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—— 5-[(3S)-1-[(2R)-2-methylbutanoyl]piperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H32N6O2
5-[(3S)-1-[(2R)-2-methylbutanoyl]piperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5E)-5-{5-chloro-2-[(3-chlorobenzyl)oxy]benzylidene}-3-(3,4-dimethylphenyl)-2-thioxo-1,3-thiazolidin-4-one —— C25H19Cl2NO2S2
(5E)-5-{5-chloro-2-[(3-chlorobenzyl)oxy]benzylidene}-3-(3,4-dimethylphenyl)-2-thioxo-1,3-thiazolidin-4-one
—— 5-[(3S)-1-butanoylpiperidin-3-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H33N5O3
5-[(3S)-1-butanoylpiperidin-3-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(Cyclohexylmethyl)piperidin-4-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H37N5O2
5-[1-(Cyclohexylmethyl)piperidin-4-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5Z)-5-{[3-(4-bromophenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-3-(tetrahydrofuran-2-ylmethyl)-2-thioxo-1,3-thiazolidin-4-one —— C24H20BrN3O2S2
(5Z)-5-{[3-(4-bromophenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-3-(tetrahydrofuran-2-ylmethyl)-2-thioxo-1,3-thiazolidin-4-one
—— (5E)-5-[[5-(2-nitrophenyl)furan-2-yl]methylidene]-2-phenylimino-1,3-thiazolidin-4-one —— C20H13N3O4S
(5E)-5-[[5-(2-nitrophenyl)furan-2-yl]methylidene]-2-phenylimino-1,3-thiazolidin-4-one
—— 5-(4-chlorophenyl)-3-hydroxy-4-[(3-methyl-4-propoxyphenyl)carbonyl]-1-[3-(morpholin-4-yl)propyl]-1,5-dihydro-2H-pyrrol-2-one —— C28H33ClN2O5
5-(4-chlorophenyl)-3-hydroxy-4-[(3-methyl-4-propoxyphenyl)carbonyl]-1-[3-(morpholin-4-yl)propyl]-1,5-dihydro-2H-pyrrol-2-one
—— 5-[(3R)-1-(cyclobutanecarbonyl)piperidin-3-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[(3R)-1-(cyclobutanecarbonyl)piperidin-3-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H31N5O4
5-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-propanoylpiperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H28N6O2
5-[(3R)-1-propanoylpiperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[4-(4-bromophenyl)sulfonylpiperazin-1-yl]-2-nitro-N-[(2S)-4-phenylbutan-2-yl]aniline —— C26H29BrN4O4S
5-[4-(4-bromophenyl)sulfonylpiperazin-1-yl]-2-nitro-N-[(2S)-4-phenylbutan-2-yl]aniline
—— 5-[(3R)-1-[(2R)-2-methylbutanoyl]piperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H32N6O2
5-[(3R)-1-[(2R)-2-methylbutanoyl]piperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H33N5O2
5-[(3R)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-(cyclobutanecarbonyl)piperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H30N6O2
5-[(3S)-1-(cyclobutanecarbonyl)piperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[[(1S)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[1-[[(1S)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-11-(2-methoxyacetyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-11-(2-methoxyacetyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[[(1S)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H35N5O2
5-[1-[[(1S)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(Cyclohexylmethyl)piperidin-4-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H35N5O3
5-[1-(Cyclohexylmethyl)piperidin-4-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-4-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H31N5O4
5-[1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-4-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-(cyclobutanecarbonyl)piperidin-3-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[(3S)-1-(cyclobutanecarbonyl)piperidin-3-yl]-11-(oxan-4-yl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[4-(4-bromophenyl)sulfonylpiperazin-1-yl]-2-nitro-N-[(2R)-4-phenylbutan-2-yl]aniline —— C26H29BrN4O4S
5-[4-(4-bromophenyl)sulfonylpiperazin-1-yl]-2-nitro-N-[(2R)-4-phenylbutan-2-yl]aniline
—— 5-[1-(Cyclopropylmethyl)piperidin-4-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C21H29N5O3
5-[1-(Cyclopropylmethyl)piperidin-4-yl]-12-(2-methoxyacetyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(2,4-dimethylanilino)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C13H13N3O2S
5-[(2,4-dimethylanilino)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-4-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-4-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-4-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-4-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-(1-propan-2-ylpiperidin-4-yl)-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H30N6O2
5-(1-propan-2-ylpiperidin-4-yl)-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[1-(Cyclohexylmethyl)piperidin-4-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H37N5O2
5-[1-(Cyclohexylmethyl)piperidin-4-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[(1S,6S)-bicyclo[4.1.0]heptane-7-carbonyl]piperidin-4-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H35N5O2
5-[1-[(1S,6S)-bicyclo[4.1.0]heptane-7-carbonyl]piperidin-4-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H33N5O2
5-[(3S)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-11-(cyclopropanecarbonyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H35N5O2
5-[1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-11-(2-methylpropanoyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-(1,3-benzodioxol-5-yl)-N-(4-ethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H21F3N4O4
5-(1,3-benzodioxol-5-yl)-N-(4-ethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[1-[[(1S)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-11-(2-methoxyacetyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H33N5O3
5-[1-[[(1S)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-11-(2-methoxyacetyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H35N5O2
5-[1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-4-yl]-12-(2-methylpropanoyl)-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-(cyclopropanecarbonyl)piperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H28N6O2
5-[(3S)-1-(cyclopropanecarbonyl)piperidin-3-yl]-11-(pyridin-4-ylmethyl)-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5Z)-5-{[3-(4-ethoxy-3-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-2-thioxo-1,3-thiazolidin-4-one —— C21H16FN3O2S2
(5Z)-5-{[3-(4-ethoxy-3-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-2-thioxo-1,3-thiazolidin-4-one
—— 5-(1-propan-2-ylpiperidin-4-yl)-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H30N6O2
5-(1-propan-2-ylpiperidin-4-yl)-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5E)-5-[[3-bromo-5-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C25H19BrFNO3S2
(5E)-5-[[3-bromo-5-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[(2,4-dihydroxyphenyl)methylidene]-3-[(4-methoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H15NO4S2
(5E)-5-[(2,4-dihydroxyphenyl)methylidene]-3-[(4-methoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[3-chloro-5-ethoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H22ClNO3S2
(5E)-5-[[3-chloro-5-ethoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[3-bromo-4-[(2,4-dichlorophenyl)methoxy]-5-ethoxyphenyl]methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C22H18BrCl2NO3S2
(5E)-5-[[3-bromo-4-[(2,4-dichlorophenyl)methoxy]-5-ethoxyphenyl]methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-methyl-N-[(Z)-thiophen-2-ylmethylideneamino]thiophene-3-carboxamide —— C11H10N2OS2
5-methyl-N-[(Z)-thiophen-2-ylmethylideneamino]thiophene-3-carboxamide
—— (5Z)-5-[[3-chloro-5-ethoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H22ClNO3S2
(5Z)-5-[[3-chloro-5-ethoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-benzyl-5-[(3-bromo-5-ethoxy-4-phenylmethoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H22BrNO3S2
(5Z)-3-benzyl-5-[(3-bromo-5-ethoxy-4-phenylmethoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[[3-bromo-4-[(2-chlorophenyl)methoxy]-5-ethoxyphenyl]methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C25H19BrClNO3S2
(5Z)-5-[[3-bromo-4-[(2-chlorophenyl)methoxy]-5-ethoxyphenyl]methylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(2,5-dimethylthiophen-3-yl)-2-methyl-1H-pyrazol-3-one —— C10H12N2OS
5-(2,5-dimethylthiophen-3-yl)-2-methyl-1H-pyrazol-3-one
—— (5E)-3-benzyl-2-benzylimino-5-[[3-bromo-5-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]methylidene]-1,3-thiazolidin-4-one —— C34H31BrN2O3S
(5E)-3-benzyl-2-benzylimino-5-[[3-bromo-5-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]methylidene]-1,3-thiazolidin-4-one
—— (5E)-5-[[3-bromo-5-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]methylidene]-3-phenyl-2-phenylimino-1,3-thiazolidin-4-one —— C32H27BrN2O3S
(5E)-5-[[3-bromo-5-ethoxy-4-[(4-methylphenyl)methoxy]phenyl]methylidene]-3-phenyl-2-phenylimino-1,3-thiazolidin-4-one
—— (5E)-3-(4-chlorophenyl)-5-(3-methylbutylidene)-2-sulfanylidene-1,3-thiazolidin-4-one —— C14H14ClNOS2
(5E)-3-(4-chlorophenyl)-5-(3-methylbutylidene)-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[(3,5-ditert-butyl-4-hydroxyphenyl)methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C19H23N3O2S
(5E)-5-[(3,5-ditert-butyl-4-hydroxyphenyl)methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— (5Z)-3-benzyl-5-[[3-bromo-5-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H21BrFNO3S2
(5Z)-3-benzyl-5-[[3-bromo-5-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one