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—— (5S,9R)-7,7,9-trimethyl-2-oxaspiro[4.5]decane-1,3-dione —— C12H18O3
(5S,9R)-7,7,9-trimethyl-2-oxaspiro[4.5]decane-1,3-dione
—— (5E)-5-[[[(1S,2S)-2-aminocyclohexyl]amino]methylidene]-1-[(2R)-butan-2-yl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C15H24N4O2S
(5E)-5-[[[(1S,2S)-2-aminocyclohexyl]amino]methylidene]-1-[(2R)-butan-2-yl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-5-[(3-bromophenyl)methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C16H17BrN2O2S
(5Z)-5-[(3-bromophenyl)methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— (5-methyl-2-oxochromen-7-yl) 2-[(1R,2S,6S,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]acetate —— C23H19NO6
(5-methyl-2-oxochromen-7-yl) 2-[(1R,2S,6S,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]acetate
—— (5-methyl-2-oxochromen-7-yl) 2-[(1R,2S,6R,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]acetate —— C23H19NO6
(5-methyl-2-oxochromen-7-yl) 2-[(1R,2S,6R,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]acetate
—— 5,5,7,7-tetramethyl-2-[[4-[methyl-[[(2R)-oxolan-2-yl]methyl]sulfamoyl]benzoyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxamide —— C25H34N4O5S2
5,5,7,7-tetramethyl-2-[[4-[methyl-[[(2R)-oxolan-2-yl]methyl]sulfamoyl]benzoyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxamide
—— 5-[(5R)-3-(6-chloro-2-oxo-4-phenylquinolin-3-ylidene)-5-(4-fluorophenyl)pyrazolidin-1-yl]-5-oxopentanoic acid —— C29H23ClFN3O4
5-[(5R)-3-(6-chloro-2-oxo-4-phenylquinolin-3-ylidene)-5-(4-fluorophenyl)pyrazolidin-1-yl]-5-oxopentanoic acid
—— (5-methyl-2-oxochromen-7-yl) 2-[(1S,2R,6S,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]acetate —— C23H19NO6
(5-methyl-2-oxochromen-7-yl) 2-[(1S,2R,6S,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]acetate
—— 5-[(5S)-3-(6-chloro-2-oxo-4-phenylquinolin-3-ylidene)-5-(4-fluorophenyl)pyrazolidin-1-yl]-5-oxopentanoic acid —— C29H23ClFN3O4
5-[(5S)-3-(6-chloro-2-oxo-4-phenylquinolin-3-ylidene)-5-(4-fluorophenyl)pyrazolidin-1-yl]-5-oxopentanoic acid
—— (5S)-5-(2,5-dimethylanilino)-3-[[4-[[(5S)-5-(2,5-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione —— C30H30N4O4S2
(5S)-5-(2,5-dimethylanilino)-3-[[4-[[(5S)-5-(2,5-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
—— 5,5,7,7-tetramethyl-2-[[4-[methyl-[[(2S)-oxolan-2-yl]methyl]sulfamoyl]benzoyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxamide —— C25H34N4O5S2
5,5,7,7-tetramethyl-2-[[4-[methyl-[[(2S)-oxolan-2-yl]methyl]sulfamoyl]benzoyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxamide
—— 5,7-dihydroxy-3-[4-[(2S,3R,4R,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]chromen-4-one —— C21H20O10
5,7-dihydroxy-3-[4-[(2S,3R,4R,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]chromen-4-one
—— (5Z)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-5-[(2-hydroxyphenyl)methylidene]-1,3-thiazol-4-one —— C16H18N2O3S
(5Z)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-5-[(2-hydroxyphenyl)methylidene]-1,3-thiazol-4-one
—— (5-methyl-2-oxochromen-7-yl) (2S)-2-[(1R,2S,6S,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]-3-phenylpropanoate —— C30H25NO6
(5-methyl-2-oxochromen-7-yl) (2S)-2-[(1R,2S,6S,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]-3-phenylpropanoate
—— (5R)-5-(2,5-dimethylanilino)-3-[[4-[[(5S)-5-(2,5-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione —— C30H30N4O4S2
(5R)-5-(2,5-dimethylanilino)-3-[[4-[[(5S)-5-(2,5-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
—— (5R)-5-(2,4-dimethylanilino)-3-[[4-[[(5R)-5-(2,4-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione —— C30H30N4O4S2
(5R)-5-(2,4-dimethylanilino)-3-[[4-[[(5R)-5-(2,4-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
—— (5R)-5-(2,5-dimethylanilino)-3-[[4-[[(5R)-5-(2,5-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione —— C30H30N4O4S2
(5R)-5-(2,5-dimethylanilino)-3-[[4-[[(5R)-5-(2,5-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
—— (5R,7R)-N-[4-[acetyl(methyl)amino]phenyl]-3-(3-bromo-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C22H26BrN5O2
(5R,7R)-N-[4-[acetyl(methyl)amino]phenyl]-3-(3-bromo-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5S,7S)-N-[4-[acetyl(methyl)amino]phenyl]-3-(3-bromo-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C22H26BrN5O2
(5S,7S)-N-[4-[acetyl(methyl)amino]phenyl]-3-(3-bromo-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5S,10bR)-2-phenylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-1,3-thiazinane]-2'-one —— C19H17N3O2S
(5S,10bR)-2-phenylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-1,3-thiazinane]-2'-one
—— (5S)-5-(2,4-dimethylanilino)-3-[[4-[[(5S)-5-(2,4-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione —— C30H30N4O4S2
(5S)-5-(2,4-dimethylanilino)-3-[[4-[[(5S)-5-(2,4-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
—— (5R)-5-(2,4-dimethylanilino)-3-[[4-[[(5S)-5-(2,4-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione —— C30H30N4O4S2
(5R)-5-(2,4-dimethylanilino)-3-[[4-[[(5S)-5-(2,4-dimethylanilino)-2,4-dioxo-1,3-thiazolidin-3-yl]methyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
—— (5-methyl-2-oxochromen-7-yl) (2S)-2-[(1R,2R,6S,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]-3-phenylpropanoate —— C30H25NO6
(5-methyl-2-oxochromen-7-yl) (2S)-2-[(1R,2R,6S,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]-3-phenylpropanoate
—— (5R,7R)-3-(3-bromo-1,2,4-triazol-1-yl)-N-[1-(2-morpholin-4-ylethyl)benzimidazol-2-yl]adamantane-1-carboxamide —— C26H32BrN7O2
(5R,7R)-3-(3-bromo-1,2,4-triazol-1-yl)-N-[1-(2-morpholin-4-ylethyl)benzimidazol-2-yl]adamantane-1-carboxamide
—— (5S,7S)-3-(3-bromo-1,2,4-triazol-1-yl)-N-[1-(2-morpholin-4-ylethyl)benzimidazol-2-yl]adamantane-1-carboxamide —— C26H32BrN7O2
(5S,7S)-3-(3-bromo-1,2,4-triazol-1-yl)-N-[1-(2-morpholin-4-ylethyl)benzimidazol-2-yl]adamantane-1-carboxamide
—— (5R,10bS)-2-(1,3-benzodioxol-5-yl)-5-(4-nitrophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17N3O5
(5R,10bS)-2-(1,3-benzodioxol-5-yl)-5-(4-nitrophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-bromo-2-[2-[(3S)-5-(3-bromophenyl)-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C22H16Br2N2O3S
5-bromo-2-[2-[(3S)-5-(3-bromophenyl)-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— (5Z)-5-[[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H28N4O4S2
(5Z)-5-[[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-bromo-2-[2-[(3R)-5-(2-chlorophenyl)-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C24H17BrCl2N2O3
5-bromo-2-[2-[(3R)-5-(2-chlorophenyl)-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— (5R)-5-(3-bromophenyl)-4-[hydroxy-(4-piperidin-1-ylsulfonylphenyl)methylidene]-1-(3-methoxypropyl)pyrrolidine-2,3-dione —— C26H29BrN2O6S
(5R)-5-(3-bromophenyl)-4-[hydroxy-(4-piperidin-1-ylsulfonylphenyl)methylidene]-1-(3-methoxypropyl)pyrrolidine-2,3-dione
—— 5-bromo-2-[2-[(3R)-5-(3-bromophenyl)-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C24H17Br2ClN2O3
5-bromo-2-[2-[(3R)-5-(3-bromophenyl)-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-bromo-2-[2-[(3S)-5-(4-bromophenyl)-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C24H17Br2ClN2O3
5-bromo-2-[2-[(3S)-5-(4-bromophenyl)-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-bromo-2-[2-[(3R)-5-(4-bromophenyl)-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C24H17Br2ClN2O3
5-bromo-2-[2-[(3R)-5-(4-bromophenyl)-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-bromo-2-[2-[(3R)-5-(3-bromophenyl)-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C22H16Br2N2O3S
5-bromo-2-[2-[(3R)-5-(3-bromophenyl)-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-chloro-1-[2-[(3R)-3-[4-(dimethylamino)phenyl]-5-naphthalen-1-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione —— C31H25ClN4O3
5-chloro-1-[2-[(3R)-3-[4-(dimethylamino)phenyl]-5-naphthalen-1-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione
—— 5-bromo-2-[2-[(3S)-3-[4-(dimethylamino)phenyl]-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C30H26BrN3O3
5-bromo-2-[2-[(3S)-3-[4-(dimethylamino)phenyl]-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— (5Z)-5-[[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H28N4O4S2
(5Z)-5-[[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-3-[(4-methoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-bromo-2-[2-[(3R)-5-naphthalen-2-yl-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C26H19BrN2O3S
5-bromo-2-[2-[(3R)-5-naphthalen-2-yl-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-chloro-1-[2-[(3R)-3-(3,4-dimethoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione —— C31H24ClN3O5
5-chloro-1-[2-[(3R)-3-(3,4-dimethoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione
—— 5-bromo-2-[2-[(3R)-5-naphthalen-1-yl-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C26H19BrN2O3S
5-bromo-2-[2-[(3R)-5-naphthalen-1-yl-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-bromo-2-[2-[(3S)-5-naphthalen-2-yl-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C26H19BrN2O3S
5-bromo-2-[2-[(3S)-5-naphthalen-2-yl-3-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-chloro-1-[2-[(3S)-5-(2-chlorophenyl)-3-(3,4-dimethoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione —— C27H21Cl2N3O5
5-chloro-1-[2-[(3S)-5-(2-chlorophenyl)-3-(3,4-dimethoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione
—— (5R)-4-[hydroxy-(4-morpholin-4-ylsulfonylphenyl)methylidene]-1-(2-methoxyethyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C30H30N2O8S
(5R)-4-[hydroxy-(4-morpholin-4-ylsulfonylphenyl)methylidene]-1-(2-methoxyethyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— 5-chloro-1-[2-[(3R)-3-(3,4-dimethoxyphenyl)-5-naphthalen-1-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione —— C31H24ClN3O5
5-chloro-1-[2-[(3R)-3-(3,4-dimethoxyphenyl)-5-naphthalen-1-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione
—— 5-bromo-2-[2-[(3S)-3-[4-(dimethylamino)phenyl]-5-naphthalen-1-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C30H26BrN3O3
5-bromo-2-[2-[(3S)-3-[4-(dimethylamino)phenyl]-5-naphthalen-1-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-chloro-1-[2-[(3R)-3-[4-(dimethylamino)phenyl]-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione —— C31H25ClN4O3
5-chloro-1-[2-[(3R)-3-[4-(dimethylamino)phenyl]-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione
—— 5-bromo-2-[2-[(3S)-3-(3,4-dimethoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C30H25BrN2O5
5-bromo-2-[2-[(3S)-3-(3,4-dimethoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-chloro-1-[2-[(3S)-5-(4-chlorophenyl)-3-(3,4-dimethoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione —— C27H21Cl2N3O5
5-chloro-1-[2-[(3S)-5-(4-chlorophenyl)-3-(3,4-dimethoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione
—— 5-bromo-2-[2-[(3R)-3-(3,4-dimethoxyphenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde —— C26H22BrFN2O5
5-bromo-2-[2-[(3R)-3-(3,4-dimethoxyphenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]benzaldehyde
—— 5-chloro-1-[2-[(3S)-3-[4-(dimethylamino)phenyl]-5-naphthalen-1-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione —— C31H25ClN4O3
5-chloro-1-[2-[(3S)-3-[4-(dimethylamino)phenyl]-5-naphthalen-1-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione