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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R,4R,5S)-3-methyl-2,6-dioxo-N-[[(2S)-oxolan-2-yl]methyl]-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C18H20N2O4
(3R,4R,5S)-3-methyl-2,6-dioxo-N-[[(2S)-oxolan-2-yl]methyl]-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-N-[[(3S)-oxan-3-yl]methyl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C19H22N2O4
(3R,4R,5S)-3-methyl-N-[[(3S)-oxan-3-yl]methyl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R)-1-[(3S,4R,5S)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carbonyl]piperidine-3-carboxamide —— C19H21N3O4
(3R)-1-[(3S,4R,5S)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carbonyl]piperidine-3-carboxamide
—— (3R,4R,5S)-3-methyl-2,6-dioxo-N-(2-pyrrolidin-1-ylethyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C19H23N3O3
(3R,4R,5S)-3-methyl-2,6-dioxo-N-(2-pyrrolidin-1-ylethyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-2,6-dioxo-N-(2-pyridin-4-ylethyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C20H19N3O3
(3R,4R,5S)-3-methyl-2,6-dioxo-N-(2-pyridin-4-ylethyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-N-[(3R)-1-methylpiperidin-3-yl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C19H23N3O3
(3R,4R,5S)-3-methyl-N-[(3R)-1-methylpiperidin-3-yl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-N-(1H-imidazol-2-ylmethyl)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C17H16N4O3
(3R,4R,5S)-N-(1H-imidazol-2-ylmethyl)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-2,6-dioxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C19H21N3O4
(3R,4R,5S)-3-methyl-2,6-dioxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-2,6-dioxo-N-[2-(pyridine-4-carbonylamino)ethyl]-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C21H20N4O4
(3R,4R,5S)-3-methyl-2,6-dioxo-N-[2-(pyridine-4-carbonylamino)ethyl]-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-N-[2-[[(2S)-oxan-2-yl]methoxy]ethyl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C21H26N2O5
(3R,4R,5S)-3-methyl-N-[2-[[(2S)-oxan-2-yl]methoxy]ethyl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-3-methyl-2,6-dioxo-N-[[(2R)-oxolan-2-yl]methyl]-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C18H20N2O4
(3R,4R,5S)-3-methyl-2,6-dioxo-N-[[(2R)-oxolan-2-yl]methyl]-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5S)-N-(2-imidazol-1-ylethyl)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C18H18N4O3
(3R,4R,5S)-N-(2-imidazol-1-ylethyl)-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3S,4R,5S)-3-methyl-4-(piperidine-1-carbonyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-2,6-dione —— C18H20N2O3
(3S,4R,5S)-3-methyl-4-(piperidine-1-carbonyl)-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-2,6-dione
—— (3R,4R,5S)-3-methyl-N-[(1-methylimidazol-2-yl)methyl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C18H18N4O3
(3R,4R,5S)-3-methyl-N-[(1-methylimidazol-2-yl)methyl]-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3aS,10aS)-10a-methyl-2-(thiophen-2-ylmethyl)-1,3,3a,4-tetrahydropyrrolo[3,4-c][2]benzazepine-5,10-dione —— C18H18N2O2S
(3aS,10aS)-10a-methyl-2-(thiophen-2-ylmethyl)-1,3,3a,4-tetrahydropyrrolo[3,4-c][2]benzazepine-5,10-dione
—— (3R,4R,5S)-N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C20H22N4O3
(3R,4R,5S)-N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3R,4R,5R)-N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide —— C20H22N4O3
(3R,4R,5R)-N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-3-methyl-2,6-dioxo-7-azatricyclo[6.4.0.03,5]dodeca-1(12),8,10-triene-4-carboxamide
—— (3S)-1'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H24N4O2
(3S)-1'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[2-(4-methylsulfonylphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H24N2O4S
(3R)-1'-[2-(4-methylsulfonylphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H24N4O2
(3R)-1'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H26N4O3
(3R)-1'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H26N4O3
(3S)-1'-[2-(3,5-dimethylpyrazol-1-yl)acetyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(2-methoxypyrimidin-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H22N4O2
(3S)-1'-[(2-methoxypyrimidin-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2-methoxypyrimidin-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C19H22N4O2
(3R)-1'-[(2-methoxypyrimidin-5-yl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(4-methoxy-3-methylphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O2
(3S)-1'-[(4-methoxy-3-methylphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(4-methoxy-3-methylphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O2
(3R)-1'-[(4-methoxy-3-methylphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[2-(2-methoxyphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H24N2O3
(3S)-1'-[2-(2-methoxyphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— 3-[[5-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C19H18N4O2S
3-[[5-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— (3R)-1'-[2-(2-methoxyphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H24N2O3
(3R)-1'-[2-(2-methoxyphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— 1-(3-{3-[(methoxycarbonyl)amino]-10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl}-3-oxopropyl)piperidinium —— C24H30N3O3+
1-(3-{3-[(methoxycarbonyl)amino]-10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl}-3-oxopropyl)piperidinium
—— (3S)-1'-[(2,3-dimethoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O3
(3S)-1'-[(2,3-dimethoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(2,6-dimethoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O3
(3S)-1'-[(2,6-dimethoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2,3-dimethoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O3
(3R)-1'-[(2,3-dimethoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(2,6-dimethoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O3
(3R)-1'-[(2,6-dimethoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-8-methoxy-1'-[(3-methoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H26N2O3
(3S)-8-methoxy-1'-[(3-methoxyphenyl)methyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[2-(3-methoxyphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H24N2O3
(3S)-1'-[2-(3-methoxyphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[2-(3-methoxyphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C22H24N2O3
(3R)-1'-[2-(3-methoxyphenyl)acetyl]spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C14H18N2O2
(3S)-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-8-methoxy-1'-(pyridine-3-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21N3O3
(3R)-8-methoxy-1'-(pyridine-3-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-8-methoxy-1'-(pyridine-2-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21N3O3
(3S)-8-methoxy-1'-(pyridine-2-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-8-methoxy-1'-(pyridin-2-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O2
(3S)-8-methoxy-1'-(pyridin-2-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(4-fluorophenyl)methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H23FN2O2
(3S)-1'-[(4-fluorophenyl)methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(3,4-difluorophenyl)methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H22F2N2O2
(3R)-1'-[(3,4-difluorophenyl)methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-8-methoxy-1'-(pyridin-2-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O2
(3R)-8-methoxy-1'-(pyridin-2-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-1'-[(4-fluorophenyl)methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H23FN2O2
(3R)-1'-[(4-fluorophenyl)methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-8-methoxy-1'-(pyridin-3-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O2
(3R)-8-methoxy-1'-(pyridin-3-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-8-methoxy-1'-(pyridin-4-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H23N3O2
(3R)-8-methoxy-1'-(pyridin-4-ylmethyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-8-methoxy-1'-(pyridine-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21N3O3
(3S)-8-methoxy-1'-(pyridine-4-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3S)-1'-[(3,4-difluorophenyl)methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C21H22F2N2O2
(3S)-1'-[(3,4-difluorophenyl)methyl]-8-methoxyspiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one
—— (3R)-8-methoxy-1'-(pyridine-2-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one —— C20H21N3O3
(3R)-8-methoxy-1'-(pyridine-2-carbonyl)spiro[4,5-dihydro-2H-2-benzazepine-3,3'-pyrrolidine]-1-one