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—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-(4-oxoquinazolin-3-yl)acetate —— C20H14ClN3O4
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-(4-oxoquinazolin-3-yl)acetate
—— (5S)-1-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-(1,5-dimethylpyrazol-4-yl)-4-[hydroxy-(1,3,5-trimethylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione —— C25H33N5O3
(5S)-1-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-(1,5-dimethylpyrazol-4-yl)-4-[hydroxy-(1,3,5-trimethylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione
—— 5-chloro-N-[(4S)-3,4-dihydro-2H-chromen-4-yl]thiophene-2-carboxamide —— C14H12ClNO2S
5-chloro-N-[(4S)-3,4-dihydro-2H-chromen-4-yl]thiophene-2-carboxamide
—— 5-bromo-N-[(4-ethoxyphenyl)methyl]-N-methylthiophene-2-sulfonamide —— C14H16BrNO3S2
5-bromo-N-[(4-ethoxyphenyl)methyl]-N-methylthiophene-2-sulfonamide
—— 5-bromo-2-chloro-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]benzamide —— C16H13BrClNO2
5-bromo-2-chloro-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]benzamide
—— (5R)-1-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-(1,5-dimethylpyrazol-4-yl)-4-[hydroxy-(1,3,5-trimethylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione —— C25H33N5O3
(5R)-1-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-(1,5-dimethylpyrazol-4-yl)-4-[hydroxy-(1,3,5-trimethylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione
—— (5E)-5-[[4-(4-benzylpiperazine-1-carbonyl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C22H21N3O3S
(5E)-5-[[4-(4-benzylpiperazine-1-carbonyl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— 5-[[(1R)-2-(2,2-dimethylpropanoyl)-1-(3-fluorophenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide —— C32H38FN3O4
5-[[(1R)-2-(2,2-dimethylpropanoyl)-1-(3-fluorophenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide
—— 5-[[(1S)-2-(furan-2-carbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide —— C32H32N2O6
5-[[(1S)-2-(furan-2-carbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide
—— (5S)-1-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-(1,5-dimethylpyrazol-4-yl)-4-[hydroxy-(1,3,5-trimethylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione —— C25H33N5O3
(5S)-1-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-(1,5-dimethylpyrazol-4-yl)-4-[hydroxy-(1,3,5-trimethylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione
—— 5-[[(1S)-2-(furan-2-carbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide —— C32H32N2O6
5-[[(1S)-2-(furan-2-carbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide
—— 5-[[(1S)-2-(2,2-dimethylpropanoyl)-1-(3-fluorophenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide —— C32H38FN3O4
5-[[(1S)-2-(2,2-dimethylpropanoyl)-1-(3-fluorophenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide
—— 5-[[(1S)-2-(cyclopentanecarbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide —— C34H41N3O4
5-[[(1S)-2-(cyclopentanecarbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide
—— 5-bromo-2-chloro-N-[(4S)-3,4-dihydro-2H-chromen-4-yl]benzamide —— C16H13BrClNO2
5-bromo-2-chloro-N-[(4S)-3,4-dihydro-2H-chromen-4-yl]benzamide
—— 5-[[(1R)-2-(furan-2-carbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide —— C32H32N2O6
5-[[(1R)-2-(furan-2-carbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide
—— (5S)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-7-methyl-N-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C29H35N5O2S
(5S)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-7-methyl-N-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— [5-[[(1R)-1-phenyl-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]furan-2-yl]-thiomorpholin-4-ylmethanone —— C30H28N2O4S2
[5-[[(1R)-1-phenyl-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]furan-2-yl]-thiomorpholin-4-ylmethanone
—— 5-[[(1R)-2-(furan-2-carbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide —— C32H32N2O6
5-[[(1R)-2-(furan-2-carbonyl)-1-(3-methylphenyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide
—— 5-bromo-2-ethoxy-N-[(4-methoxyphenyl)methyl]-N-methylbenzenesulfonamide —— C17H20BrNO4S
5-bromo-2-ethoxy-N-[(4-methoxyphenyl)methyl]-N-methylbenzenesulfonamide
—— (5R)-5-(4-chlorophenyl)-N,N,7-trimethyl-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H27ClN4O2S
(5R)-5-(4-chlorophenyl)-N,N,7-trimethyl-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-[[6-[2-(2-fluorophenoxy)acetyl]-3-oxo-1,4-benzoxazin-4-yl]methyl]-N-[(1S)-1-phenylethyl]furan-2-carboxamide —— C30H25FN2O6
5-[[6-[2-(2-fluorophenoxy)acetyl]-3-oxo-1,4-benzoxazin-4-yl]methyl]-N-[(1S)-1-phenylethyl]furan-2-carboxamide
—— (5S)-5-(4-chlorophenyl)-3-[2-(cyclopropylamino)-2-oxoethyl]-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C21H23ClN4O2S
(5S)-5-(4-chlorophenyl)-3-[2-(cyclopropylamino)-2-oxoethyl]-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-(7-Thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanylmethyl)-3-thiophen-2-yl-1,2,4-oxadiazole —— C16H12N4OS3
5-(7-Thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanylmethyl)-3-thiophen-2-yl-1,2,4-oxadiazole
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-[(3,5-dimethoxybenzoyl)amino]acetate —— C20H21N3O7
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-[(3,5-dimethoxybenzoyl)amino]acetate
—— 5-(4-Chlorophenyl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanylmethyl)-1,3-oxazole —— C16H11ClN4OS
5-(4-Chlorophenyl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanylmethyl)-1,3-oxazole
—— (5S)-3-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C23H27F3N4O2S
(5S)-3-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S)-5-(4-chlorophenyl)-3-[2-[ethyl(methyl)amino]-2-oxoethyl]-7-methyl-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C25H25ClN4O2S
(5S)-5-(4-chlorophenyl)-3-[2-[ethyl(methyl)amino]-2-oxoethyl]-7-methyl-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S,6S,7S)-7-(1,5-dimethylpyrazol-4-yl)-5-hydroxy-5-methyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C12H17N7O2
(5S,6S,7S)-7-(1,5-dimethylpyrazol-4-yl)-5-hydroxy-5-methyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (5S,10bR)-9-bromo-2-(4-methoxyphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-1,3-thiazolidine]-2'-one —— C19H16BrN3O3S
(5S,10bR)-9-bromo-2-(4-methoxyphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-1,3-thiazolidine]-2'-one
—— (5R)-3-[2-(cyclopropylamino)-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C22H23F3N4O2S
(5R)-3-[2-(cyclopropylamino)-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-chlorophenyl)-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C25H25ClN4O2S
(5R)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-chlorophenyl)-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— [5-[[(1S)-1-phenyl-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]furan-2-yl]-thiomorpholin-4-ylmethanone —— C30H28N2O4S2
[5-[[(1S)-1-phenyl-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-isoquinolin-7-yl]oxymethyl]furan-2-yl]-thiomorpholin-4-ylmethanone
—— 5,6-dimethyl-2-[(4-methyl-6-phenylpyrimidin-2-yl)sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C20H18N4OS2
5,6-dimethyl-2-[(4-methyl-6-phenylpyrimidin-2-yl)sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-[(3-methoxybenzoyl)amino]acetate —— C20H17ClN2O5
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-[(3-methoxybenzoyl)amino]acetate
—— (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C22H23F3N4O2S
(5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-chlorophenyl)-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C25H25ClN4O2S
(5S)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-chlorophenyl)-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S)-5-(2,5-dimethylphenyl)-7-methyl-3-(2-oxo-2-pyrrolidin-1-ylethyl)-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H30N4O2S
(5S)-5-(2,5-dimethylphenyl)-7-methyl-3-(2-oxo-2-pyrrolidin-1-ylethyl)-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R,7R)-3-acetamido-N-[(4-methoxyphenyl)methyl]adamantane-1-carboxamide —— C21H28N2O3
(5R,7R)-3-acetamido-N-[(4-methoxyphenyl)methyl]adamantane-1-carboxamide
—— 5-(butylsulfonylamino)-2-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[(1S)-1-phenylethyl]benzenesulfonamide —— C29H38N4O5S2
5-(butylsulfonylamino)-2-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[(1S)-1-phenylethyl]benzenesulfonamide
—— (5S)-5-(4-chlorophenyl)-N,N,7-trimethyl-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H27ClN4O2S
(5S)-5-(4-chlorophenyl)-N,N,7-trimethyl-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C23H27F3N4O2S
(5S)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-5-(4-chlorophenyl)-N,N,7-trimethyl-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H27ClN4O2S
(5R)-5-(4-chlorophenyl)-N,N,7-trimethyl-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-5-(4-chlorophenyl)-3-[2-(cyclopropylamino)-2-oxoethyl]-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C21H23ClN4O2S
(5R)-5-(4-chlorophenyl)-3-[2-(cyclopropylamino)-2-oxoethyl]-N,N,7-trimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-7-methyl-N-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C29H35N5O2S
(5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-7-methyl-N-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S)-5-(4-chlorophenyl)-N,N,7-trimethyl-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H27ClN4O2S
(5S)-5-(4-chlorophenyl)-N,N,7-trimethyl-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-5-(2,5-dimethylphenyl)-7-methyl-3-(2-oxo-2-pyrrolidin-1-ylethyl)-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H30N4O2S
(5R)-5-(2,5-dimethylphenyl)-7-methyl-3-(2-oxo-2-pyrrolidin-1-ylethyl)-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-[[5-(4-Fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C18H14FN5OS2
5-[[5-(4-Fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— (5S,10bS)-9-bromo-2-(4-methoxyphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-1,3-thiazolidine]-2'-one —— C19H16BrN3O3S
(5S,10bS)-9-bromo-2-(4-methoxyphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-1,3-thiazolidine]-2'-one
—— (5R)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C23H27F3N4O2S
(5R)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-N,N,7-trimethyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S,7S)-3-acetamido-N-[(4-methoxyphenyl)methyl]adamantane-1-carboxamide —— C21H28N2O3
(5S,7S)-3-acetamido-N-[(4-methoxyphenyl)methyl]adamantane-1-carboxamide