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—— 5-(3,5-Dimethoxyphenyl)-3-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-1,3,4-oxadiazole-2-thione —— C20H23N3O3S
5-(3,5-Dimethoxyphenyl)-3-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-1,3,4-oxadiazole-2-thione
—— [(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H27F3N4OS
[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— [5-[(1S)-1-(2-fluorophenoxy)ethyl]-2-sulfanylidene-1,3,4-oxadiazol-3-yl]methyl-methyl-[(2-methylphenyl)methyl]azanium —— C20H23FN3O2S+
[5-[(1S)-1-(2-fluorophenoxy)ethyl]-2-sulfanylidene-1,3,4-oxadiazol-3-yl]methyl-methyl-[(2-methylphenyl)methyl]azanium
—— 5-(4-Chlorophenyl)-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-4-methyl-1,2,4-triazole-3-thione —— C18H18ClFN4S
5-(4-Chlorophenyl)-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-4-methyl-1,2,4-triazole-3-thione
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (2R)-2-(4-cyanophenoxy)propanoate —— C19H17N3O5
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (2R)-2-(4-cyanophenoxy)propanoate
—— 5-chloro-N-[[(5S,7S)-3-chloro-1-adamantyl]methyl]-1-methylimidazole-4-sulfonamide —— C15H21Cl2N3O2S
5-chloro-N-[[(5S,7S)-3-chloro-1-adamantyl]methyl]-1-methylimidazole-4-sulfonamide
—— [(5S,7R)-5-(4-chlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2S)-2-ethylpiperidin-1-yl]methanone —— C21H24ClF3N4O
[(5S,7R)-5-(4-chlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2S)-2-ethylpiperidin-1-yl]methanone
—— 5-[(4-Methoxyphenoxy)methyl]-4-methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-1,2,4-triazole-3-thione —— C21H26N4O2S
5-[(4-Methoxyphenoxy)methyl]-4-methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-1,2,4-triazole-3-thione
—— 5-Fluoro-1-[[methyl-[(2-methylphenyl)methyl]amino]methyl]indole-2,3-dione —— C18H17FN2O2
5-Fluoro-1-[[methyl-[(2-methylphenyl)methyl]amino]methyl]indole-2,3-dione
—— [(5S,7R)-5-(4-chlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2R)-2-ethylpiperidin-1-yl]methanone —— C21H24ClF3N4O
[(5S,7R)-5-(4-chlorophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2R)-2-ethylpiperidin-1-yl]methanone
—— (5R,7R)-N-[3-[(1S)-1-hydroxyethyl]phenyl]-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H23F3N4O2
(5R,7R)-N-[3-[(1S)-1-hydroxyethyl]phenyl]-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H27F3N4OS
[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 5-chloro-N-[[(5R,7R)-3-chloro-1-adamantyl]methyl]-1-methylimidazole-4-sulfonamide —— C15H21Cl2N3O2S
5-chloro-N-[[(5R,7R)-3-chloro-1-adamantyl]methyl]-1-methylimidazole-4-sulfonamide
—— 5-(4-Chlorophenyl)-2-[[5-(furan-2-yl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazole —— C17H13ClN4O2S
5-(4-Chlorophenyl)-2-[[5-(furan-2-yl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazole
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-1,4-dimethylpyrazole-3-carboxylic acid —— C25H27F3N4O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-1,4-dimethylpyrazole-3-carboxylic acid
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 4-acetamidobenzoate —— C18H17N3O5
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 4-acetamidobenzoate
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-methoxy-4-propan-2-yloxyphenyl)prop-2-enoate —— C22H24N2O6
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-methoxy-4-propan-2-yloxyphenyl)prop-2-enoate
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(3-chlorophenoxy)acetate —— C17H15ClN2O5
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(3-chlorophenoxy)acetate
—— (5R,7S)-N-[6-[(1S)-1-hydroxyethyl]-1,3-benzodioxol-5-yl]-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H23F3N4O4
(5R,7S)-N-[6-[(1S)-1-hydroxyethyl]-1,3-benzodioxol-5-yl]-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-[[(1R)-2,2-dichlorocyclopropyl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C9H11Cl2N3S2
5-[[(1R)-2,2-dichlorocyclopropyl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— (5S,7R)-3-bromo-N-[4-chloro-2-[(S)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H21BrClF3N4O2
(5S,7R)-3-bromo-N-[4-chloro-2-[(S)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H27F3N4OS
[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— [(5S,7S)-3-bromo-1-adamantyl]-[4-[3-(3,5-dimethylpyrazol-1-yl)-4-nitrophenyl]piperazin-1-yl]methanone —— C26H32BrN5O3
[(5S,7S)-3-bromo-1-adamantyl]-[4-[3-(3,5-dimethylpyrazol-1-yl)-4-nitrophenyl]piperazin-1-yl]methanone
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-1,4-dimethylpyrazole-3-carboxylic acid —— C25H27F3N4O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-1,4-dimethylpyrazole-3-carboxylic acid
—— [(5R,7R)-3-bromo-1-adamantyl]-[4-[3-(3,5-dimethylpyrazol-1-yl)-4-nitrophenyl]piperazin-1-yl]methanone —— C26H32BrN5O3
[(5R,7R)-3-bromo-1-adamantyl]-[4-[3-(3,5-dimethylpyrazol-1-yl)-4-nitrophenyl]piperazin-1-yl]methanone
—— (5R,7R)-3-chloro-N-[4-[(1S)-1-hydroxyethyl]phenyl]-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H22ClF3N4O2
(5R,7R)-3-chloro-N-[4-[(1S)-1-hydroxyethyl]phenyl]-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[[5-(4-Chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-ethylphenyl)-1,2,4-oxadiazole —— C20H18ClN5OS
5-[[5-(4-Chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-ethylphenyl)-1,2,4-oxadiazole
—— 5-[2-(4-chlorophenyl)sulfanylethylsulfanyl]-2-indol-3-ylidene-3H-1,3,4-oxadiazole —— C18H14ClN3OS2
5-[2-(4-chlorophenyl)sulfanylethylsulfanyl]-2-indol-3-ylidene-3H-1,3,4-oxadiazole
—— [(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(1R,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C22H27F3N4OS
[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(1R,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 3-(thiophene-2-carbonylamino)benzoate —— C22H16N2O4S
(5-Phenyl-1,2-oxazol-3-yl)methyl 3-(thiophene-2-carbonylamino)benzoate
—— (5R,7R)-3-bromo-N-[4-chloro-2-[(S)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H21BrClF3N4O2
(5R,7R)-3-bromo-N-[4-chloro-2-[(S)-hydroxy(phenyl)methyl]phenyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-[6-[(1S)-1-hydroxyethyl]-1,3-benzodioxol-5-yl]-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H23F3N4O4
(5R,7R)-N-[6-[(1S)-1-hydroxyethyl]-1,3-benzodioxol-5-yl]-5-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate —— C21H17N3O3S
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate
—— 5,6-bis(4-methylphenyl)-3-[[(2S)-oxolan-2-yl]methylsulfanyl]-1,2,4-triazine —— C22H23N3OS
5,6-bis(4-methylphenyl)-3-[[(2S)-oxolan-2-yl]methylsulfanyl]-1,2,4-triazine
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 4-methoxynaphthalene-1-carboxylate —— C22H18N2O4
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 4-methoxynaphthalene-1-carboxylate
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,5-difluorophenyl)sulfanylacetate —— C17H11ClF2N2O3S
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,5-difluorophenyl)sulfanylacetate
—— (5-methyl-1,2-oxazol-3-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C15H14FNO4
(5-methyl-1,2-oxazol-3-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— (5S,7R)-3-chloro-N-[1-[2-[[(2S)-1-methoxypropan-2-yl]amino]-2-oxoethyl]pyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H25ClF3N7O3
(5S,7R)-3-chloro-N-[1-[2-[[(2S)-1-methoxypropan-2-yl]amino]-2-oxoethyl]pyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,5-difluorophenyl)sulfanylacetate —— C15H10F2N2O4S
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,5-difluorophenyl)sulfanylacetate
—— [(5S,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2R,6R)-2,4,6-trimethylpiperidin-1-yl]methanone —— C20H25F3N4O2
[(5S,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2R,6R)-2,4,6-trimethylpiperidin-1-yl]methanone
—— (5S,7R)-3-chloro-N-[1-[2-[[(2R)-1-methoxypropan-2-yl]amino]-2-oxoethyl]pyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H25ClF3N7O3
(5S,7R)-3-chloro-N-[1-[2-[[(2R)-1-methoxypropan-2-yl]amino]-2-oxoethyl]pyrazol-4-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2R,4Z)-2-tert-butyl-4-(thiophen-2-ylmethylidene)-2,3-dihydro-1H-acridine-9-carboxylate —— C32H29N3O3S
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2R,4Z)-2-tert-butyl-4-(thiophen-2-ylmethylidene)-2,3-dihydro-1H-acridine-9-carboxylate
—— [(5S,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2S,6S)-2,4,6-trimethylpiperidin-1-yl]methanone —— C20H25F3N4O2
[(5S,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2S,6S)-2,4,6-trimethylpiperidin-1-yl]methanone
—— 5-[[5-(2-Chlorophenyl)tetrazol-2-yl]methyl]-3-(2-methoxyphenyl)-1,2,4-oxadiazole —— C17H13ClN6O2
5-[[5-(2-Chlorophenyl)tetrazol-2-yl]methyl]-3-(2-methoxyphenyl)-1,2,4-oxadiazole
—— [(5S,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2S,6R)-2,4,6-trimethylpiperidin-1-yl]methanone —— C20H25F3N4O2
[(5S,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-[(2S,6R)-2,4,6-trimethylpiperidin-1-yl]methanone
—— 5-[[5-(2-Chlorophenyl)tetrazol-2-yl]methyl]-3-(2-methylphenyl)-1,2,4-oxadiazole —— C17H13ClN6O
5-[[5-(2-Chlorophenyl)tetrazol-2-yl]methyl]-3-(2-methylphenyl)-1,2,4-oxadiazole
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2S,4Z)-2-tert-butyl-4-(thiophen-2-ylmethylidene)-2,3-dihydro-1H-acridine-9-carboxylate —— C32H29N3O3S
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (2S,4Z)-2-tert-butyl-4-(thiophen-2-ylmethylidene)-2,3-dihydro-1H-acridine-9-carboxylate
—— (5S,7R)-5-(1,3-benzodioxol-5-yl)-N-[(6S)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H28F3N5O3S
(5S,7R)-5-(1,3-benzodioxol-5-yl)-N-[(6S)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [(5R)-3-(2-chloro-6-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-[(2S,6S)-2,6-dimethylpiperidin-1-yl]methanone —— C17H20ClFN2O2
[(5R)-3-(2-chloro-6-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-[(2S,6S)-2,6-dimethylpiperidin-1-yl]methanone
—— [(5R)-3-(2-chloro-6-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-[(2R,6R)-2,6-dimethylpiperidin-1-yl]methanone —— C17H20ClFN2O2
[(5R)-3-(2-chloro-6-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-[(2R,6R)-2,6-dimethylpiperidin-1-yl]methanone