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—— (5S,10bS)-9-bromo-5-(3-bromo-4-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Br2FN2O2
(5S,10bS)-9-bromo-5-(3-bromo-4-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-7,9-dibromo-5-(2,3-dimethoxyphenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H22Br2N2O4
(5R,10bR)-7,9-dibromo-5-(2,3-dimethoxyphenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-7,9-dibromo-5-(3-fluorophenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H17Br2FN2O
(5S,10bS)-7,9-dibromo-5-(3-fluorophenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-7,9-dibromo-5-(3-nitrophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H13Br2N3O3S
(5S,10bS)-7,9-dibromo-5-(3-nitrophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-7,9-dibromo-5-(3,4-dimethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H18Br2N2O3S
(5R,10bR)-7,9-dibromo-5-(3,4-dimethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-9-bromo-5-(3-bromo-4-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Br2FN2O2
(5S,10bR)-9-bromo-5-(3-bromo-4-methoxyphenyl)-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,6R)-3-[(E)-2-acetamidoethenyl]sulfinyl-6-[(1S)-1-hydroxyethyl]-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid —— C13H16N2O6S
(5R,6R)-3-[(E)-2-acetamidoethenyl]sulfinyl-6-[(1S)-1-hydroxyethyl]-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
—— (5S,10bR)-7,9-dibromo-5-(3,4-dimethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H18Br2N2O3S
(5S,10bR)-7,9-dibromo-5-(3,4-dimethoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-propan-2-yl-N-[[4-(2-propan-2-yl-5-pyridin-4-ylpyrimidin-4-yl)cyclohexyl]methyl]-1,2-oxazole-3-carboxamide —— C26H33N5O2
5-propan-2-yl-N-[[4-(2-propan-2-yl-5-pyridin-4-ylpyrimidin-4-yl)cyclohexyl]methyl]-1,2-oxazole-3-carboxamide
—— (5S,10bR)-7,9-dibromo-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H13Br2ClN2OS
(5S,10bR)-7,9-dibromo-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-9-bromo-2-(3-methoxyphenyl)-5-propan-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H21BrN2O2
(5R,10bR)-9-bromo-2-(3-methoxyphenyl)-5-propan-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-methyl-N-[[4-[2-methyl-5-(3-methylpyridin-4-yl)pyrimidin-4-yl]cyclohexyl]methyl]thiophene-3-carboxamide —— C24H28N4OS
5-methyl-N-[[4-[2-methyl-5-(3-methylpyridin-4-yl)pyrimidin-4-yl]cyclohexyl]methyl]thiophene-3-carboxamide
—— (5S,10bR)-7,9-dibromo-5-(3-nitrophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H13Br2N3O3S
(5S,10bR)-7,9-dibromo-5-(3-nitrophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-7,9-dibromo-5-(2-methoxyphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C27H20Br2N2O2
(5R,10bR)-7,9-dibromo-5-(2-methoxyphenyl)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-ethyl-N-[[4-[2-methyl-5-(3-methylpyridin-4-yl)pyrimidin-4-yl]cyclohexyl]methyl]-1,2-oxazole-3-carboxamide —— C24H29N5O2
5-ethyl-N-[[4-[2-methyl-5-(3-methylpyridin-4-yl)pyrimidin-4-yl]cyclohexyl]methyl]-1,2-oxazole-3-carboxamide
—— (5S,10bR)-2-(4-chlorophenyl)-7-methoxy-5-(2-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H21ClN2O3
(5S,10bR)-2-(4-chlorophenyl)-7-methoxy-5-(2-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5,6-dimethyl-N-[[4-(2-methyl-5-pyridin-4-ylpyrimidin-4-yl)cyclohexyl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C25H29N5O2
5,6-dimethyl-N-[[4-(2-methyl-5-pyridin-4-ylpyrimidin-4-yl)cyclohexyl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (5S,10bS)-9-chloro-5-(2,4-dimethoxyphenyl)-2-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H23ClN2O4
(5S,10bS)-9-chloro-5-(2,4-dimethoxyphenyl)-2-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-9-chloro-2-(3-methoxyphenyl)-5-propan-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H21ClN2O2
(5R,10bR)-9-chloro-2-(3-methoxyphenyl)-5-propan-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-9-chloro-5-(2,4-dimethoxyphenyl)-2-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H23ClN2O4
(5S,10bR)-9-chloro-5-(2,4-dimethoxyphenyl)-2-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-7-methoxy-5-(2-methoxyphenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H22N2O3
(5S,10bR)-7-methoxy-5-(2-methoxyphenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— [5-[2-amino-8-[(Z)-(3,8-dimethyl-3aH-imidazo[4,5-f]quinoxalin-2-ylidene)amino]-6-oxo-1H-purin-9-yl]-2-(phosphonooxymethyl)oxolan-3-yl] dihydrogen phosphate —— C21H24N10O10P2
[5-[2-amino-8-[(Z)-(3,8-dimethyl-3aH-imidazo[4,5-f]quinoxalin-2-ylidene)amino]-6-oxo-1H-purin-9-yl]-2-(phosphonooxymethyl)oxolan-3-yl] dihydrogen phosphate
—— (5Z)-5-[[9-methyl-2-(2-morpholin-4-ylethylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(1S)-1-phenylethyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H29N5O3S2
(5Z)-5-[[9-methyl-2-(2-morpholin-4-ylethylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(1S)-1-phenylethyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[3-(4-bromophenyl)-1-phenylpyrazol-4-yl]methylidene]-3-[(3S)-1,1-dioxothiolan-3-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C23H18BrN3O3S3
(5E)-5-[[3-(4-bromophenyl)-1-phenylpyrazol-4-yl]methylidene]-3-[(3S)-1,1-dioxothiolan-3-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-1-[2-(diethylamino)ethyl]-4-[hydroxy-(2-methyl-4-prop-2-enoxyphenyl)methylidene]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C33H36N2O5
(5S)-1-[2-(diethylamino)ethyl]-4-[hydroxy-(2-methyl-4-prop-2-enoxyphenyl)methylidene]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— (5E,8Z,11Z,13Z)-15-hydroperoxyicosa-5,8,11,13-tetraenoic acid —— C20H32O4
(5E,8Z,11Z,13Z)-15-hydroperoxyicosa-5,8,11,13-tetraenoic acid
—— (5E)-5-[[3-(4-bromophenyl)-1-phenylpyrazol-4-yl]methylidene]-3-[(3R)-1,1-dioxothiolan-3-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C23H18BrN3O3S3
(5E)-5-[[3-(4-bromophenyl)-1-phenylpyrazol-4-yl]methylidene]-3-[(3R)-1,1-dioxothiolan-3-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[[9-methyl-2-(2-morpholin-4-ylethylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(1R)-1-phenylethyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H29N5O3S2
(5Z)-5-[[9-methyl-2-(2-morpholin-4-ylethylamino)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(1R)-1-phenylethyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-[2-(3,4-dimethoxyphenyl)ethyl]-5-[[4-oxo-2-[[(2R)-oxolan-2-yl]methylamino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H28N4O5S2
(5Z)-3-[2-(3,4-dimethoxyphenyl)ethyl]-5-[[4-oxo-2-[[(2R)-oxolan-2-yl]methylamino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,10bR)-7-methoxy-5-(4-methylphenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H22N2O2
(5S,10bR)-7-methoxy-5-(4-methylphenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5Z)-5-[(3aR,4R,5R,6aR)-4-[(E,3S)-3-hydroxyoct-1-enyl]-5-methoxy-3,3a,4,5,6,6a-hexahydrocyclopenta[b]furan-2-ylidene]pentanoic acid —— C21H34O5
(5Z)-5-[(3aR,4R,5R,6aR)-4-[(E,3S)-3-hydroxyoct-1-enyl]-5-methoxy-3,3a,4,5,6,6a-hexahydrocyclopenta[b]furan-2-ylidene]pentanoic acid
—— 5-(4-chloro-1-ethylpyrazol-3-yl)-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18ClN5O2
5-(4-chloro-1-ethylpyrazol-3-yl)-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5Z)-3-[2-(3,4-dimethoxyphenyl)ethyl]-5-[[4-oxo-2-[[(2S)-oxolan-2-yl]methylamino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H28N4O5S2
(5Z)-3-[2-(3,4-dimethoxyphenyl)ethyl]-5-[[4-oxo-2-[[(2S)-oxolan-2-yl]methylamino]pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethyl]-2-ethyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H24N6O
5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethyl]-2-ethyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
5-(1-ethyl-3-methylpyrazol-4-yl)-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(4-chloro-1-ethylpyrazol-3-yl)-3-(3,4-dimethoxyphenyl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H20ClN5O3
5-(4-chloro-1-ethylpyrazol-3-yl)-3-(3,4-dimethoxyphenyl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R)-5-(3,4-dimethoxyphenyl)-4-[hydroxy-(3-methyl-4-propoxyphenyl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C30H38N2O7
(5R)-5-(3,4-dimethoxyphenyl)-4-[hydroxy-(3-methyl-4-propoxyphenyl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— 5-[2-(3-chlorophenyl)ethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C14H12ClN3O
5-[2-(3-chlorophenyl)ethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
5-(1-ethyl-3-methylpyrazol-4-yl)-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(4-(Trifluoromethyl)phenethyl)pyrazolo[1,5-a]pyrimidin-7-ol —— C15H12F3N3O
5-(4-(Trifluoromethyl)phenethyl)pyrazolo[1,5-a]pyrimidin-7-ol
—— (5R)-1-[2-(diethylamino)ethyl]-4-[hydroxy-(2-methyl-4-prop-2-enoxyphenyl)methylidene]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C33H36N2O5
(5R)-1-[2-(diethylamino)ethyl]-4-[hydroxy-(2-methyl-4-prop-2-enoxyphenyl)methylidene]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-4-[hydroxy-(3-methyl-4-propoxyphenyl)methylidene]-1-(2-morpholin-4-ylethyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C33H36N2O6
(5S)-4-[hydroxy-(3-methyl-4-propoxyphenyl)methylidene]-1-(2-morpholin-4-ylethyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— 5-(1-ethylpyrazol-3-yl)-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H17N5O
5-(1-ethylpyrazol-3-yl)-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethyl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H22N6O
5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethyl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(3,4-Difluorophenethyl)pyrazolo[1,5-a]pyrimidin-7-ol —— C14H11F2N3O
5-(3,4-Difluorophenethyl)pyrazolo[1,5-a]pyrimidin-7-ol
—— 5-(4-chloro-1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H20ClN5O3
5-(4-chloro-1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H14FN5O
5-(1-ethylpyrazol-3-yl)-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O3
5-(1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
5-(1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H15N5O
5-(1-ethylpyrazol-3-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one