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—— (5R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-3-[2-[ethyl(methyl)amino]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H29ClN4O2S
(5R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-3-[2-[ethyl(methyl)amino]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-chloro-2-hydroxybenzoate —— C16H10ClN3O6
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-chloro-2-hydroxybenzoate
—— (5E)-5-[(4-bromophenyl)methylidene]-2-[(2E)-2-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one —— C20H22BrN3OS
(5E)-5-[(4-bromophenyl)methylidene]-2-[(2E)-2-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-chloro-2-hydroxybenzoate —— C14H9ClN2O5
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-chloro-2-hydroxybenzoate
—— 5-[(3-fluorophenyl)methyl]-2-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one —— C24H29FN4O2
5-[(3-fluorophenyl)methyl]-2-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one
—— (5R,7R)-3-chloro-N-[2-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]ethyl]adamantane-1-carboxamide —— C23H27ClN2OS
(5R,7R)-3-chloro-N-[2-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]ethyl]adamantane-1-carboxamide
—— (5R,7R)-N-(2-anilino-2-oxoethyl)-3-bromo-N-methyladamantane-1-carboxamide —— C20H25BrN2O2
(5R,7R)-N-(2-anilino-2-oxoethyl)-3-bromo-N-methyladamantane-1-carboxamide
—— 5-(2-methoxyphenyl)-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]-1,2-oxazole-3-carboxamide —— C21H24N2O3
5-(2-methoxyphenyl)-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]-1,2-oxazole-3-carboxamide
—— 5-[(3-fluorophenyl)methyl]-2-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one —— C24H29FN4O2
5-[(3-fluorophenyl)methyl]-2-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one
—— [5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-[[(2R)-oxolan-2-yl]methoxy]benzoate —— C21H19ClN2O5
[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-[[(2R)-oxolan-2-yl]methoxy]benzoate
—— (5S,7S)-N-(2-anilino-2-oxoethyl)-3-bromo-N-methyladamantane-1-carboxamide —— C20H25BrN2O2
(5S,7S)-N-(2-anilino-2-oxoethyl)-3-bromo-N-methyladamantane-1-carboxamide
—— 5-[[4-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-methyl-1,2-oxazole —— C23H27FN4O2S
5-[[4-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-methyl-1,2-oxazole
—— 5-[[4-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-methyl-1,2-oxazole —— C23H27FN4O2S
5-[[4-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-methyl-1,2-oxazole
—— 5-(4-methylphenyl)-2-[2-oxo-2-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl]sulfanyl-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one —— C28H33N3O2S2
5-(4-methylphenyl)-2-[2-oxo-2-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl]sulfanyl-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one
—— 5-(2-methoxyphenyl)-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]-1,2-oxazole-3-carboxamide —— C21H24N2O3
5-(2-methoxyphenyl)-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]-1,2-oxazole-3-carboxamide
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 3-hydroxynaphthalene-2-carboxylate —— C21H16N2O4
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 3-hydroxynaphthalene-2-carboxylate
—— (5S,7S)-3-chloro-N-[2-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]ethyl]adamantane-1-carboxamide —— C23H27ClN2OS
(5S,7S)-3-chloro-N-[2-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]ethyl]adamantane-1-carboxamide
—— [5-[[[(2R)-butan-2-yl]-(2-chlorobenzoyl)amino]methyl]-2-methoxyphenyl] 3-(trifluoromethyl)benzenesulfonate —— C26H25ClF3NO5S
[5-[[[(2R)-butan-2-yl]-(2-chlorobenzoyl)amino]methyl]-2-methoxyphenyl] 3-(trifluoromethyl)benzenesulfonate
—— (5S,7S)-3-chloro-N-[2-(4-methoxyphenyl)ethyl]adamantane-1-carboxamide —— C20H26ClNO2
(5S,7S)-3-chloro-N-[2-(4-methoxyphenyl)ethyl]adamantane-1-carboxamide
—— (5R,7R)-3-chloro-N-[2-(4-methoxyphenyl)ethyl]adamantane-1-carboxamide —— C20H26ClNO2
(5R,7R)-3-chloro-N-[2-(4-methoxyphenyl)ethyl]adamantane-1-carboxamide
—— 5-[[4-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-methyl-1,2-oxazole —— C23H27FN4O2S
5-[[4-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-methyl-1,2-oxazole
—— (5R,7R)-3-chloro-N-[2-(pyrazin-2-ylamino)ethyl]adamantane-1-carboxamide —— C17H23ClN4O
(5R,7R)-3-chloro-N-[2-(pyrazin-2-ylamino)ethyl]adamantane-1-carboxamide
—— (5S,7S)-3-bromo-N-[2-(pyrazin-2-ylamino)ethyl]adamantane-1-carboxamide —— C17H23BrN4O
(5S,7S)-3-bromo-N-[2-(pyrazin-2-ylamino)ethyl]adamantane-1-carboxamide
—— 5-(4-methylphenyl)-2-[2-oxo-2-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl]sulfanyl-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one —— C28H33N3O2S2
5-(4-methylphenyl)-2-[2-oxo-2-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl]sulfanyl-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one
—— (5R)-5-(2,5-dimethylphenyl)-7-methyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C31H31N5O2S
(5R)-5-(2,5-dimethylphenyl)-7-methyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R,7R)-3-bromo-N-[2-(pyrazin-2-ylamino)ethyl]adamantane-1-carboxamide —— C17H23BrN4O
(5R,7R)-3-bromo-N-[2-(pyrazin-2-ylamino)ethyl]adamantane-1-carboxamide
—— 5-oxo-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C17H19N3O2S
5-oxo-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S,7S)-3-chloro-N-[2-(pyrazin-2-ylamino)ethyl]adamantane-1-carboxamide —— C17H23ClN4O
(5S,7S)-3-chloro-N-[2-(pyrazin-2-ylamino)ethyl]adamantane-1-carboxamide
—— 5-[(4-bromobenzoyl)amino]-2-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H33BrN4O4
5-[(4-bromobenzoyl)amino]-2-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— (5S)-5-(2,5-dimethylphenyl)-7-methyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C31H31N5O2S
(5S)-5-(2,5-dimethylphenyl)-7-methyl-3-[2-oxo-2-(2-pyridin-2-ylethylamino)ethyl]-N-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-5-(4-fluorophenyl)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H28F2N4O2S
(5R)-5-(4-fluorophenyl)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5-Phenyl-1,2-oxazol-3-yl)methyl pyridine-3-carboxylate —— C16H12N2O3
(5-Phenyl-1,2-oxazol-3-yl)methyl pyridine-3-carboxylate
—— 5-[[5-benzyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(3S)-4-(2-methoxybenzoyl)-3-methylpiperazin-1-yl]pentan-1-one —— C34H39N5O3S
5-[[5-benzyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(3S)-4-(2-methoxybenzoyl)-3-methylpiperazin-1-yl]pentan-1-one
—— (5S,7S)-3-(4-methylphenyl)-N-(1H-pyrazol-4-yl)adamantane-1-carboxamide —— C21H25N3O
(5S,7S)-3-(4-methylphenyl)-N-(1H-pyrazol-4-yl)adamantane-1-carboxamide
—— (5S)-5-(4-fluorophenyl)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C27H28F2N4O2S
(5S)-5-(4-fluorophenyl)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-[[5-benzyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(3R)-4-(2-methoxybenzoyl)-3-methylpiperazin-1-yl]pentan-1-one —— C34H39N5O3S
5-[[5-benzyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(3R)-4-(2-methoxybenzoyl)-3-methylpiperazin-1-yl]pentan-1-one
—— 5-oxo-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C17H19N3O2S
5-oxo-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-[(4-bromobenzoyl)amino]-2-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C30H33BrN4O4
5-[(4-bromobenzoyl)amino]-2-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— [5-(5-Bromothiophen-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-chlorobenzoate —— C14H8BrClN2O3S
[5-(5-Bromothiophen-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-chlorobenzoate
—— (5R,7R)-3-(4-methylphenyl)-N-(1H-pyrazol-4-yl)adamantane-1-carboxamide —— C21H25N3O
(5R,7R)-3-(4-methylphenyl)-N-(1H-pyrazol-4-yl)adamantane-1-carboxamide
—— 5-methyl-4-nitro-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]thiophene-2-carboxamide —— C16H20N2O3S
5-methyl-4-nitro-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]thiophene-2-carboxamide
—— 5-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C22H18N4O4
5-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(3,5-dimethylphenoxy)acetate —— C20H20N2O4
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(3,5-dimethylphenoxy)acetate
—— 5,7-Dimethyl-3-[(1-propyltetrazol-5-yl)methylsulfanyl]-[1,2,4]triazolo[4,3-a]pyrimidine —— C12H16N8S
5,7-Dimethyl-3-[(1-propyltetrazol-5-yl)methylsulfanyl]-[1,2,4]triazolo[4,3-a]pyrimidine
—— 5-[(5-Bromo-2-methoxyphenyl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C19H15BrN4O2
5-[(5-Bromo-2-methoxyphenyl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— 5,6-dimethyl-3-(2-methylpropyl)-2-[[(2R)-oxolan-2-yl]methylsulfanyl]thieno[2,3-d]pyrimidin-4-one —— C17H24N2O2S2
5,6-dimethyl-3-(2-methylpropyl)-2-[[(2R)-oxolan-2-yl]methylsulfanyl]thieno[2,3-d]pyrimidin-4-one
—— 5-[2-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C22H25N5O2
5-[2-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2,6-dimethoxybenzoate —— C18H15N3O7
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2,6-dimethoxybenzoate
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 3,5-dimethoxybenzoate —— C16H14N2O6
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 3,5-dimethoxybenzoate
—— 5-methyl-4-nitro-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]thiophene-2-carboxamide —— C16H20N2O3S
5-methyl-4-nitro-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]thiophene-2-carboxamide