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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 7,12-Dihydroindolo[3,2-d][1]benzazepine-9-carbonitrile —— C17H11N3
7,12-Dihydroindolo[3,2-d][1]benzazepine-9-carbonitrile
—— 9-(3-Pyrrolidin-1-ylpropyl)-5,7-dihydropyrimido[5,4-d][1]benzazepin-6-one —— C19H22N4O
9-(3-Pyrrolidin-1-ylpropyl)-5,7-dihydropyrimido[5,4-d][1]benzazepin-6-one
—— Ethane;(3-methyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl) trifluoromethanesulfonate —— C14H20F3NO3S
Ethane;(3-methyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl) trifluoromethanesulfonate
—— N'-[(1R,3S,12R,16R)-9-bromo-4-(cyclopropylmethyl)-3-(hydroxymethyl)-8-methoxy-16-methyl-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-14-yl]-4-methoxybenzenesulfonohydrazide —— C29H36BrN3O6S
N'-[(1R,3S,12R,16R)-9-bromo-4-(cyclopropylmethyl)-3-(hydroxymethyl)-8-methoxy-16-methyl-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-14-yl]-4-methoxybenzenesulfonohydrazide
—— 10-bromo-7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-2-(trifluoromethyl)-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine —— C28H26BrF3N6OS
10-bromo-7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-2-(trifluoromethyl)-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine
—— 8-(5-Chloropent-1-enyl)-5,5-dimethyl-1,2,3,4-tetrahydro-1-benzazepine —— C17H24ClN
8-(5-Chloropent-1-enyl)-5,5-dimethyl-1,2,3,4-tetrahydro-1-benzazepine
—— [1-[[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-[(2,4-difluorophenyl)methyl]carbamate —— C26H23F2N3O4
[1-[[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-[(2,4-difluorophenyl)methyl]carbamate
—— 1-[2-[(3-Cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-3,4-dihydropyridin-5-yl]propan-1-one —— C22H28N2O2
1-[2-[(3-Cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-3,4-dihydropyridin-5-yl]propan-1-one
—— 2-(trifluoromethyl)-7,8,9,10-tetrahydro-6H-[1,3]oxazolo[4,5-g][1]benzazepine —— C12H11F3N2O
2-(trifluoromethyl)-7,8,9,10-tetrahydro-6H-[1,3]oxazolo[4,5-g][1]benzazepine
—— 9-Methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepine-1-carboxylic acid —— C13H14F3NO2
9-Methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepine-1-carboxylic acid
—— 2-[[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]amino]-7H-pyrimido[5,4-i][1]benzazepin-6-ol —— C22H22ClN5O
2-[[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]amino]-7H-pyrimido[5,4-i][1]benzazepin-6-ol
—— N-(7H-benzo[d][1]benzazepin-7-yl)formamide —— C15H12N2O
N-(7H-benzo[d][1]benzazepin-7-yl)formamide
—— 2-(cyclopropylmethyl)-7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine —— C31H34N6OS
2-(cyclopropylmethyl)-7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine
—— Tert-butyl 7-ethyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepine-1-carboxylate —— C18H24F3NO2
Tert-butyl 7-ethyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepine-1-carboxylate
—— Oxan-4-yl 7-methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepine-1-carboxylate —— C18H22F3NO3
Oxan-4-yl 7-methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepine-1-carboxylate
—— Methyl 19-cyclohexyl-15-[2-[[cyclopropyl(methyl)sulfamoyl]amino]-2-hydroxyethyl]-5-methoxy-12-azapentacyclo[10.7.0.02,7.08,10.013,18]nonadeca-1(19),2(7),3,5,13(18),14,16-heptaene-10-carboxylate —— C33H41N3O6S
Methyl 19-cyclohexyl-15-[2-[[cyclopropyl(methyl)sulfamoyl]amino]-2-hydroxyethyl]-5-methoxy-12-azapentacyclo[10.7.0.02,7.08,10.013,18]nonadeca-1(19),2(7),3,5,13(18),14,16-heptaene-10-carboxylate
—— 1-[3-(Cyclobutadienyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]-3-phenylpropan-2-one —— C23H23NO
1-[3-(Cyclobutadienyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]-3-phenylpropan-2-one
—— 5-[3-[3-[3-(2-Hydroxyethyl)-3-methyloxiran-2-yl]-1,2,4,5-tetrahydro-3-benzazepin-7-yl]-1,2,4-oxadiazol-5-yl]-2-propan-2-yloxybenzonitrile —— C27H30N4O4
5-[3-[3-[3-(2-Hydroxyethyl)-3-methyloxiran-2-yl]-1,2,4,5-tetrahydro-3-benzazepin-7-yl]-1,2,4-oxadiazol-5-yl]-2-propan-2-yloxybenzonitrile
—— 13-Fluoro-5-methyl-4-prop-2-enyl-11-oxa-4-azapentacyclo[8.7.0.01,6.03,16.012,17]heptadeca-7,12,14,16-tetraen-9-ol —— C19H20FNO2
13-Fluoro-5-methyl-4-prop-2-enyl-11-oxa-4-azapentacyclo[8.7.0.01,6.03,16.012,17]heptadeca-7,12,14,16-tetraen-9-ol
—— (6-methoxy-6,11-dihydrobenzo[b][1]benzazepin-5-ylidene)methanone —— C16H13NO2
(6-methoxy-6,11-dihydrobenzo[b][1]benzazepin-5-ylidene)methanone
—— (1R)-2-methyl-1-[2-(4-methylsulfanylphenoxy)ethyl]-1,3-dihydro-2-benzazepine —— C20H23NOS
(1R)-2-methyl-1-[2-(4-methylsulfanylphenoxy)ethyl]-1,3-dihydro-2-benzazepine
—— [7-[Amino(hydroxy)methyl]-1,3,4,5-tetrahydro-2-benzazepin-2-yl]-(1-benzothiophen-3-yl)methanone —— C20H20N2O2S
[7-[Amino(hydroxy)methyl]-1,3,4,5-tetrahydro-2-benzazepin-2-yl]-(1-benzothiophen-3-yl)methanone
—— 6-[7-[5-(3-Cyano-4-propan-2-yloxyphenyl)-1,2,4-oxadiazol-3-yl]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]hexanamide —— C28H33N5O3
6-[7-[5-(3-Cyano-4-propan-2-yloxyphenyl)-1,2,4-oxadiazol-3-yl]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]hexanamide
—— 2-(2-bicyclo[2.2.1]heptanyl)-6-methoxy-4,5-dihydro-3H-1-benzazepine-9-carboxylic acid —— C19H23NO3
2-(2-bicyclo[2.2.1]heptanyl)-6-methoxy-4,5-dihydro-3H-1-benzazepine-9-carboxylic acid
—— [(1R,3S,12R,16R)-9-bromo-8-methoxy-14-methoxyimino-16-methyl-4-undecyl-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17)-trien-3-yl]methanol —— C30H47BrN2O4
[(1R,3S,12R,16R)-9-bromo-8-methoxy-14-methoxyimino-16-methyl-4-undecyl-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17)-trien-3-yl]methanol
—— 2-(4,4-difluoro-2,3-dihydro-1H-1-benzazepin-5-ylidene)acetamide —— C12H12F2N2O
2-(4,4-difluoro-2,3-dihydro-1H-1-benzazepin-5-ylidene)acetamide
—— 7-(2-aminoethyl)-5,5-dimethyl-3,4-dihydro-1H-1-benzazepin-2-one —— C14H20N2O
7-(2-aminoethyl)-5,5-dimethyl-3,4-dihydro-1H-1-benzazepin-2-one
—— 3-[7,9-difluoro-13-hexyl-4-methyl-2-(2-methylprop-2-enyl)-8-(trifluoromethyl)-1-azoniatetracyclo[9.4.0.02,4.05,10]pentadeca-1(11),5,7,9,12,14-hexaen-3-yl]-6-methyl-3H-imidazo[1,5-c][1,3]oxazol-6-ium-1-one —— C32H34F5N3O2+2
3-[7,9-difluoro-13-hexyl-4-methyl-2-(2-methylprop-2-enyl)-8-(trifluoromethyl)-1-azoniatetracyclo[9.4.0.02,4.05,10]pentadeca-1(11),5,7,9,12,14-hexaen-3-yl]-6-methyl-3H-imidazo[1,5-c][1,3]oxazol-6-ium-1-one
—— 2,2,2-trifluoro-1-[(4S)-8-hydroxy-4-methyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]ethanone —— C13H14F3NO2
2,2,2-trifluoro-1-[(4S)-8-hydroxy-4-methyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]ethanone
—— 9-Methyl-1,3-diazatricyclo[6.4.1.04,13]trideca-4,6,8(13)-trien-2-one —— C12H14N2O
9-Methyl-1,3-diazatricyclo[6.4.1.04,13]trideca-4,6,8(13)-trien-2-one
—— [(1R,3S,12R,16R)-9-bromo-8-methoxy-14-methoxyimino-16-methyl-4-(3-methylsulfanylpropyl)-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17)-trien-3-yl]methanol —— C23H33BrN2O4S
[(1R,3S,12R,16R)-9-bromo-8-methoxy-14-methoxyimino-16-methyl-4-(3-methylsulfanylpropyl)-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17)-trien-3-yl]methanol
—— 6-fluoro-3-[4-[6-methoxy-1-(1,2-oxazol-4-yl)hepta-2,4-dien-4-yl]pyrazol-1-yl]-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one —— C26H26F4N4O3
6-fluoro-3-[4-[6-methoxy-1-(1,2-oxazol-4-yl)hepta-2,4-dien-4-yl]pyrazol-1-yl]-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one
—— tert-butyl N-[[3-[[7-methoxy-8-[[4-(trifluoromethyl)cyclohexen-1-yl]carbamoyl]-4,5-dihydro-3H-1-benzazepin-2-yl]amino]-4-(trifluoromethyl)phenyl]methyl]carbamate —— C32H36F6N4O4
tert-butyl N-[[3-[[7-methoxy-8-[[4-(trifluoromethyl)cyclohexen-1-yl]carbamoyl]-4,5-dihydro-3H-1-benzazepin-2-yl]amino]-4-(trifluoromethyl)phenyl]methyl]carbamate
—— (E)-4-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-1,1,1-trifluorobut-3-en-2-one —— C18H14F3NO
(E)-4-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-1,1,1-trifluorobut-3-en-2-one
—— 11-Pentylpyrido[3,2-c][2]benzazepin-6-one —— C18H18N2O
11-Pentylpyrido[3,2-c][2]benzazepin-6-one
—— 6,6-Diethyl-10,12-difluoro-2-methyl-11-(trifluoromethyl)pyrido[2,1-a][2]benzazepin-5-ium —— C20H19F5N+
6,6-Diethyl-10,12-difluoro-2-methyl-11-(trifluoromethyl)pyrido[2,1-a][2]benzazepin-5-ium
—— 9-Cyclohexyl-8-ethylidene-14-methoxy-7-[3-(morpholin-4-ylsulfinylamino)-3-oxopropylidene]-6-azatetracyclo[9.4.0.02,4.06,10]pentadeca-1(11),9,12,14-tetraene-4-carboxylic acid —— C31H39N3O6S
9-Cyclohexyl-8-ethylidene-14-methoxy-7-[3-(morpholin-4-ylsulfinylamino)-3-oxopropylidene]-6-azatetracyclo[9.4.0.02,4.06,10]pentadeca-1(11),9,12,14-tetraene-4-carboxylic acid
—— [3-[3-(1,3-Benzoxazol-2-ylsulfanyl)propyl]-1,2,4,5-tetrahydro-3-benzazepin-7-yl]methanesulfonic acid —— C21H24N2O4S2
[3-[3-(1,3-Benzoxazol-2-ylsulfanyl)propyl]-1,2,4,5-tetrahydro-3-benzazepin-7-yl]methanesulfonic acid
—— ethane;2-methylsulfonyl-3,4-dihydro-1H-2-benzazepin-5-one —— C13H19NO3S
ethane;2-methylsulfonyl-3,4-dihydro-1H-2-benzazepin-5-one
—— 10-bromo-2-methyl-7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine —— C28H29BrN6OS
10-bromo-2-methyl-7-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine
—— [(5R)-11-carbamoyl-5,6-dihydrobenzo[b][1]benzazepin-5-yl] pyridine-3-carboxylate —— C21H17N3O3
[(5R)-11-carbamoyl-5,6-dihydrobenzo[b][1]benzazepin-5-yl] pyridine-3-carboxylate
—— ethane;(4Z)-4-ethylidene-1H-1-benzazepine-2,5-dione —— C14H17NO2
ethane;(4Z)-4-ethylidene-1H-1-benzazepine-2,5-dione
—— 2,5-dimethyl-4,5-dihydro-1H-1-benzazepine —— C12H15N
2,5-dimethyl-4,5-dihydro-1H-1-benzazepine
—— 2,5-Dimethyl-4,5-dihydro-1-benzazepin-1-ide —— C12H14N-
2,5-Dimethyl-4,5-dihydro-1-benzazepin-1-ide
—— 6,8-dimethoxy-2,5,5-trimethyl-1'-(3-phenylprop-2-enyl)spiro[10H-imidazo[1,5-b][2]benzazepine-3,4'-piperidine]-1-one —— C30H37N3O3
6,8-dimethoxy-2,5,5-trimethyl-1'-(3-phenylprop-2-enyl)spiro[10H-imidazo[1,5-b][2]benzazepine-3,4'-piperidine]-1-one
—— 3-[3-[1-(3,4-dimethoxy-7-bicyclo[4.2.0]octa-1,3,5-trienyl)ethenyl-methylamino]propyl]-7,8-dimethoxy-2,5-dihydro-1H-3-benzazepin-4-one —— C28H36N2O5
3-[3-[1-(3,4-dimethoxy-7-bicyclo[4.2.0]octa-1,3,5-trienyl)ethenyl-methylamino]propyl]-7,8-dimethoxy-2,5-dihydro-1H-3-benzazepin-4-one
—— 2H-pyrazolo[3,4-a][3]benzazepin-3-one —— C11H7N3O
2H-pyrazolo[3,4-a][3]benzazepin-3-one
—— 2,8-dimethyl-4,6-dihydro-3H-imidazo[4,5-d][2]benzazepin-5-amine —— C13H16N4
2,8-dimethyl-4,6-dihydro-3H-imidazo[4,5-d][2]benzazepin-5-amine
—— 2-(2,5-dimethylpyrazol-3-yl)-8-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-7,8,9,10-tetrahydro-6H-[1,3]oxazolo[4,5-g][1]benzazepine —— C32H34N8OS
2-(2,5-dimethylpyrazol-3-yl)-8-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-7,8,9,10-tetrahydro-6H-[1,3]oxazolo[4,5-g][1]benzazepine
—— N-(2-hydroxyethyl)-2-[4,4,7-trifluoro-1-[4-[(2S)-2-fluoropropoxy]-2-(trifluoromethyl)benzoyl]-2,3-dihydro-1-benzazepin-5-ylidene]acetamide —— C25H23F7N2O4
N-(2-hydroxyethyl)-2-[4,4,7-trifluoro-1-[4-[(2S)-2-fluoropropoxy]-2-(trifluoromethyl)benzoyl]-2,3-dihydro-1-benzazepin-5-ylidene]acetamide