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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-1'-[(2-morpholin-4-ylpyrimidin-4-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H27N5O2
(3S)-1'-[(2-morpholin-4-ylpyrimidin-4-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— N-[3-oxo-3-[(3R)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1'-yl]propyl]pyridine-3-carboxamide —— C22H24N4O3
N-[3-oxo-3-[(3R)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1'-yl]propyl]pyridine-3-carboxamide
—— (3S)-1'-(quinoxalin-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H22N4O
(3S)-1'-(quinoxalin-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[2-(4-fluorophenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H21FN2O2
(3S)-1'-[2-(4-fluorophenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(3,4-difluorophenyl)sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H18F2N2O3S
(3S)-1'-(3,4-difluorophenyl)sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(6-morpholin-4-ylpyridin-3-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C23H28N4O2
(3S)-1'-[(6-morpholin-4-ylpyridin-3-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(2-pyridin-4-ylethylsulfonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O3S
(3R)-1'-(2-pyridin-4-ylethylsulfonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(E)-3-pyridin-3-ylprop-2-enyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H23N3O
(3S)-1'-[(E)-3-pyridin-3-ylprop-2-enyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(2-fluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21FN2O
(3S)-1'-[(2-fluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— N-[3-oxo-3-[(3S)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1'-yl]propyl]pyridine-3-carboxamide —— C22H24N4O3
N-[3-oxo-3-[(3S)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1'-yl]propyl]pyridine-3-carboxamide
—— (3R)-1'-(quinoxalin-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H22N4O
(3R)-1'-(quinoxalin-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(4-fluorophenyl)sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H19FN2O3S
(3R)-1'-(4-fluorophenyl)sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(pyridin-3-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H21N3O
(3R)-1'-(pyridin-3-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[[2-(trifluoromethyl)phenyl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H21F3N2O
(3S)-1'-[[2-(trifluoromethyl)phenyl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(pyridine-3-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H19N3O2
(3R)-1'-(pyridine-3-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(6-chloro-1,3-benzodioxol-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H21ClN2O3
(3S)-1'-[(6-chloro-1,3-benzodioxol-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C13H16N2O
(3R)-spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2-piperidin-1-ylpyrimidin-4-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C23H29N5O
(3R)-1'-[(2-piperidin-1-ylpyrimidin-4-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2-morpholin-4-ylpyrimidin-4-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H27N5O2
(3R)-1'-[(2-morpholin-4-ylpyrimidin-4-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(4-fluorobenzoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H19FN2O2
(3S)-1'-(4-fluorobenzoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[3-(3,4-difluorophenyl)propanoyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H22F2N2O2
(3S)-1'-[3-(3,4-difluorophenyl)propanoyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[[5-(morpholin-4-ylmethyl)furan-2-yl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C23H29N3O3
(3S)-1'-[[5-(morpholin-4-ylmethyl)furan-2-yl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(2-pyridin-4-ylethylsulfonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O3S
(3S)-1'-(2-pyridin-4-ylethylsulfonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[3-(trifluoromethyl)phenyl]sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H19F3N2O3S
(3R)-1'-[3-(trifluoromethyl)phenyl]sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2,3-difluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H20F2N2O
(3R)-1'-[(2,3-difluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(2-phenoxyethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H24N2O2
(3R)-1'-(2-phenoxyethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(2-phenoxyethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H24N2O2
(3S)-1'-(2-phenoxyethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(3-phenoxypropyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O2
(3S)-1'-(3-phenoxypropyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-benzyl-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H24N2O2
(3S,4'R)-1'-benzyl-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-benzylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H22N2O
(3S)-1'-benzylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-benzylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H22N2O
(3R)-1'-benzylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— 1-[(5R)-8-fluoro-5-(4-fluorophenyl)-2,3,4,5-tetrahydro-1-benzazepin-1-yl]-2-[4-(2-hydroxyethyl)piperazin-1-yl]ethanone —— C24H29F2N3O2
1-[(5R)-8-fluoro-5-(4-fluorophenyl)-2,3,4,5-tetrahydro-1-benzazepin-1-yl]-2-[4-(2-hydroxyethyl)piperazin-1-yl]ethanone
—— (3R,3'S)-N,N-dimethyl-1'-(1-methylpyrazole-4-carbonyl)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H25N5O3
(3R,3'S)-N,N-dimethyl-1'-(1-methylpyrazole-4-carbonyl)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3S)-1'-[(2-methylpyrimidin-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H22N4O
(3S)-1'-[(2-methylpyrimidin-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2-methylpyrimidin-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H22N4O
(3R)-1'-[(2-methylpyrimidin-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(3-methylpyridin-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O
(3S)-1'-[(3-methylpyridin-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(3-methylpyridin-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O
(3R)-1'-[(3-methylpyridin-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[[2-(2-methylphenyl)pyrimidin-5-yl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C25H26N4O
(3S)-1'-[[2-(2-methylphenyl)pyrimidin-5-yl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(6-methylpyridin-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O
(3R)-1'-[(6-methylpyridin-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(6-methylpyridin-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O
(3S)-1'-[(6-methylpyridin-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(2-methoxy-3-methylphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O2
(3S)-1'-[(2-methoxy-3-methylphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2-methoxy-3-methylphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O2
(3R)-1'-[(2-methoxy-3-methylphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— N-[3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)propyl]-N-methyl-4-(4-nitrophenyl)-1,3-thiazol-2-amine —— C27H26N4O2S
N-[3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)propyl]-N-methyl-4-(4-nitrophenyl)-1,3-thiazol-2-amine
—— (3aS,10aS)-10a-methyl-2-[(5-methylthiophen-2-yl)methyl]-1,3,3a,4-tetrahydropyrrolo[3,4-c][2]benzazepine-5,10-dione —— C19H20N2O2S
(3aS,10aS)-10a-methyl-2-[(5-methylthiophen-2-yl)methyl]-1,3,3a,4-tetrahydropyrrolo[3,4-c][2]benzazepine-5,10-dione
—— (3S,4'R)-4'-(hydroxymethyl)-1'-[(5-methylthiophen-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H24N2O2S
(3S,4'R)-4'-(hydroxymethyl)-1'-[(5-methylthiophen-2-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R,3'S)-N,N-dimethyl-1'-(3-methyl-1,2-oxazole-5-carbonyl)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H24N4O4
(3R,3'S)-N,N-dimethyl-1'-(3-methyl-1,2-oxazole-5-carbonyl)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3S)-8-methoxy-1'-(3-methyl-1,2-oxazole-5-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H21N3O4
(3S)-8-methoxy-1'-(3-methyl-1,2-oxazole-5-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-8-methoxy-1'-(3-methyl-1,2-oxazole-5-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H21N3O4
(3R)-8-methoxy-1'-(3-methyl-1,2-oxazole-5-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,3'R)-N-tert-butyl-1'-methyl-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide —— C19H27N3O2
(3S,3'R)-N-tert-butyl-1'-methyl-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,4'-pyrrolidine]-3'-carboxamide
—— N-[4-[(3S,4'R)-4'-(hydroxymethyl)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1'-yl]sulfonylphenyl]acetamide —— C22H25N3O5S
N-[4-[(3S,4'R)-4'-(hydroxymethyl)-1-oxospiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1'-yl]sulfonylphenyl]acetamide