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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [1-(5-Chloro-3-methylpyridin-2-yl)piperidin-4-yl]-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone —— C22H25Cl2N3O
[1-(5-Chloro-3-methylpyridin-2-yl)piperidin-4-yl]-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone
—— (7-chlorospiro[3,4-dihydro-2H-1-benzazepine-5,1'-cyclopropane]-1-yl)-(1-pyridin-2-ylpiperidin-4-yl)methanone —— C23H26ClN3O
(7-chlorospiro[3,4-dihydro-2H-1-benzazepine-5,1'-cyclopropane]-1-yl)-(1-pyridin-2-ylpiperidin-4-yl)methanone
—— [1-(5-Chloropyrimidin-2-yl)piperidin-4-yl]-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone —— C20H22Cl2N4O
[1-(5-Chloropyrimidin-2-yl)piperidin-4-yl]-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone
—— (7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(6,7-dihydro-5H-cyclopenta[c]pyridin-3-yl)piperidin-4-yl]methanone —— C24H28ClN3O
(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(6,7-dihydro-5H-cyclopenta[c]pyridin-3-yl)piperidin-4-yl]methanone
—— 2-[4-(7-Chloro-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)piperidin-1-yl]pyridine-3-carbonitrile —— C22H23ClN4O
2-[4-(7-Chloro-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)piperidin-1-yl]pyridine-3-carbonitrile
—— (7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(3-fluoro-5-methylpyridin-2-yl)piperidin-4-yl]methanone —— C22H25ClFN3O
(7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(3-fluoro-5-methylpyridin-2-yl)piperidin-4-yl]methanone
—— 2-(2-Chloropyridine-3-carbonyl)-2-azatricyclo[9.4.0.0,3,8]pentadeca-1(11),3(8),4,6,12,14-hexaene —— C20H15ClN2O
2-(2-Chloropyridine-3-carbonyl)-2-azatricyclo[9.4.0.0,3,8]pentadeca-1(11),3(8),4,6,12,14-hexaene
—— 3-[4-[2-amino-4-(dipropylcarbamoyl)-3H-1-benzazepin-8-yl]phenyl]propanoic acid —— C26H31N3O3
3-[4-[2-amino-4-(dipropylcarbamoyl)-3H-1-benzazepin-8-yl]phenyl]propanoic acid
—— (7-Cyano-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)carbamic acid —— C12H11N3O3
(7-Cyano-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)carbamic acid
—— (7-bromo-1-methyl-2-oxo-4,5-dihydro-3H-1-benzazepin-3-yl)carbamic acid —— C12H13BrN2O3
(7-bromo-1-methyl-2-oxo-4,5-dihydro-3H-1-benzazepin-3-yl)carbamic acid
—— 3-Amino-5-methyl-1-oxido-1,2,3,5-tetrahydro-1-benzazepin-1-ium-4-one —— C11H14N2O2
3-Amino-5-methyl-1-oxido-1,2,3,5-tetrahydro-1-benzazepin-1-ium-4-one
—— 7-(2H-tetrazol-5-yl)-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C11H11N5O
7-(2H-tetrazol-5-yl)-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— [2-oxo-7-(2H-tetrazol-5-yl)-1,3,4,5-tetrahydro-1-benzazepin-3-yl]carbamic acid —— C12H12N6O3
[2-oxo-7-(2H-tetrazol-5-yl)-1,3,4,5-tetrahydro-1-benzazepin-3-yl]carbamic acid
—— N-benzyl-N-(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)-1H-1,2,4-triazole-5-carboxamide —— C20H19N5O2
N-benzyl-N-(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)-1H-1,2,4-triazole-5-carboxamide
—— [2-Oxo-8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1,3,4,5-tetrahydro-1-benzazepin-3-yl]carbamic acid —— C17H23BN2O5
[2-Oxo-8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1,3,4,5-tetrahydro-1-benzazepin-3-yl]carbamic acid
—— 5-benzyl-N-(5-methyl-1,4-dioxo-3,5-dihydro-2H-1-benzazepin-1-ium-3-yl)-1,2-oxazole-3-carboxamide —— C22H20N3O4+
5-benzyl-N-(5-methyl-1,4-dioxo-3,5-dihydro-2H-1-benzazepin-1-ium-3-yl)-1,2-oxazole-3-carboxamide
—— 7-chloro-9-fluoro-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one —— C10H9ClFNO
7-chloro-9-fluoro-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one
—— 3-amino-5-methyl-1-oxo-3,5-dihydro-2H-1-benzazepin-1-ium-4-one —— C11H13N2O2+
3-amino-5-methyl-1-oxo-3,5-dihydro-2H-1-benzazepin-1-ium-4-one
—— (8-Hydroxy-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)carbamic acid —— C11H12N2O4
(8-Hydroxy-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)carbamic acid
—— [2-oxo-8-(2-pyrrolidin-1-ylethoxy)-4,5-dihydro-3H-1-benzazepin-1-yl]carbamic acid —— C17H23N3O4
[2-oxo-8-(2-pyrrolidin-1-ylethoxy)-4,5-dihydro-3H-1-benzazepin-1-yl]carbamic acid
—— 3-amino-5-methyl-1-oxido-3,5-dihydro-2H-1-benzazepin-4-one —— C11H13N2O2-
3-amino-5-methyl-1-oxido-3,5-dihydro-2H-1-benzazepin-4-one
—— (1-Methyl-2,5-dioxo-3,4-dihydro-1-benzazepin-3-yl) carbamate —— C12H12N2O4
(1-Methyl-2,5-dioxo-3,4-dihydro-1-benzazepin-3-yl) carbamate
—— 3-amino-1-methyl-7-(2,2,2-trifluoro-1,1-dihydroxyethyl)-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one —— C13H15F3N2O3
3-amino-1-methyl-7-(2,2,2-trifluoro-1,1-dihydroxyethyl)-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one
—— [2-Oxo-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1,3,4,5-tetrahydro-1-benzazepin-3-yl]carbamic acid —— C17H23BN2O5
[2-Oxo-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1,3,4,5-tetrahydro-1-benzazepin-3-yl]carbamic acid
—— [4-[(2-amino-2-oxoethyl)-propylcarbamoyl]-8-bromo-3H-1-benzazepin-2-yl]carbamic acid —— C17H19BrN4O4
[4-[(2-amino-2-oxoethyl)-propylcarbamoyl]-8-bromo-3H-1-benzazepin-2-yl]carbamic acid
—— [13-cyclohexyl-3-methoxy-6-[methyl-[2-[2-[methyl(sulfamoyl)amino]ethoxy]ethyl]carbamoyl]-7H-indolo[2,1-a][2]benzazepin-10-yl] hydrogen carbonate —— C32H40N4O8S
[13-cyclohexyl-3-methoxy-6-[methyl-[2-[2-[methyl(sulfamoyl)amino]ethoxy]ethyl]carbamoyl]-7H-indolo[2,1-a][2]benzazepin-10-yl] hydrogen carbonate
—— 2-benzyl-3-ethyl-5-[(4-fluorophenyl)methyl]-4-oxo-N-(3-pyrrolidin-1-ylpropyl)-3,5-dihydro-1-benzazepine-7-carboxamide —— C34H38FN3O2
2-benzyl-3-ethyl-5-[(4-fluorophenyl)methyl]-4-oxo-N-(3-pyrrolidin-1-ylpropyl)-3,5-dihydro-1-benzazepine-7-carboxamide
—— tert-butyl (3-(7-((4-((2-acrylamidophenyl)amino)-5-chloropyrimidin-2-yl)amino)-6-methoxy-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)propyl)carbamate 1622000-58-1 C32H38ClN7O5
tert-butyl (3-(7-((4-((2-acrylamidophenyl)amino)-5-chloropyrimidin-2-yl)amino)-6-methoxy-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)propyl)carbamate
—— 9-methyl-2,5-dihydro-1H-1-benzazepine —— C11H13N
9-methyl-2,5-dihydro-1H-1-benzazepine
—— 9-methyl-2,3-dihydro-1H-1-benzazepine —— C11H13N
9-methyl-2,3-dihydro-1H-1-benzazepine
—— 8-(4-Fluorophenyl)-3,14-dimethyl-10,14-diazatetracyclo[8.7.1.05,18.011,17]octadeca-1,3,5(18),7,11(17)-pentaene —— C24H25FN2
8-(4-Fluorophenyl)-3,14-dimethyl-10,14-diazatetracyclo[8.7.1.05,18.011,17]octadeca-1,3,5(18),7,11(17)-pentaene
—— 8-(4-Fluorophenyl)-3,14-dimethyl-10,14-diazatetracyclo[8.7.1.05,18.011,17]octadeca-1,3,5(18),11(17)-tetraene —— C24H27FN2
8-(4-Fluorophenyl)-3,14-dimethyl-10,14-diazatetracyclo[8.7.1.05,18.011,17]octadeca-1,3,5(18),11(17)-tetraene
—— 3,7,14-Trimethyl-7-pyridin-4-yl-10,14-diazatetracyclo[8.7.1.05,18.011,17]octadeca-1,3,5(18),11(17)-tetraene —— C24H29N3
3,7,14-Trimethyl-7-pyridin-4-yl-10,14-diazatetracyclo[8.7.1.05,18.011,17]octadeca-1,3,5(18),11(17)-tetraene
—— [4-(Azepan-1-ylsulfonyl)phenyl]-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)methanone —— C27H28N2O3S
[4-(Azepan-1-ylsulfonyl)phenyl]-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)methanone
—— 1-O-[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] 4-O-methyl (2R)-2-[4-(furan-2-carbonyloxy)-4-methylpentyl]-2-hydroxybutanedioate —— C35H45NO11
1-O-[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] 4-O-methyl (2R)-2-[4-(furan-2-carbonyloxy)-4-methylpentyl]-2-hydroxybutanedioate
—— 1-O-[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] 4-O-methyl (2R)-2-hydroxy-2-[4-methyl-4-(2-phenylacetyl)oxypentyl]butanedioate —— C38H49NO10
1-O-[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] 4-O-methyl (2R)-2-hydroxy-2-[4-methyl-4-(2-phenylacetyl)oxypentyl]butanedioate
—— 1-O-[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] 4-O-methyl (2R)-2-hydroxy-2-[4-methyl-4-(5-methyl-1,2-oxazole-4-carbonyl)oxypentyl]butanedioate —— C35H46N2O11
1-O-[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] 4-O-methyl (2R)-2-hydroxy-2-[4-methyl-4-(5-methyl-1,2-oxazole-4-carbonyl)oxypentyl]butanedioate
—— 2-[(2R)-4-[(1R)-1-(carboxymethylamino)ethyl]-7-(3-chlorophenyl)-2,3-dihydro-1H-3-benzazepin-2-yl]acetic acid —— C22H23ClN2O4
2-[(2R)-4-[(1R)-1-(carboxymethylamino)ethyl]-7-(3-chlorophenyl)-2,3-dihydro-1H-3-benzazepin-2-yl]acetic acid
—— 3-[(3S)-1-[2-(3,4-dimethoxyphenyl)ethyl]piperidin-3-yl]-7,8-dimethoxy-5-methyl-2,5-dihydro-1H-3-benzazepin-4-one —— C28H38N2O5
3-[(3S)-1-[2-(3,4-dimethoxyphenyl)ethyl]piperidin-3-yl]-7,8-dimethoxy-5-methyl-2,5-dihydro-1H-3-benzazepin-4-one
—— N-(2-((5-chloro-2-((1-ethyl-6-methoxy-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidin-4-yl)amino)phenyl)propionamide 1622002-04-3 C26H29ClN6O3
N-(2-((5-chloro-2-((1-ethyl-6-methoxy-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidin-4-yl)amino)phenyl)propionamide
—— 7-amino-6-methoxy-1-(2-morpholin-4-ylethyl)-4,5-dihydro-3H-1-benzazepin-2-one —— C17H25N3O3
7-amino-6-methoxy-1-(2-morpholin-4-ylethyl)-4,5-dihydro-3H-1-benzazepin-2-one
—— 7-amino-6-methoxy-1-(3-morpholin-4-ylpropyl)-4,5-dihydro-3H-1-benzazepin-2-one —— C18H27N3O3
7-amino-6-methoxy-1-(3-morpholin-4-ylpropyl)-4,5-dihydro-3H-1-benzazepin-2-one
—— N-(2-((2-((1-(3-aminopropyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)-5-chloropyrimidin-4-yl)amino)phenyl)propionamide 1622002-03-2 C26H30ClN7O2
N-(2-((2-((1-(3-aminopropyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)-5-chloropyrimidin-4-yl)amino)phenyl)propionamide
—— 4-((2-acrylamidophenyl)amino)-2-((6-methoxy-1-(2-morpholinoethyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidine-5-carboxamide 1622001-63-1 C31H36N8O5
4-((2-acrylamidophenyl)amino)-2-((6-methoxy-1-(2-morpholinoethyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidine-5-carboxamide
—— N-(2-((2-((1-(3-aminopropyl)-6-methoxy-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)-5-chloropyrimidin-4-yl)amino)phenyl)acrylamide 1622000-59-2 C27H30ClN7O3
N-(2-((2-((1-(3-aminopropyl)-6-methoxy-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)-5-chloropyrimidin-4-yl)amino)phenyl)acrylamide
—— N-(2-((5-chloro-2-((6-methoxy-1-(3-morpholinopropyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide 1622000-57-0 C31H36ClN7O4
N-(2-((5-chloro-2-((6-methoxy-1-(3-morpholinopropyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide
—— 3-(7-amino-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-1-yl)propylcarbamic acid —— C15H21N3O4
3-(7-amino-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-1-yl)propylcarbamic acid
—— 4-((2-acrylamidophenyl)amino)-2-((6-methoxy-1-(3-morpholinopropyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidine-5-carboxamide 1622001-62-0 C32H38N8O5
4-((2-acrylamidophenyl)amino)-2-((6-methoxy-1-(3-morpholinopropyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidine-5-carboxamide
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-naphthalen-1-ylethanone —— C26H21NO
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-naphthalen-1-ylethanone
—— 1-ethyl-3-[6-(4-fluorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]urea —— C21H19FN4O2
1-ethyl-3-[6-(4-fluorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]urea