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—— 5-[2-(2-chloro-6-fluorophenyl)propan-2-yl]-1,2-oxazole-3-carboxylic acid —— C13H11ClFNO3
5-[2-(2-chloro-6-fluorophenyl)propan-2-yl]-1,2-oxazole-3-carboxylic acid
—— (5R,7S)-5-(4-bromophenyl)-N-cyclohexyl-N-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H24BrF3N4O
(5R,7S)-5-(4-bromophenyl)-N-cyclohexyl-N-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5Z)-2-amino-5-(6-chloro-7-methyl-2-oxo-1H-indol-3-ylidene)-1,3-thiazol-4-one —— C12H8ClN3O2S
(5Z)-2-amino-5-(6-chloro-7-methyl-2-oxo-1H-indol-3-ylidene)-1,3-thiazol-4-one
—— (5Z)-5-[[4-(difluoromethoxy)phenyl]methylidene]-3-prop-2-enyl-2-sulfanylideneimidazolidin-4-one —— C14H12F2N2O2S
(5Z)-5-[[4-(difluoromethoxy)phenyl]methylidene]-3-prop-2-enyl-2-sulfanylideneimidazolidin-4-one
—— (5R,7S)-5-(4-methylphenyl)-7-(trifluoromethyl)-N-(3,4,5-trimethoxyphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H25F3N4O4
(5R,7S)-5-(4-methylphenyl)-7-(trifluoromethyl)-N-(3,4,5-trimethoxyphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5E)-5-[(6-ethoxy-1,3-benzodioxol-5-yl)methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-phenylimino-1,3-thiazolidin-4-one —— C24H24N2O5S
(5E)-5-[(6-ethoxy-1,3-benzodioxol-5-yl)methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-phenylimino-1,3-thiazolidin-4-one
—— [5-cyclopropyl-2-(2,3-dichlorophenyl)-1,2,4-triazol-3-yl]methanamine —— C12H12Cl2N4
[5-cyclopropyl-2-(2,3-dichlorophenyl)-1,2,4-triazol-3-yl]methanamine
—— (5R,7S)-N-(3-hydroxyphenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H15F3N4O2S
(5R,7S)-N-(3-hydroxyphenyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[6-(2-aminoethylamino)-2-methylpyrimidin-4-yl]-1,3-dihydroindol-2-one —— C15H17N5O
5-[6-(2-aminoethylamino)-2-methylpyrimidin-4-yl]-1,3-dihydroindol-2-one
—— (5S,7R)-N-(3-chloro-4-fluorophenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H13ClF4N4O2
(5S,7R)-N-(3-chloro-4-fluorophenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5E)-5-[(2,3-dimethylanilino)methylidene]-1-(2-fluorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C19H16FN3O2S
(5E)-5-[(2,3-dimethylanilino)methylidene]-1-(2-fluorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-amino-3-(5-chloro-2-methoxyphenyl)-2-oxo-1H-imidazole-4-carboxylic acid —— C11H10ClN3O4
5-amino-3-(5-chloro-2-methoxyphenyl)-2-oxo-1H-imidazole-4-carboxylic acid
—— 5-[2-(2-methyl-1H-indol-3-yl)propan-2-yl]-1H-pyrazole-3-carboxylic acid —— C16H17N3O2
5-[2-(2-methyl-1H-indol-3-yl)propan-2-yl]-1H-pyrazole-3-carboxylic acid
—— (5Z)-5-[(E)-3-(furan-2-yl)prop-2-enylidene]-2-(4-methoxyphenyl)imino-1,3-thiazolidin-4-one —— C17H14N2O3S
(5Z)-5-[(E)-3-(furan-2-yl)prop-2-enylidene]-2-(4-methoxyphenyl)imino-1,3-thiazolidin-4-one
—— (5E)-5-(4-methoxybenzylidene)-3-{[4-(4-methylphenyl)piperazin-1-yl]methyl}-1,3-thiazolidine-2,4-dione —— C23H25N3O3S
(5E)-5-(4-methoxybenzylidene)-3-{[4-(4-methylphenyl)piperazin-1-yl]methyl}-1,3-thiazolidine-2,4-dione
—— (5-bromo-4-{(Z)-[1-(2-chlorophenyl)-3-methyl-5-oxo-1,5-dihydro-4H-pyrazol-4-ylidene]methyl}-2-methoxyphenoxy)acetic acid —— C20H16BrClN2O5
(5-bromo-4-{(Z)-[1-(2-chlorophenyl)-3-methyl-5-oxo-1,5-dihydro-4H-pyrazol-4-ylidene]methyl}-2-methoxyphenoxy)acetic acid
—— (5E)-5-[(2-bromo-4-ethoxy-5-methoxyphenyl)methylidene]-3-[(4-fluorophenyl)methyl]-1,3-thiazolidine-2,4-dione —— C20H17BrFNO4S
(5E)-5-[(2-bromo-4-ethoxy-5-methoxyphenyl)methylidene]-3-[(4-fluorophenyl)methyl]-1,3-thiazolidine-2,4-dione
—— [5-(trifluoromethyl)-3-(2,4,6-trimethylphenyl)-1H-pyrazol-4-yl]methanamine —— C14H16F3N3
[5-(trifluoromethyl)-3-(2,4,6-trimethylphenyl)-1H-pyrazol-4-yl]methanamine
—— (5R,7S)-N-(3-chloro-4-fluorophenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H13ClF4N4O2
(5R,7S)-N-(3-chloro-4-fluorophenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[2-(5-chloro-2-fluorophenyl)propan-2-yl]-1,2-oxazole-3-carboxylic acid —— C13H11ClFNO3
5-[2-(5-chloro-2-fluorophenyl)propan-2-yl]-1,2-oxazole-3-carboxylic acid
—— (5-chloro-2-methoxy-4-methylphenyl)-(4-hydroxypiperidin-1-yl)methanone —— C14H18ClNO3
(5-chloro-2-methoxy-4-methylphenyl)-(4-hydroxypiperidin-1-yl)methanone
—— (5R,7S)-5-(4-chlorophenyl)-N-methyl-N-(2-pyridin-2-ylethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H21ClF3N5O
(5R,7S)-5-(4-chlorophenyl)-N-methyl-N-(2-pyridin-2-ylethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5Z)-5-[[1-(2,3-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-ethyl-2-sulfanylideneimidazolidin-4-one —— C20H23N3OS
(5Z)-5-[[1-(2,3-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-ethyl-2-sulfanylideneimidazolidin-4-one
—— (5E)-3-ethyl-5-[[4-methoxy-3-(morpholin-4-ylmethyl)phenyl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H22N2O3S2
(5E)-3-ethyl-5-[[4-methoxy-3-(morpholin-4-ylmethyl)phenyl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R,7S)-N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H22F3N5O2S
(5R,7S)-N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(3,4-dimethylphenyl)-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methanamine —— C14H16F3N3
[5-(3,4-dimethylphenyl)-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methanamine
—— 5-[2-(4-tert-butyl-6-methylpyrimidin-2-yl)ethyl]-2-methylaniline —— C18H25N3
5-[2-(4-tert-butyl-6-methylpyrimidin-2-yl)ethyl]-2-methylaniline
—— (5E)-5-[(2,5-dimethoxy-4-pyrrolidin-1-ylphenyl)methylidene]-3-[(4-methylphenyl)methyl]-1,3-thiazolidine-2,4-dione —— C24H26N2O4S
(5E)-5-[(2,5-dimethoxy-4-pyrrolidin-1-ylphenyl)methylidene]-3-[(4-methylphenyl)methyl]-1,3-thiazolidine-2,4-dione
—— [5-(2-methyl-1H-indol-3-yl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]methanamine —— C14H13N5S
[5-(2-methyl-1H-indol-3-yl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]methanamine
—— 5-(5-methoxy-3-methyl-1,3-benzothiazol-2(3H)-ylidene)-3-methyl-2-(6-quinolinylimino)-1,3-thiazolidin-4-one —— C22H18N4O2S2
5-(5-methoxy-3-methyl-1,3-benzothiazol-2(3H)-ylidene)-3-methyl-2-(6-quinolinylimino)-1,3-thiazolidin-4-one
—— [5-(1-methylindol-3-yl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]methanamine —— C14H13N5S
[5-(1-methylindol-3-yl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]methanamine
—— 5-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1,3,3-trimethylindol-2-one —— C15H17N5O
5-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1,3,3-trimethylindol-2-one
—— [5-cyclopropyl-2-(3,4-dichlorophenyl)-1,2,4-triazol-3-yl]methanamine —— C12H12Cl2N4
[5-cyclopropyl-2-(3,4-dichlorophenyl)-1,2,4-triazol-3-yl]methanamine
—— (5Z)-5-[(2-methyl-1H-indol-3-yl)methylidene]-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3-thiazolidine-2,4-dione —— C19H19N3O3S
(5Z)-5-[(2-methyl-1H-indol-3-yl)methylidene]-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3-thiazolidine-2,4-dione
—— [5-(2,5-dimethylphenyl)-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methanamine —— C14H16F3N3
[5-(2,5-dimethylphenyl)-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methanamine
—— 5-[6-(2-aminoethylamino)pyrimidin-4-yl]-1-methyl-3H-indol-2-one —— C15H17N5O
5-[6-(2-aminoethylamino)pyrimidin-4-yl]-1-methyl-3H-indol-2-one
—— [5-(trifluoromethyl)-3-(2,4,5-trimethylphenyl)-1H-pyrazol-4-yl]methanamine —— C14H16F3N3
[5-(trifluoromethyl)-3-(2,4,5-trimethylphenyl)-1H-pyrazol-4-yl]methanamine
—— [5-(2,4-dimethylphenyl)-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methanamine —— C14H16F3N3
[5-(2,4-dimethylphenyl)-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methanamine
—— 5-[4-(2-aminoethyl)-6-methyl-1,3,5-triazin-2-yl]-1-methyl-3H-indol-2-one —— C15H17N5O
5-[4-(2-aminoethyl)-6-methyl-1,3,5-triazin-2-yl]-1-methyl-3H-indol-2-one
—— 5-[2-(1-methylindol-3-yl)propan-2-yl]-1H-pyrazole-3-carboxylic acid —— C16H17N3O2
5-[2-(1-methylindol-3-yl)propan-2-yl]-1H-pyrazole-3-carboxylic acid
—— 5-(5-chloro-2-methoxy-3-methylphenyl)thiophene-3-carboxylic acid —— C13H11ClO3S
5-(5-chloro-2-methoxy-3-methylphenyl)thiophene-3-carboxylic acid
—— [5-cyclopropyl-2-(3,5-dichlorophenyl)-1,2,4-triazol-3-yl]methanamine —— C12H12Cl2N4
[5-cyclopropyl-2-(3,5-dichlorophenyl)-1,2,4-triazol-3-yl]methanamine
—— 5-(1,2-dimethylindol-3-yl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-amine —— C14H13N5S
5-(1,2-dimethylindol-3-yl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-amine
—— [5-(4-ethylphenyl)-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methanamine —— C14H16F3N3
[5-(4-ethylphenyl)-1-methyl-3-(trifluoromethyl)pyrazol-4-yl]methanamine
—— [5-cyclopropyl-2-(2,5-dichlorophenyl)-1,2,4-triazol-3-yl]methanamine —— C12H12Cl2N4
[5-cyclopropyl-2-(2,5-dichlorophenyl)-1,2,4-triazol-3-yl]methanamine
—— 5-[2-(5-chloro-2-fluorophenyl)propan-2-yl]-1H-pyrazole-3-carboxylic acid —— C13H12ClFN2O2
5-[2-(5-chloro-2-fluorophenyl)propan-2-yl]-1H-pyrazole-3-carboxylic acid
—— (5S,7R)-N-(2,3-dimethylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H19F3N4O2
(5S,7R)-N-(2,3-dimethylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-5-(furan-2-yl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H15F3N4O2
(5S,7S)-5-(furan-2-yl)-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7S)-5-(3-methoxyphenyl)-N-[[(2R)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H23F3N4O3
(5R,7S)-5-(3-methoxyphenyl)-N-[[(2R)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7R)-5-(furan-2-yl)-N-[(2-methoxyphenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H19F3N4O3
(5R,7R)-5-(furan-2-yl)-N-[(2-methoxyphenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide