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—— 5-[(2R)-1-[(2R)-2-methylbutanoyl]pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H33N5O3
5-[(2R)-1-[(2R)-2-methylbutanoyl]pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-[(2S)-2-methylbutanoyl]piperidin-3-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H33N5O3
5-[(3S)-1-[(2S)-2-methylbutanoyl]piperidin-3-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-[(2S)-2-methylbutanoyl]piperidin-3-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H31N5O3
5-[(3S)-1-[(2S)-2-methylbutanoyl]piperidin-3-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]pyrrolidin-2-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H31N5O3
5-[(2R)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]pyrrolidin-2-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-butanoylpiperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H29N5O3
5-[(3S)-1-butanoylpiperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(4-fluorophenyl)methyl]pyrrolidin-2-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H28FN5O2
5-[(2S)-1-[(4-fluorophenyl)methyl]pyrrolidin-2-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-(cyclopentanecarbonyl)piperidin-3-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H31N5O3
5-[(3S)-1-(cyclopentanecarbonyl)piperidin-3-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5Z)-5-[(1,3-benzodioxol-5-ylamino)methylidene]-1-(3-chlorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H12ClN3O4S
(5Z)-5-[(1,3-benzodioxol-5-ylamino)methylidene]-1-(3-chlorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-5-{[3-(4-methoxy-3-nitrophenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-2-(4-methylphenyl)[1,3]thiazolo[3,2-b][1,2,4]triazol-6(5H)-one —— C28H20N6O4S
(5Z)-5-{[3-(4-methoxy-3-nitrophenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-2-(4-methylphenyl)[1,3]thiazolo[3,2-b][1,2,4]triazol-6(5H)-one
—— 5-[(2S)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H26FN5O2
5-[(2S)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H28FN5O2
5-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H31N5O3
5-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H28FN5O2
5-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[2-(dimethylamino)acetyl]pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H32N6O3
5-[(2R)-1-[2-(dimethylamino)acetyl]pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H29N5O2
5-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-butanoylpiperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H29N5O3
5-[(3R)-1-butanoylpiperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(2-hydroxy-4-methylphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O3
5-[(2R)-1-[(2-hydroxy-4-methylphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(2-hydroxyphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H29N5O3
5-[(2S)-1-[(2-hydroxyphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H31N5O3
5-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(4-methoxyphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O3
5-[(2R)-1-[(4-methoxyphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-(4-fluorobenzoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H28FN5O2
5-[(2S)-1-(4-fluorobenzoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(5-methylthiophen-2-yl)methyl]piperidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H29N5O2S
5-[(2R)-1-[(5-methylthiophen-2-yl)methyl]piperidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(5-methylthiophen-3-yl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H29N5O2S
5-[(2R)-1-[(5-methylthiophen-3-yl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-(2,2-dimethylpropanoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H33N5O2
5-[(2R)-1-(2,2-dimethylpropanoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-(cyclopentanecarbonyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H33N5O2
5-[(2S)-1-(cyclopentanecarbonyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-(2-methylpropanoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C21H31N5O2
5-[(2R)-1-(2-methylpropanoyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5Z)-5-[(5-bromothiophen-2-yl)methylidene]-1-prop-2-enyl-1,3-diazinane-2,4,6-trione —— C12H9BrN2O3S
(5Z)-5-[(5-bromothiophen-2-yl)methylidene]-1-prop-2-enyl-1,3-diazinane-2,4,6-trione
—— 5-[(2R)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H28FN5O2
5-[(2R)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3-{2-Nitrophenyl}-2-propenylidene)amino]-2-(4-methoxyphenyl)-1,3-benzoxazole —— C23H17N3O4
5-[(3-{2-Nitrophenyl}-2-propenylidene)amino]-2-(4-methoxyphenyl)-1,3-benzoxazole
—— 5-[(2R)-1-[(3-methoxyphenyl)methyl]piperidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O3
5-[(2R)-1-[(3-methoxyphenyl)methyl]piperidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(5-methylthiophen-2-yl)methyl]piperidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H29N5O2S
5-[(2S)-1-[(5-methylthiophen-2-yl)methyl]piperidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-butanoylpiperidin-2-yl]-11-(thiophen-2-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H29N5O2S
5-[(2S)-1-butanoylpiperidin-2-yl]-11-(thiophen-2-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(2R)-2-methylbutanoyl]piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H33N5O2
5-[(2R)-1-[(2R)-2-methylbutanoyl]piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-[(2R)-2-methylbutanoyl]piperidin-3-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H31N5O3
5-[(3R)-1-[(2R)-2-methylbutanoyl]piperidin-3-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5R,7R)-3-acetamido-N-spiro[1,3-benzodioxole-2,1'-cyclohexane]-5-yladamantane-1-carboxamide —— C25H32N2O4
(5R,7R)-3-acetamido-N-spiro[1,3-benzodioxole-2,1'-cyclohexane]-5-yladamantane-1-carboxamide
—— 5-[(2R)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C21H29N5O4
5-[(2R)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(5-methylthiophen-2-yl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H29N5O2S
5-[(2R)-1-[(5-methylthiophen-2-yl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5Z)-5-{[5-(3-Methyl-4-nitrophenyl)furan-2-YL]methylidene}-1,3-thiazolidine-2,4-dione —— C15H10N2O5S
(5Z)-5-{[5-(3-Methyl-4-nitrophenyl)furan-2-YL]methylidene}-1,3-thiazolidine-2,4-dione
—— 5-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H29N5O3
5-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-(4-methylbenzoyl)pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H29N5O2
5-[(2S)-1-(4-methylbenzoyl)pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-(cyclohexylmethyl)pyrrolidin-2-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H35N5O2
5-[(2R)-1-(cyclohexylmethyl)pyrrolidin-2-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(2S)-2-methylbutanoyl]pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H33N5O3
5-[(2S)-1-[(2S)-2-methylbutanoyl]pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H28FN5O2
5-[(2S)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(3-fluorophenyl)methyl]pyrrolidin-2-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H28FN5O2
5-[(2R)-1-[(3-fluorophenyl)methyl]pyrrolidin-2-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-(5-ethyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H28N6O3
5-[(2S)-1-(5-ethyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H29N5O2
5-[(2S)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-12-propan-2-yl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(2-methoxyphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O3
5-[(2S)-1-[(2-methoxyphenyl)methyl]piperidin-2-yl]-11-propanoyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2S)-1-[(2R)-2-methylbutanoyl]pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H33N5O3
5-[(2S)-1-[(2R)-2-methylbutanoyl]pyrrolidin-2-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2R)-1-[(5-methylthiophen-3-yl)methyl]piperidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H29N5O2S
5-[(2R)-1-[(5-methylthiophen-3-yl)methyl]piperidin-2-yl]-12-propanoyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-(cyclobutanecarbonyl)piperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H29N5O3
5-[(3R)-1-(cyclobutanecarbonyl)piperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one