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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-methyl-2,3-dihydro-1H-3-benzazepin-2-one 425386-56-7 C11H11NO
3-methyl-2,3-dihydro-1H-3-benzazepin-2-one
—— 1,1-Dimethylethyl 7-{(3S)-3-[{[(E)-2-(5-chloro-2-thienyl)ethenyl]sulfonyl}(2-hydroxyethyl)amino]-2-oxo-1-pyrrolidinyl}-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate 939043-46-6 C27H34ClN3O6S2
1,1-Dimethylethyl 7-{(3S)-3-[{[(E)-2-(5-chloro-2-thienyl)ethenyl]sulfonyl}(2-hydroxyethyl)amino]-2-oxo-1-pyrrolidinyl}-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate
—— 1,1-Dimethylethyl 7-((3S)-3-{[(3-chloro-1H-indol-6-yl)sulfonyl]-amino}-2-oxo-1-pyrrolidinyl)-1,2,4,5-tetrahydro-3H-3-benzazepine-3-carboxylate 939043-39-7 C27H31ClN4O5S
1,1-Dimethylethyl 7-((3S)-3-{[(3-chloro-1H-indol-6-yl)sulfonyl]-amino}-2-oxo-1-pyrrolidinyl)-1,2,4,5-tetrahydro-3H-3-benzazepine-3-carboxylate
—— 1,1-dimethylethyl 7-[(3S)-3-amino-2-oxo-1-pyrrolidinyl]-1,2,4,5-tetrahydro-3H-3-benzazepine-3-carboxylate 939043-38-6 C19H27N3O3
1,1-dimethylethyl 7-[(3S)-3-amino-2-oxo-1-pyrrolidinyl]-1,2,4,5-tetrahydro-3H-3-benzazepine-3-carboxylate
—— 1,1-dimethylethyl 7-((3S)-3-{[(3-chloro-1H-indol-6-yl)sulfonyl]amino}-2-oxo-1-pyrrolidinyl)-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate 939043-37-5 C27H31ClN4O5S
1,1-dimethylethyl 7-((3S)-3-{[(3-chloro-1H-indol-6-yl)sulfonyl]amino}-2-oxo-1-pyrrolidinyl)-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate
—— 1,1-Dimethylethyl 7-{(3S)-3-[{[(E)-2-(5-chloro-2-thienyl)ethenyl]sulfonyl}(methyl)amino]-2-oxo-1-pyrrolidinyl}-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate 939043-44-4 C26H32ClN3O5S2
1,1-Dimethylethyl 7-{(3S)-3-[{[(E)-2-(5-chloro-2-thienyl)ethenyl]sulfonyl}(methyl)amino]-2-oxo-1-pyrrolidinyl}-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate
—— 1,1-Dimethylethyl 7-[(3S)-2-oxo-3-({[(phenylmethyl)oxy]carbonyl}amino)-1-pyrrolidinyl]-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate 939043-34-2 C27H33N3O5
1,1-Dimethylethyl 7-[(3S)-2-oxo-3-({[(phenylmethyl)oxy]carbonyl}amino)-1-pyrrolidinyl]-1,3,4,5-tetrahydro-2H-2-benzazepine-2-carboxylate
—— 7-Brom-2,3,-dihydro-5-hydroxy-2-oxo-1H-1-benzazepin-4-carbonsaeureethylester 137046-57-2 C13H12BrNO4
7-Brom-2,3,-dihydro-5-hydroxy-2-oxo-1H-1-benzazepin-4-carbonsaeureethylester
—— 7-Bromo-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[d]azepine 833480-19-6 C11H12BrN
7-Bromo-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[d]azepine
—— 5-(11-Carbamoylbenzo[b][1]benzazepin-3-yl)oxypentanoic acid 1335422-97-3 C20H20N2O4
5-(11-Carbamoylbenzo[b][1]benzazepin-3-yl)oxypentanoic acid
—— 6,7,8,9-tetrahydro-2-amino-7-((1-[<sup>13</sup>C]methyl-1H-[<sup>13</sup>N<sub>2</sub>]pyrazol-4-yl)[<sup>13</sup>C]methyl)-5H-thiazolo[4,5-h][3]benzazepine 1403324-99-1 C16H19N5S
6,7,8,9-tetrahydro-2-amino-7-((1-[<sup>13</sup>C]methyl-1H-[<sup>13</sup>N<sub>2</sub>]pyrazol-4-yl)[<sup>13</sup>C]methyl)-5H-thiazolo[4,5-h][3]benzazepine
—— tert-butyl 4-{1-[6-fluoro-2-oxo-1-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-1-benzazepin-3-yl]-1H-1,2,3-triazol-4-yl}piperidine-1-carboxylate 1231192-17-8 C24H29F4N5O3
tert-butyl 4-{1-[6-fluoro-2-oxo-1-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-1-benzazepin-3-yl]-1H-1,2,3-triazol-4-yl}piperidine-1-carboxylate
—— N-[(R)-4-chloro-8-oxo-9-(2,2,2-trifluoroethyl)-3,6,7,8,9,10-hexahydro-azepino[3,4-e]indazol-7-yl]-4-(2-oxo-2,3-dihydro-imidazo[4,5-b]pyridin-1-yl)-piperidine-1-carboxamide 1038866-29-3 C25H24ClF3N8O3
N-[(R)-4-chloro-8-oxo-9-(2,2,2-trifluoroethyl)-3,6,7,8,9,10-hexahydro-azepino[3,4-e]indazol-7-yl]-4-(2-oxo-2,3-dihydro-imidazo[4,5-b]pyridin-1-yl)-piperidine-1-carboxamide
—— N-[(R)-4-chloro-8-oxo-9-(2,2,2-trifluoroethyl)-3,6,7,8,9,10-hexahydro-azepino[3,4-e]indazol-7-yl]-2'-oxo-1',2'-dihydro-1H-spiro[piperidine-4,4'-pyrido[2,3-d][1,3]oxazine]-1-carboxamide 1038866-30-6 C25H23ClF3N7O4
N-[(R)-4-chloro-8-oxo-9-(2,2,2-trifluoroethyl)-3,6,7,8,9,10-hexahydro-azepino[3,4-e]indazol-7-yl]-2'-oxo-1',2'-dihydro-1H-spiro[piperidine-4,4'-pyrido[2,3-d][1,3]oxazine]-1-carboxamide
—— ethyl 8-[2-(imidazo [1,2-a]pyrimidin-2-yl)ethoxy]-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetra-hydro-1H-2-benzazepin-4-acetate 1152636-75-3 C24H25F3N4O4
ethyl 8-[2-(imidazo [1,2-a]pyrimidin-2-yl)ethoxy]-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetra-hydro-1H-2-benzazepin-4-acetate
—— 3-tert-butoxycarbonyl-7-chloro-6-(4-trifluoromethoxy-benzylthio)-2,3,4,5-tetrahydro-1H-benzo[d]azepine 1133340-46-1 C23H25ClF3NO3S
3-tert-butoxycarbonyl-7-chloro-6-(4-trifluoromethoxy-benzylthio)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
—— ethyl 3-oxo-8-[2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-2-yl)ethoxy]-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepin-4-acetate hydrochloride 1152635-67-0 C24H29F3N4O4*ClH
ethyl 3-oxo-8-[2-(5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-2-yl)ethoxy]-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepin-4-acetate hydrochloride
—— 8-[2-(imidazo [1,2-b][1,2,4]triazin-6-yl)ethoxy]-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepin-4-acetic acid 1152636-81-1 C21H20F3N5O4
8-[2-(imidazo [1,2-b][1,2,4]triazin-6-yl)ethoxy]-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepin-4-acetic acid
—— Ethyl 8-[2-(imidazo[1,2-b][1,2,4]triazin-6-yl)ethoxy]-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepin-4-acetate 1152636-78-6 C23H24F3N5O4
Ethyl 8-[2-(imidazo[1,2-b][1,2,4]triazin-6-yl)ethoxy]-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepin-4-acetate
—— ethyl 8-hydroxy-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepin-4-acetate 1029477-74-4 C16H18F3NO4
ethyl 8-hydroxy-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepin-4-acetate
—— tert-butyl 7-amino-8-nitro-1,2,4,5-tetrahydro-3H-benzo[d]azepine-3-carboxylate 1241841-12-2 C15H21N3O4
tert-butyl 7-amino-8-nitro-1,2,4,5-tetrahydro-3H-benzo[d]azepine-3-carboxylate
—— 2-[2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)-5-methyl-pyrimidin-4-ylamino]-N-methyl-benzamide 1022964-09-5 C25H30N6O
2-[2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)-5-methyl-pyrimidin-4-ylamino]-N-methyl-benzamide
—— 1028486-06-7 C27H20ClFN4NaO4
—— rel-(3aR,10bS)-8-(2,6-Difluorophenyl)-2,3,3a,4,5,10b-hexahydropyrrolo[3,4-d][2]benzazepin-6(1H)-one 1256600-00-6 C18H16F2N2O
rel-(3aR,10bS)-8-(2,6-Difluorophenyl)-2,3,3a,4,5,10b-hexahydropyrrolo[3,4-d][2]benzazepin-6(1H)-one
—— 2-{5-chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]-pyrimidin-4-ylamino}-5,N-dimethyl-benzamide 1022969-61-4 C26H31ClN6O2
2-{5-chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]-pyrimidin-4-ylamino}-5,N-dimethyl-benzamide
—— 2-(5-chloro-2-{1-[2-(4-methyl-piperazin-1-yl)-2-oxo-ethyl]-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-ylamino}-pyrimidin-4-ylamino)-N-methyl-benzenesulfonamide 1022954-77-3 C28H33ClN8O4S
2-(5-chloro-2-{1-[2-(4-methyl-piperazin-1-yl)-2-oxo-ethyl]-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-ylamino}-pyrimidin-4-ylamino)-N-methyl-benzenesulfonamide
—— 3-ethyl-8-methoxy-1,3,4,5-tetrahydro-benzo[d]azepin-2-one 1022966-84-2 C13H17NO2
3-ethyl-8-methoxy-1,3,4,5-tetrahydro-benzo[d]azepin-2-one
—— (5R)-7-chloro-3,5-dimethyl-1,2,4,5-tetrahydro-3-benzazepine 616202-93-8 C12H16ClN
(5R)-7-chloro-3,5-dimethyl-1,2,4,5-tetrahydro-3-benzazepine
—— 4-dimethylaminomethylene-7-methoxy-3,4-dihydro-1H-benzo[b]azepine-2,5-dione 884196-33-2 C14H16N2O3
4-dimethylaminomethylene-7-methoxy-3,4-dihydro-1H-benzo[b]azepine-2,5-dione
—— 5-(4-chlorophenyl)-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1H-benzo[c]azepine 921218-89-5 C18H20ClNO
5-(4-chlorophenyl)-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1H-benzo[c]azepine
—— 5-(4-fluorophenyl)-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1H-benzo[c]azepine 921436-04-6 C18H20FNO
5-(4-fluorophenyl)-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1H-benzo[c]azepine
—— 5-(1-Benzothiophen-5-yl)-8-methoxy-2-methyl-1,3,4,5-tetrahydro-2-benzazepine —— C20H21NOS
5-(1-Benzothiophen-5-yl)-8-methoxy-2-methyl-1,3,4,5-tetrahydro-2-benzazepine
—— t-butyl 5-cyclopropyl-6-methyl-3,4,6,7,9,10-hexahydro[1,4]oxazino[2,3-h][3]benzazepine-8(2H)-carboxylate 1334433-47-4 C21H30N2O3
t-butyl 5-cyclopropyl-6-methyl-3,4,6,7,9,10-hexahydro[1,4]oxazino[2,3-h][3]benzazepine-8(2H)-carboxylate
—— 1-methyl-1,3,4,6,7,8,9,10-octahydro-2H-azepino[4,5-g]quinolin-2-one monohydrochloride 1334438-77-5 C14H18N2O*ClH
1-methyl-1,3,4,6,7,8,9,10-octahydro-2H-azepino[4,5-g]quinolin-2-one monohydrochloride
—— t-butyl 6-methyl-3,4,6,7,9,10-hexahydro[1,4]oxazino[2,3-h][3]benzazepine-8(2H)-carboxylate 1334434-52-4 C18H26N2O3
t-butyl 6-methyl-3,4,6,7,9,10-hexahydro[1,4]oxazino[2,3-h][3]benzazepine-8(2H)-carboxylate
—— t-butyl 3,4,6,7,9,10-hexahydro[1,4]oxazino[2,3-h][3]benzazepine-8(2H)-carboxylate 871501-47-2 C17H24N2O3
t-butyl 3,4,6,7,9,10-hexahydro[1,4]oxazino[2,3-h][3]benzazepine-8(2H)-carboxylate
—— 4-methyl-7-amino-1,3,4,5-tetrahydro-1-benzazepin-2-one 1023317-34-1 C11H14N2O
4-methyl-7-amino-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 4-methyl-7-nitro-1,3,4,5-tetrahydro-1-benzazepin-2-one 1023317-32-9 C11H12N2O3
4-methyl-7-nitro-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-chloro-5-methyl-1,3,4,5-tetrahydro-1-benzazepin-2-one 1023317-41-0 C11H12ClNO
7-chloro-5-methyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-fluoro-4-methyl-1,3,4,5-tetrahydro-1-benzazepin-2-one 1023317-36-3 C11H12FNO
7-fluoro-4-methyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 5-methyl-7-nitro-1,3,4,5-tetrahydro-1-benzazepin-2-one 104479-29-0 C11H12N2O3
5-methyl-7-nitro-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 8-trifluoromethyl-1,2,3,4-tetrahydrobenzo[b]azepin-5-one 920334-40-3 C11H10F3NO
8-trifluoromethyl-1,2,3,4-tetrahydrobenzo[b]azepin-5-one
—— 5,5-Dimethyl-2,3,4,5-tetrahydro-1H-2-benzoazepin-1-one 1279622-00-2 C12H15NO
5,5-Dimethyl-2,3,4,5-tetrahydro-1H-2-benzoazepin-1-one
—— 3-(dimethylamino)propyl 2-(4-((1E,4E)-2-(tert-butoxycarbonylamino)-4-((3-(tert-butyldimethylsilyloxy)propyl)(propyl)carbamoyl)-3H-benzo[b]azepin-8-yl)phenyl)acetate 1268465-38-8 C41H62N4O6Si
3-(dimethylamino)propyl 2-(4-((1E,4E)-2-(tert-butoxycarbonylamino)-4-((3-(tert-butyldimethylsilyloxy)propyl)(propyl)carbamoyl)-3H-benzo[b]azepin-8-yl)phenyl)acetate
—— propyl 2-(4-((1E,4E)-2-(tert-butoxycarbonylamino)-4-((3-(tert-butyldimethylsilyloxy)propyl)(propyl)carbamoyl)-3H-benzo[b]azepin-8-yl)phenyl)acetate 1268465-25-3 C39H57N3O6Si
propyl 2-(4-((1E,4E)-2-(tert-butoxycarbonylamino)-4-((3-(tert-butyldimethylsilyloxy)propyl)(propyl)carbamoyl)-3H-benzo[b]azepin-8-yl)phenyl)acetate
—— benzyl 2-(4-((1E,4E)-2-amino-4-(dipropylcarbamoyl)-3H-benzo[b]azepin-8-yl)phenyl)acetate 1268465-09-3 C32H35N3O3
benzyl 2-(4-((1E,4E)-2-amino-4-(dipropylcarbamoyl)-3H-benzo[b]azepin-8-yl)phenyl)acetate
—— butyl 2-(4-((1E,4E)-2-(tert-butoxycarbonylamino)-4-((3-(tert-butyldimethylsilyloxy)propyl)(propyl)carbamoyl)-3H-benzo[b]azepin-8-yl)phenyl)acetate 1268465-27-5 C40H59N3O6Si
butyl 2-(4-((1E,4E)-2-(tert-butoxycarbonylamino)-4-((3-(tert-butyldimethylsilyloxy)propyl)(propyl)carbamoyl)-3H-benzo[b]azepin-8-yl)phenyl)acetate
—— 1-(4-(3-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-2-oxopropyl)piperidin-1-yl)propan-1-one 1204828-92-1 C25H36N2O2
1-(4-(3-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)-2-oxopropyl)piperidin-1-yl)propan-1-one
—— 7-(1-methoxy-3-(1-methyl-1H-pyrazol-3-yl)propyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepinium chloride 1204828-84-1 C18H25N3O*ClH
7-(1-methoxy-3-(1-methyl-1H-pyrazol-3-yl)propyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepinium chloride
—— 1-(4-(hydroxy(2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)methyl)piperidin-1-yl)ethanone 1204829-18-4 C18H26N2O2
1-(4-(hydroxy(2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)methyl)piperidin-1-yl)ethanone