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—— [5-(5-chloro-4-ethoxy-2-methylphenyl)-2-methyl-1,2,4-triazol-3-yl]methanamine —— C13H17ClN4O
[5-(5-chloro-4-ethoxy-2-methylphenyl)-2-methyl-1,2,4-triazol-3-yl]methanamine
—— [5-(3-chloro-6-methoxy-2,4-dimethylphenyl)-2-methyl-1,2,4-triazol-3-yl]methanamine —— C13H17ClN4O
[5-(3-chloro-6-methoxy-2,4-dimethylphenyl)-2-methyl-1,2,4-triazol-3-yl]methanamine
—— (5R,7S)-5-(1,3-benzodioxol-5-yl)-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H20F3N5O3S
(5R,7S)-5-(1,3-benzodioxol-5-yl)-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-3-bromo-N-(furan-2-ylmethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H18BrF3N4O3
(5R,7S)-3-bromo-N-(furan-2-ylmethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H22F3N5O2S
(5R,7S)-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-oxo-4-(4-phenylphenyl)-1,2-dihydropyrazole-3-carboxylic acid —— C16H12N2O3
5-oxo-4-(4-phenylphenyl)-1,2-dihydropyrazole-3-carboxylic acid
—— [5-[(Z)-[(3-chlorobenzoyl)hydrazinylidene]methyl]-2-methoxyphenyl] benzoate —— C22H17ClN2O4
[5-[(Z)-[(3-chlorobenzoyl)hydrazinylidene]methyl]-2-methoxyphenyl] benzoate
—— (5R,7S)-N-[1-[(4-bromophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C26H24BrF3N6O
(5R,7S)-N-[1-[(4-bromophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(2-aminoethyl)-N-(3,4-dimethoxyphenyl)-1,3,4-thiadiazol-2-amine —— C12H16N4O2S
5-(2-aminoethyl)-N-(3,4-dimethoxyphenyl)-1,3,4-thiadiazol-2-amine
—— [(5S,7S)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-piperidin-1-ylmethanone —— C19H21F3N4O
[(5S,7S)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-piperidin-1-ylmethanone
—— 5-(3-chloro-4-methoxyphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-amine —— C11H9ClN4OS
5-(3-chloro-4-methoxyphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-amine
—— (5R,7S)-5-(1,3-benzodioxol-5-yl)-N-[(5-chloro-1H-indol-2-yl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H19ClF3N5O3
(5R,7S)-5-(1,3-benzodioxol-5-yl)-N-[(5-chloro-1H-indol-2-yl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(3-fluoro-4-propan-2-yloxyphenyl)thiophene-3-carboxylic acid —— C14H13FO3S
5-(3-fluoro-4-propan-2-yloxyphenyl)thiophene-3-carboxylic acid
—— (5S,7R)-5-(4-bromophenyl)-N-(thiophen-2-ylmethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H16BrF3N4OS
(5S,7R)-5-(4-bromophenyl)-N-(thiophen-2-ylmethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7R)-N-[4-[(1S)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-5-(3,4,5-trimethoxyphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H27F3N4O5
(5S,7R)-N-[4-[(1S)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-5-(3,4,5-trimethoxyphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [5-(4-ethylsulfonylphenyl)-2-methyl-1,2,4-triazol-3-yl]methanamine —— C12H16N4O2S
[5-(4-ethylsulfonylphenyl)-2-methyl-1,2,4-triazol-3-yl]methanamine
—— 5-(3-chloro-4-methoxyphenyl)-1,3-dimethylpyrazole-4-carboxylic acid —— C13H13ClN2O3
5-(3-chloro-4-methoxyphenyl)-1,3-dimethylpyrazole-4-carboxylic acid
—— (5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H24ClF3N6O3
(5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-7-(difluoromethyl)-N-(furan-2-ylmethyl)-5-(4-methylphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H20F2N4O2
(5S,7S)-7-(difluoromethyl)-N-(furan-2-ylmethyl)-5-(4-methylphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-[2-(1,2,4-benzotriazin-3-yl)ethyl]-2-methoxyaniline —— C16H16N4O
5-[2-(1,2,4-benzotriazin-3-yl)ethyl]-2-methoxyaniline
—— (5S,7R)-7-(difluoromethyl)-5-(4-methylphenyl)-N-[1-[(2-methylphenyl)methyl]pyrazol-4-yl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H26F2N6O
(5S,7R)-7-(difluoromethyl)-5-(4-methylphenyl)-N-[1-[(2-methylphenyl)methyl]pyrazol-4-yl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7S)-3-bromo-5-(5-bromofuran-2-yl)-7-(trifluoromethyl)-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H19Br2F3N6O2
(5S,7S)-3-bromo-5-(5-bromofuran-2-yl)-7-(trifluoromethyl)-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-[(5-chloro-1H-indol-2-yl)methyl]-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C25H23ClF3N5O3
(5R,7R)-N-[(5-chloro-1H-indol-2-yl)methyl]-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-3-bromo-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H17BrF3N5O2S
(5R,7S)-3-bromo-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-cyclohexyl-5-(3,4-dichlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H21Cl2F3N4O
(5R,7R)-N-cyclohexyl-5-(3,4-dichlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-methyl-5-phenyl-7-(trifluoromethyl)-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H25F3N6O
(5S,7S)-N-methyl-5-phenyl-7-(trifluoromethyl)-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7R)-N-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H28ClF3N6O3
(5R,7R)-N-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-5-(3,4-dimethoxyphenyl)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H25F3N6O3
(5R,7S)-5-(3,4-dimethoxyphenyl)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-N-[(1,3-dimethylpyrazol-4-yl)methyl]-N-methyl-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H25F3N6O
(5R,7S)-N-[(1,3-dimethylpyrazol-4-yl)methyl]-N-methyl-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [(5S,7R)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-piperidin-1-ylmethanone —— C19H21F3N4O
[(5S,7R)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-piperidin-1-ylmethanone
—— (5R,7S)-5-(1,3-benzodioxol-5-yl)-N-(2-methylsulfanylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H19F3N4O3S
(5R,7S)-5-(1,3-benzodioxol-5-yl)-N-(2-methylsulfanylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-5-(3,4-dimethoxyphenyl)-N-methyl-7-(trifluoromethyl)-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H29F3N6O3
(5S,7S)-5-(3,4-dimethoxyphenyl)-N-methyl-7-(trifluoromethyl)-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [5-(5-chloro-4-ethoxy-2-methylphenyl)-3-methyl-1,2-oxazol-4-yl]methanamine —— C14H17ClN2O2
[5-(5-chloro-4-ethoxy-2-methylphenyl)-3-methyl-1,2-oxazol-4-yl]methanamine
—— [5-(3-Chloro-6-methoxy-2,4-dimethylphenyl)-1-methylpyrazol-3-yl]methanamine —— C14H18ClN3O
[5-(3-Chloro-6-methoxy-2,4-dimethylphenyl)-1-methylpyrazol-3-yl]methanamine
—— [5-(3-chloro-4-propan-2-yloxyphenyl)-2-methyl-1,2,4-triazol-3-yl]methanamine —— C13H17ClN4O
[5-(3-chloro-4-propan-2-yloxyphenyl)-2-methyl-1,2,4-triazol-3-yl]methanamine
—— (5S,7R)-5-(3,4-dimethoxyphenyl)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H25F3N6O3
(5S,7R)-5-(3,4-dimethoxyphenyl)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7S)-3-bromo-N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H21BrF3N5O2S
(5R,7S)-3-bromo-N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-5-(1,3-benzodioxol-5-yl)-N-[(4-pyrazol-1-ylphenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C25H21F3N6O3
(5S,7S)-5-(1,3-benzodioxol-5-yl)-N-[(4-pyrazol-1-ylphenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-5-(4-bromophenyl)-3-chloro-N-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H19BrClF3N4O3
(5R,7R)-5-(4-bromophenyl)-3-chloro-N-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(4-methanesulfonylphenyl)-1-methyl-1H-pyrazole-4-carboxylic acid —— C12H12N2O4S
5-(4-methanesulfonylphenyl)-1-methyl-1H-pyrazole-4-carboxylic acid
—— 5-chloro-N-(2-hydroxyethyl)-4-methoxy-2-methylbenzenesulfonamide —— C10H14ClNO4S
5-chloro-N-(2-hydroxyethyl)-4-methoxy-2-methylbenzenesulfonamide
—— 5-chloro-N-(2-hydroxyethyl)-2-methoxy-3-methylbenzenesulfonamide —— C10H14ClNO4S
5-chloro-N-(2-hydroxyethyl)-2-methoxy-3-methylbenzenesulfonamide
—— [5-methyl-4-(4-phenylphenyl)thiophen-3-yl]methanamine —— C18H17NS
[5-methyl-4-(4-phenylphenyl)thiophen-3-yl]methanamine
—— (5Z)-5-[[5-(3-fluorophenyl)furan-2-yl]methylidene]-3-phenylimidazolidine-2,4-dione —— C20H13FN2O3
(5Z)-5-[[5-(3-fluorophenyl)furan-2-yl]methylidene]-3-phenylimidazolidine-2,4-dione
—— (5E)-3-benzyl-5-(3-hydroxy-4-methoxybenzylidene)imidazolidine-2,4-dione —— C18H16N2O4
(5E)-3-benzyl-5-(3-hydroxy-4-methoxybenzylidene)imidazolidine-2,4-dione
—— (5S)-5-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]-2,9-dimethyl-3,5-dihydropyrazolo[1,5-c]quinazoline —— C28H25N5O
(5S)-5-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]-2,9-dimethyl-3,5-dihydropyrazolo[1,5-c]quinazoline
—— (5Z)-5-[(3,4-dimethoxyphenyl)methylidene]-3-ethylimidazolidine-2,4-dione —— C14H16N2O4
(5Z)-5-[(3,4-dimethoxyphenyl)methylidene]-3-ethylimidazolidine-2,4-dione
—— 5-tert-butyl-N-(3-hydroxypropyl)-4-methoxy-2-methylbenzamide —— C16H25NO3
5-tert-butyl-N-(3-hydroxypropyl)-4-methoxy-2-methylbenzamide
—— (5E)-5-[(7-ethyl-1H-indol-3-yl)methylidene]-3-methyl-2-sulfanylideneimidazolidin-4-one —— C15H15N3OS
(5E)-5-[(7-ethyl-1H-indol-3-yl)methylidene]-3-methyl-2-sulfanylideneimidazolidin-4-one
—— [5-methyl-4-(4-phenoxyphenyl)-1H-imidazol-2-yl]methanamine —— C17H17N3O
[5-methyl-4-(4-phenoxyphenyl)-1H-imidazol-2-yl]methanamine