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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7S,10R,11R,12S)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-10,17-diamine —— C23H23FN8O
(7S,10R,11R,12S)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-10,17-diamine
—— (7S,11S,12S)-15-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,10,21-pentazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaen-17-amine —— C22H21FN8O
(7S,11S,12S)-15-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,10,21-pentazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaen-17-amine
—— (7R,8S,11S,12S)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-8,17-diamine —— C23H23FN8O
(7R,8S,11S,12S)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-8,17-diamine
—— (8S,9S,10S,11S)-14-fluoro-16-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,20-tetrazahexacyclo[15.2.1.18,10.05,19.06,11.013,18]henicosa-1(19),2,4,13,15,17-hexaene-9,16-diamine —— C23H23FN8O
(8S,9S,10S,11S)-14-fluoro-16-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,20-tetrazahexacyclo[15.2.1.18,10.05,19.06,11.013,18]henicosa-1(19),2,4,13,15,17-hexaene-9,16-diamine
—— (7R,11S,12S)-15-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,8,21-pentazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaen-17-amine —— C22H21FN8O
(7R,11S,12S)-15-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,8,21-pentazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaen-17-amine
—— (8S,9R,10S,11S)-14-fluoro-16-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,20-tetrazahexacyclo[15.2.1.18,10.05,19.06,11.013,18]henicosa-1(19),2,4,13,15,17-hexaene-9,16-diamine —— C23H23FN8O
(8S,9R,10S,11S)-14-fluoro-16-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,20-tetrazahexacyclo[15.2.1.18,10.05,19.06,11.013,18]henicosa-1(19),2,4,13,15,17-hexaene-9,16-diamine
—— (7S,10R,11R,13R)-16-fluoro-18-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,22-tetrazahexacyclo[17.2.1.05,21.06,13.07,11.015,20]docosa-1(21),2,4,15,17,19-hexaene-10,18-diamine —— C24H25FN8O
(7S,10R,11R,13R)-16-fluoro-18-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,22-tetrazahexacyclo[17.2.1.05,21.06,13.07,11.015,20]docosa-1(21),2,4,15,17,19-hexaene-10,18-diamine
—— (7S,12R,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,11,22-pentazahexacyclo[17.2.1.05,21.06,13.07,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine —— C23H23FN8O
(7S,12R,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,11,22-pentazahexacyclo[17.2.1.05,21.06,13.07,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine
—— (7R,11S,12S)-15-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,21-pentazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaen-17-amine —— C22H21FN8O
(7R,11S,12S)-15-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,21-pentazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaen-17-amine
—— (7S,12S,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,10,22-pentazahexacyclo[17.2.1.05,21.06,13.07,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine —— C23H23FN8O
(7S,12S,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,10,22-pentazahexacyclo[17.2.1.05,21.06,13.07,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine
—— N-cyclohexyl-3-(4-methoxyphenyl)-1H-1-benzazepine-5-carboxamide —— C24H26N2O2
N-cyclohexyl-3-(4-methoxyphenyl)-1H-1-benzazepine-5-carboxamide
—— 3-[[4-[1-[4-(2,3-dimethylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]-N-(3-hydroxypropyl)benzamide —— C36H42N4O4
3-[[4-[1-[4-(2,3-dimethylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]-N-(3-hydroxypropyl)benzamide
—— 7-chloro-N-[[4-(cyclopropylmethylamino)phenyl]methyl]-N-pyrazol-1-yl-2,3,4,5-tetrahydro-1H-3-benzazepin-6-amine —— C24H28ClN5
7-chloro-N-[[4-(cyclopropylmethylamino)phenyl]methyl]-N-pyrazol-1-yl-2,3,4,5-tetrahydro-1H-3-benzazepin-6-amine
—— 2-amino-2-[4-[[(7-chloro-2,3,4,5-tetrahydro-1H-3-benzazepin-6-yl)amino]methyl]phenyl]-1-cyclopropylethanone;butanedioic acid —— C26H32ClN3O5
2-amino-2-[4-[[(7-chloro-2,3,4,5-tetrahydro-1H-3-benzazepin-6-yl)amino]methyl]phenyl]-1-cyclopropylethanone;butanedioic acid
—— (E)-7-chloro-6-{[6-(2-cyclohexyl-vinyl)-pyridin-3-ylmethyl]-amino}-2,3,4,5-tetrahydro-1H-benzo[d]azepine succinate —— C4H6O4*C24H30ClN3
(E)-7-chloro-6-{[6-(2-cyclohexyl-vinyl)-pyridin-3-ylmethyl]-amino}-2,3,4,5-tetrahydro-1H-benzo[d]azepine succinate
—— 7-chloro-N-[[6-(cyclohexyloxymethyl)pyridin-3-yl]methyl]-2,3,4,5-tetrahydro-1H-3-benzazepin-6-amine —— C23H30ClN3O
7-chloro-N-[[6-(cyclohexyloxymethyl)pyridin-3-yl]methyl]-2,3,4,5-tetrahydro-1H-3-benzazepin-6-amine
—— 7-chloro-N-[[6-(cyclopentyloxymethyl)pyridin-3-yl]methyl]-2,3,4,5-tetrahydro-1H-3-benzazepin-6-amine —— C22H28ClN3O
7-chloro-N-[[6-(cyclopentyloxymethyl)pyridin-3-yl]methyl]-2,3,4,5-tetrahydro-1H-3-benzazepin-6-amine
—— 1-amino-1-[4-[[(7-chloro-2,3,4,5-tetrahydro-1H-3-benzazepin-6-yl)amino]methyl]phenyl]-3,3-dimethylbutan-2-one —— C23H30ClN3O
1-amino-1-[4-[[(7-chloro-2,3,4,5-tetrahydro-1H-3-benzazepin-6-yl)amino]methyl]phenyl]-3,3-dimethylbutan-2-one
—— (E)-7-chloro-6-{[5-(2-cyclohexyl-vinyl)-pyridin-2-ylmethyl]-amino}-2,3,4,5-tetrahydro-1H-benzo[d]azepine succinate —— C4H6O4*C24H30ClN3
(E)-7-chloro-6-{[5-(2-cyclohexyl-vinyl)-pyridin-2-ylmethyl]-amino}-2,3,4,5-tetrahydro-1H-benzo[d]azepine succinate
—— 2-amino-2-[4-[[(7-chloro-2,3,4,5-tetrahydro-1H-3-benzazepin-6-yl)amino]methyl]phenyl]-1-cyclopropylethanone —— C22H26ClN3O
2-amino-2-[4-[[(7-chloro-2,3,4,5-tetrahydro-1H-3-benzazepin-6-yl)amino]methyl]phenyl]-1-cyclopropylethanone
—— 6-(2-Fluoro-5-nitrophenyl)benzo[d][2]benzazepine-5,7-dione —— C20H11FN2O4
6-(2-Fluoro-5-nitrophenyl)benzo[d][2]benzazepine-5,7-dione
—— 1-(5,7-Dihydrobenzo[b][1]benzazepin-11-yl)-3-(dimethylamino)propan-2-ol —— C19H24N2O
1-(5,7-Dihydrobenzo[b][1]benzazepin-11-yl)-3-(dimethylamino)propan-2-ol
—— 1-(5,7-dihydrobenzo[b][1]benzazepin-11-yl)-3-fluoro-N,N-dimethylpropan-2-amine —— C19H23FN2
1-(5,7-dihydrobenzo[b][1]benzazepin-11-yl)-3-fluoro-N,N-dimethylpropan-2-amine
—— N-[(1S,5R)-8-methyl-8-azoniabicyclo[3.2.1]octan-3-yl]-5,6-dihydrobenzo[b][1]benzazepine-11-carboxamide —— C23H28N3O+
N-[(1S,5R)-8-methyl-8-azoniabicyclo[3.2.1]octan-3-yl]-5,6-dihydrobenzo[b][1]benzazepine-11-carboxamide
—— 1-(Tert-butylamino)-3-(5,7-dihydrobenzo[b][1]benzazepin-11-yl)propan-2-ol —— C21H28N2O
1-(Tert-butylamino)-3-(5,7-dihydrobenzo[b][1]benzazepin-11-yl)propan-2-ol
—— 6-(2-Methoxy-4-nitrophenyl)benzo[d][2]benzazepine-5,7-dione —— C21H14N2O5
6-(2-Methoxy-4-nitrophenyl)benzo[d][2]benzazepine-5,7-dione
—— 3-(3-chloropropyl)-7,8-dimethoxy-5-propyl-1H-3-benzazepin-2-one —— C18H24ClNO3
3-(3-chloropropyl)-7,8-dimethoxy-5-propyl-1H-3-benzazepin-2-one
—— (5,5-dimethyl-4,5-dihydrospiro[2-benzazepine-3,1'-cyclohexan]-2(1H)-yl)(morpholin-4-yl)methanone —— C22H32N2O2
(5,5-dimethyl-4,5-dihydrospiro[2-benzazepine-3,1'-cyclohexan]-2(1H)-yl)(morpholin-4-yl)methanone
—— 3,5-dichloro-N-[3-(3-chloro-10,11-dihydrobenzo[d][1]benzazepin-5-yl)propyl]-2-hydroxybenzamide —— C24H21Cl3N2O2
3,5-dichloro-N-[3-(3-chloro-10,11-dihydrobenzo[d][1]benzazepin-5-yl)propyl]-2-hydroxybenzamide
—— 2-(Dicyclohexylamino)-1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)ethanone —— C28H36N2O
2-(Dicyclohexylamino)-1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)ethanone
—— Dicyclohexyl-[2-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-oxoethyl]azanium —— C28H37N2O+
Dicyclohexyl-[2-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-oxoethyl]azanium
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[4-(3-methoxyphenyl)piperazin-1-ium-1-yl]ethanone —— C27H30N3O2+
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[4-(3-methoxyphenyl)piperazin-1-ium-1-yl]ethanone
—— 1-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-2-[4-(3-methoxyphenyl)piperazin-1-yl]ethanone —— C27H29N3O2
1-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-2-[4-(3-methoxyphenyl)piperazin-1-yl]ethanone
—— 3-(5,7-dihydrobenzo[b][1]benzazepin-11-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpropan-1-amine —— C28H34N2O2
3-(5,7-dihydrobenzo[b][1]benzazepin-11-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpropan-1-amine
—— 4-[(3-carboxy-2-hydroxynaphthalen-1-yl)methyl]-3-hydroxynaphthalene-2-carboxylic acid;3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-N,N-dimethylpropan-1-amine;2-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-methylphenol —— C64H71N3O7
4-[(3-carboxy-2-hydroxynaphthalen-1-yl)methyl]-3-hydroxynaphthalene-2-carboxylic acid;3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-N,N-dimethylpropan-1-amine;2-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-methylphenol
—— (4-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)methanesulfonic acid 1404422-78-1 C34H38N4O6S
(4-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)methanesulfonic acid
—— [[4-[[4-[1-[4-(2,3-Dimethylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino] methanesulfonate —— C34H38N4O6S
[[4-[[4-[1-[4-(2,3-Dimethylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino] methanesulfonate
—— 3-[[4-[1-[4-(3-Chloro-2-methylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoic acid —— C32H32ClN3O4
3-[[4-[1-[4-(3-Chloro-2-methylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoic acid
—— 2-(4-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)ethanesulfonic acid 1404422-79-2 C35H40N4O6S
2-(4-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)ethanesulfonic acid
—— (3-((4-( 1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)methanesulfonic acid 1404422-70-3 C34H38N4O6S
(3-((4-( 1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)methanesulfonic acid
—— 2-(3-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)ethanesulfonic acid 1404422-71-4 C35H40N4O6S
2-(3-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)ethanesulfonic acid
—— 2-[[4-[[4-[(1aR,7bS)-3-[4-(2,3-dimethylphenoxy)butanoyl]-1,1a,2,7b-tetrahydrocyclopropa[c]quinolin-7-yl]pyrazol-1-yl]methyl]-3-chloro-5-fluorobenzoyl]amino]ethyl-trimethylazanium —— C38H44ClFN5O3+
2-[[4-[[4-[(1aR,7bS)-3-[4-(2,3-dimethylphenoxy)butanoyl]-1,1a,2,7b-tetrahydrocyclopropa[c]quinolin-7-yl]pyrazol-1-yl]methyl]-3-chloro-5-fluorobenzoyl]amino]ethyl-trimethylazanium
—— [[3-[[4-[1-[4-(2,3-Dimethylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino] methanesulfonate —— C34H38N4O6S
[[3-[[4-[1-[4-(2,3-Dimethylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino] methanesulfonate
—— 4-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzoic acid 1404420-62-7 C33H35N3O4
4-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzoic acid
—— 3-(4-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid 1404422-33-8 C36H40N4O5
3-(4-((4-(1-(4-(2,3-dimethylphenoxy)butanoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-6-yl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
—— 2-[[3-[[4-[1-[4-(3-Chloro-2-methylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino]ethanesulfonic acid —— C34H37ClN4O6S
2-[[3-[[4-[1-[4-(3-Chloro-2-methylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino]ethanesulfonic acid
—— [[3-[[4-[1-[4-(3-Chloro-2-methylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino]methanesulfonic acid —— C33H35ClN4O6S
[[3-[[4-[1-[4-(3-Chloro-2-methylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino]methanesulfonic acid
—— 2-[[3-[[4-[1-[4-(3-Chloro-2-methylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino]ethyl-trimethylazanium —— C37H45ClN5O3+
2-[[3-[[4-[1-[4-(3-Chloro-2-methylphenoxy)butanoyl]-2,3,4,5-tetrahydro-1-benzazepin-6-yl]pyrazol-1-yl]methyl]benzoyl]amino]ethyl-trimethylazanium
—— (1R,2R,3S,4S)-3-(3,3,5,5-tetramethyl-1,4-dihydro-2-benzazepine-2-carbonyl)bicyclo[2.2.1]hept-5-ene-2-carboxylate —— C23H28NO3-
(1R,2R,3S,4S)-3-(3,3,5,5-tetramethyl-1,4-dihydro-2-benzazepine-2-carbonyl)bicyclo[2.2.1]hept-5-ene-2-carboxylate
—— 2-(6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-N'-(2,2,3,3,3-pentafluoropropyl)propanediamide —— C20H16F5N3O3
2-(6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-N'-(2,2,3,3,3-pentafluoropropyl)propanediamide