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—— [(5S)-5-(piperidin-1-ylmethyl)-1,4-thiazepan-4-yl]-thiophen-2-ylmethanone —— C16H24N2OS2
[(5S)-5-(piperidin-1-ylmethyl)-1,4-thiazepan-4-yl]-thiophen-2-ylmethanone
—— (5R)-4-(3-chloro-4-fluorophenyl)sulfonyl-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane —— C16H22ClFN2O2S2
(5R)-4-(3-chloro-4-fluorophenyl)sulfonyl-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane
—— (5S)-5-(pyrrolidin-1-ylmethyl)-N-[2-(trifluoromethyl)phenyl]-1,4-thiazepane-4-carboxamide —— C18H24F3N3OS
(5S)-5-(pyrrolidin-1-ylmethyl)-N-[2-(trifluoromethyl)phenyl]-1,4-thiazepane-4-carboxamide
—— [(5R)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]-[4-(trifluoromethyl)phenyl]methanone —— C18H23F3N2O2S
[(5R)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]-[4-(trifluoromethyl)phenyl]methanone
—— (5S)-4-methylsulfonyl-5-(piperidin-1-ylmethyl)-1,4-thiazepane —— C12H24N2O2S2
(5S)-4-methylsulfonyl-5-(piperidin-1-ylmethyl)-1,4-thiazepane
—— (5R)-N-(4-methoxyphenyl)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide —— C18H27N3O2S
(5R)-N-(4-methoxyphenyl)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide
—— (5S)-N-(2-methylphenyl)-5-(piperidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide —— C19H29N3OS
(5S)-N-(2-methylphenyl)-5-(piperidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide
—— (5-methyl-1-phenylpyrazol-4-yl)-[(5R)-5-(piperidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C22H30N4OS
(5-methyl-1-phenylpyrazol-4-yl)-[(5R)-5-(piperidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— [(5S)-5-[(dimethylamino)methyl]-1,4-thiazepan-4-yl]-(7-methoxy-1-benzofuran-2-yl)methanone —— C18H24N2O3S
[(5S)-5-[(dimethylamino)methyl]-1,4-thiazepan-4-yl]-(7-methoxy-1-benzofuran-2-yl)methanone
—— (5R)-N-(2-methylphenyl)-5-(piperidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide —— C19H29N3OS
(5R)-N-(2-methylphenyl)-5-(piperidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide
—— [(5R)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]-(4-phenylphenyl)methanone —— C23H28N2O2S
[(5R)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]-(4-phenylphenyl)methanone
—— (5R)-4-pyridin-3-ylsulfonyl-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane —— C15H23N3O2S2
(5R)-4-pyridin-3-ylsulfonyl-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane
—— (5S)-5-(pyrrolidin-1-ylmethyl)-4-thiophen-2-ylsulfonyl-1,4-thiazepane —— C14H22N2O2S3
(5S)-5-(pyrrolidin-1-ylmethyl)-4-thiophen-2-ylsulfonyl-1,4-thiazepane
—— (5R)-4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane —— C18H26N2O4S2
(5R)-4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane
—— (5S)-N-[2-(4-methoxyphenyl)ethyl]-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide —— C20H31N3O2S
(5S)-N-[2-(4-methoxyphenyl)ethyl]-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide
—— (5S)-N-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide —— C19H29N3OS
(5S)-N-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide
—— (5S)-4-[(4-chlorophenyl)methylsulfonyl]-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane —— C17H25ClN2O2S2
(5S)-4-[(4-chlorophenyl)methylsulfonyl]-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane
—— (5S)-4-(3-fluoro-4-methoxyphenyl)sulfonyl-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane —— C17H25FN2O3S2
(5S)-4-(3-fluoro-4-methoxyphenyl)sulfonyl-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane
—— [(5S)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]-[4-(trifluoromethoxy)phenyl]methanone —— C18H23F3N2O2S
[(5S)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]-[4-(trifluoromethoxy)phenyl]methanone
—— (5R)-N-benzyl-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide —— C18H27N3OS
(5R)-N-benzyl-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepane-4-carboxamide
—— [(5S)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]-(4-phenylphenyl)methanone —— C23H28N2O2S
[(5S)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]-(4-phenylphenyl)methanone
—— (5-chlorothiophen-2-yl)-[(5R)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C15H21ClN2O2S2
(5-chlorothiophen-2-yl)-[(5R)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— 5-[2-[5-(4-fluorophenyl)tetrazol-2-yl]acetyl]-1-methyl-3H-indol-2-one —— C18H14FN5O2
5-[2-[5-(4-fluorophenyl)tetrazol-2-yl]acetyl]-1-methyl-3H-indol-2-one
—— [(5S)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]-[4-(trifluoromethoxy)phenyl]methanone —— C18H23F3N2O3S
[(5S)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]-[4-(trifluoromethoxy)phenyl]methanone
—— (5R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-methyl-3-[2-(2-morpholin-4-ylethylamino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C30H34ClN5O3S
(5R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-methyl-3-[2-(2-morpholin-4-ylethylamino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-5-(3-chlorophenyl)-N-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H30ClN5O3S
(5R)-5-(3-chlorophenyl)-N-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-[2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-1-methyl-3H-indol-2-one —— C19H14FN3O3S
5-[2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-1-methyl-3H-indol-2-one
—— (5S)-5-(3-chlorophenyl)-N-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H30ClN5O3S
(5S)-5-(3-chlorophenyl)-N-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-(2-methoxyethyl)-4-methyl-1-phenylpyrazole-3-carboxamide —— C24H29N5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-(2-methoxyethyl)-4-methyl-1-phenylpyrazole-3-carboxamide
—— (5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-N,N-diethyl-7-methyl-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C30H37N5O3S
(5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-N,N-diethyl-7-methyl-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3-(1,3-benzothiazol-2-ylsulfanyl)propanoate —— C19H15N3O3S2
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3-(1,3-benzothiazol-2-ylsulfanyl)propanoate
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-(2-methoxyethyl)-4-methyl-1-phenylpyrazole-3-carboxamide —— C24H29N5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-(2-methoxyethyl)-4-methyl-1-phenylpyrazole-3-carboxamide
—— (5S)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-methyl-3-[2-(2-morpholin-4-ylethylamino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C30H34ClN5O3S
(5S)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-methyl-3-[2-(2-morpholin-4-ylethylamino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S,7S)-N-(benzimidazol-1-yl)-3-(4-methoxyphenyl)adamantane-1-carboxamide —— C25H27N3O2
(5S,7S)-N-(benzimidazol-1-yl)-3-(4-methoxyphenyl)adamantane-1-carboxamide
—— (5R,7R)-N-(benzimidazol-1-yl)-3-(4-methoxyphenyl)adamantane-1-carboxamide —— C25H27N3O2
(5R,7R)-N-(benzimidazol-1-yl)-3-(4-methoxyphenyl)adamantane-1-carboxamide
—— (5S)-5-(4-fluorophenyl)-N,7-dimethyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H30FN5O2S
(5S)-5-(4-fluorophenyl)-N,7-dimethyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-5-(4-fluorophenyl)-N,7-dimethyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H30FN5O2S
(5R)-5-(4-fluorophenyl)-N,7-dimethyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H31N5O3S
(5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-[(3-methoxyphenyl)methyl]-2-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one —— C25H32N4O3
5-[(3-methoxyphenyl)methyl]-2-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one
—— (5S)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-N-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C30H35N5O2S
(5S)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-N-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H31N5O3S
(5S)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-N-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C30H35N5O2S
(5R)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-N-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C31H30ClN5O2S
(5R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S,7S)-3-bromo-N-[[3-(1,2,4-triazol-1-ylmethyl)phenyl]methyl]adamantane-1-carboxamide —— C21H25BrN4O
(5S,7S)-3-bromo-N-[[3-(1,2,4-triazol-1-ylmethyl)phenyl]methyl]adamantane-1-carboxamide
—— 5-[(3-methoxyphenyl)methyl]-2-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one —— C25H32N4O3
5-[(3-methoxyphenyl)methyl]-2-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (E)-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enoate —— C21H14N6O3
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (E)-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enoate
—— (5-Acetyl-2-methoxyphenyl)methyl 2-(4-fluorophenoxy)-2-methylpropanoate —— C20H21FO5
(5-Acetyl-2-methoxyphenyl)methyl 2-(4-fluorophenoxy)-2-methylpropanoate
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2S)-2-(4-nitrophenyl)sulfanylpropanoate —— C18H15N3O5S
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2S)-2-(4-nitrophenyl)sulfanylpropanoate
—— (5S)-7-methyl-5-(3-methylphenyl)-3-[2-(2-morpholin-4-ylethylamino)-2-oxoethyl]-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C29H33N5O3S
(5S)-7-methyl-5-(3-methylphenyl)-3-[2-(2-morpholin-4-ylethylamino)-2-oxoethyl]-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S)-5-(3-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H31N5O3S
(5S)-5-(3-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide