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—— [5-(5-chloro-4-ethoxy-2-methylphenyl)-1-methyl-1,2,4-triazol-3-yl]methanamine —— C13H17ClN4O
[5-(5-chloro-4-ethoxy-2-methylphenyl)-1-methyl-1,2,4-triazol-3-yl]methanamine
—— (5S,7R)-3-chloro-N-cyclohexyl-N-methyl-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H22ClF3N4OS
(5S,7R)-3-chloro-N-cyclohexyl-N-methyl-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(2-aminoethyl)-N-(2,5-dimethoxyphenyl)-1,3,4-thiadiazol-2-amine —— C12H16N4O2S
5-(2-aminoethyl)-N-(2,5-dimethoxyphenyl)-1,3,4-thiadiazol-2-amine
—— (5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-(3,4-dimethylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H24ClF3N4O3
(5R,7R)-3-chloro-5-(3,4-dimethoxyphenyl)-N-(3,4-dimethylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-N-[(Z)-(4-fluorophenyl)methylideneamino]-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide —— C20H25FN4O
(5R)-N-[(Z)-(4-fluorophenyl)methylideneamino]-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
—— [5-(3-chloro-4-propan-2-yloxyphenyl)-3-methyl-1,2-oxazol-4-yl]methanamine —— C14H17ClN2O2
[5-(3-chloro-4-propan-2-yloxyphenyl)-3-methyl-1,2-oxazol-4-yl]methanamine
—— 5-(2-Bromo-4-hydroxy-5-methoxybenzylidene)-3-(4-methoxyphenyl)-2-thioxo-4-imidazolidinone —— C18H15BrN2O4S
5-(2-Bromo-4-hydroxy-5-methoxybenzylidene)-3-(4-methoxyphenyl)-2-thioxo-4-imidazolidinone
—— (5S,7S)-N-(4-chlorophenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H16ClF3N4O
(5S,7S)-N-(4-chlorophenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-(3-chlorophenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H18ClF3N4O2
(5S,7R)-N-(3-chlorophenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-(3-chloro-6-methoxy-2,4-dimethylphenyl)thiophene-2-carbaldehyde —— C14H13ClO2S
5-(3-chloro-6-methoxy-2,4-dimethylphenyl)thiophene-2-carbaldehyde
—— (5R,7S)-N-(5-chloro-2-methoxyphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H16ClF3N4O3
(5R,7S)-N-(5-chloro-2-methoxyphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-chloro-2-(5-morpholin-4-yl-1,3,4-oxadiazol-2-yl)aniline —— C12H13ClN4O2
5-chloro-2-(5-morpholin-4-yl-1,3,4-oxadiazol-2-yl)aniline
—— (5S,7S)-3-chloro-N-cyclohexyl-N-methyl-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H22ClF3N4OS
(5S,7S)-3-chloro-N-cyclohexyl-N-methyl-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-3-chloro-N-(2,3-dichlorophenyl)-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H18Cl3F3N4O3
(5R,7R)-3-chloro-N-(2,3-dichlorophenyl)-5-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-3-bromo-N-[(4-methoxyphenyl)methyl]-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H18BrF3N4O2S
(5R,7R)-3-bromo-N-[(4-methoxyphenyl)methyl]-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-3-bromo-N-(2-hydroxy-5-methylphenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H16BrF3N4O2S
(5R,7R)-3-bromo-N-(2-hydroxy-5-methylphenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-5-(4-chlorophenyl)-N-[(4-fluorophenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H17ClF4N4O
(5S,7S)-5-(4-chlorophenyl)-N-[(4-fluorophenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-3-bromo-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxylic acid —— C14H11BrF3N3O2
(5S,7R)-3-bromo-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxylic acid
—— (5S,7R)-5-(furan-2-yl)-N-[4-(trifluoromethoxy)phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H14F6N4O3
(5S,7R)-5-(furan-2-yl)-N-[4-(trifluoromethoxy)phenyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [5-methyl-2-(4-phenoxyphenyl)-1,2,4-triazol-3-yl]methanamine —— C16H16N4O
[5-methyl-2-(4-phenoxyphenyl)-1,2,4-triazol-3-yl]methanamine
—— 5-chloro-N-{4-[N-(phenylsulfonyl)ethanehydrazonoyl]phenyl}-2-thiophenecarboxamide —— C19H16ClN3O3S2
5-chloro-N-{4-[N-(phenylsulfonyl)ethanehydrazonoyl]phenyl}-2-thiophenecarboxamide
—— (5S,7S)-3-chloro-5-(4-methoxyphenyl)-N-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H20ClF3N4O2
(5S,7S)-3-chloro-5-(4-methoxyphenyl)-N-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-bromo-N'-[1-(4-chlorophenyl)propylidene]-2-furohydrazide —— C14H12BrClN2O2
5-bromo-N'-[1-(4-chlorophenyl)propylidene]-2-furohydrazide
—— (5S,7S)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-N-methyl-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H25F3N6O
(5S,7S)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-N-methyl-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(2-aminoethyl)-N-(2,4-dimethoxyphenyl)-1,3,4-thiadiazol-2-amine —— C12H16N4O2S
5-(2-aminoethyl)-N-(2,4-dimethoxyphenyl)-1,3,4-thiadiazol-2-amine
—— (5R,7S)-3-bromo-N-(2-methylsulfanylphenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H16BrF3N4OS2
(5R,7S)-3-bromo-N-(2-methylsulfanylphenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(4-ethylsulfonylphenyl)-1H-pyrazole-4-carboxylic acid —— C12H12N2O4S
5-(4-ethylsulfonylphenyl)-1H-pyrazole-4-carboxylic acid
—— (5R,7R)-3-chloro-N-[(1,5-dimethylpyrazol-4-yl)methyl]-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H18ClF3N6OS
(5R,7R)-3-chloro-N-[(1,5-dimethylpyrazol-4-yl)methyl]-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-(5-bromopyridin-2-yl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H15BrF3N5O
(5S,7S)-N-(5-bromopyridin-2-yl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-3-bromo-N-(2-methylsulfanylphenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H18BrF3N4OS
(5S,7R)-3-bromo-N-(2-methylsulfanylphenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-benzyl-3-chloro-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H20ClF3N4O2
(5S,7S)-N-benzyl-3-chloro-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-cyclohexyl-N-methyl-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H27F3N4O
(5R,7R)-N-cyclohexyl-N-methyl-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [5-(4-ethylsulfonylphenyl)-3-methyl-1,2-oxazol-4-yl]methanamine —— C13H16N2O3S
[5-(4-ethylsulfonylphenyl)-3-methyl-1,2-oxazol-4-yl]methanamine
—— 5-amino-4-(3-fluoro-4-propan-2-yloxyphenyl)-1,2-oxazole-3-carboxylic acid —— C13H13FN2O4
5-amino-4-(3-fluoro-4-propan-2-yloxyphenyl)-1,2-oxazole-3-carboxylic acid
—— (5R,7R)-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxylic acid —— C12H9ClF3N3O2S
(5R,7R)-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxylic acid
—— (5S,7R)-N-(2,4-dimethoxyphenyl)-5-(4-fluorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H20F4N4O3
(5S,7R)-N-(2,4-dimethoxyphenyl)-5-(4-fluorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-3-bromo-N-(4-bromophenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H15Br2F3N4O
(5R,7S)-3-bromo-N-(4-bromophenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-3-bromo-N-[(4-fluorophenyl)methyl]-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H15BrF4N4OS
(5R,7S)-3-bromo-N-[(4-fluorophenyl)methyl]-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-5-(4-fluorophenyl)-N-[(4-methoxyphenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H20F4N4O2
(5S,7S)-5-(4-fluorophenyl)-N-[(4-methoxyphenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7R)-3-chloro-N-[(1,3-dimethylpyrazol-4-yl)methyl]-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H18ClF3N6OS
(5S,7R)-3-chloro-N-[(1,3-dimethylpyrazol-4-yl)methyl]-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[(4-chloro-5-methyl-3-nitropyrazol-1-yl)methyl]-N-[(E)-1-[3-[(2-fluorobenzoyl)amino]phenyl]ethylideneamino]furan-2-carboxamide —— C25H20ClFN6O5
5-[(4-chloro-5-methyl-3-nitropyrazol-1-yl)methyl]-N-[(E)-1-[3-[(2-fluorobenzoyl)amino]phenyl]ethylideneamino]furan-2-carboxamide
—— 5-bromo-N'-(2-isopropoxy-3-methoxybenzylidene)-1-benzofuran-2-carbohydrazide —— C20H19BrN2O4
5-bromo-N'-(2-isopropoxy-3-methoxybenzylidene)-1-benzofuran-2-carbohydrazide
—— [5-(4-propan-2-ylsulfonylphenyl)-1,2-oxazol-3-yl]methanamine —— C13H16N2O3S
[5-(4-propan-2-ylsulfonylphenyl)-1,2-oxazol-3-yl]methanamine
—— (5S,7R)-3-chloro-N-(3-chloro-4-fluorophenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H14Cl2F4N4O
(5S,7R)-3-chloro-N-(3-chloro-4-fluorophenyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(4-ethylsulfonylphenyl)-1-methyl-1,2,4-triazol-3-yl]methanamine —— C12H16N4O2S
[5-(4-ethylsulfonylphenyl)-1-methyl-1,2,4-triazol-3-yl]methanamine
—— 5-bromo-N-[4-[(Z)-N-(cyclopropanecarbonylamino)-C-methylcarbonimidoyl]phenyl]furan-2-carboxamide —— C17H16BrN3O3
5-bromo-N-[4-[(Z)-N-(cyclopropanecarbonylamino)-C-methylcarbonimidoyl]phenyl]furan-2-carboxamide
—— (5R,7R)-N-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H27F3N6O
(5R,7R)-N-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(3-Chloro-4-propan-2-yloxyphenyl)-1-methylpyrazol-3-yl]methanamine —— C14H18ClN3O
[5-(3-Chloro-4-propan-2-yloxyphenyl)-1-methylpyrazol-3-yl]methanamine
—— 5-[6-(cyclopropylamino)-2-methylpyrimidin-4-yl]-1,3-dihydroindol-2-one —— C16H16N4O
5-[6-(cyclopropylamino)-2-methylpyrimidin-4-yl]-1,3-dihydroindol-2-one
—— 5-(2-chloro-4-methoxyphenyl)-1,3-dimethylpyrazole-4-carboxylic acid —— C13H13ClN2O3
5-(2-chloro-4-methoxyphenyl)-1,3-dimethylpyrazole-4-carboxylic acid