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—— 5-methoxy-2-[[(1R,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]phenol —— C20H22N4O2
5-methoxy-2-[[(1R,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]phenol
—— 5-methoxy-2-[[(1S,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]phenol —— C20H22N4O2
5-methoxy-2-[[(1S,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]phenol
—— (5R)-3-[2-(5-methoxy-2-methyl-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one —— C29H34N2O3
(5R)-3-[2-(5-methoxy-2-methyl-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one
—— (5R)-2-butanoyl-3-[2-(2-methyl-5-phenylmethoxy-1H-indol-3-yl)ethylamino]-5-phenylcyclohex-2-en-1-one —— C34H36N2O3
(5R)-2-butanoyl-3-[2-(2-methyl-5-phenylmethoxy-1H-indol-3-yl)ethylamino]-5-phenylcyclohex-2-en-1-one
—— (5R)-3-[2-(2-methyl-5-phenylmethoxy-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one —— C35H38N2O3
(5R)-3-[2-(2-methyl-5-phenylmethoxy-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one
—— (5S)-3-[2-(5-methoxy-2-methyl-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one —— C29H34N2O3
(5S)-3-[2-(5-methoxy-2-methyl-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one
—— (5R)-2-butanoyl-3-[2-[2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl]ethylamino]-5-phenylcyclohex-2-en-1-one —— C28H29F3N2O3
(5R)-2-butanoyl-3-[2-[2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl]ethylamino]-5-phenylcyclohex-2-en-1-one
—— (5R)-3-[2-(2-methyl-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one —— C28H32N2O2
(5R)-3-[2-(2-methyl-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one
—— (5S)-3-[2-(2-methyl-5-phenylmethoxy-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one —— C35H38N2O3
(5S)-3-[2-(2-methyl-5-phenylmethoxy-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one
—— 5-(3,4-dichlorophenyl)-4-(4-ethoxybenzoyl)-1-(2-furylmethyl)-3-hydroxy-1,5-dihydro-2H-pyrrol-2-one —— C24H19Cl2NO5
5-(3,4-dichlorophenyl)-4-(4-ethoxybenzoyl)-1-(2-furylmethyl)-3-hydroxy-1,5-dihydro-2H-pyrrol-2-one
—— (5E)-3-ethyl-5-[[7-ethyl-1-(2-morpholin-4-yl-2-oxoethyl)indol-3-yl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C22H26N4O3S
(5E)-3-ethyl-5-[[7-ethyl-1-(2-morpholin-4-yl-2-oxoethyl)indol-3-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5S)-3-[2-(2-methyl-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one —— C28H32N2O2
(5S)-3-[2-(2-methyl-1H-indol-3-yl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one
—— 5-ethyl-2-[(2S)-1-(4-methylthiadiazole-5-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C16H18N6O2S
5-ethyl-2-[(2S)-1-(4-methylthiadiazole-5-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2S)-1-[(5S,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22F3N7O2
5-methyl-2-[(2S)-1-[(5S,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-Butyl-2-oxoindolin-3-ylidene)-3-hexyl-2-thioxothiazolidin-4-one 611185-67-2 C21H26N2O2S2
5-(1-Butyl-2-oxoindolin-3-ylidene)-3-hexyl-2-thioxothiazolidin-4-one
—— 5-methyl-2-[(2S)-1-(2-morpholin-4-ylacetyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H23N5O3
5-methyl-2-[(2S)-1-(2-morpholin-4-ylacetyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5Z)-5-{3-ethoxy-4-[(2-nitrobenzyl)oxy]benzylidene}-3-(4-nitrobenzyl)-1,3-thiazolidine-2,4-dione —— C26H21N3O8S
(5Z)-5-{3-ethoxy-4-[(2-nitrobenzyl)oxy]benzylidene}-3-(4-nitrobenzyl)-1,3-thiazolidine-2,4-dione
—— 5-methyl-2-[(2R)-1-[(5S,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22F3N7O2
5-methyl-2-[(2R)-1-[(5S,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2R)-1-(2-morpholin-4-ylacetyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H23N5O3
5-methyl-2-[(2R)-1-(2-morpholin-4-ylacetyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5,6-dimethyl-2-[(2R)-1-(1-methylsulfonylpiperidine-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H27N5O4S
5,6-dimethyl-2-[(2R)-1-(1-methylsulfonylpiperidine-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-6-[(2R)-2-(5-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-2-yl)pyrrolidine-1-carbonyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C19H18N6O3S
5-methyl-6-[(2R)-2-(5-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-2-yl)pyrrolidine-1-carbonyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-methyl-2-[(2R)-1-(1-methylsulfonyl-2,3-dihydroindole-5-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O4S
5-methyl-2-[(2R)-1-(1-methylsulfonyl-2,3-dihydroindole-5-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-ethyl-2-[(2R)-1-[(1S,3S)-3-methoxycyclohexanecarbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H28N4O3
5-ethyl-2-[(2R)-1-[(1S,3S)-3-methoxycyclohexanecarbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-ethyl-2-[(2R)-1-(4-methylthiadiazole-5-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C16H18N6O2S
5-ethyl-2-[(2R)-1-(4-methylthiadiazole-5-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5,6-dimethyl-2-[(2S)-1-(2H-triazole-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C15H17N7O2
5,6-dimethyl-2-[(2S)-1-(2H-triazole-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2S)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O5
5-methyl-2-[(2S)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2R)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O5
5-methyl-2-[(2R)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S)-3-[2-(3,4-diethoxyphenyl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one —— C29H37NO4
(5S)-3-[2-(3,4-diethoxyphenyl)ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one
—— 5,6-dimethyl-2-[(2S)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N4O5
5,6-dimethyl-2-[(2S)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5,6-dimethyl-2-[(2R)-1-(2H-triazole-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C15H17N7O2
5,6-dimethyl-2-[(2R)-1-(2H-triazole-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5Z)-3-(5-chloro-1,3-benzothiazol-2-yl)-5-[(2-hydroxyphenyl)methylidene]-2-phenylimidazol-4-one —— C23H14ClN3O2S
(5Z)-3-(5-chloro-1,3-benzothiazol-2-yl)-5-[(2-hydroxyphenyl)methylidene]-2-phenylimidazol-4-one
—— [(5E)-5-hydrazinylidene-7,8-dihydro-6H-naphthalen-1-yl]-trimethylazanium —— C13H20N3+
[(5E)-5-hydrazinylidene-7,8-dihydro-6H-naphthalen-1-yl]-trimethylazanium
—— 5-(2-chlorophenyl)-4-(4-fluorobenzoyl)-3-hydroxy-1-(thiazol-2-yl)-1H-pyrrol-2(5H)-one —— C20H12ClFN2O3S
5-(2-chlorophenyl)-4-(4-fluorobenzoyl)-3-hydroxy-1-(thiazol-2-yl)-1H-pyrrol-2(5H)-one
—— 5-methyl-N-[(E)-pyridin-4-ylmethylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C16H17N3OS
5-methyl-N-[(E)-pyridin-4-ylmethylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5Z)-3-ethyl-5-({1-[3-(2-methylphenoxy)propyl]-1H-indol-3-yl}methylidene)-2-thioxoimidazolidin-4-one —— C24H25N3O2S
(5Z)-3-ethyl-5-({1-[3-(2-methylphenoxy)propyl]-1H-indol-3-yl}methylidene)-2-thioxoimidazolidin-4-one
—— (5Z)-5-[(4-chlorophenyl)hydrazinylidene]-1-(4-methoxyphenyl)-3-(2-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C24H19ClN4O3S
(5Z)-5-[(4-chlorophenyl)hydrazinylidene]-1-(4-methoxyphenyl)-3-(2-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5E)-5-benzylidene-9-phenyl-5,6,7,8-tetrahydro[1,2,4]triazolo[5,1-b]quinazoline —— C22H18N4
(5E)-5-benzylidene-9-phenyl-5,6,7,8-tetrahydro[1,2,4]triazolo[5,1-b]quinazoline
—— 5,6-dimethyl-2-[(2S)-1-[2-(4-methylsulfonylphenyl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4S
5,6-dimethyl-2-[(2S)-1-[2-(4-methylsulfonylphenyl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2R)-1-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22F3N7O2
5-methyl-2-[(2R)-1-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2R)-1-[2-(3,4,5-trimethoxyphenyl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N4O5
5-methyl-2-[(2R)-1-[2-(3,4,5-trimethoxyphenyl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2S)-1-[1-(thiophene-2-carbonyl)piperidine-4-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H25N5O3S
5-methyl-2-[(2S)-1-[1-(thiophene-2-carbonyl)piperidine-4-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2R)-1-[1-(thiophene-2-carbonyl)piperidine-4-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H25N5O3S
5-methyl-2-[(2R)-1-[1-(thiophene-2-carbonyl)piperidine-4-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R)-3-[2-[2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl]ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one —— C29H31F3N2O3
(5R)-3-[2-[2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl]ethylamino]-2-pentanoyl-5-phenylcyclohex-2-en-1-one
—— 5,6-dimethyl-2-[(3R)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H21N5O3
5,6-dimethyl-2-[(3R)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(3R)-1-[(2S)-2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H25N5O3
5-methyl-2-[(3R)-1-[(2S)-2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(3R)-1-[2-(4-methylsulfonylphenyl)acetyl]piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4S
5-methyl-2-[(3R)-1-[2-(4-methylsulfonylphenyl)acetyl]piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(2S)-1-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22F3N7O2
5-methyl-2-[(2S)-1-[(5R,7R)-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(3S)-1-[3-(6-methylpyridin-2-yl)propanoyl]piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H25N5O2
5-methyl-2-[(3S)-1-[3-(6-methylpyridin-2-yl)propanoyl]piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-2-[(3S)-1-[(3R)-3-(3,4,5-trimethylpyrazol-1-yl)butanoyl]piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H30N6O2
5-methyl-2-[(3S)-1-[(3R)-3-(3,4,5-trimethylpyrazol-1-yl)butanoyl]piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[[(Z)-(3-methyl-1-naphthalen-1-yl-5-oxopyrazol-4-ylidene)methyl]amino]isoindole-1,3-dione —— C23H16N4O3
5-[[(Z)-(3-methyl-1-naphthalen-1-yl-5-oxopyrazol-4-ylidene)methyl]amino]isoindole-1,3-dione