cyclohexyl]methyl]-1H-pyrazole-3-carboxamide —— C23H30N6O
5-ethyl-4-methyl-N-[[4-(1-methyl-4-pyridin-4-ylpyrazol-3-yl)cyclohexyl]methyl]-1H-pyrazole-3-carboxamide
—— 5-[(1R)-1-[(3-fluorophenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H22FN5O
5-[(1R)-1-[(3-fluorophenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1R)-1-[(3-methoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H25N5O2
5-[(1R)-1-[(3-methoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1R)-1-[(4-fluorophenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H22FN5O
5-[(1R)-1-[(4-fluorophenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1R)-1-[(3,4-dimethoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H27N5O3
5-[(1R)-1-[(3,4-dimethoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1S)-1-[(4-fluorophenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H22FN5O
5-[(1S)-1-[(4-fluorophenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1S)-1-[(4-methoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H25N5O2
5-[(1S)-1-[(4-methoxyphenyl)methylamino]-2-methylpropyl]-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5Z)-3-[4-(4-chlorophenoxy)phenyl]-5-(1H-indol-2-ylmethylidene)-2-methylimidazol-4-one —— C25H18ClN3O2
(5Z)-3-[4-(4-chlorophenoxy)phenyl]-5-(1H-indol-2-ylmethylidene)-2-methylimidazol-4-one
—— (5Z)-3-[4-(4-fluorophenoxy)phenyl]-5-(1H-indol-2-ylmethylidene)-2-phenylimidazol-4-one —— C30H20FN3O2
(5Z)-3-[4-(4-fluorophenoxy)phenyl]-5-(1H-indol-2-ylmethylidene)-2-phenylimidazol-4-one
—— 5-ethyl-3-methyl-N-[[4-[1-methyl-4-(3-methyl-1,2-oxazol-5-yl)pyrazol-3-yl]cyclohexyl]methyl]-1,2-oxazole-4-carboxamide —— C22H29N5O3
5-ethyl-3-methyl-N-[[4-[1-methyl-4-(3-methyl-1,2-oxazol-5-yl)pyrazol-3-yl]cyclohexyl]methyl]-1,2-oxazole-4-carboxamide
—— [(5R,7R)-2,2-dichloroadamantane-1-carbonyl] (5S,7R)-2,2-dichloroadamantane-1-carboxylate —— C22H26Cl4O3
[(5R,7R)-2,2-dichloroadamantane-1-carbonyl] (5S,7R)-2,2-dichloroadamantane-1-carboxylate
—— 5-ethyl-3-methyl-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]cyclohexyl]methyl]-1,2-oxazole-4-carboxamide —— C23H29N5O3
5-ethyl-3-methyl-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]cyclohexyl]methyl]-1,2-oxazole-4-carboxamide
—— [(5R,7R)-2,2-dichloroadamantane-1-carbonyl] (5R,7R)-2,2-dichloroadamantane-1-carboxylate —— C22H26Cl4O3
[(5R,7R)-2,2-dichloroadamantane-1-carbonyl] (5R,7R)-2,2-dichloroadamantane-1-carboxylate
—— [(5R,7R)-2,2-dichloroadamantane-1-carbonyl] (5S,7S)-2,2-dichloroadamantane-1-carboxylate —— C22H26Cl4O3
[(5R,7R)-2,2-dichloroadamantane-1-carbonyl] (5S,7S)-2,2-dichloroadamantane-1-carboxylate
—— 5-ethyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]cyclohexyl]methyl]-1,2-oxazole-3-carboxamide —— C24H31N5O3
5-ethyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]cyclohexyl]methyl]-1,2-oxazole-3-carboxamide
—— 5-methoxy-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]cyclohexyl]methyl]thiophene-2-carboxamide —— C22H26N4O3S
5-methoxy-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]cyclohexyl]methyl]thiophene-2-carboxamide
—— 5-methyl-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]cyclohexyl]methyl]thiophene-3-carboxamide —— C22H26N4O2S
5-methyl-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]cyclohexyl]methyl]thiophene-3-carboxamide
—— 5-[(4-phenyl-1,3,5-triazin-2-yl)amino]-2-[(E)-2-[4-[(4-phenyl-1,3,5-triazin-2-yl)amino]-2-sulfophenyl]ethenyl]benzenesulfonic acid —— C32H24N8O6S2
5-[(4-phenyl-1,3,5-triazin-2-yl)amino]-2-[(E)-2-[4-[(4-phenyl-1,3,5-triazin-2-yl)amino]-2-sulfophenyl]ethenyl]benzenesulfonic acid
—— 5,6-dimethyl-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]cyclohexyl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C24H29N5O3
5,6-dimethyl-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]cyclohexyl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— 5-ethyl-2-[(3S)-1-[(2-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O2
5-ethyl-2-[(3S)-1-[(2-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5,6-dimethyl-2-[(3S)-1-[(2S)-2-phenylpropyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O
5,6-dimethyl-2-[(3S)-1-[(2S)-2-phenylpropyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R)-5-[(3,4-dimethoxyphenyl)methyl]-1-(4-methoxyphenyl)-5-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione —— C32H34N4O7
(5R)-5-[(3,4-dimethoxyphenyl)methyl]-1-(4-methoxyphenyl)-5-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-diazinane-2,4,6-trione
—— 5-ethyl-2-[(3R)-1-[(2-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O2
5-ethyl-2-[(3R)-1-[(2-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R,10bS)-7,9-dibromo-5-(3-fluorophenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Br2FN2O2
(5R,10bS)-7,9-dibromo-5-(3-fluorophenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-7,9-dibromo-5-(3-fluorophenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Br2FN2O2
(5R,10bR)-7,9-dibromo-5-(3-fluorophenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-7,9-dibromo-5-(3-fluorophenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H17Br2FN2O
(5S,10bR)-7,9-dibromo-5-(3-fluorophenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-7,9-dibromo-5-(2,4-dimethylphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C28H22Br2N2O
(5S,10bR)-7,9-dibromo-5-(2,4-dimethylphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-7,9-dibromo-5-(2,4-dimethylphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C28H22Br2N2O
(5S,10bS)-7,9-dibromo-5-(2,4-dimethylphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-9-bromo-5-(5-bromo-2-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Br2FN2O2
(5R,10bS)-9-bromo-5-(5-bromo-2-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-7,9-dibromo-5-(2-methoxyphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C27H20Br2N2O2
(5R,10bS)-7,9-dibromo-5-(2-methoxyphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-7,9-dibromo-5-(2-methoxyphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C27H20Br2N2O2
(5S,10bR)-7,9-dibromo-5-(2-methoxyphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-7,9-dibromo-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H13Br2ClN2OS
(5R,10bS)-7,9-dibromo-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-7,9-dibromo-5-(2-fluorophenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H17Br2FN2O
(5S,10bR)-7,9-dibromo-5-(2-fluorophenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-9-bromo-5-(3-bromo-4-methoxyphenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H20Br2N2O3
(5R,10bS)-9-bromo-5-(3-bromo-4-methoxyphenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-cyclopropyl-2-methyl-N-[[4-[2-methyl-5-(3-methylpyridin-4-yl)pyrimidin-4-yl]cyclohexyl]methyl]furan-3-carboxamide —— C27H32N4O2
5-cyclopropyl-2-methyl-N-[[4-[2-methyl-5-(3-methylpyridin-4-yl)pyrimidin-4-yl]cyclohexyl]methyl]furan-3-carboxamide
—— (5R,10bR)-9-bromo-5-(3-bromo-4-methoxyphenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H20Br2N2O3
(5R,10bR)-9-bromo-5-(3-bromo-4-methoxyphenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-9-bromo-5-(5-bromo-2-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Br2FN2O2
(5S,10bR)-9-bromo-5-(5-bromo-2-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-9-bromo-5-(5-bromo-2-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Br2FN2O2
(5R,10bR)-9-bromo-5-(5-bromo-2-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-9-bromo-5-(5-bromo-2-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Br2FN2O2
(5S,10bS)-9-bromo-5-(5-bromo-2-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-7,9-dibromo-5-(2-methoxyphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C27H20Br2N2O2
(5S,10bS)-7,9-dibromo-5-(2-methoxyphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-9-chloro-5-(2-chlorophenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H18Cl2N2O
(5S,10bS)-9-chloro-5-(2-chlorophenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-7,9-dibromo-5-(3,4-dimethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H18Br2N2O3S
(5R,10bS)-7,9-dibromo-5-(3,4-dimethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-7,9-dibromo-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H13Br2ClN2OS
(5S,10bS)-7,9-dibromo-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-9-chloro-5-(3-fluorophenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H15ClF2N2O
(5S,10bR)-9-chloro-5-(3-fluorophenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-7,9-dibromo-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H13Br2ClN2OS
(5R,10bR)-7,9-dibromo-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-7,9-dibromo-5-(3,4-dimethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H18Br2N2O3S
(5S,10bS)-7,9-dibromo-5-(3,4-dimethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine