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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,3,3a,5,10,10a-hexahydro-1H-cyclopenta[c][1]benzazepin-4-one —— C13H15NO
2,3,3a,5,10,10a-hexahydro-1H-cyclopenta[c][1]benzazepin-4-one
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[3-(3-methylbutoxy)phenoxy]ethanone —— C27H29NO3
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[3-(3-methylbutoxy)phenoxy]ethanone
—— 9-Ethoxy-2-[(3-hydroxyphenyl)methyl]-1,3,4,5-tetrahydro-2-benzazepine-7-carboxamide —— C20H24N2O3
9-Ethoxy-2-[(3-hydroxyphenyl)methyl]-1,3,4,5-tetrahydro-2-benzazepine-7-carboxamide
—— 2-Fluoro-8-hydroxy-4-methoxy-11-oxa-5-azatetracyclo[8.6.1.01,12.06,17]heptadeca-2,4,6(17),7,9-pentaene-15-carbaldehyde —— C17H16FNO4
2-Fluoro-8-hydroxy-4-methoxy-11-oxa-5-azatetracyclo[8.6.1.01,12.06,17]heptadeca-2,4,6(17),7,9-pentaene-15-carbaldehyde
—— Propan-2-ylsulfinyl 19-cyclohexyl-5-methoxy-9-methyl-10-(3-oxa-7,10-diazatricyclo[3.3.3.01,5]undecane-7-carbonyl)-12-azapentacyclo[10.7.0.02,7.08,10.013,18]nonadeca-1(19),2(7),3,5,14,16-hexaene-15-carboxylate —— C39H49N3O6S
Propan-2-ylsulfinyl 19-cyclohexyl-5-methoxy-9-methyl-10-(3-oxa-7,10-diazatricyclo[3.3.3.01,5]undecane-7-carbonyl)-12-azapentacyclo[10.7.0.02,7.08,10.013,18]nonadeca-1(19),2(7),3,5,14,16-hexaene-15-carboxylate
—— 2-(2,4,6-Trifluorobenzoyl)-1,3,4,5-tetrahydro-2-benzazepine-7-carboxamide —— C18H15F3N2O2
2-(2,4,6-Trifluorobenzoyl)-1,3,4,5-tetrahydro-2-benzazepine-7-carboxamide
—— 3-[3-[(4-ethyl-3-methoxy-7-bicyclo[4.2.0]octa-1,3,5-trienyl)methyl-methylamino]propyl]-7-methoxy-8-methyl-2,5-dihydro-1H-3-benzazepin-4-one —— C28H38N2O3
3-[3-[(4-ethyl-3-methoxy-7-bicyclo[4.2.0]octa-1,3,5-trienyl)methyl-methylamino]propyl]-7-methoxy-8-methyl-2,5-dihydro-1H-3-benzazepin-4-one
—— (3S)-2-butyl-3-(cyclopropylmethyl)-N'-[(7S)-5-[[3-(2,4-dichlorophenyl)phenyl]methyl]-6-oxo-7H-benzo[d][1]benzazepin-7-yl]butanediamide —— C39H39Cl2N3O3
(3S)-2-butyl-3-(cyclopropylmethyl)-N'-[(7S)-5-[[3-(2,4-dichlorophenyl)phenyl]methyl]-6-oxo-7H-benzo[d][1]benzazepin-7-yl]butanediamide
—— 2',2',5,6',6',11a-Hexamethyl-4,6,7,11a-tetrahydrospiro[1,3-oxazolo[3',4':1,2]azepino[5,4,3-cd]indole-11,4'-piperidin]-9-one —— C23H31N3O2
2',2',5,6',6',11a-Hexamethyl-4,6,7,11a-tetrahydrospiro[1,3-oxazolo[3',4':1,2]azepino[5,4,3-cd]indole-11,4'-piperidin]-9-one
—— 2-[2-(4-methoxyphenoxy)ethylsulfanyl]-4,5-dimethyl-4,5-dihydro-3H-1-benzazepine —— C21H25NO2S
2-[2-(4-methoxyphenoxy)ethylsulfanyl]-4,5-dimethyl-4,5-dihydro-3H-1-benzazepine
—— 4-[[2-(2,2-dimethylpropyl)-5-[(4-hydroxyoxan-4-yl)methyl]-4,5-dihydro-3H-1-benzazepin-8-yl]sulfonyl]piperidine-1-carboxamide —— C27H41N3O5S
4-[[2-(2,2-dimethylpropyl)-5-[(4-hydroxyoxan-4-yl)methyl]-4,5-dihydro-3H-1-benzazepin-8-yl]sulfonyl]piperidine-1-carboxamide
—— tert-butyl 2-[3-[2-[3-(4,5-dihydro-1H-imidazol-2-yl)propylamino]-2-oxoethyl]-4-oxo-2,5-dihydro-1H-3-benzazepin-5-yl]acetate —— C24H34N4O4
tert-butyl 2-[3-[2-[3-(4,5-dihydro-1H-imidazol-2-yl)propylamino]-2-oxoethyl]-4-oxo-2,5-dihydro-1H-3-benzazepin-5-yl]acetate
—— Ethyl 2-(2-ethoxy-2-oxoethylidene)-5,5-dimethyl-3-(2,2,7-trimethyl-1,3-dihydro-3-benzazepin-4-yl)pyrrolidine-3-carboxylate —— C26H36N2O4
Ethyl 2-(2-ethoxy-2-oxoethylidene)-5,5-dimethyl-3-(2,2,7-trimethyl-1,3-dihydro-3-benzazepin-4-yl)pyrrolidine-3-carboxylate
—— 2-[[(1R,3S,12R,16R)-4-(benzylcarbamoyl)-9-bromo-3-(hydroxymethyl)-8-methoxy-16-methyl-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-14-yl]amino]acetic acid —— C28H32BrN3O6
2-[[(1R,3S,12R,16R)-4-(benzylcarbamoyl)-9-bromo-3-(hydroxymethyl)-8-methoxy-16-methyl-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-14-yl]amino]acetic acid
—— Ethyl 2-(2-ethoxy-2-oxoethylidene)-5,5-dimethyl-3-(2,2,7-trimethyl-1,3-dihydro-3-benzazepin-3-ium-4-yl)pyrrolidine-3-carboxylate —— C26H37N2O4+
Ethyl 2-(2-ethoxy-2-oxoethylidene)-5,5-dimethyl-3-(2,2,7-trimethyl-1,3-dihydro-3-benzazepin-3-ium-4-yl)pyrrolidine-3-carboxylate
—— 6-Ethyl-6-pentan-2-ylpyrido[2,1-a][2]benzazepin-5-ium —— C21H26N+
6-Ethyl-6-pentan-2-ylpyrido[2,1-a][2]benzazepin-5-ium
—— 2-[(5-Butyl-2-methylpyridin-3-yl)amino]-9-(trifluoromethyl)-5,7-dihydropyrimido[5,4-d][1]benzazepin-6-one —— C23H22F3N5O
2-[(5-Butyl-2-methylpyridin-3-yl)amino]-9-(trifluoromethyl)-5,7-dihydropyrimido[5,4-d][1]benzazepin-6-one
—— Methyl 2-[1-[4-bromo-2-(trifluoromethyl)benzoyl]-4,4-difluoro-2,3-dihydro-1-benzazepin-5-ylidene]acetate —— C21H15BrF5NO3
Methyl 2-[1-[4-bromo-2-(trifluoromethyl)benzoyl]-4,4-difluoro-2,3-dihydro-1-benzazepin-5-ylidene]acetate
—— (2S)-2-fluoro-2-methyl-3-oxo-3-[[6-oxo-5-(2-phenylmethoxyethyl)-7H-benzo[d][1]benzazepin-7-yl]amino]propanoic acid —— C27H25FN2O5
(2S)-2-fluoro-2-methyl-3-oxo-3-[[6-oxo-5-(2-phenylmethoxyethyl)-7H-benzo[d][1]benzazepin-7-yl]amino]propanoic acid
—— 2-(1-benzyl-4,5-didehydro-3,6-dihydro-2H-pyridin-2-yl)-1-(2,3,4,5-tetrahydro-1H-1-benzazepin-8-yl)propan-1-one —— C25H28N2O
2-(1-benzyl-4,5-didehydro-3,6-dihydro-2H-pyridin-2-yl)-1-(2,3,4,5-tetrahydro-1H-1-benzazepin-8-yl)propan-1-one
—— 8,8-Diethyl-9,10-dihydroisoquinolino[1,2-a][2]benzazepin-7-ium —— C22H24N+
8,8-Diethyl-9,10-dihydroisoquinolino[1,2-a][2]benzazepin-7-ium
—— (3S)-2-butyl-3-(cyclobutylmethyl)-N'-[(7S)-6-oxo-5-[(3-phenoxyphenyl)methyl]-7H-benzo[d][1]benzazepin-7-yl]butanediamide —— C40H43N3O4
(3S)-2-butyl-3-(cyclobutylmethyl)-N'-[(7S)-6-oxo-5-[(3-phenoxyphenyl)methyl]-7H-benzo[d][1]benzazepin-7-yl]butanediamide
—— methyl 2-[5-methyl-6-oxo-3-[3-(pyridin-2-ylamino)propoxy]-11H-benzo[c][1]benzazepin-11-yl]acetate —— C26H27N3O4
methyl 2-[5-methyl-6-oxo-3-[3-(pyridin-2-ylamino)propoxy]-11H-benzo[c][1]benzazepin-11-yl]acetate
—— tert-butyl N-methyl-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)carbamate —— C16H24N2O2
tert-butyl N-methyl-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)carbamate
—— tert-butyl 4-methyl-3-oxo-7,8,9,10-tetrahydro-6H-[1,4]oxazino[2,3-h][1]benzazepine-8-carboxylate —— C18H24N2O4
tert-butyl 4-methyl-3-oxo-7,8,9,10-tetrahydro-6H-[1,4]oxazino[2,3-h][1]benzazepine-8-carboxylate
—— 8-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-4-methylsulfonyl-3,6,7,8,9,10-hexahydro-2H-[1,4]oxazino[2,3-h][1]benzazepine —— C29H34N6O3S2
8-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-4-methylsulfonyl-3,6,7,8,9,10-hexahydro-2H-[1,4]oxazino[2,3-h][1]benzazepine
—— 2-chloro-5-fluoro-N-[5-(2'-nitrosospiro[3,5-dihydro-2H-1-benzazepine-4,1'-cyclopentane]-1-carbonyl)pyridin-2-yl]benzamide —— C27H24ClFN4O3
2-chloro-5-fluoro-N-[5-(2'-nitrosospiro[3,5-dihydro-2H-1-benzazepine-4,1'-cyclopentane]-1-carbonyl)pyridin-2-yl]benzamide
—— 1-[4-Chloro-9-(1-phenylethylamino)-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C20H20ClF3N2O
1-[4-Chloro-9-(1-phenylethylamino)-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— (1R,2S)-2-[formyl(piperazin-1-yl)amino]-N-[(3S)-5-methyl-2-oxo-1-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)hexan-3-yl]cyclohexane-1-carboxamide —— C29H45N5O3
(1R,2S)-2-[formyl(piperazin-1-yl)amino]-N-[(3S)-5-methyl-2-oxo-1-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)hexan-3-yl]cyclohexane-1-carboxamide
—— 7-[(5S)-5-acetamido-2-oxo-1,3-oxazolidin-3-yl]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxylic acid —— C16H19N3O5
7-[(5S)-5-acetamido-2-oxo-1,3-oxazolidin-3-yl]-1,2,4,5-tetrahydro-3-benzazepine-3-carboxylic acid
—— methyl 10-butanoyl-13-cyclohexyl-3-methoxy-7H-indolo[2,1-a][2]benzazepine-6-carboxylate —— C30H33NO4
methyl 10-butanoyl-13-cyclohexyl-3-methoxy-7H-indolo[2,1-a][2]benzazepine-6-carboxylate
—— 4-[fluoro-[7-(2-fluorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid —— C25H16F2N4O2
4-[fluoro-[7-(2-fluorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid
—— 3H-1-benzazepine-2-carbonitrile —— C11H8N2
3H-1-benzazepine-2-carbonitrile
—— 7-Methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepin-1-ium 1-oxide —— C12H13F3NO+
7-Methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepin-1-ium 1-oxide
—— 3,6,10-Trioxa-13-azapentacyclo[10.8.1.02,7.09,20.014,19]henicosa-1(20),2(7),8,11,14,16,18-heptaene —— C17H13NO3
3,6,10-Trioxa-13-azapentacyclo[10.8.1.02,7.09,20.014,19]henicosa-1(20),2(7),8,11,14,16,18-heptaene
—— 3-methyl-5-nitroso-2,5-dihydro-1H-3-benzazepin-4-one —— C11H12N2O2
3-methyl-5-nitroso-2,5-dihydro-1H-3-benzazepin-4-one
—— 3-[2-(4-Chlorophenoxy)ethyl]-6-fluoro-1,2,4,5-tetrahydro-3-benzazepine-8-carboxamide —— C19H20ClFN2O2
3-[2-(4-Chlorophenoxy)ethyl]-6-fluoro-1,2,4,5-tetrahydro-3-benzazepine-8-carboxamide
—— 4-[7-[2-(3-cyano-4-propan-2-yloxyphenyl)-4,5-dihydro-1,3-oxazol-4-yl]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-N,N-dimethylbutanamide —— C29H36N4O3
4-[7-[2-(3-cyano-4-propan-2-yloxyphenyl)-4,5-dihydro-1,3-oxazol-4-yl]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-N,N-dimethylbutanamide
—— 2-ethylidene-5-propan-2-yl-1-propyl-4,5-dihydro-3H-1-benzazepine —— C18H27N
2-ethylidene-5-propan-2-yl-1-propyl-4,5-dihydro-3H-1-benzazepine
—— 5-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(4-methoxyphenyl)pentanal —— C26H27NO2
5-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(4-methoxyphenyl)pentanal
—— 3-ethyl-5-nitroso-2,5-dihydro-1H-3-benzazepin-4-one —— C12H14N2O2
3-ethyl-5-nitroso-2,5-dihydro-1H-3-benzazepin-4-one
—— 2-[3-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)propyl-methylamino]-3-[[1-[2,5-dioxo-1-(2-oxo-2-phosphanylethyl)pyrrolidin-3-yl]-3-sulfanylpropyl]amino]-3-oxopropanoic acid —— C30H37N4O6PS
2-[3-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)propyl-methylamino]-3-[[1-[2,5-dioxo-1-(2-oxo-2-phosphanylethyl)pyrrolidin-3-yl]-3-sulfanylpropyl]amino]-3-oxopropanoic acid
—— 1-[8-[(5-bromo-2,3-dihydroindol-1-yl)sulfonyl]-2,3,4,5-tetrahydro-1H-3-benzazepin-5-yl]ethanone —— C20H21BrN2O3S
1-[8-[(5-bromo-2,3-dihydroindol-1-yl)sulfonyl]-2,3,4,5-tetrahydro-1H-3-benzazepin-5-yl]ethanone
—— 1,2,3,5,5a,9a-Hexahydro-3-benzazepin-4-one —— C10H13NO
1,2,3,5,5a,9a-Hexahydro-3-benzazepin-4-one
—— 2-(trifluoromethyl)-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine —— C12H11F3N2O
2-(trifluoromethyl)-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine
—— (2S)-2-[[(2R)-2-hydroxy-3-morpholin-4-ylpropyl]amino]-N-(7-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-1-yl)propanamide —— C25H32N4O4
(2S)-2-[[(2R)-2-hydroxy-3-morpholin-4-ylpropyl]amino]-N-(7-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-1-yl)propanamide
—— 4-methylsulfonyl-3,6,7,8,9,10-hexahydro-2H-[1,4]oxazino[2,3-h][1]benzazepine —— C13H18N2O3S
4-methylsulfonyl-3,6,7,8,9,10-hexahydro-2H-[1,4]oxazino[2,3-h][1]benzazepine
—— [13-cyclohexyl-3-methoxy-6-[4-(morpholin-4-ylmethyl)-2-propan-2-ylpyrazol-3-yl]-7H-indolo[2,1-a][2]benzazepin-10-yl]methyl formate —— C37H44N4O4
[13-cyclohexyl-3-methoxy-6-[4-(morpholin-4-ylmethyl)-2-propan-2-ylpyrazol-3-yl]-7H-indolo[2,1-a][2]benzazepin-10-yl]methyl formate
—— 6-fluoro-3-[4-[2-fluoro-6-(1H-pyridin-4-ylidene)hexa-2,4-dien-3-yl]triazol-1-yl]-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one —— C25H22F5N5O
6-fluoro-3-[4-[2-fluoro-6-(1H-pyridin-4-ylidene)hexa-2,4-dien-3-yl]triazol-1-yl]-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one
—— (2Z)-2-(1-acetyl-4,4-difluoro-2,3-dihydro-1-benzazepin-5-ylidene)-N-(2-morpholin-4-ylethyl)acetamide;ethane;toluene —— C29H39F2N3O3
(2Z)-2-(1-acetyl-4,4-difluoro-2,3-dihydro-1-benzazepin-5-ylidene)-N-(2-morpholin-4-ylethyl)acetamide;ethane;toluene