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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— propan-2-ylsulfonyl 10-[3a-(methoxymethyl)-3,4,6,6a-tetrahydro-1H-furo[3,4-c]pyrrole-5-carbonyl]-19-cyclohexyl-5-hydroxy-18-methyl-12-azatetracyclo[10.7.0.02,7.08,10]nonadeca-1(19),2(7),3,5,14,16-hexaene-15-carboxylate —— C38H50N2O8S
propan-2-ylsulfonyl 10-[3a-(methoxymethyl)-3,4,6,6a-tetrahydro-1H-furo[3,4-c]pyrrole-5-carbonyl]-19-cyclohexyl-5-hydroxy-18-methyl-12-azatetracyclo[10.7.0.02,7.08,10]nonadeca-1(19),2(7),3,5,14,16-hexaene-15-carboxylate
—— (2S)-2-[[(2R)-2-hydroxybutyl]amino]-N-(7-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-1-yl)propanamide —— C22H27N3O3
(2S)-2-[[(2R)-2-hydroxybutyl]amino]-N-(7-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-1-yl)propanamide
—— 2-(5-chlorothiophen-2-yl)-N-[5-oxo-1-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)-2H-pyrrol-4-yl]ethanesulfonamide —— C20H22ClN3O3S2
2-(5-chlorothiophen-2-yl)-N-[5-oxo-1-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)-2H-pyrrol-4-yl]ethanesulfonamide
—— Ethyl 3-carbamoylimino-2-cyano-3-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)propanoate —— C17H20N4O3
Ethyl 3-carbamoylimino-2-cyano-3-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)propanoate
—— (3S,5S)-N-[3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-hydroxypropyl]-N-methyl-5-[(4-methylphenyl)sulfonylamino]piperidine-3-carboxamide —— C31H38N4O4S
(3S,5S)-N-[3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-hydroxypropyl]-N-methyl-5-[(4-methylphenyl)sulfonylamino]piperidine-3-carboxamide
—— 1,4-dimethyl-3,4-dihydro-2H-1-benzazepin-5-one;ethane —— C14H21NO
1,4-dimethyl-3,4-dihydro-2H-1-benzazepin-5-one;ethane
—— Ethane;8-methyl-10-azatetracyclo[8.7.1.02,7.014,18]octadeca-1(17),2,4,6,14(18),15-hexaen-9-one —— C22H29NO
Ethane;8-methyl-10-azatetracyclo[8.7.1.02,7.014,18]octadeca-1(17),2,4,6,14(18),15-hexaen-9-one
—— 9-Chloro-2-[[2-methyl-6-[4-(methylamino)piperidin-1-yl]pyridin-3-yl]amino]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione —— C24H26ClN7S
9-Chloro-2-[[2-methyl-6-[4-(methylamino)piperidin-1-yl]pyridin-3-yl]amino]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione
—— 4-methyl-8-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-7,8,9,10-tetrahydro-6H-[1,4]oxazino[2,3-h][1]benzazepin-3-one —— C29H32N6O2S
4-methyl-8-[3-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-7,8,9,10-tetrahydro-6H-[1,4]oxazino[2,3-h][1]benzazepin-3-one
—— N-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)methyl]-6-(2-methoxyethoxy)pyridine-3-carboxamide —— C24H31N3O3
N-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)methyl]-6-(2-methoxyethoxy)pyridine-3-carboxamide
—— 8-[(2-Fluorophenyl)methoxy]-1,2,3,3a,4,5-hexahydropyrrolo[3,4-d][2]benzazepine —— C19H19FN2O
8-[(2-Fluorophenyl)methoxy]-1,2,3,3a,4,5-hexahydropyrrolo[3,4-d][2]benzazepine
—— ethane;2,3,4,5-tetrahydro-1H-1-benzazepine —— C12H19N
ethane;2,3,4,5-tetrahydro-1H-1-benzazepine
—— 7-(2-methylprop-2-enyl)-2,3,4,5-tetrahydro-1H-1-benzazepin-3-ol —— C14H19NO
7-(2-methylprop-2-enyl)-2,3,4,5-tetrahydro-1H-1-benzazepin-3-ol
—— Ethane;3-methyl-1,2,4,5-tetrahydro-3-benzazepine —— C13H21N
Ethane;3-methyl-1,2,4,5-tetrahydro-3-benzazepine
—— 7-(2-bromophenyl)-9-chloro-5H-pyrimido[5,4-d][2]benzazepine —— C18H11BrClN3
7-(2-bromophenyl)-9-chloro-5H-pyrimido[5,4-d][2]benzazepine
—— [1-[[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-[(2-chlorophenyl)methyl]carbamate —— C26H24ClN3O4
[1-[[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-[(2-chlorophenyl)methyl]carbamate
—— 1-(Cyclopropylmethyl)-7-methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepin-5-amine —— C16H21F3N2
1-(Cyclopropylmethyl)-7-methyl-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepin-5-amine
—— 13-cyclohexyl-3-methoxy-7H-indolo[2,1-a][2]benzazepine-6-carboxylic acid —— C25H25NO3
13-cyclohexyl-3-methoxy-7H-indolo[2,1-a][2]benzazepine-6-carboxylic acid
—— (2S)-2-hydroxy-2-methyl-N-[6-oxo-5-(2-phenylmethoxyethyl)-7H-benzo[d][1]benzazepin-7-yl]-N'-(3,3,4,4,4-pentafluorobutyl)propanediamide —— C31H30F5N3O5
(2S)-2-hydroxy-2-methyl-N-[6-oxo-5-(2-phenylmethoxyethyl)-7H-benzo[d][1]benzazepin-7-yl]-N'-(3,3,4,4,4-pentafluorobutyl)propanediamide
—— (6aS,13bR)-11-chloro-7-methyl-5,6,6a,8,9,13b-hexahydronaphtho[1,2-a][3]benzazepin-12-ol;N-methylacetamide —— C22H27ClN2O2
(6aS,13bR)-11-chloro-7-methyl-5,6,6a,8,9,13b-hexahydronaphtho[1,2-a][3]benzazepin-12-ol;N-methylacetamide
—— 9-Chloro-10-[3-(methylamino)propyl]-2-[(2-methylpyridin-3-yl)amino]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione —— C22H23ClN6S
9-Chloro-10-[3-(methylamino)propyl]-2-[(2-methylpyridin-3-yl)amino]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione
—— 8,8-Diethyl-5-(trifluoromethyl)-11-azoniatetracyclo[9.8.0.02,7.012,17]nonadeca-1(11),2(7),3,5,12,14,16,18-octaene —— C23H23F3N+
8,8-Diethyl-5-(trifluoromethyl)-11-azoniatetracyclo[9.8.0.02,7.012,17]nonadeca-1(11),2(7),3,5,12,14,16,18-octaene
—— 3-[1-(3-prop-2-enylideneoxolan-2-ylidene)propan-2-yl]-2,3,4,5-tetrahydro-1H-1-benzazepine —— C20H25NO
3-[1-(3-prop-2-enylideneoxolan-2-ylidene)propan-2-yl]-2,3,4,5-tetrahydro-1H-1-benzazepine
—— 9-fluoro-5a,9a-dihydro-1H-3-benzazepine-5-carboxylic acid —— C11H10FNO2
9-fluoro-5a,9a-dihydro-1H-3-benzazepine-5-carboxylic acid
—— [1-[[(7R)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-(2,2,3,3,3-pentafluoropropyl)carbamate —— C22H20F5N3O4
[1-[[(7R)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]amino]-1-oxopropan-2-yl] N-(2,2,3,3,3-pentafluoropropyl)carbamate
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[(7-methyl-10-thia-3,4,6,8-tetrazatetracyclo[7.7.0.02,6.011,16]hexadeca-1(9),2,4,7,11(16)-pentaen-5-yl)sulfanyl]ethanone —— C28H25N5OS2
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[(7-methyl-10-thia-3,4,6,8-tetrazatetracyclo[7.7.0.02,6.011,16]hexadeca-1(9),2,4,7,11(16)-pentaen-5-yl)sulfanyl]ethanone
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(2-ethyl-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylethanone —— C26H25N3OS2
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(2-ethyl-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylethanone
—— [(1R,3S,12R,16R)-9-bromo-8-methoxy-16-methyl-14-phenylmethoxyimino-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17)-trien-3-yl]methanol —— C25H29BrN2O4
[(1R,3S,12R,16R)-9-bromo-8-methoxy-16-methyl-14-phenylmethoxyimino-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17)-trien-3-yl]methanol
—— 1-Ethyl-1,2-dimethyl-3,4-dihydro-2-benzazepin-5-one —— C14H19NO
1-Ethyl-1,2-dimethyl-3,4-dihydro-2-benzazepin-5-one
—— 5-(5,8,14-Triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2,4,6,8,10-pentaen-13-yl)pentane-2,3-diol —— C18H23N3O2
5-(5,8,14-Triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2,4,6,8,10-pentaen-13-yl)pentane-2,3-diol
—— 3-[10-cyclohexyl-4-[11-(2,2-difluoropropyl)-7,11-diazatetracyclo[6.4.0.01,5.05,9]dodecane-7-carbonyl]-9-ethylidene-15-methoxy-6-azatetracyclo[10.4.0.02,4.06,11]hexadeca-1(12),10,13,15-tetraen-8-ylidene]-N-(dimethylsulfamoyl)-2-methylpropanamide —— C44H59F2N5O5S
3-[10-cyclohexyl-4-[11-(2,2-difluoropropyl)-7,11-diazatetracyclo[6.4.0.01,5.05,9]dodecane-7-carbonyl]-9-ethylidene-15-methoxy-6-azatetracyclo[10.4.0.02,4.06,11]hexadeca-1(12),10,13,15-tetraen-8-ylidene]-N-(dimethylsulfamoyl)-2-methylpropanamide
—— 9-chloro-7-(2-fluorophenyl)-N-[2-(methylaminomethyl)benzimidazol-1-yl]-5H-pyrimido[5,4-d][2]benzazepin-2-amine —— C27H21ClFN7
9-chloro-7-(2-fluorophenyl)-N-[2-(methylaminomethyl)benzimidazol-1-yl]-5H-pyrimido[5,4-d][2]benzazepin-2-amine
—— 2,8-dimethyl-4,5-dihydro-3H-imidazo[4,5-d][1]benzazepin-6-amine —— C13H16N4
2,8-dimethyl-4,5-dihydro-3H-imidazo[4,5-d][1]benzazepin-6-amine
—— ethane;4-methyl-3-(methylamino)-1-phenyl-4,5-dihydro-3H-1-benzazepin-2-one —— C20H26N2O
ethane;4-methyl-3-(methylamino)-1-phenyl-4,5-dihydro-3H-1-benzazepin-2-one
—— benzyl N-[9-(3,3-dimethylbutyl)-8-oxo-3,6,7,10-tetrahydropyrazolo[3,4-i][2]benzazepin-7-yl]carbamate —— C25H30N4O3
benzyl N-[9-(3,3-dimethylbutyl)-8-oxo-3,6,7,10-tetrahydropyrazolo[3,4-i][2]benzazepin-7-yl]carbamate
—— (7-Bromo-8-methoxy-1,2,4,5-tetrahydro-3-benzazepin-3-yl)methanol —— C12H16BrNO2
(7-Bromo-8-methoxy-1,2,4,5-tetrahydro-3-benzazepin-3-yl)methanol
—— Methyl 8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepine-1-carboxylate —— C13H14F3NO2
Methyl 8-(trifluoromethyl)-2,3,4,5-tetrahydro-1-benzazepine-1-carboxylate
—— 2-[1-(2-hydroxyethyl)-2-oxo-4,5-dihydro-3H-1-benzazepin-5-yl]-3,3-dimethylbutanoic acid —— C18H25NO4
2-[1-(2-hydroxyethyl)-2-oxo-4,5-dihydro-3H-1-benzazepin-5-yl]-3,3-dimethylbutanoic acid
—— 3-(10-Cyclohexyl-15-methoxy-5-methoxycarbonyl-9-propylidene-7-azatetracyclo[10.4.0.02,5.07,11]hexadeca-1(12),10,13,15-tetraen-8-ylidene)propanoic acid —— C30H37NO5
3-(10-Cyclohexyl-15-methoxy-5-methoxycarbonyl-9-propylidene-7-azatetracyclo[10.4.0.02,5.07,11]hexadeca-1(12),10,13,15-tetraen-8-ylidene)propanoic acid
—— 5,7-dimethyl-7H-benzo[d][1]benzazepin-6-one;ethane —— C22H33NO
5,7-dimethyl-7H-benzo[d][1]benzazepin-6-one;ethane
—— 2,6-Dimethyl-4-[4-(5,6,8,9-tetrahydrobenzo[b][1]benzazepin-11-yl)butyl]morpholine —— C24H34N2O
2,6-Dimethyl-4-[4-(5,6,8,9-tetrahydrobenzo[b][1]benzazepin-11-yl)butyl]morpholine
—— 1-[2-[3-(2,3-Dihydroindol-1-yl)-3-oxopropyl]-9-fluoro-1,3,4,5-tetrahydro-2-benzazepin-7-yl]-4-hydroxybutan-1-one —— C25H29FN2O3
1-[2-[3-(2,3-Dihydroindol-1-yl)-3-oxopropyl]-9-fluoro-1,3,4,5-tetrahydro-2-benzazepin-7-yl]-4-hydroxybutan-1-one
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[(2-propan-2-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)sulfanyl]ethanone —— C29H29N3OS2
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[(2-propan-2-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)sulfanyl]ethanone
—— 2-[(2-Cyclopropyl-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)sulfanyl]-1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)ethanone —— C30H29N3OS2
2-[(2-Cyclopropyl-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)sulfanyl]-1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)ethanone
—— 1-[(4S)-7-chloro-4-methyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C13H13ClF3NO
1-[(4S)-7-chloro-4-methyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— 3-[4-(Benzylamino)pyrimidin-2-yl]-1,2,4,5-tetrahydro-3-benzazepine-7-carboxamide —— C22H23N5O
3-[4-(Benzylamino)pyrimidin-2-yl]-1,2,4,5-tetrahydro-3-benzazepine-7-carboxamide
—— 2-[[5-[(2-Anilino-1,3-thiazol-4-yl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]-1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)ethanone —— C28H23N5O2S2
2-[[5-[(2-Anilino-1,3-thiazol-4-yl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]-1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)ethanone
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(5,6-dimethyl-2-propan-2-ylthieno[2,3-d]pyrimidin-4-yl)sulfanylethanone —— C27H27N3OS2
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(5,6-dimethyl-2-propan-2-ylthieno[2,3-d]pyrimidin-4-yl)sulfanylethanone
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(2,5,6-trimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylethanone —— C25H23N3OS2
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-(2,5,6-trimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylethanone
—— 1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[[5-[[2-(4-ethoxyanilino)-1,3-thiazol-4-yl]methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethanone —— C30H27N5O3S2
1-(5,6-Dihydrobenzo[b][1]benzazepin-11-yl)-2-[[5-[[2-(4-ethoxyanilino)-1,3-thiazol-4-yl]methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethanone