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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-Bromo-2,3,4,5-tetrahydro-1H-1-benzazepine-9-carboxylic acid benzyl ester 133433-69-9 C18H18BrNO2
7-Bromo-2,3,4,5-tetrahydro-1H-1-benzazepine-9-carboxylic acid benzyl ester
—— 8-(Methoxymethyl)-5-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-ol 113080-87-8 C18H21NO2
8-(Methoxymethyl)-5-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-ol
—— 8-chloro-1-(2-chlorophenyl)-4-dimethylaminomethylene-3,4-dihydro-2-benzazepin-5-one 58582-31-3 C19H16Cl2N2O
8-chloro-1-(2-chlorophenyl)-4-dimethylaminomethylene-3,4-dihydro-2-benzazepin-5-one
—— 1-butyl-3-[(3-dimethylcarbamoyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl) sulfonyl]urea 57846-54-5 C18H28N4O4S
1-butyl-3-[(3-dimethylcarbamoyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl) sulfonyl]urea
—— 1-Hydroxy-3-methanesulfonyl-7-methoxy-4-methyl-1,2,4,5-tetrahydro-3H,3-benzazepine 76208-86-1 C13H19NO4S
1-Hydroxy-3-methanesulfonyl-7-methoxy-4-methyl-1,2,4,5-tetrahydro-3H,3-benzazepine
—— (S)-8-[3-(4-methylpyridin-2-ylamino)-1-propyloxy]-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepine-4-acetic acid 205678-28-0 C23H26F3N3O4
(S)-8-[3-(4-methylpyridin-2-ylamino)-1-propyloxy]-3-oxo-2-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1H-2-benzazepine-4-acetic acid
—— methyl (R)-(+)-8-hydroxy-3-oxo-2,3,4,5-tetrahydro-1H-2-benzazepine-4-acetate 205676-79-5 C13H15NO4
methyl (R)-(+)-8-hydroxy-3-oxo-2,3,4,5-tetrahydro-1H-2-benzazepine-4-acetate
—— methyl (S)-(-)-8-hydroxy-3-oxo-2,3,4,5-tetrahydro-1H-2-benzazepine-4-acetate 205676-80-8 C13H15NO4
methyl (S)-(-)-8-hydroxy-3-oxo-2,3,4,5-tetrahydro-1H-2-benzazepine-4-acetate
—— 8-Chloro-4-[1-dimethylamino-meth-(E)-ylidene]-1-phenyl-3,4-dihydro-benzo[c]azepin-5-one 58582-16-4 C19H17ClN2O
8-Chloro-4-[1-dimethylamino-meth-(E)-ylidene]-1-phenyl-3,4-dihydro-benzo[c]azepin-5-one
—— 4-Cyano-10-aza-tricyclo[6.3.1.02,7]dodeca-2(7),3,5-triene-10-carboxylic acid tert-butyl ester 230615-79-9 C17H20N2O2
4-Cyano-10-aza-tricyclo[6.3.1.02,7]dodeca-2(7),3,5-triene-10-carboxylic acid tert-butyl ester
—— 6-Methyl-7-isobutyl-5,7,13-triazatetracyclo[9.3.1.02,10.04,8]pentadeca-2(10),3,5,8-tetraene-13-carboxylic acid tert-butyl ester 230615-68-6 C22H31N3O2
6-Methyl-7-isobutyl-5,7,13-triazatetracyclo[9.3.1.02,10.04,8]pentadeca-2(10),3,5,8-tetraene-13-carboxylic acid tert-butyl ester
—— Methyl (S)-8-methoxy-3-oxo-2-(4-trifluoromethylbenzyl)-2,3,4,5-tetrahydro-1 H-2-benzazepine-4-acetate 205677-00-5 C22H22F3NO4
Methyl (S)-8-methoxy-3-oxo-2-(4-trifluoromethylbenzyl)-2,3,4,5-tetrahydro-1 H-2-benzazepine-4-acetate
—— ethyl (R)-(1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyrazino[1,2-a]azepin-2-yl)carboxylate 136224-83-4 C20H22N2O2
ethyl (R)-(1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyrazino[1,2-a]azepin-2-yl)carboxylate
—— 8-Chlor-2H-2-benzazepin-1,3(2H)-dion 56820-61-2 C10H6ClNO2
8-Chlor-2H-2-benzazepin-1,3(2H)-dion
—— 3-(hydroxy)-2,3,4,5-tetrahydro-1H-1-benzazepin-2-one 187107-82-0 C10H11NO2
3-(hydroxy)-2,3,4,5-tetrahydro-1H-1-benzazepin-2-one
—— phenylmethyl-7-[5-(aminomethyl)-2-oxo-1,3-oxazolidin-3-yl]-2H,3H,4H,5H-benzo[f]azaperhydroepinecarboxylate 740842-83-5 C22H25N3O4
phenylmethyl-7-[5-(aminomethyl)-2-oxo-1,3-oxazolidin-3-yl]-2H,3H,4H,5H-benzo[f]azaperhydroepinecarboxylate
—— N,N-dimethyl-3-[9-(trifluoromethylsulfanyl)-5,6-dihydropyrrolo[1,2-c][3]benzazepin-11-ylidene]propan-1-amine 62542-10-3 C19H21F3N2S
N,N-dimethyl-3-[9-(trifluoromethylsulfanyl)-5,6-dihydropyrrolo[1,2-c][3]benzazepin-11-ylidene]propan-1-amine
—— (3S)-7,8-dimethoxy-17,19-dioxa-11-azapentacyclo[12.7.0.03,11.04,9.016,20]henicosa-1(21),4(9),5,7,14,16(20)-hexaene 1383957-75-2 C20H21NO4
(3S)-7,8-dimethoxy-17,19-dioxa-11-azapentacyclo[12.7.0.03,11.04,9.016,20]henicosa-1(21),4(9),5,7,14,16(20)-hexaene
—— 8-methoxy-4-methyl-2-propyl-4,5-dihydro-1H-2-benzazepin-3-one 1173893-68-9 C15H21NO2
8-methoxy-4-methyl-2-propyl-4,5-dihydro-1H-2-benzazepin-3-one
—— 2-butyl-8-methoxy-4-methyl-4,5-dihydro-1H-2-benzazepin-3-one 1173893-69-0 C16H23NO2
2-butyl-8-methoxy-4-methyl-4,5-dihydro-1H-2-benzazepin-3-one
—— 1-Methyl-2,3-dihydro-1-benzazepine;hydrobromide 54620-91-6 C11H14BrN
1-Methyl-2,3-dihydro-1-benzazepine;hydrobromide
—— 5-phenyl-2,3,4,5-tetrahydro-1H-1-benzazepine;hydrochloride 16140-93-5 C16H18ClN
5-phenyl-2,3,4,5-tetrahydro-1H-1-benzazepine;hydrochloride
—— 4-Hydroxy-2,5-dihydro-1H-1-benzazepin-2,5-dion 22757-74-0 C10H7NO3
4-Hydroxy-2,5-dihydro-1H-1-benzazepin-2,5-dion
—— 2,3,4,5-tetrahydro-1H-benzo[b]azepine hydrochloride 112610-03-4 C10H13N*ClH
2,3,4,5-tetrahydro-1H-benzo[b]azepine hydrochloride
—— 9-Ethyl-2,3,4,5-tetrahydro-1H-1-benzazepin-5-amine 886367-44-8 C12H18N2
9-Ethyl-2,3,4,5-tetrahydro-1H-1-benzazepin-5-amine
—— 7-Ethyl-2,3,4,5-tetrahydro-1H-benzo[B]azepin-5-ylamine 886367-65-3 C12H18N2
7-Ethyl-2,3,4,5-tetrahydro-1H-benzo[B]azepin-5-ylamine
—— 7-Methyl-2,3,4,5-tetrahydro-1H-benzo[b]azepin-5-amine 886367-51-7 C11H16N2
7-Methyl-2,3,4,5-tetrahydro-1H-benzo[b]azepin-5-amine
—— 7-Ethyl-1,2,3,4-tetrahydro-benzo[B]azepin-5-one 886366-97-8 C12H15NO
7-Ethyl-1,2,3,4-tetrahydro-benzo[B]azepin-5-one
—— 9-Chloro-2,3,4,5-tetrahydro-1H-1-benzazepin-5-amine 886367-30-2 C10H13ClN2
9-Chloro-2,3,4,5-tetrahydro-1H-1-benzazepin-5-amine
—— 3,4,5,6-Tetrahydroimidazo[4,5-d][2]benzazepine 1214875-37-2 C11H11N3
3,4,5,6-Tetrahydroimidazo[4,5-d][2]benzazepine
—— 2,3-dihydro-[1H]-2-benzazepine 1043927-17-8 C10H11N
2,3-dihydro-[1H]-2-benzazepine
—— Ditert-butyl 11-[3-(dimethylamino)propyl]-5,6-dihydrobenzo[b][1]benzazepine-2,9-dicarboxylate 1338085-85-0 C29H40N2O4
Ditert-butyl 11-[3-(dimethylamino)propyl]-5,6-dihydrobenzo[b][1]benzazepine-2,9-dicarboxylate
—— 11-[3-(Dimethylamino)propyl]-5,6-dihydrobenzo[b][1]benzazepine-2,9-dicarboxylic acid;hydrochloride 1338085-90-7 C21H24N2O4*ClH
11-[3-(Dimethylamino)propyl]-5,6-dihydrobenzo[b][1]benzazepine-2,9-dicarboxylic acid;hydrochloride
—— 2-O-tert-butyl 9-O-ethyl 11-[3-(dimethylamino)propyl]-5,6-dihydrobenzo[b][1]benzazepine-2,9-dicarboxylate 1338085-97-4 C27H36N2O4
2-O-tert-butyl 9-O-ethyl 11-[3-(dimethylamino)propyl]-5,6-dihydrobenzo[b][1]benzazepine-2,9-dicarboxylate
—— Tert-butyl 11-[3-(dimethylamino)propyl]-9-(hydroxymethyl)-5,6-dihydrobenzo[b][1]benzazepine-2-carboxylate 1338085-98-5 C25H34N2O3
Tert-butyl 11-[3-(dimethylamino)propyl]-9-(hydroxymethyl)-5,6-dihydrobenzo[b][1]benzazepine-2-carboxylate
—— 8-β-D-galactopyranosyloxy-2H-dibenz[b,f]azepin-2-one 149322-40-7 C20H19NO7
8-β-D-galactopyranosyloxy-2H-dibenz[b,f]azepin-2-one
—— ethyl 6,7-dihydro-5H-imidazo[2,1-a][2]benzazepine-3-carboxylate 1333169-44-0 C15H16N2O2
ethyl 6,7-dihydro-5H-imidazo[2,1-a][2]benzazepine-3-carboxylate
—— N-{(1R,2R)-2-[5-chloro-2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)pyrimidin-4-ylamino]cyclohexyl}acetamide 1022973-31-4 C24H33ClN6O
N-{(1R,2R)-2-[5-chloro-2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)pyrimidin-4-ylamino]cyclohexyl}acetamide
—— N-{(1R,2R)-2-[5-chloro-2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)pyrimidin-4-ylamino]cyclohexyl}-2,2,2-trifluoroacetamide 1022973-33-6 C24H30ClF3N6O
N-{(1R,2R)-2-[5-chloro-2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)pyrimidin-4-ylamino]cyclohexyl}-2,2,2-trifluoroacetamide
—— 5,7-Dioxa-14-azapentacyclo[12.8.0.02,10.04,8.016,21]docosa-1(22),2,4(8),9,11,16,18,20-octaen-15-one 1338475-52-7 C19H13NO3
5,7-Dioxa-14-azapentacyclo[12.8.0.02,10.04,8.016,21]docosa-1(22),2,4(8),9,11,16,18,20-octaen-15-one
—— N-((1R,2R)-2-{5-chloro-2-[8-methoxy-3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]pyrimidin-4-ylamino}cyclohexyl)-N-ethylmethanesulfonamide 1022955-52-7 C27H41ClN6O4S
N-((1R,2R)-2-{5-chloro-2-[8-methoxy-3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]pyrimidin-4-ylamino}cyclohexyl)-N-ethylmethanesulfonamide
—— 2,2,2-trifluoroethanesulfonic acid ((1R,2R)-2-{5-chloro-2-[3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]pyrimidin-4-ylamino}cyclohexyl)amide 1022973-46-1 C25H34ClF3N6O3S
2,2,2-trifluoroethanesulfonic acid ((1R,2R)-2-{5-chloro-2-[3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]pyrimidin-4-ylamino}cyclohexyl)amide
—— N-((1R,2R)-2-{5-chloro-2-[3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]-pyrimidin-4-ylamino}cyclohexyl)methanesulfonamide 1022956-07-5 C24H35ClN6O3S
N-((1R,2R)-2-{5-chloro-2-[3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]-pyrimidin-4-ylamino}cyclohexyl)methanesulfonamide
—— N-((1R,2R)-2-{5-chloro-2-[8-methoxy-3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]pyrimidin-4-ylamino}cyclohexyl)-N-methyl-methanesulfonamide 1022955-49-2 C26H39ClN6O4S
N-((1R,2R)-2-{5-chloro-2-[8-methoxy-3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]pyrimidin-4-ylamino}cyclohexyl)-N-methyl-methanesulfonamide
—— N-{(1R,2R)-2-[5-chloro-2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)pyrimidin-4-ylamino]cyclohexyl}methanesulfonamide 1022973-19-8 C23H33ClN6O2S
N-{(1R,2R)-2-[5-chloro-2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)pyrimidin-4-ylamino]cyclohexyl}methanesulfonamide
—— 3-{(1R,2R)-2-[5-chloro-2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)pyrimidin-4-ylamino]cyclohexyl}-1,1-dimethylurea 1022973-37-0 C25H36ClN7O
3-{(1R,2R)-2-[5-chloro-2-(3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino)pyrimidin-4-ylamino]cyclohexyl}-1,1-dimethylurea
—— propane-2-sulfonic acid ((1R,2R)-2-{5-chloro-2-[3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]pyrimidin-4-ylamino}cyclohexyl)amide 1022973-51-8 C26H39ClN6O3S
propane-2-sulfonic acid ((1R,2R)-2-{5-chloro-2-[3-(2-methoxyethyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ylamino]pyrimidin-4-ylamino}cyclohexyl)amide
—— 2-Hydroxy-2,3,4,5-tetrahydro-1H-3-benzazepin 19301-10-1 C10H13NO
2-Hydroxy-2,3,4,5-tetrahydro-1H-3-benzazepin
—— 10,11-Dihydro-5-(2-(octahydro-2H-pyrido(1,2-a)pyrazin-2-yl)ethyl)-5H-dibenz(b,f)azepine 34790-38-0 C24H31N3
10,11-Dihydro-5-(2-(octahydro-2H-pyrido(1,2-a)pyrazin-2-yl)ethyl)-5H-dibenz(b,f)azepine
—— Alisertib Sodium 1208255-63-3 C27H21ClFN4NaO5
Alisertib Sodium