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—— 5-[(1R)-1-[(2-methoxyacetyl)amino]ethyl]thiophene-2-sulfonyl chloride —— C9H12ClNO4S2
5-[(1R)-1-[(2-methoxyacetyl)amino]ethyl]thiophene-2-sulfonyl chloride
—— (5S,7R)-3-bromo-5-(5-bromofuran-2-yl)-N-(2-methoxyethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C15H15Br2F3N4O3
(5S,7R)-3-bromo-5-(5-bromofuran-2-yl)-N-(2-methoxyethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H23F3N4OS
[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— (5E)-3-methyl-1-phenyl-5-(1,3,3-trimethylindol-2-ylidene)pyrazolo[3,4-b][1,4]azaphosphinin-4-ium 4-oxide —— C23H22N4OP+
(5E)-3-methyl-1-phenyl-5-(1,3,3-trimethylindol-2-ylidene)pyrazolo[3,4-b][1,4]azaphosphinin-4-ium 4-oxide
—— (5R,7S)-3-bromo-5-(5-bromofuran-2-yl)-N-(2-methoxyethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C15H15Br2F3N4O3
(5R,7S)-3-bromo-5-(5-bromofuran-2-yl)-N-(2-methoxyethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[(1R)-1-(3-methylbutanoylamino)ethyl]thiophene-2-sulfonyl chloride —— C11H16ClNO3S2
5-[(1R)-1-(3-methylbutanoylamino)ethyl]thiophene-2-sulfonyl chloride
—— 5-[(1S)-1-[[(1R,2S)-2-methylcyclopropanecarbonyl]amino]ethyl]thiophene-2-sulfonyl chloride —— C11H14ClNO3S2
5-[(1S)-1-[[(1R,2S)-2-methylcyclopropanecarbonyl]amino]ethyl]thiophene-2-sulfonyl chloride
—— (5R,7R)-3-(carboxymethylsulfanyl)adamantane-1-carboxylic acid —— C13H18O4S
(5R,7R)-3-(carboxymethylsulfanyl)adamantane-1-carboxylic acid
—— 5-[(1S)-1-[[(2S)-2-methylbutanoyl]amino]ethyl]thiophene-2-sulfonyl chloride —— C11H16ClNO3S2
5-[(1S)-1-[[(2S)-2-methylbutanoyl]amino]ethyl]thiophene-2-sulfonyl chloride
—— 5-[(1R)-1-(2-methylpropanoylamino)ethyl]thiophene-2-sulfonyl chloride —— C10H14ClNO3S2
5-[(1R)-1-(2-methylpropanoylamino)ethyl]thiophene-2-sulfonyl chloride
—— 5-[(1S)-1-[[(1R,2R)-2-methylcyclopropanecarbonyl]amino]ethyl]thiophene-2-sulfonyl chloride —— C11H14ClNO3S2
5-[(1S)-1-[[(1R,2R)-2-methylcyclopropanecarbonyl]amino]ethyl]thiophene-2-sulfonyl chloride
—— 5-[(1R)-1-[[(2S)-2-methylbutanoyl]amino]ethyl]thiophene-2-sulfonyl chloride —— C11H16ClNO3S2
5-[(1R)-1-[[(2S)-2-methylbutanoyl]amino]ethyl]thiophene-2-sulfonyl chloride
—— 5-[(1S)-1-[[(1S,2S)-2-methylcyclopropanecarbonyl]amino]ethyl]thiophene-2-sulfonyl chloride —— C11H14ClNO3S2
5-[(1S)-1-[[(1S,2S)-2-methylcyclopropanecarbonyl]amino]ethyl]thiophene-2-sulfonyl chloride
—— 5-[(1R)-1-[[(2R)-2-methylbutanoyl]amino]ethyl]thiophene-2-sulfonyl chloride —— C11H16ClNO3S2
5-[(1R)-1-[[(2R)-2-methylbutanoyl]amino]ethyl]thiophene-2-sulfonyl chloride
—— [(5R,7R)-5-(3,4-dichlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(4-phenylpiperazin-1-yl)methanone —— C24H22Cl2F3N5O
[(5R,7R)-5-(3,4-dichlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(4-phenylpiperazin-1-yl)methanone
—— [5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H23F3N4OS
[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 5-[(1S)-1-(3-methylbutanoylamino)ethyl]thiophene-2-sulfonyl chloride —— C11H16ClNO3S2
5-[(1S)-1-(3-methylbutanoylamino)ethyl]thiophene-2-sulfonyl chloride
—— [5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H23F3N4OS
[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 5-[(1S)-1-[(2-methoxyacetyl)amino]ethyl]thiophene-2-sulfonyl chloride —— C9H12ClNO4S2
5-[(1S)-1-[(2-methoxyacetyl)amino]ethyl]thiophene-2-sulfonyl chloride
—— 5-[(1R)-1-(2,2-dimethylpropanoylamino)ethyl]thiophene-2-sulfonyl chloride —— C11H16ClNO3S2
5-[(1R)-1-(2,2-dimethylpropanoylamino)ethyl]thiophene-2-sulfonyl chloride
—— [5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H23F3N4OS
[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 5-[[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]-2-hydroxybenzoic acid —— C16H19NO4
5-[[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]-2-hydroxybenzoic acid
—— 5-[(1S)-1-(cyclopropanecarbonylamino)ethyl]thiophene-2-sulfonyl chloride —— C10H12ClNO3S2
5-[(1S)-1-(cyclopropanecarbonylamino)ethyl]thiophene-2-sulfonyl chloride
—— (5R,7R)-3-bromo-5-(5-bromofuran-2-yl)-N-(2-methoxyethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C15H15Br2F3N4O3
(5R,7R)-3-bromo-5-(5-bromofuran-2-yl)-N-(2-methoxyethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[(1S)-1-(2,2-dimethylpropanoylamino)ethyl]thiophene-2-sulfonyl chloride —— C11H16ClNO3S2
5-[(1S)-1-(2,2-dimethylpropanoylamino)ethyl]thiophene-2-sulfonyl chloride
—— [(5S,7S)-5-(3,4-dichlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(4-phenylpiperazin-1-yl)methanone —— C24H22Cl2F3N5O
[(5S,7S)-5-(3,4-dichlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(4-phenylpiperazin-1-yl)methanone
—— (5S)-5-butyl-5-[2-[(5-chloropyridin-2-yl)amino]acetyl]oxolan-2-one —— C15H19ClN2O3
(5S)-5-butyl-5-[2-[(5-chloropyridin-2-yl)amino]acetyl]oxolan-2-one
—— 5-[[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]-2-hydroxybenzoic acid —— C16H19NO4
5-[[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]-2-hydroxybenzoic acid
—— (5E)-5-[[2-[2-(diethylazaniumyl)ethyl]hydrazinyl]methylidene]-1-(4-fluorophenyl)-6-oxo-2-sulfanylidenepyrimidin-4-olate —— C17H22FN5O2S
(5E)-5-[[2-[2-(diethylazaniumyl)ethyl]hydrazinyl]methylidene]-1-(4-fluorophenyl)-6-oxo-2-sulfanylidenepyrimidin-4-olate
—— 5-[bis[(2R)-2-hydroxypropyl]amino]-4-(3-chlorophenyl)-11-methyl-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one —— C22H27ClN4O3S
5-[bis[(2R)-2-hydroxypropyl]amino]-4-(3-chlorophenyl)-11-methyl-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
—— 5-[(1R)-1-acetamidoethyl]thiophene-2-sulfonyl chloride —— C8H10ClNO3S2
5-[(1R)-1-acetamidoethyl]thiophene-2-sulfonyl chloride
—— (5S)-5-[(E)-2-(furan-2-yl)ethenyl]-11-methyl-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7)-dien-3-one —— C16H17N3O2S
(5S)-5-[(E)-2-(furan-2-yl)ethenyl]-11-methyl-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7)-dien-3-one
—— 5-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-2-(pyridin-3-ylmethylamino)benzoic acid —— C22H19N3O4
5-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-2-(pyridin-3-ylmethylamino)benzoic acid
—— (5E)-5-[[[(1R,2R)-2-aminocyclohexyl]amino]methylidene]-1-(3-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H22N4O3S
(5E)-5-[[[(1R,2R)-2-aminocyclohexyl]amino]methylidene]-1-(3-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R,7R)-N-[(6S)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H21ClF3N5O2S2
(5R,7R)-N-[(6S)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(4-chlorophenyl)-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C23H23ClF3N5O
[5-(4-chlorophenyl)-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— [(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H27F3N4OS
[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 5-bromo-N'-[(E)-(3-chloro-5-nitro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]pyridine-3-carbohydrazide —— C13H8BrClN4O4
5-bromo-N'-[(E)-(3-chloro-5-nitro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]pyridine-3-carbohydrazide
—— [(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H27F3N4OS
[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 5-bromo-2-hydroxy-N-[(Z)-[2-[(4-methylphenyl)sulfonylamino]phenyl]methylideneamino]benzamide —— C21H18BrN3O4S
5-bromo-2-hydroxy-N-[(Z)-[2-[(4-methylphenyl)sulfonylamino]phenyl]methylideneamino]benzamide
—— (5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[4-[(1R)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H24ClF3N4O4
(5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[4-[(1R)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[4-[(1R)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H24ClF3N4O4
(5R,7S)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[4-[(1R)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C25H17BrF3NO4
(5R)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— [5-(4-chlorophenyl)-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C23H23ClF3N5O
[5-(4-chlorophenyl)-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— (5R,7S)-N-benzyl-3-chloro-5-(4-methylphenyl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H24ClF3N4O
(5R,7S)-N-benzyl-3-chloro-5-(4-methylphenyl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-3-bromo-N-(2,4-dichlorophenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H12BrCl2F3N4OS
(5S,7S)-3-bromo-N-(2,4-dichlorophenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione —— C25H17BrF3NO4
(5S)-4-[(4-bromophenyl)-hydroxymethylidene]-5-(4-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]pyrrolidine-2,3-dione
—— 5-bromo-1-{[(1S)-6,7-dimethoxy-1-methyl-3,4-dihydroisoquinolin-2(1H)-yl]methyl}-1H-indole-2,3-dione —— C21H21BrN2O4
5-bromo-1-{[(1S)-6,7-dimethoxy-1-methyl-3,4-dihydroisoquinolin-2(1H)-yl]methyl}-1H-indole-2,3-dione
—— 5-amino-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-chlorobenzamide —— C16H21ClN2O
5-amino-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-chlorobenzamide
—— (5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[3-[(1R)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H24ClF3N4O4
(5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-[3-[(1R)-1-hydroxyethyl]phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide