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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-methyl-2-{3-[5-(4-trifluoromethyl-phenyl)-furan-2-ylmethyl]-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy}-propionic acid ethyl ester 952709-99-8 C28H30F3NO4
2-methyl-2-{3-[5-(4-trifluoromethyl-phenyl)-furan-2-ylmethyl]-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy}-propionic acid ethyl ester
—— 1-{3-[5-(4-trifluoromethyl-phenyl)-thiophen-2-ylmethyl]-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy}-cyclopropanecarboxylic acid methyl ester 952710-78-0 C27H26F3NO3S
1-{3-[5-(4-trifluoromethyl-phenyl)-thiophen-2-ylmethyl]-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy}-cyclopropanecarboxylic acid methyl ester
—— 7-ethoxycarbonylmethoxy-1,2,4,5-tetrahydro-benzo[d]azepine-3-carboxylic acid tert-butyl ester 952710-71-3 C19H27NO5
7-ethoxycarbonylmethoxy-1,2,4,5-tetrahydro-benzo[d]azepine-3-carboxylic acid tert-butyl ester
—— 2-methyl-2-(2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)-propionic acid ethyl ester 952709-88-5 C16H23NO3
2-methyl-2-(2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)-propionic acid ethyl ester
—— (S)-N-methyl-8,9-dichloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine 824430-83-3 C12H15Cl2N
(S)-N-methyl-8,9-dichloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine
—— 2-Fluoro-5-(2,3,4,5-tetrahydro-1H-1-benzoazepin-1-ylsulfonyl)-4-methoxyaniline 1073436-71-1 C17H19FN2O3S
2-Fluoro-5-(2,3,4,5-tetrahydro-1H-1-benzoazepin-1-ylsulfonyl)-4-methoxyaniline
—— 4-[2-(tert-Butyldimethylsilyloxy)ethoxy]-2-fluoro-5-(2,3,4,5-tetrahydro-1H-1-benzoazepin-1-ylsulfonyl)aniline 1073437-03-2 C24H35FN2O4SSi
4-[2-(tert-Butyldimethylsilyloxy)ethoxy]-2-fluoro-5-(2,3,4,5-tetrahydro-1H-1-benzoazepin-1-ylsulfonyl)aniline
—— 2-{[5-[3-(dimethylamino)propyl]-2-(trifluoromethyl)pyridin-3-yl]amino}-9-(trifluoromethyl)-5,7-dihydro-6H-pyrimido[5,4-d][1]benzazepin-6-one 1228962-16-0 C24H22F6N6O
2-{[5-[3-(dimethylamino)propyl]-2-(trifluoromethyl)pyridin-3-yl]amino}-9-(trifluoromethyl)-5,7-dihydro-6H-pyrimido[5,4-d][1]benzazepin-6-one
—— 2-{[5-(3-aminopropyl)-2-methylpyridin-3-yl]amino}-9-(trifluoromethyl)-5,7-dihydro-6H-pyrimido[5,4-d][1]benzazepin-6-one 1228962-12-6 C22H21F3N6O
2-{[5-(3-aminopropyl)-2-methylpyridin-3-yl]amino}-9-(trifluoromethyl)-5,7-dihydro-6H-pyrimido[5,4-d][1]benzazepin-6-one
—— 7-ethyl-5-oxo-8-trifluoromethyl-2,3,4,5-tetrahydro-benzo[b]azepine-1-carboxylic acid tert-butyl ester 872624-97-0 C18H22F3NO3
7-ethyl-5-oxo-8-trifluoromethyl-2,3,4,5-tetrahydro-benzo[b]azepine-1-carboxylic acid tert-butyl ester
—— 7-ethyl-8-trifluoromethyl-1,2,3,4-tetrahydro-benzo[b]azepin-5-one 872624-96-9 C13H14F3NO
7-ethyl-8-trifluoromethyl-1,2,3,4-tetrahydro-benzo[b]azepin-5-one
—— 1-(3,4-dihydro-1H-spiro[benzo[b]azepine-5,4'-piperidin-1-yl])-ethanone 1007566-49-5 C16H22N2O
1-(3,4-dihydro-1H-spiro[benzo[b]azepine-5,4'-piperidin-1-yl])-ethanone
—— (R)-7-ethyl-5-hydroxy-8-trifluoromethyl-2,3,4,5-tetrahydro-benzo[b]azepine-1-carboxylic acid tert-butyl ester 872624-98-1 C18H24F3NO3
(R)-7-ethyl-5-hydroxy-8-trifluoromethyl-2,3,4,5-tetrahydro-benzo[b]azepine-1-carboxylic acid tert-butyl ester
—— (R)-tert-butyl 5-hydroxy-7-methyl-8-trifluoromethyl-2,3,4,5-tetrahydrobenzo[6]azepine-1-carboxylate 872624-60-7 C17H22F3NO3
(R)-tert-butyl 5-hydroxy-7-methyl-8-trifluoromethyl-2,3,4,5-tetrahydrobenzo[6]azepine-1-carboxylate
—— 7-chloro-2-{[2-(trifluoromethyl)imidazo-[1,2-a]pyridin-3-yl]methyl}-1,2,4,5-tetrahydro-3H-2-benzazepin-3-one 1076192-22-7 C19H15ClF3N3O
7-chloro-2-{[2-(trifluoromethyl)imidazo-[1,2-a]pyridin-3-yl]methyl}-1,2,4,5-tetrahydro-3H-2-benzazepin-3-one
—— 5H-benzo[b]pyrido[4,3-f]azepin-6(11H)-one 1246547-23-8 C13H10N2O
5H-benzo[b]pyrido[4,3-f]azepin-6(11H)-one
—— (E)-6-((dimethylamino)methylene)-6,11-dihydro-5H-benzo[f]pyrido[2,3-b]azepin-5-one 1246547-21-6 C16H15N3O
(E)-6-((dimethylamino)methylene)-6,11-dihydro-5H-benzo[f]pyrido[2,3-b]azepin-5-one
—— 3-(7-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-2-{[(1,1-dimethylethyl)oxy]carbonyl}-2,3,4,5-tetrahydro-1H-2-benzazepin-1-yl)propanoic acid 1165946-33-7 C29H34ClN3O6
3-(7-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-2-{[(1,1-dimethylethyl)oxy]carbonyl}-2,3,4,5-tetrahydro-1H-2-benzazepin-1-yl)propanoic acid
—— 1,1-dimethylethyl 1-[3-(methyloxy)-3-oxopropyl]-7-[(phenylmethyl)oxy]-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate 1165946-27-9 C26H33NO5
1,1-dimethylethyl 1-[3-(methyloxy)-3-oxopropyl]-7-[(phenylmethyl)oxy]-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate
—— methyl 3-[7-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-2,3,4,5-tetrahydro-1H-2-benzazepin-1-yl]propanoate 1165946-34-8 C25H28ClN3O4
methyl 3-[7-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-2,3,4,5-tetrahydro-1H-2-benzazepin-1-yl]propanoate
—— methyl 3-{7-[(phenylmethyl)oxy]-2,3,4,5-tetrahydro-1H-2-benzazepin-1-yl}propanoate 1165946-26-8 C21H25NO3
methyl 3-{7-[(phenylmethyl)oxy]-2,3,4,5-tetrahydro-1H-2-benzazepin-1-yl}propanoate
—— ((S)-3-(3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylcarbamoyl)-tetrahydro-furan-3-yl)-carbamic acid tert-butyl ester 1037301-12-4 C21H31N3O4
((S)-3-(3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylcarbamoyl)-tetrahydro-furan-3-yl)-carbamic acid tert-butyl ester
—— 8-methoxy-3-methyl-1,3-dihydrobenzo[d]azepin-2-one 120039-18-1 C12H13NO2
8-methoxy-3-methyl-1,3-dihydrobenzo[d]azepin-2-one
—— 6-amino-5,6-dihydroimidazo[4,5,1-jk][1]benzazepine-2,7(1H,4H)-dione 1019769-46-0 C11H11N3O2
6-amino-5,6-dihydroimidazo[4,5,1-jk][1]benzazepine-2,7(1H,4H)-dione
—— [(S)-9-(2,2-dimethyl-propyl)-4-isopropyl-8-oxo-3,6,7,8,9,10-hexahydro-2,3,9-triaza-cyclohept[e]inden-7-yl]-acetic acid methyl ester 885609-69-8 C22H31N3O3
[(S)-9-(2,2-dimethyl-propyl)-4-isopropyl-8-oxo-3,6,7,8,9,10-hexahydro-2,3,9-triaza-cyclohept[e]inden-7-yl]-acetic acid methyl ester
—— 6-(2,3,4,5-Tetrahydro-1H-benzo[d]azepin-7-yloxy)nicotinamide 676496-20-1 C16H17N3O2
6-(2,3,4,5-Tetrahydro-1H-benzo[d]azepin-7-yloxy)nicotinamide
—— (R)-tert-butyl 4-amino-2-benzyl-7-methyl-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-8-ylcarbamate 885608-95-7 C23H29N3O3
(R)-tert-butyl 4-amino-2-benzyl-7-methyl-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-8-ylcarbamate
—— 7-amino-9-(4-trifluoromethyl-benzyl)-6,7,9,10-tetrahydro-3H-2,3,9-triaza-(R)-cyclohepta[e]inden-8-one 885608-41-3 C19H17F3N4O
7-amino-9-(4-trifluoromethyl-benzyl)-6,7,9,10-tetrahydro-3H-2,3,9-triaza-(R)-cyclohepta[e]inden-8-one
—— (R)-9-(1-acetylpiperidin-4-yl)-7-amino-6,7,9,10-tetrahydroazepino[3,4-e]indazol-8(3H)-one 885609-09-6 C18H23N5O2
(R)-9-(1-acetylpiperidin-4-yl)-7-amino-6,7,9,10-tetrahydroazepino[3,4-e]indazol-8(3H)-one
—— [4-methyl-9-(2,2-dimethyl-propyl)-8-oxo-3,6,7,8,9,10-hexahydro-2,3,9-triaza-(S)-cyclohepta[e]inden-7-yl]-acetic acid 885609-61-0 C19H25N3O3
[4-methyl-9-(2,2-dimethyl-propyl)-8-oxo-3,6,7,8,9,10-hexahydro-2,3,9-triaza-(S)-cyclohepta[e]inden-7-yl]-acetic acid
—— (R)-tert-butyl 2-benzyl-7-methyl-3-oxo-4-(4-(2-oxo-1,2-dihydroquinazolin-3(4H)-yl)piperidine-1-carboxamido)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-8-ylcarbamate 885608-96-8 C37H44N6O5
(R)-tert-butyl 2-benzyl-7-methyl-3-oxo-4-(4-(2-oxo-1,2-dihydroquinazolin-3(4H)-yl)piperidine-1-carboxamido)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-8-ylcarbamate
—— (R)-benzyl 8-tert-butoxycarbonylamino-2-benzyl-7-methyl-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-ylcarbamate 885608-93-5 C31H35N3O5
(R)-benzyl 8-tert-butoxycarbonylamino-2-benzyl-7-methyl-3-oxo-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-ylcarbamate
—— (R)-4-chloro-7-hydroxy-9-(2,2,2-trifluoroethyl)-6,7,9,10-tetrahydroazepino[3,4-e]indazol-8(3H)-one 912463-10-6 C13H11ClF3N3O2
(R)-4-chloro-7-hydroxy-9-(2,2,2-trifluoroethyl)-6,7,9,10-tetrahydroazepino[3,4-e]indazol-8(3H)-one
—— 6-Phenylethynyl-2,3,4,5-tetrahydro-benzo[c]azepin-1-one 873330-66-6 C18H15NO
6-Phenylethynyl-2,3,4,5-tetrahydro-benzo[c]azepin-1-one
—— 3-tert-butoxycarbonyl-7-chloro-6-(thiazol-2-ylethynyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 864265-69-0 C20H21ClN2O2S
3-tert-butoxycarbonyl-7-chloro-6-(thiazol-2-ylethynyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— 3-tert-butoxycarbonyl-7-chloro-6-(2-thiazol-2-ylethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 928830-42-6 C20H25ClN2O2S
3-tert-butoxycarbonyl-7-chloro-6-(2-thiazol-2-ylethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— 3-tert-butoxycarbonyl-7-chloro-6-ethynyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine 864265-66-7 C17H20ClNO2
3-tert-butoxycarbonyl-7-chloro-6-ethynyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— 7-acetyl-6-hydroxy-3-(2,2,2-trifluoroacetyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 864262-78-2 C14H14F3NO3
7-acetyl-6-hydroxy-3-(2,2,2-trifluoroacetyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— 7-Chloro-6-(3-hydroxyazetidin-1-yl)-3-(2,2,2-trifluoroacetyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 927829-41-2 C15H16ClF3N2O2
7-Chloro-6-(3-hydroxyazetidin-1-yl)-3-(2,2,2-trifluoroacetyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— 7-ethyl-6-hydroxy-3-(2,2,2-trifluoroacetyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 864262-79-3 C14H16F3NO2
7-ethyl-6-hydroxy-3-(2,2,2-trifluoroacetyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— 6-(2-phenylpyrrolidin-1-yl)-2,3,4,5-tetrahydro-1H-3-benzazepine 927830-37-3 C20H24N2
6-(2-phenylpyrrolidin-1-yl)-2,3,4,5-tetrahydro-1H-3-benzazepine
—— 7-chloro-6-(3-hydroxy-2,2-dimethyl-propylamino)-3-(2,2,2-trifluoroacetyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 927829-38-7 C17H22ClF3N2O2
7-chloro-6-(3-hydroxy-2,2-dimethyl-propylamino)-3-(2,2,2-trifluoroacetyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— tert-Butyl 3-(7-amino-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)pyrrolidine-1-carboxylate 1063408-73-0 C19H29N3O2
tert-Butyl 3-(7-amino-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)pyrrolidine-1-carboxylate
—— 5,5-difluoro-2,3,4,5-tetrahydro-1H-benzazepine 1422496-42-1 C10H11F2N
5,5-difluoro-2,3,4,5-tetrahydro-1H-benzazepine
—— dimethyl-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-ylmethyl)-amine 686298-27-1 C13H20N2
dimethyl-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-ylmethyl)-amine
—— 1-(1-Methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-amine 1063408-16-1 C16H25N3
1-(1-Methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-amine
—— tert-Butyl-4-(7-amino-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)piperidine-1-carboxylate 1063409-39-1 C20H31N3O2
tert-Butyl-4-(7-amino-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)piperidine-1-carboxylate
—— 6-acetyl-3-tert-butoxycarbonyl-7-chloro-2,3,4,5-tetrahydro-1H-benzo[d]azepine 928793-98-0 C17H22ClNO3
6-acetyl-3-tert-butoxycarbonyl-7-chloro-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— 3-tert-butoxycarbonyl-7-chloro-6-(1-hydroxy-ethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 928794-00-7 C17H24ClNO3
3-tert-butoxycarbonyl-7-chloro-6-(1-hydroxy-ethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— 6-(aminomethyl)-3-tert-butoxycarbonyl-7-chloro-2,3,4,5-tetrahydro-1H-benzo[d]azepine 928794-06-3 C16H23ClN2O2
6-(aminomethyl)-3-tert-butoxycarbonyl-7-chloro-2,3,4,5-tetrahydro-1H-benzo[d]azepine