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—— (5S,6R,7S)-7-(1,5-dimethylpyrazol-4-yl)-5-hydroxy-5-methyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C12H17N7O2
(5S,6R,7S)-7-(1,5-dimethylpyrazol-4-yl)-5-hydroxy-5-methyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (5S,6S,7R)-7-(1,5-dimethylpyrazol-4-yl)-5-hydroxy-5-methyl-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C12H17N7O2
(5S,6S,7R)-7-(1,5-dimethylpyrazol-4-yl)-5-hydroxy-5-methyl-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (5Z)-5-[[4-[(4-chlorophenyl)methoxy]-3-methoxyphenyl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C18H15ClN2O3S
(5Z)-5-[[4-[(4-chlorophenyl)methoxy]-3-methoxyphenyl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5Z)-5-[(3-methylphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C11H10N2OS
(5Z)-5-[(3-methylphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5S,7S)-3-(4-methoxyphenyl)-N-[[2-(pyrazol-1-ylmethyl)phenyl]methyl]adamantane-1-carboxamide —— C29H33N3O2
(5S,7S)-3-(4-methoxyphenyl)-N-[[2-(pyrazol-1-ylmethyl)phenyl]methyl]adamantane-1-carboxamide
—— [(5S)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-[(3R)-1-methylsulfonylpiperidin-3-yl]methanone —— C11H16F3N3O4S
[(5S)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-[(3R)-1-methylsulfonylpiperidin-3-yl]methanone
—— [(5S)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-[(3S)-1-methylsulfonylpiperidin-3-yl]methanone —— C11H16F3N3O4S
[(5S)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-[(3S)-1-methylsulfonylpiperidin-3-yl]methanone
—— [5-[[(2-chlorobenzoyl)-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C26H24Cl3NO6S
[5-[[(2-chlorobenzoyl)-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— (5Z)-2-cyclohexylimino-5-[[2-(difluoromethoxy)phenyl]methylidene]-1,3-thiazolidin-4-one —— C17H18F2N2O2S
(5Z)-2-cyclohexylimino-5-[[2-(difluoromethoxy)phenyl]methylidene]-1,3-thiazolidin-4-one
—— (5Z)-5-[[3-ethoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C20H20N2O4S
(5Z)-5-[[3-ethoxy-4-(2-phenoxyethoxy)phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5Z)-3-[[bis(2-hydroxyethyl)amino]methyl]-5-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-1,3-thiazolidine-2,4-dione —— C19H19ClN2O5S
(5Z)-3-[[bis(2-hydroxyethyl)amino]methyl]-5-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-1,3-thiazolidine-2,4-dione
—— (5Z)-5-[[3-ethoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C21H22N2O4S
(5Z)-5-[[3-ethoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5Z)-2-cyclohexylimino-5-[[3-(difluoromethoxy)-4-methoxyphenyl]methylidene]-1,3-thiazolidin-4-one —— C18H20F2N2O3S
(5Z)-2-cyclohexylimino-5-[[3-(difluoromethoxy)-4-methoxyphenyl]methylidene]-1,3-thiazolidin-4-one
—— (5E)-3-[4-(dimethylamino)phenyl]-5-[(4-methylphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C19H18N2OS2
(5E)-3-[4-(dimethylamino)phenyl]-5-[(4-methylphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5-phenyl-1,2-oxazol-3-yl)methyl 3-(5-cyano-2,4-dimethyl-6-oxo-1H-pyridin-3-yl)propanoate —— C21H19N3O4
(5-phenyl-1,2-oxazol-3-yl)methyl 3-(5-cyano-2,4-dimethyl-6-oxo-1H-pyridin-3-yl)propanoate
—— [5-[[3,3-dimethylbutanoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C25H31Cl2NO6S
[5-[[3,3-dimethylbutanoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— (5Z)-5-[(2-chloro-7-methylquinolin-3-yl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C14H10ClN3OS
(5Z)-5-[(2-chloro-7-methylquinolin-3-yl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— 5-(methylsulfamoyl)-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]furan-2-carboxamide —— C16H22N2O4S
5-(methylsulfamoyl)-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]furan-2-carboxamide
—— 5-(tert-butylsulfamoyl)-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]furan-2-carboxamide —— C19H28N2O4S
5-(tert-butylsulfamoyl)-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]furan-2-carboxamide
—— (5Z)-5-[[4-(difluoromethoxy)-3-methoxyphenyl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C12H10F2N2O3S
(5Z)-5-[[4-(difluoromethoxy)-3-methoxyphenyl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5Z)-5-[(4-bromo-3-nitrophenyl)methylidene]-2-cyclohexylimino-1,3-thiazolidin-4-one —— C16H16BrN3O3S
(5Z)-5-[(4-bromo-3-nitrophenyl)methylidene]-2-cyclohexylimino-1,3-thiazolidin-4-one
—— [5-[[3,3-dimethylbutanoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C25H31Cl2NO6S
[5-[[3,3-dimethylbutanoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— (5E)-3-[4-(dimethylamino)phenyl]-5-[(3-methylthiophen-2-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C17H16N2OS3
(5E)-3-[4-(dimethylamino)phenyl]-5-[(3-methylthiophen-2-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— [5-[[(2-fluorobenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C26H24Cl2FNO6S
[5-[[(2-fluorobenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— [5-[[furan-2-carbonyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C24H23Cl2NO7S
[5-[[furan-2-carbonyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— 5-(tert-butylsulfamoyl)-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]furan-2-carboxamide —— C19H28N2O4S
5-(tert-butylsulfamoyl)-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]furan-2-carboxamide
—— (5R,7R)-3-(tetrazol-2-yl)-N-(1,3-thiazol-2-yl)adamantane-1-carboxamide —— C15H18N6OS
(5R,7R)-3-(tetrazol-2-yl)-N-(1,3-thiazol-2-yl)adamantane-1-carboxamide
—— (5R)-5-(2,5-difluorophenyl)-3-[(2R)-2-hydroxy-3-morpholin-4-ylpropyl]-5-methylimidazolidine-2,4-dione —— C17H21F2N3O4
(5R)-5-(2,5-difluorophenyl)-3-[(2R)-2-hydroxy-3-morpholin-4-ylpropyl]-5-methylimidazolidine-2,4-dione
—— [5-[[(3-fluorobenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C26H24Cl2FNO6S
[5-[[(3-fluorobenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— (5Z)-5-[(4-bromothiophen-2-yl)methylidene]-2-cyclohexylimino-1,3-thiazolidin-4-one —— C14H15BrN2OS2
(5Z)-5-[(4-bromothiophen-2-yl)methylidene]-2-cyclohexylimino-1,3-thiazolidin-4-one
—— (5Z)-5-[[2-(difluoromethoxy)-3-ethoxyphenyl]methylidene]-2-sulfanylideneimidazolidin-4-one —— C13H12F2N2O3S
(5Z)-5-[[2-(difluoromethoxy)-3-ethoxyphenyl]methylidene]-2-sulfanylideneimidazolidin-4-one
—— [5-[[(2-chlorobenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C26H24Cl3NO6S
[5-[[(2-chlorobenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— 5-(methylsulfamoyl)-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]furan-2-carboxamide —— C16H22N2O4S
5-(methylsulfamoyl)-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]furan-2-carboxamide
—— (5S,7S)-3-(tetrazol-2-yl)-N-(1,3-thiazol-2-yl)adamantane-1-carboxamide —— C15H18N6OS
(5S,7S)-3-(tetrazol-2-yl)-N-(1,3-thiazol-2-yl)adamantane-1-carboxamide
—— [5-[[furan-2-carbonyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C24H23Cl2NO7S
[5-[[furan-2-carbonyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— 5,6-dichloro-2-[(3R,4R)-4-hydroxy-1,1-dioxothiolan-3-yl]isoindole-1,3-dione —— C12H9Cl2NO5S
5,6-dichloro-2-[(3R,4R)-4-hydroxy-1,1-dioxothiolan-3-yl]isoindole-1,3-dione
—— [5-[[(3-fluorobenzoyl)-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C26H24Cl2FNO6S
[5-[[(3-fluorobenzoyl)-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— [(5S)-3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[(5S,7S)-3-(tetrazol-2-yl)-1-adamantyl]methanone —— C17H20F4N6O2
[(5S)-3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[(5S,7S)-3-(tetrazol-2-yl)-1-adamantyl]methanone
—— (5R)-3-[(2S)-2-hydroxy-3-(3-methylphenoxy)propyl]-5-methyl-5-(4-propan-2-ylphenyl)imidazolidine-2,4-dione —— C23H28N2O4
(5R)-3-[(2S)-2-hydroxy-3-(3-methylphenoxy)propyl]-5-methyl-5-(4-propan-2-ylphenyl)imidazolidine-2,4-dione
—— [5-[[[(2R)-butan-2-yl]-(2-chlorobenzoyl)amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C25H24Cl3NO5S
[5-[[[(2R)-butan-2-yl]-(2-chlorobenzoyl)amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— (5S,10bS)-1'-benzyl-9-bromo-2-(4-methylphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one —— C31H24BrN3O2
(5S,10bS)-1'-benzyl-9-bromo-2-(4-methylphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one
—— [5-[[(2-chlorobenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3-(trifluoromethyl)benzenesulfonate —— C27H25ClF3NO6S
[5-[[(2-chlorobenzoyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] 3-(trifluoromethyl)benzenesulfonate
—— 5,6-dichloro-2-[(2R)-3-(2,6-dimethylphenoxy)-2-hydroxypropyl]isoindole-1,3-dione —— C19H17Cl2NO4
5,6-dichloro-2-[(2R)-3-(2,6-dimethylphenoxy)-2-hydroxypropyl]isoindole-1,3-dione
—— (5R,7R)-N-(2-methoxy-5-methylphenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C21H26N4O2
(5R,7R)-N-(2-methoxy-5-methylphenyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5E)-5-(5-bromo-1,7-dimethyl-2-oxoindol-3-ylidene)-3-(3,4-dimethylphenyl)-2-(3,4-dimethylphenyl)imino-1,3-thiazolidin-4-one —— C29H26BrN3O2S
(5E)-5-(5-bromo-1,7-dimethyl-2-oxoindol-3-ylidene)-3-(3,4-dimethylphenyl)-2-(3,4-dimethylphenyl)imino-1,3-thiazolidin-4-one
—— [5-[[[(2S)-butan-2-yl]-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate —— C25H24Cl2FNO5S
[5-[[[(2S)-butan-2-yl]-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] 3,4-dichlorobenzenesulfonate
—— (5S,7S)-N-pyridin-4-yl-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C18H21N5O
(5S,7S)-N-pyridin-4-yl-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5R,7R)-3-(3-chloro-1,2,4-triazol-1-yl)-N-propyladamantane-1-carboxamide —— C16H23ClN4O
(5R,7R)-3-(3-chloro-1,2,4-triazol-1-yl)-N-propyladamantane-1-carboxamide
—— (5S,7S)-N-(4-chloro-2-methylphenyl)-3-(3-chloro-1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C20H22Cl2N4O
(5S,7S)-N-(4-chloro-2-methylphenyl)-3-(3-chloro-1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (5S,7R)-N-[(6S)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H30F3N5O2S
(5S,7R)-N-[(6S)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide