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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R,3S)-3-hydroxy-2-phenyl-5-azatricyclo[7.4.0.02,5]trideca-1(13),9,11-trien-4-one —— C18H17NO2
(2R,3S)-3-hydroxy-2-phenyl-5-azatricyclo[7.4.0.02,5]trideca-1(13),9,11-trien-4-one
—— 8-chloro-4-(dimethylaminomethylidene)-7-ethyl-1H-1-benzazepine-2,5-dione —— C15H17ClN2O2
8-chloro-4-(dimethylaminomethylidene)-7-ethyl-1H-1-benzazepine-2,5-dione
—— 7-[4-(2-butoxyethoxy)phenyl]-1-isobutyl-N-[4-[(3-propylimidazol-4-yl)methylsulfonyl]phenyl]-2,3-dihydro-1-benzazepine-4-carboxamide; ethyl acetate —— C44H58N4O7S
7-[4-(2-butoxyethoxy)phenyl]-1-isobutyl-N-[4-[(3-propylimidazol-4-yl)methylsulfonyl]phenyl]-2,3-dihydro-1-benzazepine-4-carboxamide; ethyl acetate
—— 7-[4-(2-butoxyethoxy)phenyl]-1-isobutyl-N-[4-(pyrazin-2-ylmethylsulfinyl)phenyl]-2,3-dihydro-1-benzazepine-4-carboxamide —— C38H44N4O4S
7-[4-(2-butoxyethoxy)phenyl]-1-isobutyl-N-[4-(pyrazin-2-ylmethylsulfinyl)phenyl]-2,3-dihydro-1-benzazepine-4-carboxamide
—— 2-ethyl-3-[8-(3-fluoropiperidin-4-yl)oxyquinolin-2-yl]-4,5-dihydro-3H-1-benzazepine —— C26H28FN3O
2-ethyl-3-[8-(3-fluoropiperidin-4-yl)oxyquinolin-2-yl]-4,5-dihydro-3H-1-benzazepine
—— 5-Nitroso-1,2,3,5-tetrahydro-3-benzazepin-4-one —— C10H10N2O2
5-Nitroso-1,2,3,5-tetrahydro-3-benzazepin-4-one
—— [5-methyl-6-oxo-3-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butylcarbamoyl]-11H-benzo[c][1]benzazepin-11-yl] propanoate —— C31H34N4O4
[5-methyl-6-oxo-3-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butylcarbamoyl]-11H-benzo[c][1]benzazepin-11-yl] propanoate
—— (3S)-2-butyl-N'-[(7S)-5-(cyclohexylmethyl)-6-oxo-7H-benzo[d][1]benzazepin-7-yl]-3-(2-methylpropyl)butanediamide —— C33H45N3O3
(3S)-2-butyl-N'-[(7S)-5-(cyclohexylmethyl)-6-oxo-7H-benzo[d][1]benzazepin-7-yl]-3-(2-methylpropyl)butanediamide
—— 1-[(4S)-7-chloro-6-fluoro-4-methyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C13H12ClF4NO
1-[(4S)-7-chloro-6-fluoro-4-methyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— [4-[[9-chloro-7-(2-chlorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]morpholin-4-ium-4-yl]-phenylmethanone —— C29H24Cl2N5O2+
[4-[[9-chloro-7-(2-chlorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]morpholin-4-ium-4-yl]-phenylmethanone
—— 3-Methyl-1,2,4,5-tetrahydro-3-benzazepine-7-carbonitrile —— C12H14N2
3-Methyl-1,2,4,5-tetrahydro-3-benzazepine-7-carbonitrile
—— 4-[[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxymethyl]benzoic acid —— C29H23N7O3
4-[[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxymethyl]benzoic acid
—— 4-[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxybutanoic acid —— C25H23N7O3
4-[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxybutanoic acid
—— 2-[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxyacetic acid —— C23H19N7O3
2-[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxyacetic acid
—— 3-[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxypropanoic acid —— C24H21N7O3
3-[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxypropanoic acid
—— 11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-ol —— C21H17N7O
11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-ol
—— 5-[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxypentanoic acid —— C26H25N7O3
5-[11-[(2,4-Diaminopteridin-6-yl)methyl]benzo[b][1]benzazepin-4-yl]oxypentanoic acid
—— (2S)-2-methoxy-N-(5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl)-N'-(2,2,3,3,3-pentafluoropropyl)propanediamide —— C22H20F5N3O4
(2S)-2-methoxy-N-(5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl)-N'-(2,2,3,3,3-pentafluoropropyl)propanediamide
—— 9-(2-Piperidin-1-ylethyl)-3,6,7,10-tetrahydropyrazolo[3,4-i][2]benzazepin-8-one —— C18H24N4O
9-(2-Piperidin-1-ylethyl)-3,6,7,10-tetrahydropyrazolo[3,4-i][2]benzazepin-8-one
—— 2-[(4-chloro-2-fluoro-5-methylphenyl)methyl]-8-(2-methyl-3H-benzimidazol-5-yl)-1,3,4,5-tetrahydro-2-benzazepine —— C26H25ClFN3
2-[(4-chloro-2-fluoro-5-methylphenyl)methyl]-8-(2-methyl-3H-benzimidazol-5-yl)-1,3,4,5-tetrahydro-2-benzazepine
—— 5-Ethylidene-6-methyl-4b,6,11,11a-tetrahydroindeno[1,2-c][2]benzazepin-5-ium-12-one —— C20H20NO+
5-Ethylidene-6-methyl-4b,6,11,11a-tetrahydroindeno[1,2-c][2]benzazepin-5-ium-12-one
—— Methyl [4-(aminomethyl)-2,3-dihydro-1h-1-benzazepin-2-yl]acetate —— C14H18N2O2
Methyl [4-(aminomethyl)-2,3-dihydro-1h-1-benzazepin-2-yl]acetate
—— tert-butyl N-(1-sulfanyl-2,3,4,5-tetrahydro-1-benzazepin-4-yl)carbamate —— C15H22N2O2S
tert-butyl N-(1-sulfanyl-2,3,4,5-tetrahydro-1-benzazepin-4-yl)carbamate
—— 6-[7,9-difluoro-4-methyl-2-prop-1-en-2-yl-8-(trifluoromethyl)-1-azoniatetracyclo[9.4.0.02,4.05,10]pentadeca-1(15),5,7,9,11,13-hexaen-3-yl]-5,6-dihydro-2H-imidazo[5,1-c][1,4]oxazin-4-ium-8-one —— C25H20F5N3O2+2
6-[7,9-difluoro-4-methyl-2-prop-1-en-2-yl-8-(trifluoromethyl)-1-azoniatetracyclo[9.4.0.02,4.05,10]pentadeca-1(15),5,7,9,11,13-hexaen-3-yl]-5,6-dihydro-2H-imidazo[5,1-c][1,4]oxazin-4-ium-8-one
—— 3-cyclopentyl-5-(methylamino)-2,5-dihydro-1H-3-benzazepin-4-one;ethane —— C18H28N2O
3-cyclopentyl-5-(methylamino)-2,5-dihydro-1H-3-benzazepin-4-one;ethane
—— (4Z)-4-(hydroxymethylene)-1H-1-benzazepine-2,5-dione —— C11H9NO3
(4Z)-4-(hydroxymethylene)-1H-1-benzazepine-2,5-dione
—— 4-(4-acetylpiperazin-1-yl)-1-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)butan-1-one —— C20H29N3O2
4-(4-acetylpiperazin-1-yl)-1-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)butan-1-one
—— N-[2-(6-hydroxy-5,11-dihydropyrido[2,3-c][1]benzazepin-5-yl)ethyl]-N-methylformamide —— C17H19N3O2
N-[2-(6-hydroxy-5,11-dihydropyrido[2,3-c][1]benzazepin-5-yl)ethyl]-N-methylformamide
—— (11E)-2-chloro-11-(2-dimethylaminoethyloxyimino)-5H-benzo[c][1]benzazepine-6-thione —— C18H18ClN3OS
(11E)-2-chloro-11-(2-dimethylaminoethyloxyimino)-5H-benzo[c][1]benzazepine-6-thione
—— (11E)-2-chloro-11-methoxyimino-5H-benzo[c][1]benzazepine-6-thione —— C15H11ClN2OS
(11E)-2-chloro-11-methoxyimino-5H-benzo[c][1]benzazepine-6-thione
—— ethyl 7-methyl-2,5-dioxo-3,4-dihydro-1H-1-benzazepine-4-carboxylate —— C14H15NO4
ethyl 7-methyl-2,5-dioxo-3,4-dihydro-1H-1-benzazepine-4-carboxylate
—— 2-[(N-ethyl-4-fluoroanilino)-propan-2-ylamino]-2,3,4,5-tetrahydro-1-benzazepine-1-carboxamide —— C22H29FN4O
2-[(N-ethyl-4-fluoroanilino)-propan-2-ylamino]-2,3,4,5-tetrahydro-1-benzazepine-1-carboxamide
—— 7-Deuteriooxy-5-(2,3-dihydro-1-benzofuran-7-yl)-3-methyl-8-nitro-1,2,4,5-tetrahydro-3-benzazepine —— C19H20N2O4
7-Deuteriooxy-5-(2,3-dihydro-1-benzofuran-7-yl)-3-methyl-8-nitro-1,2,4,5-tetrahydro-3-benzazepine
—— 5-[(3,4-Dimethoxy-7-bicyclo[4.2.0]octa-1,3,5-trienyl)methylamino]-3-(7,8-dimethoxy-1,2,4,5-tetrahydro-3-benzazepin-3-yl)pentan-2-one —— C28H38N2O5
5-[(3,4-Dimethoxy-7-bicyclo[4.2.0]octa-1,3,5-trienyl)methylamino]-3-(7,8-dimethoxy-1,2,4,5-tetrahydro-3-benzazepin-3-yl)pentan-2-one
—— [1-[[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-(4-methylphenyl)carbamate —— C26H25N3O4
[1-[[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-(4-methylphenyl)carbamate
—— (3Z)-4,5-dimethoxy-3-[1-(pyridin-4-ylamino)ethylidene]-1,2-dihydro-2-benzazepine-1-carboxylic acid —— C20H21N3O4
(3Z)-4,5-dimethoxy-3-[1-(pyridin-4-ylamino)ethylidene]-1,2-dihydro-2-benzazepine-1-carboxylic acid
—— Tert-butyl 5-amino-4-(dimethylamino)-1,2,4,5-tetrahydro-3-benzazepine-3-carboxylate —— C17H27N3O2
Tert-butyl 5-amino-4-(dimethylamino)-1,2,4,5-tetrahydro-3-benzazepine-3-carboxylate
—— 1H-1-benzazepine-9-carboxamide —— C11H10N2O
1H-1-benzazepine-9-carboxamide
—— 7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-2-(trifluoromethyl)-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine —— C28H27F3N6OS
7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-2-(trifluoromethyl)-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine
—— 7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine —— C27H28N6OS
7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine
—— N-(5-acetyl-10,11-dihydro-5H-dibenzo[b,f]azepin-3-yl)-3-methylbenzamide —— C24H22N2O2
N-(5-acetyl-10,11-dihydro-5H-dibenzo[b,f]azepin-3-yl)-3-methylbenzamide
—— 1-(Adamantane-1-carbonyl)-2-methoxy-1,7b-dihydrocyclopropa[c]quinoline-1a-carbonitrile —— C23H24N2O2
1-(Adamantane-1-carbonyl)-2-methoxy-1,7b-dihydrocyclopropa[c]quinoline-1a-carbonitrile
—— [1-[[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-[(2-methylphenyl)methyl]carbamate —— C27H27N3O4
[1-[[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-[(2-methylphenyl)methyl]carbamate
—— 7-(dimethylamino)-2-(2,3-dimethylphenyl)-3H-2-benzazepin-1-one —— C20H22N2O
7-(dimethylamino)-2-(2,3-dimethylphenyl)-3H-2-benzazepin-1-one
—— 2-[4-[[(5S)-5-[[3,5-bis(trifluoromethyl)phenyl]methyl-(2-methyltetrazol-5-yl)amino]-7-methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-1-benzazepin-4-yl]methyl]piperidin-1-yl]acetic acid —— C31H34F9N7O2
2-[4-[[(5S)-5-[[3,5-bis(trifluoromethyl)phenyl]methyl-(2-methyltetrazol-5-yl)amino]-7-methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-1-benzazepin-4-yl]methyl]piperidin-1-yl]acetic acid
—— 1-cyclopentyl-3-(methylamino)-4,5-dihydro-3H-1-benzazepin-2-one;ethane —— C18H28N2O
1-cyclopentyl-3-(methylamino)-4,5-dihydro-3H-1-benzazepin-2-one;ethane
—— 5-[[7,9-Difluoro-2,4-dimethyl-8-(trifluoromethyl)-1-azoniatetracyclo[9.4.0.02,4.05,10]pentadeca-1(15),5,7,9,11,13-hexaen-3-yl]methyl]-2,3-dimethyl-5,6-dihydroimidazo[5,1-c][1,4]oxazin-2-ium-8-one —— C26H24F5N3O2+2
5-[[7,9-Difluoro-2,4-dimethyl-8-(trifluoromethyl)-1-azoniatetracyclo[9.4.0.02,4.05,10]pentadeca-1(15),5,7,9,11,13-hexaen-3-yl]methyl]-2,3-dimethyl-5,6-dihydroimidazo[5,1-c][1,4]oxazin-2-ium-8-one
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(3,5-dimethylpiperidin-1-ium-1-yl)ethanone;2-hydroxy-2-oxoacetate —— C25H30N2O5
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(3,5-dimethylpiperidin-1-ium-1-yl)ethanone;2-hydroxy-2-oxoacetate
—— (4R)-8-[2-[3-cyclopropyl-6-(methylamino)pyridin-2-yl]ethoxy]-4-ethyl-2-(2,2,2-trifluoroethyl)-4,5-dihydro-1H-2-benzazepin-3-one;2-[(4S)-3-oxo-8-(2-spiro[7,8-dihydro-6H-1,8-naphthyridine-5,1'-cyclopropane]-2-ylethoxy)-2-(2,2,2-trifluoroethyl)-4,5-dihydro-1H-2-benzazepin-4-yl]acetic acid —— C51H58F6N6O6
(4R)-8-[2-[3-cyclopropyl-6-(methylamino)pyridin-2-yl]ethoxy]-4-ethyl-2-(2,2,2-trifluoroethyl)-4,5-dihydro-1H-2-benzazepin-3-one;2-[(4S)-3-oxo-8-(2-spiro[7,8-dihydro-6H-1,8-naphthyridine-5,1'-cyclopropane]-2-ylethoxy)-2-(2,2,2-trifluoroethyl)-4,5-dihydro-1H-2-benzazepin-4-yl]acetic acid
—— 3-[4-(3-hydroxy-1,1-dioxo-2H-1,2,5-thiadiazol-5-yl)-3-phenylmethoxyphenoxy]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C25H23N3O6S
3-[4-(3-hydroxy-1,1-dioxo-2H-1,2,5-thiadiazol-5-yl)-3-phenylmethoxyphenoxy]-1,3,4,5-tetrahydro-1-benzazepin-2-one