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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(5-fluoropyridin-2-yl)piperidin-4-yl]methanone —— C21H23ClFN3O
(7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(5-fluoropyridin-2-yl)piperidin-4-yl]methanone
—— (7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(6-fluoroquinazolin-4-yl)piperidin-4-yl]methanone —— C24H24ClFN4O
(7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(6-fluoroquinazolin-4-yl)piperidin-4-yl]methanone
—— [1-(5-Chloro-3-fluoropyridin-2-yl)piperidin-4-yl]-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone —— C21H22Cl2FN3O
[1-(5-Chloro-3-fluoropyridin-2-yl)piperidin-4-yl]-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone
—— (7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(5-methylpyrimidin-2-yl)piperidin-4-yl]methanone —— C21H25ClN4O
(7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(5-methylpyrimidin-2-yl)piperidin-4-yl]methanone
—— 7-chloro-1-[1-(4,6-dimethylpyrimidin-2-yl)piperidine-4-carbonyl]-3,4-dihydro-2H-1-benzazepin-5-one —— C22H25ClN4O2
7-chloro-1-[1-(4,6-dimethylpyrimidin-2-yl)piperidine-4-carbonyl]-3,4-dihydro-2H-1-benzazepin-5-one
—— (7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-spiro[1H-2-benzofuran-3,4'-piperidine]-1'-ylmethanone —— C23H25ClN2O2
(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-spiro[1H-2-benzofuran-3,4'-piperidine]-1'-ylmethanone
—— (7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(5-fluoro-4-methylpyrimidin-2-yl)piperidin-4-yl]methanone —— C21H24ClFN4O
(7-Chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[1-(5-fluoro-4-methylpyrimidin-2-yl)piperidin-4-yl]methanone
—— 1'-(7-chloro-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)spiro[1H-3,1-benzoxazine-4,4'-piperidine]-2-one —— C23H24ClN3O3
1'-(7-chloro-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)spiro[1H-3,1-benzoxazine-4,4'-piperidine]-2-one
—— [1-(7-Chloroquinazolin-4-yl)piperidin-4-yl]-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone —— C24H24Cl2N4O
[1-(7-Chloroquinazolin-4-yl)piperidin-4-yl]-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone
—— 10-(2-Bicyclo[2.2.2]octanylmethyl)-2,3,10-triazatricyclo[6.4.1.04,13]trideca-1(13),3,5,7-tetraen-9-one —— C19H23N3O
10-(2-Bicyclo[2.2.2]octanylmethyl)-2,3,10-triazatricyclo[6.4.1.04,13]trideca-1(13),3,5,7-tetraen-9-one
—— (8-Bromo-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)carbamic acid —— C11H11BrN2O3
(8-Bromo-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)carbamic acid
—— 5-benzyl-N-(5-methyl-1-oxido-4-oxo-1,2,3,5-tetrahydro-1-benzazepin-1-ium-3-yl)-1,2-oxazole-3-carboxamide —— C22H21N3O4
5-benzyl-N-(5-methyl-1-oxido-4-oxo-1,2,3,5-tetrahydro-1-benzazepin-1-ium-3-yl)-1,2-oxazole-3-carboxamide
—— 5-benzyl-N-(5-methyl-1-oxido-4-oxo-3,5-dihydro-2H-1-benzazepin-3-yl)-1,2-oxazole-3-carboxamide —— C22H20N3O4-
5-benzyl-N-(5-methyl-1-oxido-4-oxo-3,5-dihydro-2H-1-benzazepin-3-yl)-1,2-oxazole-3-carboxamide
—— 5-benzyl-N-(1-hydroxy-5-methyl-4-oxo-3,5-dihydro-2H-1-benzazepin-3-yl)-1,2-oxazole-3-carboxamide —— C22H21N3O4
5-benzyl-N-(1-hydroxy-5-methyl-4-oxo-3,5-dihydro-2H-1-benzazepin-3-yl)-1,2-oxazole-3-carboxamide
—— 9-methyl-4,5-dihydro-1H-1-benzazepine —— C11H13N
9-methyl-4,5-dihydro-1H-1-benzazepine
—— 3-[7-[[5-chloro-4-[2-(prop-2-enoylamino)anilino]pyrimidin-2-yl]amino]-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-1-yl]propylcarbamic acid —— C28H30ClN7O5
3-[7-[[5-chloro-4-[2-(prop-2-enoylamino)anilino]pyrimidin-2-yl]amino]-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-1-yl]propylcarbamic acid
—— N-(2-((5-chloro-2-((6-methoxy-1-(2-morpholinoethyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide 1622000-56-9 C30H34ClN7O4
N-(2-((5-chloro-2-((6-methoxy-1-(2-morpholinoethyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide
—— 5,8,11a-trimethyl-6-oxo-3-propan-2-yl-7a,9,10,11-tetrahydro-7H-benzo[d][1]benzazepine-8-carbaldehyde —— C21H29NO2
5,8,11a-trimethyl-6-oxo-3-propan-2-yl-7a,9,10,11-tetrahydro-7H-benzo[d][1]benzazepine-8-carbaldehyde
—— 1-[(4S)-1-methyl-6-morpholin-4-yl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one —— C19H21N3O3
1-[(4S)-1-methyl-6-morpholin-4-yl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one
—— 1-[(4S)-8-chloro-1-methyl-6-(4-methylphenyl)-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one —— C22H19ClN2O2
1-[(4S)-8-chloro-1-methyl-6-(4-methylphenyl)-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one
—— 1-[(4S)-7-chloro-6-(4-chlorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one —— C21H16Cl2N2O2
1-[(4S)-7-chloro-6-(4-chlorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one
—— 1-[(4S)-7-chloro-1-methyl-6-pyridin-4-yl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one —— C20H16ClN3O2
1-[(4S)-7-chloro-1-methyl-6-pyridin-4-yl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one
—— 1-[(4S)-8-(6-aminopyridin-3-yl)-6-(4-fluorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one —— C26H21FN4O2
1-[(4S)-8-(6-aminopyridin-3-yl)-6-(4-fluorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one
—— 1-[(4S)-6-(4-chloro-3-methylphenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one —— C22H19ClN2O2
1-[(4S)-6-(4-chloro-3-methylphenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]propan-2-one
—— 11-[4-[2-Fluoro-4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]piperazin-1-yl]-5,11-dimethylbenzo[c][1]benzazepin-6-one —— C29H28FN5O2
11-[4-[2-Fluoro-4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]piperazin-1-yl]-5,11-dimethylbenzo[c][1]benzazepin-6-one
—— 11-[1-[2-Chloro-4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]piperidin-4-yl]-11-hydroxy-5-methylbenzo[c][1]benzazepin-6-one —— C29H27ClN4O3
11-[1-[2-Chloro-4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]piperidin-4-yl]-11-hydroxy-5-methylbenzo[c][1]benzazepin-6-one
—— 2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]-5-(1H-pyrazol-5-yl)benzonitrile —— C28H24N6O
2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]-5-(1H-pyrazol-5-yl)benzonitrile
—— N-[3-chloro-4-[(2R)-2-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)acetamide —— C32H32ClN5O3
N-[3-chloro-4-[(2R)-2-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)acetamide
—— N-[3-chloro-4-[(2R)-2-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]oxolane-3-carboxamide —— C30H31ClN4O3
N-[3-chloro-4-[(2R)-2-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]oxolane-3-carboxamide
—— N-[3-cyano-4-[4-(11-hydroxy-6-oxo-5H-benzo[c][1]benzazepin-11-yl)piperidin-1-yl]phenyl]-2,2-dimethylpropanamide —— C31H32N4O3
N-[3-cyano-4-[4-(11-hydroxy-6-oxo-5H-benzo[c][1]benzazepin-11-yl)piperidin-1-yl]phenyl]-2,2-dimethylpropanamide
—— N-[3-cyano-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)-N-methylacetamide —— C33H32N6O3
N-[3-cyano-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)-N-methylacetamide
—— N-tert-butyl-3-cyano-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]benzamide 1620770-99-1 C30H31N5O2
N-tert-butyl-3-cyano-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]benzamide
—— N,N-diethyl-4-[[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazine-1-carbothioyl]amino]benzamide —— C30H33N5O2S
N,N-diethyl-4-[[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazine-1-carbothioyl]amino]benzamide
—— 2-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]-5-(6-methylpyridin-2-yl)benzonitrile —— C32H29N5O
2-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]-5-(6-methylpyridin-2-yl)benzonitrile
—— N-[3-cyano-4-[(3R)-3-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-ethylbutanamide —— C32H35N5O2
N-[3-cyano-4-[(3R)-3-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-ethylbutanamide
—— N-[3-cyano-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-phenylpyrazole-3-carboxamide —— C35H29N7O2
N-[3-cyano-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-phenylpyrazole-3-carboxamide
—— N-[3-cyano-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-3-phenyl-1,2-oxazole-4-carboxamide —— C35H28N6O3
N-[3-cyano-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-3-phenyl-1,2-oxazole-4-carboxamide
—— N-[3-cyano-4-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2,2-dimethylpropanamide —— C31H33N5O2
N-[3-cyano-4-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2,2-dimethylpropanamide
—— 5-Methyl-2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]benzonitrile —— C26H24N4O
5-Methyl-2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]benzonitrile
—— N-[3-cyano-4-[4-(11-hydroxy-5-methyl-6-oxobenzo[c][1]benzazepin-11-yl)piperidin-1-yl]phenyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)acetamide —— C34H33N5O4
N-[3-cyano-4-[4-(11-hydroxy-5-methyl-6-oxobenzo[c][1]benzazepin-11-yl)piperidin-1-yl]phenyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)acetamide
—— 2-[4-(11-fluoro-6-oxo-5H-benzo[c][1]benzazepin-11-yl)piperidin-1-yl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)benzonitrile —— C29H24FN5O2
2-[4-(11-fluoro-6-oxo-5H-benzo[c][1]benzazepin-11-yl)piperidin-1-yl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)benzonitrile
—— N-[3-fluoro-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2,2-dimethylbutanamide —— C30H33FN4O2
N-[3-fluoro-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2,2-dimethylbutanamide
—— 5-(3-Methylimidazol-4-yl)-2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]benzonitrile —— C29H26N6O
5-(3-Methylimidazol-4-yl)-2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]benzonitrile
—— N-[3-chloro-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-ethylbutanamide —— C30H33ClN4O2
N-[3-chloro-4-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-ethylbutanamide
—— 11-[4-[2-fluoro-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]piperazin-1-yl]-5-methyl-11H-benzo[c][1]benzazepin-6-one —— C28H26FN5O2
11-[4-[2-fluoro-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]piperazin-1-yl]-5-methyl-11H-benzo[c][1]benzazepin-6-one
—— N-[5-chloro-6-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]pyridin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide —— C30H29ClN6O3
N-[5-chloro-6-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]pyridin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
—— 2-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[6-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]pyridin-3-yl]acetamide —— C31H32N6O3
2-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[6-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]pyridin-3-yl]acetamide
—— 5-(2,3-dimethylimidazol-4-yl)-2-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]benzonitrile —— C31H30N6O
5-(2,3-dimethylimidazol-4-yl)-2-[4-(5-methyl-6-oxo-11H-benzo[c][1]benzazepin-11-yl)piperazin-1-yl]benzonitrile
—— N-[3-cyano-4-[(2S)-2-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-ethylbutanamide —— C32H35N5O2
N-[3-cyano-4-[(2S)-2-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2-ethylbutanamide
—— N-[3-chloro-4-[(2R)-2-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2,2-dimethylpropanamide —— C30H33ClN4O2
N-[3-chloro-4-[(2R)-2-methyl-4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]phenyl]-2,2-dimethylpropanamide