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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (11R)-5-[(4-ethenylphenyl)methyl]-11-phenylsulfanyl-11H-benzo[c][1]benzazepin-6-one —— C29H23NOS
(11R)-5-[(4-ethenylphenyl)methyl]-11-phenylsulfanyl-11H-benzo[c][1]benzazepin-6-one
—— (11S)-5-[(4-fluorophenyl)methyl]-11-phenylsulfanyl-11H-benzo[c][1]benzazepin-6-one —— C27H20FNOS
(11S)-5-[(4-fluorophenyl)methyl]-11-phenylsulfanyl-11H-benzo[c][1]benzazepin-6-one
—— 7-[(3S)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C23H31N3O6S
7-[(3S)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— (3R)-N-(2-methylphenyl)-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carboxamide —— C23H27N3O4S
(3R)-N-(2-methylphenyl)-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carboxamide
—— ethyl 1-[(3R)-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carbonyl]piperidine-4-carboxylate —— C24H33N3O6S
ethyl 1-[(3R)-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carbonyl]piperidine-4-carboxylate
—— 7-[(3S)-3-(azepane-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C22H31N3O4S
7-[(3S)-3-(azepane-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— (3S)-N-(2-fluorophenyl)-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carboxamide —— C22H24FN3O4S
(3S)-N-(2-fluorophenyl)-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carboxamide
—— 7-[(3S)-3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C22H31N3O4S
7-[(3S)-3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(3R)-3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C22H31N3O4S
7-[(3R)-3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— ethyl 4-[[(11R)-11-morpholin-4-yl-6,11-dihydrobenzo[c][1]benzazepine-5-carbonyl]amino]benzoate —— C28H29N3O4
ethyl 4-[[(11R)-11-morpholin-4-yl-6,11-dihydrobenzo[c][1]benzazepine-5-carbonyl]amino]benzoate
—— N-[4-[[(2R)-butan-2-yl]carbamoyl]phenyl]-2,3,4,5-tetrahydro-1-benzazepine-1-carboxamide —— C22H27N3O2
N-[4-[[(2R)-butan-2-yl]carbamoyl]phenyl]-2,3,4,5-tetrahydro-1-benzazepine-1-carboxamide
—— 3-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonylamino]-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]propanamide —— C23H27N3O4S
3-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonylamino]-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]propanamide
—— (3R)-N-[2-(4-chlorophenyl)ethyl]-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carboxamide —— C24H28ClN3O4S
(3R)-N-[2-(4-chlorophenyl)ethyl]-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carboxamide
—— (3S)-N-[2-(4-chlorophenyl)ethyl]-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carboxamide —— C24H28ClN3O4S
(3S)-N-[2-(4-chlorophenyl)ethyl]-1-[(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-7-yl)sulfonyl]piperidine-3-carboxamide
—— 2-(2-oxo-4,5-dihydro-3H-1-benzazepin-1-yl)-N-[(2R)-2-phenylpropyl]acetamide —— C21H24N2O2
2-(2-oxo-4,5-dihydro-3H-1-benzazepin-1-yl)-N-[(2R)-2-phenylpropyl]acetamide
—— (3R,3'S)-8-methoxy-N,N-dimethyl-1'-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C23H30N4O5
(3R,3'S)-8-methoxy-N,N-dimethyl-1'-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R)-1'-[[2-(dimethylamino)pyrimidin-5-yl]methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H27N5O2
(3R)-1'-[[2-(dimethylamino)pyrimidin-5-yl]methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-methyl-4'-(morpholine-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H25N3O3
(3S,4'R)-1'-methyl-4'-(morpholine-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[[2-(dimethylamino)pyrimidin-5-yl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H25N5O
(3R)-1'-[[2-(dimethylamino)pyrimidin-5-yl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R,3'S)-1'-(3,6-dihydro-2H-pyran-5-ylmethyl)-8-methoxy-N,N-dimethyl-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C23H31N3O4
(3R,3'S)-1'-(3,6-dihydro-2H-pyran-5-ylmethyl)-8-methoxy-N,N-dimethyl-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3S,4'R)-4'-[(dimethylamino)methyl]-1'-(pyridine-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N4O2
(3S,4'R)-4'-[(dimethylamino)methyl]-1'-(pyridine-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R,3'S)-N,N-dimethyl-1-oxo-1'-(pyrimidine-5-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H23N5O3
(3R,3'S)-N,N-dimethyl-1-oxo-1'-(pyrimidine-5-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3S,3'S)-N,N-dimethyl-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C16H21N3O2
(3S,3'S)-N,N-dimethyl-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3S)-1'-(3,5-dimethyl-1,2-oxazole-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H21N3O3
(3S)-1'-(3,5-dimethyl-1,2-oxazole-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1-[(3S,4R,5S)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carbonyl]piperidine-3-carboxamide —— C19H21N3O4
(3S)-1-[(3S,4R,5S)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carbonyl]piperidine-3-carboxamide
—— (3S,4R,5S)-3,7-dimethyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxylic acid —— C14H13NO4
(3S,4R,5S)-3,7-dimethyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxylic acid
—— (3R,4R,5S)-3-methyl-N-[2-[[(2R)-oxan-2-yl]methoxy]ethyl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C21H26N2O5
(3R,4R,5S)-3-methyl-N-[2-[[(2R)-oxan-2-yl]methoxy]ethyl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3S,4R,5S)-3-methyl-N-(2-methyl-1-morpholin-4-ylpropan-2-yl)-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C21H27N3O4
(3S,4R,5S)-3-methyl-N-(2-methyl-1-morpholin-4-ylpropan-2-yl)-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-N-[(3,4-dimethoxyphenyl)methyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C22H22N2O5
(3R,4R,5S)-N-[(3,4-dimethoxyphenyl)methyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C17H18N2O5S
(3R,4R,5S)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-2,6-dioxo-N-(pyridin-4-ylmethyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C19H17N3O3
(3R,4R,5S)-3-methyl-2,6-dioxo-N-(pyridin-4-ylmethyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-N-[(2,3-dimethoxyphenyl)methyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C22H22N2O5
(3R,4R,5S)-N-[(2,3-dimethoxyphenyl)methyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-N-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C17H18N2O5S
(3R,4R,5S)-N-[(3R)-1,1-dioxothiolan-3-yl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-2,6-dioxo-N-(pyridin-3-ylmethyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C19H17N3O3
(3R,4R,5S)-3-methyl-2,6-dioxo-N-(pyridin-3-ylmethyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3aS,10aS)-2-cyclopentyl-10a-methyl-1,3,3a,4-tetrahydropyrrolo[3,4-c][2]benzazepine-5,10-dione —— C18H22N2O2
(3aS,10aS)-2-cyclopentyl-10a-methyl-1,3,3a,4-tetrahydropyrrolo[3,4-c][2]benzazepine-5,10-dione
—— (3S)-1'-[2-(4-methylsulfonylphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H24N2O4S
(3S)-1'-[2-(4-methylsulfonylphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R,4R,5S)-N-[(3-methoxyphenyl)methyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C21H20N2O4
(3R,4R,5S)-N-[(3-methoxyphenyl)methyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R)-8-methoxy-1'-[(3-methoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O3
(3R)-8-methoxy-1'-[(3-methoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-benzyl-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H24N2O2
(3S)-1'-benzyl-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[2-(4-methoxyphenoxy)ethyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O3
(3S)-1'-[2-(4-methoxyphenoxy)ethyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(4-methoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H24N2O2
(3S)-1'-[(4-methoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R,3'S)-1'-(2,4-dimethyl-1,3-oxazole-5-carbonyl)-N,N-dimethyl-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C22H26N4O4
(3R,3'S)-1'-(2,4-dimethyl-1,3-oxazole-5-carbonyl)-N,N-dimethyl-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R)-1'-(3,4,5-trimethoxybenzoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C23H26N2O5
(3R)-1'-(3,4,5-trimethoxybenzoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— ethyl (3S,4R,5S)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxylate —— C15H15NO4
ethyl (3S,4R,5S)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxylate
—— (3R,3'S)-N,N-diethyl-1'-[(2-methoxypyrimidin-5-yl)methyl]-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C24H31N5O3
(3R,3'S)-N,N-diethyl-1'-[(2-methoxypyrimidin-5-yl)methyl]-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,4R,5S)-N-[(2S)-butan-2-yl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C17H20N2O3
(3R,4R,5S)-N-[(2S)-butan-2-yl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5R)-N-[(2R)-butan-2-yl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C17H20N2O3
(3R,4R,5R)-N-[(2R)-butan-2-yl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R)-1'-[(2S)-1-(3,4-dimethoxyphenyl)propan-2-yl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C25H32N2O4
(3R)-1'-[(2S)-1-(3,4-dimethoxyphenyl)propan-2-yl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R,4R,5R)-N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C23H24N2O5
(3R,4R,5R)-N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3S)-8-methoxy-1'-(1-propan-2-ylpyrazole-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H26N4O3
(3S)-8-methoxy-1'-(1-propan-2-ylpyrazole-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one