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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R)-8-methoxy-1'-[(3S)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H29N3O4
(3R)-8-methoxy-1'-[(3S)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-8-methoxy-1'-[(3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H29N3O4
(3S)-8-methoxy-1'-[(3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-8-methoxy-1'-[(3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H29N3O4
(3R)-8-methoxy-1'-[(3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-8-methoxy-1'-[(3S)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H29N3O4
(3S)-8-methoxy-1'-[(3S)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-[(2-fluorophenyl)methyl]-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H23FN2O2
(3S,4'R)-1'-[(2-fluorophenyl)methyl]-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(6-chloro-1,3-benzodioxol-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H21ClN2O3
(3R)-1'-[(6-chloro-1,3-benzodioxol-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(1-benzofuran-2-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H22N2O2
(3S)-1'-(1-benzofuran-2-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-[[(1R)-cyclohex-3-en-1-yl]methyl]-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H28N2O2
(3S,4'R)-1'-[[(1R)-cyclohex-3-en-1-yl]methyl]-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-(4-fluorophenyl)sulfonyl-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21FN2O4S
(3S,4'R)-1'-(4-fluorophenyl)sulfonyl-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-4'-(hydroxymethyl)-1'-(thiophen-3-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H22N2O2S
(3S,4'R)-4'-(hydroxymethyl)-1'-(thiophen-3-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(1-benzofuran-2-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H22N2O2
(3R)-1'-(1-benzofuran-2-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H24N2O6S
(3S,4'R)-1'-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-(2-fluorophenyl)sulfonyl-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21FN2O4S
(3S,4'R)-1'-(2-fluorophenyl)sulfonyl-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(3-pyrazol-1-ylpropanoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H22N4O2
(3R)-1'-(3-pyrazol-1-ylpropanoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-[[(1S)-cyclohex-3-en-1-yl]methyl]-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H28N2O2
(3S,4'R)-1'-[[(1S)-cyclohex-3-en-1-yl]methyl]-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(6-morpholin-4-ylpyridin-3-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C23H28N4O2
(3R)-1'-[(6-morpholin-4-ylpyridin-3-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-4'-(hydroxymethyl)-1'-pyridin-3-ylsulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H21N3O4S
(3S,4'R)-4'-(hydroxymethyl)-1'-pyridin-3-ylsulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-4'-(hydroxymethyl)-1'-thiophen-2-ylsulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C18H20N2O4S2
(3S,4'R)-4'-(hydroxymethyl)-1'-thiophen-2-ylsulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(pyridin-4-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H21N3O
(3R)-1'-(pyridin-4-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H24N2O3
(3S)-1'-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(3,4-difluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H20F2N2O
(3R)-1'-[(3,4-difluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[4-(2-oxopyrrolidin-1-yl)butanoyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H27N3O3
(3R)-1'-[4-(2-oxopyrrolidin-1-yl)butanoyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[[5-(morpholin-4-ylmethyl)furan-2-yl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C23H29N3O3
(3R)-1'-[[5-(morpholin-4-ylmethyl)furan-2-yl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[2-(2-fluorophenoxy)ethyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H23FN2O2
(3S)-1'-[2-(2-fluorophenoxy)ethyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(pyridine-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H19N3O2
(3R)-1'-(pyridine-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(3-pyrazol-1-ylpropanoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H22N4O2
(3S)-1'-(3-pyrazol-1-ylpropanoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[3-(trifluoromethyl)phenyl]sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H19F3N2O3S
(3S)-1'-[3-(trifluoromethyl)phenyl]sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C13H16N2O
(3S)-spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[3-(2-fluorophenoxy)propyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H25FN2O2
(3R)-1'-[3-(2-fluorophenoxy)propyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[[2-(trifluoromethyl)phenyl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H21F3N2O
(3R)-1'-[[2-(trifluoromethyl)phenyl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(pyridine-3-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H19N3O2
(3S)-1'-(pyridine-3-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2-fluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21FN2O
(3R)-1'-[(2-fluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(3,4-dihydro-2H-chromen-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C23H26N2O2
(3S)-1'-(3,4-dihydro-2H-chromen-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(3,4-difluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H20F2N2O
(3S)-1'-[(3,4-difluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(pyridine-2-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H19N3O2
(3R)-1'-(pyridine-2-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(4-fluorobenzoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H19FN2O2
(3R)-1'-(4-fluorobenzoyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(pyridine-2-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H19N3O2
(3S)-1'-(pyridine-2-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(3,4-dihydro-2H-chromen-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C23H26N2O2
(3R)-1'-(3,4-dihydro-2H-chromen-6-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2-piperidin-1-yl-1,3-thiazol-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H28N4OS
(3R)-1'-[(2-piperidin-1-yl-1,3-thiazol-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S,4'R)-1'-(3-fluorophenyl)sulfonyl-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21FN2O4S
(3S,4'R)-1'-(3-fluorophenyl)sulfonyl-4'-(hydroxymethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(E)-3-pyridin-3-ylprop-2-enyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H23N3O
(3R)-1'-[(E)-3-pyridin-3-ylprop-2-enyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(cyclohexylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H28N2O
(3R)-1'-(cyclohexylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(pyridin-4-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H21N3O
(3S)-1'-(pyridin-4-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(4-fluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21FN2O
(3S)-1'-[(4-fluorophenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C24H27N3O2
(3S)-1'-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[4-(2-oxopyrrolidin-1-yl)butanoyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H27N3O3
(3S)-1'-[4-(2-oxopyrrolidin-1-yl)butanoyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C24H27N3O2
(3R)-1'-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[3-(2-fluorophenoxy)propyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H25FN2O2
(3S)-1'-[3-(2-fluorophenoxy)propyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-(3,4-difluorophenyl)sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H18F2N2O3S
(3R)-1'-(3,4-difluorophenyl)sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-(4-fluorophenyl)sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H19FN2O3S
(3S)-1'-(4-fluorophenyl)sulfonylspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one