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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(1R)-1-(2-methoxyphenoxy)ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H19N3O3
5-[(1R)-1-(2-methoxyphenoxy)ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19ClN4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[[3-(4-fluorophenyl)-1-methylpyrazol-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H16FN5O
5-[[3-(4-fluorophenyl)-1-methylpyrazol-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— {5-[1-[3-(2-Morpholin-4-yl-2-oxo-1-phenyl-ethoxy)-4-phenethyloxy-phenyl]-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid —— C32H30N2O7S2
{5-[1-[3-(2-Morpholin-4-yl-2-oxo-1-phenyl-ethoxy)-4-phenethyloxy-phenyl]-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid
—— 5-[[3-(phenylmethoxy)-4-[(4-methylphenyl)methoxy]phenyl]methylene]-4-oxo-2-thioxo-3-thiazolidineacetic acid —— C27H23NO5S2
5-[[3-(phenylmethoxy)-4-[(4-methylphenyl)methoxy]phenyl]methylene]-4-oxo-2-thioxo-3-thiazolidineacetic acid
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(4-ethoxyphenyl)methyl]-2,2-dimethyl-5-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-dioxane-4,6-dione —— C27H32N2O6
5-[(4-ethoxyphenyl)methyl]-2,2-dimethyl-5-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]-1,3-dioxane-4,6-dione
—— [(5S,7S)-3-(4-methoxyphenyl)-1-adamantyl]-(4-pyrimidin-2-ylpiperazin-1-yl)methanone —— C26H32N4O2
[(5S,7S)-3-(4-methoxyphenyl)-1-adamantyl]-(4-pyrimidin-2-ylpiperazin-1-yl)methanone
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5Z)-5-benzylidene-3-[2-(2-methyl-5-nitro-imidazol-1-yl)ethyl]thiazolidine-2,4-dione —— C16H14N4O4S
(5Z)-5-benzylidene-3-[2-(2-methyl-5-nitro-imidazol-1-yl)ethyl]thiazolidine-2,4-dione
—— {5-[1-[4-Benzyloxy-3-(3-chloro-benzyloxy)-phenyl]-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid —— C26H20ClNO5S2
{5-[1-[4-Benzyloxy-3-(3-chloro-benzyloxy)-phenyl]-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid
—— 5-[(1S)-1-(2-methoxyphenoxy)ethyl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H21N3O3
5-[(1S)-1-(2-methoxyphenoxy)ethyl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-naphthalen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H22N6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-naphthalen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R,7R)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-(4-methoxyphenyl)adamantane-1-carboxamide —— C22H27N3O2S
(5R,7R)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-(4-methoxyphenyl)adamantane-1-carboxamide
—— 5-[(1R)-1-(2-methoxyphenoxy)ethyl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H21N3O3
5-[(1R)-1-(2-methoxyphenoxy)ethyl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H22N4O3
5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N6O
5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S,7S)-3-(4-methoxyphenyl)-N-propyladamantane-1-carboxamide —— C21H29NO2
(5S,7S)-3-(4-methoxyphenyl)-N-propyladamantane-1-carboxamide
—— {5-[1-[3-(2-Methyl-1-phenyl-propoxy)-4-phenethyloxy-phenyl]-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid —— C30H29NO5S2
{5-[1-[3-(2-Methyl-1-phenyl-propoxy)-4-phenethyloxy-phenyl]-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H22N4O2
5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(4-Chloro-2-fluorophenyl)methylene]-3-[(phenylsulfonyl)amino]-2-thioxo-1,3-thiazolidin-4-one —— C16H10ClFN2O3S3
5-[(4-Chloro-2-fluorophenyl)methylene]-3-[(phenylsulfonyl)amino]-2-thioxo-1,3-thiazolidin-4-one
—— 5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-2-(benzotriazol-1-yl)propyl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H22N6O2
5-[(2S)-2-(benzotriazol-1-yl)propyl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R,7R)-3-(4-methoxyphenyl)-N-propyladamantane-1-carboxamide —— C21H29NO2
(5R,7R)-3-(4-methoxyphenyl)-N-propyladamantane-1-carboxamide
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(benzotriazol-1-yl)propyl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H20N6O
5-[(2R)-2-(benzotriazol-1-yl)propyl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S,7S)-3-acetamido-N-[(2S)-4-(4-fluorophenyl)butan-2-yl]adamantane-1-carboxamide —— C23H31FN2O2
(5S,7S)-3-acetamido-N-[(2S)-4-(4-fluorophenyl)butan-2-yl]adamantane-1-carboxamide
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3,4-Dichlorophenyl)methylene]-3-{[(4-methoxyphenyl)sulfonyl]amino}-2-thioxo-1,3-thiazolidin-4-one —— C17H12Cl2N2O4S3
5-[(3,4-Dichlorophenyl)methylene]-3-{[(4-methoxyphenyl)sulfonyl]amino}-2-thioxo-1,3-thiazolidin-4-one
—— 5-[(3,4-Dichlorophenyl)methylene]-3-[(butylsulfonyl)amino]-2-thioxo-1,3-thiazolidin-4-one —— C14H14Cl2N2O3S3
5-[(3,4-Dichlorophenyl)methylene]-3-[(butylsulfonyl)amino]-2-thioxo-1,3-thiazolidin-4-one
—— (5S,7R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-cyclopropyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H27F3N4O
(5S,7R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-cyclopropyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[(3-Hydroxy-4-nitrophenyl)methylene]-3-[(phenylsulfonyl)amino]-2-thioxo-1,3-thiazolidin-4-one —— C16H11N3O6S3
5-[(3-Hydroxy-4-nitrophenyl)methylene]-3-[(phenylsulfonyl)amino]-2-thioxo-1,3-thiazolidin-4-one
—— (5S,7S)-N-[(1S)-1-(3,4-dihydro-2H-chromen-6-yl)ethyl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C24H30N4O2
(5S,7S)-N-[(1S)-1-(3,4-dihydro-2H-chromen-6-yl)ethyl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5Z)-9,12-dimethoxy-11,11-dimethyl-bicyclo[7.3.1]trideca-1(12),5-dien-3,7-diyn-2-ol —— C17H20O3
(5Z)-9,12-dimethoxy-11,11-dimethyl-bicyclo[7.3.1]trideca-1(12),5-dien-3,7-diyn-2-ol
—— 5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19ClN4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S,7S)-N-[(2R)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C24H33N5O
(5S,7S)-N-[(2R)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5S,7S)-N-[(2R)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]-3-(3-methyl-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C25H35N5O
(5S,7S)-N-[(2R)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]-3-(3-methyl-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— 5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H18N4O2
5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-N-(4-methylphenyl)-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H19N5O3
5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-N-(4-methylphenyl)-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-[(2R)-2-(benzotriazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H17FN6O
5-[(2R)-2-(benzotriazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H20N4O3S
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R,7R)-N-cyclopentyl-3-(4-methoxyphenyl)adamantane-1-carboxamide —— C23H31NO2
(5R,7R)-N-cyclopentyl-3-(4-methoxyphenyl)adamantane-1-carboxamide
—— 5-[(2S)-2-(benzotriazol-1-yl)propyl]-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H17FN6O
5-[(2S)-2-(benzotriazol-1-yl)propyl]-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-7-oxo-N-phenyl-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H17N5O3
5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-7-oxo-N-phenyl-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5E)-5-[(3,5-difluorophenyl)methylene]-2-thioxo-imidazolidin-4-one —— C10H6F2N2OS
(5E)-5-[(3,5-difluorophenyl)methylene]-2-thioxo-imidazolidin-4-one