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—— (5R,7R)-5-(furan-2-yl)-N-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H17F3N4O2
(5R,7R)-5-(furan-2-yl)-N-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H21F3N6O2S
(5R,7S)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7S)-N-(3-hydroxyphenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H19F3N4O3
(5R,7S)-N-(3-hydroxyphenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-amino-4-(5-chloro-4-methoxy-2-methylphenyl)-1,2-oxazole-3-carboxylic acid —— C12H11ClN2O4
5-amino-4-(5-chloro-4-methoxy-2-methylphenyl)-1,2-oxazole-3-carboxylic acid
—— [5-(5-chloro-2-fluorophenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]methanamine —— C11H8ClFN4S
[5-(5-chloro-2-fluorophenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]methanamine
—— (5R,7R)-N-[(3,4-dimethoxyphenyl)methyl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H21F3N4O4
(5R,7R)-N-[(3,4-dimethoxyphenyl)methyl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-3-chloro-5-(4-methylphenyl)-N-(2-methylpropyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H22ClF3N4O
(5R,7S)-3-chloro-5-(4-methylphenyl)-N-(2-methylpropyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-5-(furan-2-yl)-N-(2-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H17F3N4O2
(5R,7S)-5-(furan-2-yl)-N-(2-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(5-bromothiophen-2-yl)-N-[(Z)-(3,4-dimethoxyphenyl)methylideneamino]-1H-pyrazole-3-carboxamide —— C17H15BrN4O3S
5-(5-bromothiophen-2-yl)-N-[(Z)-(3,4-dimethoxyphenyl)methylideneamino]-1H-pyrazole-3-carboxamide
—— [(5R,7R)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-(4-methylpiperidin-1-yl)methanone —— C21H25F3N4O2
[(5R,7R)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-(4-methylpiperidin-1-yl)methanone
—— (5S,7S)-N-propan-2-yl-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C15H17F3N4OS
(5S,7S)-N-propan-2-yl-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-(3,5-dimethylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H19F3N4O2
(5S,7S)-N-(3,5-dimethylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [(5R,7R)-3-bromo-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(3,4-dihydro-2H-quinolin-1-yl)methanone —— C21H18BrF3N4OS
[(5R,7R)-3-bromo-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(3,4-dihydro-2H-quinolin-1-yl)methanone
—— (5R,7S)-N-tert-butyl-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H23F3N4O2
(5R,7S)-N-tert-butyl-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7S)-N-[1-[(2-methylphenyl)methyl]pyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C25H23F3N6O
(5R,7S)-N-[1-[(2-methylphenyl)methyl]pyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-benzyl-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H21F3N4O2
(5S,7R)-N-benzyl-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-bromo-N-[(Z)-(3-bromophenyl)methylideneamino]pyridine-3-carboxamide —— C13H9Br2N3O
5-bromo-N-[(Z)-(3-bromophenyl)methylideneamino]pyridine-3-carboxamide
—— (5S,7R)-3-chloro-N-[(4-chlorophenyl)methyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H17Cl2F3N4O
(5S,7R)-3-chloro-N-[(4-chlorophenyl)methyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-N-cyclopentyl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H21F3N4O
(5R,7S)-N-cyclopentyl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxylic acid —— C16H16F3N3O4
(5S,7R)-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxylic acid
—— (5S,7R)-N-tert-butyl-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H23F3N4O2
(5S,7R)-N-tert-butyl-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-(3,4-dimethoxyphenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H23F3N4O4
(5S,7R)-N-(3,4-dimethoxyphenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7R)-N-(2-ethoxyphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H19F3N4O3
(5S,7R)-N-(2-ethoxyphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-benzyl-5-(3,4-dimethoxyphenyl)-N-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H25F3N4O3
(5S,7R)-N-benzyl-5-(3,4-dimethoxyphenyl)-N-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7S)-5-(furan-2-yl)-N-[1-[(4-methylphenyl)methyl]pyrazol-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H21F3N6O2
(5R,7S)-5-(furan-2-yl)-N-[1-[(4-methylphenyl)methyl]pyrazol-3-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-naphthalen-1-yl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H19F3N4O
(5S,7R)-N-naphthalen-1-yl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-(5-bromothiophen-2-yl)-N-[(Z)-(3-methoxyphenyl)methylideneamino]-1H-pyrazole-3-carboxamide —— C16H13BrN4O2S
5-(5-bromothiophen-2-yl)-N-[(Z)-(3-methoxyphenyl)methylideneamino]-1H-pyrazole-3-carboxamide
—— (5S,7S)-N-(3-fluoro-4-methylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H16F4N4O2
(5S,7S)-N-(3-fluoro-4-methylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-5-(4-methoxyphenyl)-N-(thiophen-2-ylmethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H19F3N4O2S
(5R,7S)-5-(4-methoxyphenyl)-N-(thiophen-2-ylmethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-5-(furan-2-yl)-N-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H17F3N4O3
(5R,7S)-5-(furan-2-yl)-N-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(5-chlorothiophen-2-yl)-N-[(Z)-(4-methoxyphenyl)methylideneamino]-1H-pyrazole-3-carboxamide —— C16H13ClN4O2S
5-(5-chlorothiophen-2-yl)-N-[(Z)-(4-methoxyphenyl)methylideneamino]-1H-pyrazole-3-carboxamide
—— (5R,7S)-3-chloro-N-cyclopentyl-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C17H18ClF3N4O2
(5R,7S)-3-chloro-N-cyclopentyl-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[2-(3-chloro-4-fluorophenyl)propan-2-yl]-1H-pyrazole-3-carboxylic acid —— C13H12ClFN2O2
5-[2-(3-chloro-4-fluorophenyl)propan-2-yl]-1H-pyrazole-3-carboxylic acid
—— (5S,7S)-3-chloro-N-(4-ethylphenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H18ClF3N4OS
(5S,7S)-3-chloro-N-(4-ethylphenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-3-chloro-5-(furan-2-yl)-7-(trifluoromethyl)-N-(3,4,5-trimethoxyphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H20ClF3N4O5
(5R,7R)-3-chloro-5-(furan-2-yl)-7-(trifluoromethyl)-N-(3,4,5-trimethoxyphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-amino-4-(3-chloro-4-ethoxyphenyl)-1,2-oxazole-3-carboxylic acid —— C12H11ClN2O4
5-amino-4-(3-chloro-4-ethoxyphenyl)-1,2-oxazole-3-carboxylic acid
—— (5S,7R)-N-(4-ethylphenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H21F3N4O
(5S,7R)-N-(4-ethylphenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-5-(3-methoxyphenyl)-N-[(2R)-1-methoxypropan-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H23F3N4O3
(5R,7S)-5-(3-methoxyphenyl)-N-[(2R)-1-methoxypropan-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-amino-4-(5-chloro-2-methoxy-4-methylphenyl)-1,2-oxazole-3-carboxylic acid —— C12H11ClN2O4
5-amino-4-(5-chloro-2-methoxy-4-methylphenyl)-1,2-oxazole-3-carboxylic acid
—— 5-(2-aminoethyl)-N-(2-chloro-4,6-dimethylphenyl)-1,3,4-thiadiazol-2-amine —— C12H15ClN4S
5-(2-aminoethyl)-N-(2-chloro-4,6-dimethylphenyl)-1,3,4-thiadiazol-2-amine
—— 5-(5-chloro-2-methoxy-4-methylphenyl)thiophene-3-carboxylic acid —— C13H11ClO3S
5-(5-chloro-2-methoxy-4-methylphenyl)thiophene-3-carboxylic acid
—— (5E)-5-(5-bromo-2-oxo-1H-indol-3-ylidene)-4-(4-methoxyanilino)-1,3-thiazol-2-one —— C18H12BrN3O3S
(5E)-5-(5-bromo-2-oxo-1H-indol-3-ylidene)-4-(4-methoxyanilino)-1,3-thiazol-2-one
—— 5-[2-(3-amino-4-chlorophenyl)ethyl]-N,N-dimethyl-1,3,4-thiadiazol-2-amine —— C12H15ClN4S
5-[2-(3-amino-4-chlorophenyl)ethyl]-N,N-dimethyl-1,3,4-thiadiazol-2-amine
—— 5-Methoxy-2-(3-propan-2-ylimidazo[4,5-b]pyridin-2-yl)aniline —— C16H18N4O
5-Methoxy-2-(3-propan-2-ylimidazo[4,5-b]pyridin-2-yl)aniline
—— [5-(3-chloro-4-fluorophenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]methanamine —— C11H8ClFN4S
[5-(3-chloro-4-fluorophenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]methanamine
—— 5-[3-(aminomethyl)pyrazin-2-yl]-1,3,3-trimethylindol-2-one —— C16H18N4O
5-[3-(aminomethyl)pyrazin-2-yl]-1,3,3-trimethylindol-2-one
—— 5-[2-(2-chloro-6-fluorophenyl)propan-2-yl]-1H-pyrazole-3-carboxylic acid —— C13H12ClFN2O2
5-[2-(2-chloro-6-fluorophenyl)propan-2-yl]-1H-pyrazole-3-carboxylic acid
—— 5-(2-aminoethylsulfonyl)-1,3,3-trimethylindol-2-one —— C13H18N2O3S
5-(2-aminoethylsulfonyl)-1,3,3-trimethylindol-2-one
—— 5-amino-4-(5-chloro-2-methoxy-3-methylphenyl)-1,2-oxazole-3-carboxylic acid —— C12H11ClN2O4
5-amino-4-(5-chloro-2-methoxy-3-methylphenyl)-1,2-oxazole-3-carboxylic acid
—— 5-[2-(aminomethyl)-6-methylpyrimidin-4-yl]-3,3-dimethyl-1H-indol-2-one —— C16H18N4O
5-[2-(aminomethyl)-6-methylpyrimidin-4-yl]-3,3-dimethyl-1H-indol-2-one