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—— 5-[[3-[3-[(2R,4R,6S)-4-[(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C41H46N2O8
5-[[3-[3-[(2R,4R,6S)-4-[(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C37H37N5O7S
5-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[(1R,2S,3S,5S,6R,7S,9S,10S,11S)-11-bromo-8-pentacyclo[5.4.0.02,6.03,10.05,9]undecanylidene]-2,2-dimethyl-1,3-dioxane-4,6-dione —— C17H17BrO4
5-[(1R,2S,3S,5S,6R,7S,9S,10S,11S)-11-bromo-8-pentacyclo[5.4.0.02,6.03,10.05,9]undecanylidene]-2,2-dimethyl-1,3-dioxane-4,6-dione
—— 5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C37H39NO7S
5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C30H31N5O6S
5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C28H30N2O7S
5-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[4-[(2R,4R,6S)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C30H31N3O6
5-[4-[(2R,4R,6S)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C37H39NO7S
5-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-5-oxopentanoic acid —— C34H42N2O7
5-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C33H35N3O6S2
5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C29H31NO6S
5-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[(1R,2S,3S,5R,6R,7S,9R,10S,11S)-11-bromo-8-pentacyclo[5.4.0.02,6.03,10.05,9]undecanylidene]-2,2-dimethyl-1,3-dioxane-4,6-dione —— C17H17BrO4
5-[(1R,2S,3S,5R,6R,7S,9R,10S,11S)-11-bromo-8-pentacyclo[5.4.0.02,6.03,10.05,9]undecanylidene]-2,2-dimethyl-1,3-dioxane-4,6-dione
—— 5-[[2-[4-[(2R,4R,6S)-4-(azocan-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C37H46N2O6
5-[[2-[4-[(2R,4R,6S)-4-(azocan-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[3-[(2R,4R,6S)-4-(azocan-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C30H40N2O6
5-[3-[(2R,4R,6S)-4-(azocan-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C35H42N2O7
5-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[[3-[4-[(2R,4R,6S)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C38H46N2O6
5-[[3-[4-[(2R,4R,6S)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— (5R,6R)-5,6-dibromo-1,1,1-trichloro-6-phenylhexane-2,4-dione —— C12H9Br2Cl3O2
(5R,6R)-5,6-dibromo-1,1,1-trichloro-6-phenylhexane-2,4-dione
—— 5-[(1R,2S,3S,5R,6R,7S,9S,10S,11S)-11-bromo-8-pentacyclo[5.4.0.02,6.03,10.05,9]undecanylidene]-2,2-dimethyl-1,3-dioxane-4,6-dione —— C17H17BrO4
5-[(1R,2S,3S,5R,6R,7S,9S,10S,11S)-11-bromo-8-pentacyclo[5.4.0.02,6.03,10.05,9]undecanylidene]-2,2-dimethyl-1,3-dioxane-4,6-dione
—— 5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C28H30N2O7S
5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(pyridin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C35H36N2O6S
5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(pyridin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C30H38N2O8
5-[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[[2-[4-[(2R,4R,6S)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C37H37N3O6
5-[[2-[4-[(2R,4R,6S)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C26H30N4O6S
5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(morpholin-4-ylmethyl)-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C27H34N2O7
5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(morpholin-4-ylmethyl)-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C38H43N3O6
5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C34H40N2O6
5-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— 5-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C32H35N5O6S
5-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— (5S,7S)-1-bromo-3-[[(5R,7R)-3-bromo-1-adamantyl]-chlorophosphoryl]adamantane —— C20H28Br2ClOP
(5S,7S)-1-bromo-3-[[(5R,7R)-3-bromo-1-adamantyl]-chlorophosphoryl]adamantane
—— 5-[[2-[4-[(2R,4R,6S)-4-(2-hydroxyethylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C32H37NO7S
5-[[2-[4-[(2R,4R,6S)-4-(2-hydroxyethylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— (5S,6S)-5,6-dibromo-1,1,1-trichloro-6-phenylhexane-2,4-dione —— C12H9Br2Cl3O2
(5S,6S)-5,6-dibromo-1,1,1-trichloro-6-phenylhexane-2,4-dione
—— 5-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid —— C36H44N2O7
5-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-5-oxopentanoic acid
—— (5S,6R)-5,6-dibromo-1,1,1-trichloro-6-phenylhexane-2,4-dione —— C12H9Br2Cl3O2
(5S,6R)-5,6-dibromo-1,1,1-trichloro-6-phenylhexane-2,4-dione
—— 5-Tosyloxy-bicyclo<2.2.0>hept-2-en —— C14H16O3S
5-Tosyloxy-bicyclo<2.2.0>hept-2-en
—— (5S,7S)-1-bromo-3-[[(5S,7R)-3-bromo-1-adamantyl]-chlorophosphoryl]adamantane —— C20H28Br2ClOP
(5S,7S)-1-bromo-3-[[(5S,7R)-3-bromo-1-adamantyl]-chlorophosphoryl]adamantane
—— (5R,6S)-5,6-dibromo-1,1,1-trichloro-6-phenylhexane-2,4-dione —— C12H9Br2Cl3O2
(5R,6S)-5,6-dibromo-1,1,1-trichloro-6-phenylhexane-2,4-dione
—— (5S,7S)-1-bromo-3-[[(5S,7S)-3-bromo-1-adamantyl]-chlorophosphoryl]adamantane —— C20H28Br2ClOP
(5S,7S)-1-bromo-3-[[(5S,7S)-3-bromo-1-adamantyl]-chlorophosphoryl]adamantane
—— 5-chloro-2-methyl-3-[(1R,5R)-8-methyl-8-azabicyclo[3.2.1]oct-2-en-3-yl]-1H-indole —— C17H19ClN2
5-chloro-2-methyl-3-[(1R,5R)-8-methyl-8-azabicyclo[3.2.1]oct-2-en-3-yl]-1H-indole
—— 5-chloro-2-methyl-3-[(1S,5S)-8-methyl-8-azabicyclo[3.2.1]oct-2-en-3-yl]-1H-indole —— C17H19ClN2
5-chloro-2-methyl-3-[(1S,5S)-8-methyl-8-azabicyclo[3.2.1]oct-2-en-3-yl]-1H-indole
—— (5E)-1,6-dimethylcycloocta-1,3,5-triene —— C10H14
(5E)-1,6-dimethylcycloocta-1,3,5-triene
—— (5R,7R)-5,7-dichloro-1,11-dimethyl-5,7-dihydrobenzo[d][2]benzothiepine 6,6-dioxide —— C16H14Cl2O2S
(5R,7R)-5,7-dichloro-1,11-dimethyl-5,7-dihydrobenzo[d][2]benzothiepine 6,6-dioxide
—— (5S,7S)-5,7-dichloro-1,11-dimethyl-5,7-dihydrobenzo[d][2]benzothiepine 6,6-dioxide —— C16H14Cl2O2S
(5S,7S)-5,7-dichloro-1,11-dimethyl-5,7-dihydrobenzo[d][2]benzothiepine 6,6-dioxide
—— (5S,7S)-3-chloro-N-(6-methoxy-1,3-benzothiazol-2-yl)adamantane-1-carboxamide —— C19H21ClN2O2S
(5S,7S)-3-chloro-N-(6-methoxy-1,3-benzothiazol-2-yl)adamantane-1-carboxamide
—— (5R,7R)-3-chloro-N-(6-methoxy-1,3-benzothiazol-2-yl)adamantane-1-carboxamide —— C19H21ClN2O2S
(5R,7R)-3-chloro-N-(6-methoxy-1,3-benzothiazol-2-yl)adamantane-1-carboxamide
—— (5S,7S)-3-chloro-N-(4,5-dihydro-1,3-thiazol-2-yl)adamantane-1-carboxamide —— C14H19ClN2OS
(5S,7S)-3-chloro-N-(4,5-dihydro-1,3-thiazol-2-yl)adamantane-1-carboxamide
—— (5Z)-5-[[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H32N4O3S2
(5Z)-5-[[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,7R)-5,7-dichloro-1,11-dimethyl-5,7-dihydrobenzo[d][2]benzothiepine 6,6-dioxide —— C16H14Cl2O2S
(5S,7R)-5,7-dichloro-1,11-dimethyl-5,7-dihydrobenzo[d][2]benzothiepine 6,6-dioxide
—— 5-[[(5S,7S)-3-bromo-1-adamantyl]methyl]-3-(methoxymethyl)-1,2,4-oxadiazole —— C15H21BrN2O2
5-[[(5S,7S)-3-bromo-1-adamantyl]methyl]-3-(methoxymethyl)-1,2,4-oxadiazole
—— (5Z)-5-[[2-[[(2S)-2-hydroxy-2-phenylethyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C28H32N4O3S2
(5Z)-5-[[2-[[(2S)-2-hydroxy-2-phenylethyl]amino]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5RS)-(Z)-4-[5-(Furan-2-yl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-4-oxobut-2-enoic acid —— C17H14N2O4
(5RS)-(Z)-4-[5-(Furan-2-yl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-4-oxobut-2-enoic acid
—— 5-[[(5R,7R)-3-bromo-1-adamantyl]methyl]-3-(methoxymethyl)-1,2,4-oxadiazole —— C15H21BrN2O2
5-[[(5R,7R)-3-bromo-1-adamantyl]methyl]-3-(methoxymethyl)-1,2,4-oxadiazole