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—— (5-methyl-2-propan-2-ylphenyl) (10R,11S,15S,16S)-13-(1,3-benzodioxol-5-yl)-12,14-dioxo-1,13-diazatetracyclo[8.6.0.02,7.011,15]hexadeca-2,4,6,8-tetraene-16-carboxylate —— C32H28N2O6
(5-methyl-2-propan-2-ylphenyl) (10R,11S,15S,16S)-13-(1,3-benzodioxol-5-yl)-12,14-dioxo-1,13-diazatetracyclo[8.6.0.02,7.011,15]hexadeca-2,4,6,8-tetraene-16-carboxylate
—— 5-amino-3-[(2-hydroxy-5-sulfophenyl)hydrazinylidene]-4-oxonaphthalene-2,7-disulfonic acid —— C16H13N3O11S3
5-amino-3-[(2-hydroxy-5-sulfophenyl)hydrazinylidene]-4-oxonaphthalene-2,7-disulfonic acid
—— (5R)-4-(3H-1,3-benzothiazol-2-ylidene)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-5-(4-ethylphenyl)pyrrolidine-2,3-dione —— C28H22N4O2S3
(5R)-4-(3H-1,3-benzothiazol-2-ylidene)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-5-(4-ethylphenyl)pyrrolidine-2,3-dione
—— 5-[(1R,2S,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylphenyl)-2-piperidin-1-ylbenzamide —— C28H29N3O3
5-[(1R,2S,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylphenyl)-2-piperidin-1-ylbenzamide
—— (5R)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(3-methoxyphenyl)-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione —— C32H24FN3O4S2
(5R)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(3-methoxyphenyl)-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione
—— (5R)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione —— C31H21F2N3O3S2
(5R)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione
—— (5S)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione —— C31H21F2N3O3S2
(5S)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione
—— (5-methyl-2-propan-2-ylphenyl) (10R,11S,15S,16R)-13-(1,3-benzodioxol-5-yl)-12,14-dioxo-1,13-diazatetracyclo[8.6.0.02,7.011,15]hexadeca-2,4,6,8-tetraene-16-carboxylate —— C32H28N2O6
(5-methyl-2-propan-2-ylphenyl) (10R,11S,15S,16R)-13-(1,3-benzodioxol-5-yl)-12,14-dioxo-1,13-diazatetracyclo[8.6.0.02,7.011,15]hexadeca-2,4,6,8-tetraene-16-carboxylate
—— 5-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylphenyl)-2-piperidin-1-ylbenzamide —— C28H29N3O3
5-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylphenyl)-2-piperidin-1-ylbenzamide
—— (5S)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]-5-(4-nitrophenyl)pyrrolidine-2,3-dione —— C31H21FN4O5S2
(5S)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]-5-(4-nitrophenyl)pyrrolidine-2,3-dione
—— (5Z)-3-(furan-2-ylmethyl)-5-[(2-methoxyanilino)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C16H14N2O3S2
(5Z)-3-(furan-2-ylmethyl)-5-[(2-methoxyanilino)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-5-(4-chlorophenyl)-3-[2-(ethylamino)-2-oxoethyl]-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C20H23ClN4O2S
(5S)-5-(4-chlorophenyl)-3-[2-(ethylamino)-2-oxoethyl]-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5Z)-5-[[2-(dimethylamino)ethylamino]methylidene]-1-(2-methoxyphenyl)-3-phenyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C22H24N4O3S
(5Z)-5-[[2-(dimethylamino)ethylamino]methylidene]-1-(2-methoxyphenyl)-3-phenyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5-fluoro-1H-indol-2-yl)-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C19H23FN2O
(5-fluoro-1H-indol-2-yl)-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 5-[3-carboxy-4-[[(2Z,4E)-hexa-2,4-dienoyl]amino]phenyl]-2-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]benzoic acid —— C26H24N2O6
5-[3-carboxy-4-[[(2Z,4E)-hexa-2,4-dienoyl]amino]phenyl]-2-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]benzoic acid
—— 5-bromo-N-[(2R)-1-oxo-1-[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-3-phenylpropan-2-yl]thiophene-2-sulfonamide —— C24H24BrN3O4S2
5-bromo-N-[(2R)-1-oxo-1-[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-3-phenylpropan-2-yl]thiophene-2-sulfonamide
—— 5-[2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]pyridin-4-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H20N4O
5-[2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]pyridin-4-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5E)-5-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-3-[(4-nitrophenyl)methyl]-1,3-thiazolidine-2,4-dione —— C29H22N2O6S
(5E)-5-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-3-[(4-nitrophenyl)methyl]-1,3-thiazolidine-2,4-dione
—— 5-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylphenyl)-2-morpholin-4-ylbenzamide —— C27H27N3O4
5-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylphenyl)-2-morpholin-4-ylbenzamide
—— 5-[(1R,2S,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylphenyl)-2-morpholin-4-ylbenzamide —— C27H27N3O4
5-[(1R,2S,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(4-methylphenyl)-2-morpholin-4-ylbenzamide
—— (5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione —— C37H46N2O6
(5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione
—— 5-[2-[(3S)-3-(2,5-dihydropyrrol-1-yl)pyrrolidin-1-yl]pyridin-3-yl]-3-methyl-1,2,4-oxadiazole —— C16H19N5O
5-[2-[(3S)-3-(2,5-dihydropyrrol-1-yl)pyrrolidin-1-yl]pyridin-3-yl]-3-methyl-1,2,4-oxadiazole
—— (5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]-5-(4-propoxyphenyl)pyrrolidine-2,3-dione —— C34H40N2O5
(5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]-5-(4-propoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-5-(4-chlorophenyl)-3-[2-(ethylamino)-2-oxoethyl]-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C20H23ClN4O2S
(5R)-5-(4-chlorophenyl)-3-[2-(ethylamino)-2-oxoethyl]-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(3-methoxyphenyl)pyrrolidine-2,3-dione —— C33H38N2O5
(5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(3-methoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-5-(4-butoxyphenyl)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]pyrrolidine-2,3-dione —— C36H44N2O5
(5R)-5-(4-butoxyphenyl)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]pyrrolidine-2,3-dione
—— (5-fluoro-1H-indol-2-yl)-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C19H23FN2O
(5-fluoro-1H-indol-2-yl)-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— (5R)-1-[5-[(2-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(4-nitrophenyl)pyrrolidine-2,3-dione —— C27H18ClFN4O5S2
(5R)-1-[5-[(2-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(4-nitrophenyl)pyrrolidine-2,3-dione
—— 5-[2-[(3R)-3-(2,5-dihydropyrrol-1-yl)pyrrolidin-1-yl]pyridin-3-yl]-3-methyl-1,2,4-oxadiazole —— C16H19N5O
5-[2-[(3R)-3-(2,5-dihydropyrrol-1-yl)pyrrolidin-1-yl]pyridin-3-yl]-3-methyl-1,2,4-oxadiazole
—— (5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(3-methoxy-4-pentoxyphenyl)pyrrolidine-2,3-dione —— C38H48N2O6
(5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(3-methoxy-4-pentoxyphenyl)pyrrolidine-2,3-dione
—— (5E)-5-[[4-(dimethylamino)phenyl]methylidene]-4-methyl-2,6-dioxo-1-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carbonitrile —— C21H23N3O3
(5E)-5-[[4-(dimethylamino)phenyl]methylidene]-4-methyl-2,6-dioxo-1-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carbonitrile
—— (5R)-5-(2-fluorophenyl)-4-[hydroxy-(4-pyrrolidin-1-ylsulfonylphenyl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C28H32FN3O6S
(5R)-5-(2-fluorophenyl)-4-[hydroxy-(4-pyrrolidin-1-ylsulfonylphenyl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— (5R)-5-(2,5-dimethoxyphenyl)-4-[hydroxy-(4-pyrrolidin-1-ylsulfonylphenyl)methylidene]-1-(pyridin-3-ylmethyl)pyrrolidine-2,3-dione —— C29H29N3O7S
(5R)-5-(2,5-dimethoxyphenyl)-4-[hydroxy-(4-pyrrolidin-1-ylsulfonylphenyl)methylidene]-1-(pyridin-3-ylmethyl)pyrrolidine-2,3-dione
—— 5,6-dimethyl-3-[(E)-[2-(trifluoromethyl)phenyl]methylideneamino]thieno[2,3-d]pyrimidin-4-one —— C16H12F3N3OS
5,6-dimethyl-3-[(E)-[2-(trifluoromethyl)phenyl]methylideneamino]thieno[2,3-d]pyrimidin-4-one
—— (5S)-5-(3-bromo-4-hydroxy-5-methoxyphenyl)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C26H28BrFN2O6
(5S)-5-(3-bromo-4-hydroxy-5-methoxyphenyl)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— 5-[2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]pyridin-3-yl]-3-methyl-1,2,4-oxadiazole —— C14H16N4O
5-[2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]pyridin-3-yl]-3-methyl-1,2,4-oxadiazole
—— (5E)-1-[2-(3,4-dimethoxyphenyl)ethyl]-5-[[3-[(2R)-2,7-dimethyl-2,3-dihydro-1-benzofuran-5-yl]-1-phenylpyrazol-4-yl]methylidene]-4-methyl-2,6-dioxopyridine-3-carbonitrile —— C37H34N4O5
(5E)-1-[2-(3,4-dimethoxyphenyl)ethyl]-5-[[3-[(2R)-2,7-dimethyl-2,3-dihydro-1-benzofuran-5-yl]-1-phenylpyrazol-4-yl]methylidene]-4-methyl-2,6-dioxopyridine-3-carbonitrile
—— (5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(3-methoxy-4-pentoxyphenyl)pyrrolidine-2,3-dione —— C38H48N2O6
(5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(3-methoxy-4-pentoxyphenyl)pyrrolidine-2,3-dione
—— 5-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-2-chlorobenzoic acid —— C15H12ClNO4
5-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-2-chlorobenzoic acid
—— (5R)-1-[5-[(2-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-5-[4-(dimethylamino)phenyl]-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]pyrrolidine-2,3-dione —— C29H24ClFN4O3S2
(5R)-1-[5-[(2-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-5-[4-(dimethylamino)phenyl]-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]pyrrolidine-2,3-dione
—— (5S)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-1-(furan-2-ylmethyl)-5-(3-methoxy-4-phenylmethoxyphenyl)pyrrolidine-2,3-dione —— C31H26FNO7
(5S)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-1-(furan-2-ylmethyl)-5-(3-methoxy-4-phenylmethoxyphenyl)pyrrolidine-2,3-dione
—— (5S,7S)-N-(2-ethoxyphenyl)-3-(4-methylphenyl)adamantane-1-carboxamide —— C26H31NO2
(5S,7S)-N-(2-ethoxyphenyl)-3-(4-methylphenyl)adamantane-1-carboxamide
—— (5R)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(3-methoxy-4-phenylmethoxyphenyl)-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C33H35FN2O6
(5R)-4-[(3-fluoro-4-methylphenyl)-hydroxymethylidene]-5-(3-methoxy-4-phenylmethoxyphenyl)-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— 5-[3-carboxy-4-[[(2E,4Z)-hexa-2,4-dienoyl]amino]phenyl]-2-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]benzoic acid —— C26H24N2O6
5-[3-carboxy-4-[[(2E,4Z)-hexa-2,4-dienoyl]amino]phenyl]-2-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]benzoic acid
—— 5-[3-carboxy-4-[[(2E,4E)-hexa-2,4-dienoyl]amino]phenyl]-2-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]benzoic acid —— C26H24N2O6
5-[3-carboxy-4-[[(2E,4E)-hexa-2,4-dienoyl]amino]phenyl]-2-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]benzoic acid
—— (5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(4-phenylmethoxyphenyl)pyrrolidine-2,3-dione —— C39H42N2O5
(5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(4-phenylmethoxyphenyl)pyrrolidine-2,3-dione
—— (5E)-5-[[5-(4-acetylphenyl)furan-2-yl]methylidene]-4-methyl-2,6-dioxo-1-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carbonitrile —— C25H22N2O5
(5E)-5-[[5-(4-acetylphenyl)furan-2-yl]methylidene]-4-methyl-2,6-dioxo-1-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carbonitrile
—— (5R)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-1-(furan-2-ylmethyl)-5-(3-methoxy-4-phenylmethoxyphenyl)pyrrolidine-2,3-dione —— C31H26FNO7
(5R)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-1-(furan-2-ylmethyl)-5-(3-methoxy-4-phenylmethoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione —— C38H48N2O6
(5R)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione
—— (5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(4-phenylmethoxyphenyl)pyrrolidine-2,3-dione —— C39H42N2O5
(5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(4-phenylmethoxyphenyl)pyrrolidine-2,3-dione