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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-(3,4-Dimethylphenyl)-8,14-diethyl-8-methyl-14-azoniatricyclo[8.3.1.02,7]tetradeca-1(13),2(7),3,5,10(14),11-hexaene —— C26H30N+
4-(3,4-Dimethylphenyl)-8,14-diethyl-8-methyl-14-azoniatricyclo[8.3.1.02,7]tetradeca-1(13),2(7),3,5,10(14),11-hexaene
—— 7-[7-(1,1-difluoropropyl)-4,5-dihydro-3H-1-benzazepin-2-yl]-2-[(4-fluorophenyl)methylamino]-4-(2-phenylethyl)-3,4,5a,6,8,9-hexahydro-2H-pyrido[4,3-b]azepin-5-one —— C37H41F3N4O
7-[7-(1,1-difluoropropyl)-4,5-dihydro-3H-1-benzazepin-2-yl]-2-[(4-fluorophenyl)methylamino]-4-(2-phenylethyl)-3,4,5a,6,8,9-hexahydro-2H-pyrido[4,3-b]azepin-5-one
—— 11-(7'-ethenyl-4,4'a-dimethylspiro[1,3,4,5-tetrahydroindene-2,9'-9aH-fluorene]-2'-yl)-5,6-dihydrobenzo[b][1]benzazepine —— C39H37N
11-(7'-ethenyl-4,4'a-dimethylspiro[1,3,4,5-tetrahydroindene-2,9'-9aH-fluorene]-2'-yl)-5,6-dihydrobenzo[b][1]benzazepine
—— 2-[2-[4-(Pyrazin-2-ylamino)butylcarbamoyl]-2-benzazepin-5-yl]acetic acid —— C21H23N5O3
2-[2-[4-(Pyrazin-2-ylamino)butylcarbamoyl]-2-benzazepin-5-yl]acetic acid
—— 2,2-dicyano-N-(2-methyl-1-benzofuran-5-yl)-N'-[2-oxo-1-(2-oxo-2-pyrrolidin-1-ylethyl)-4,5-dihydro-3H-1-benzazepin-3-yl]ethanimidamide —— C29H28N6O3
2,2-dicyano-N-(2-methyl-1-benzofuran-5-yl)-N'-[2-oxo-1-(2-oxo-2-pyrrolidin-1-ylethyl)-4,5-dihydro-3H-1-benzazepin-3-yl]ethanimidamide
—— 2-[4-chloro-N-[(8-chloro-3-methyl-4,5-dihydro-3H-1-benzazepin-2-yl)methyl]anilino]acetic acid —— C20H20Cl2N2O2
2-[4-chloro-N-[(8-chloro-3-methyl-4,5-dihydro-3H-1-benzazepin-2-yl)methyl]anilino]acetic acid
—— 1-(9-Butan-2-yl-2-cyclopropylpurin-6-yl)-2-(difluoromethyl)-4,5-dihydro-1-benzazepine —— C23H25F2N5
1-(9-Butan-2-yl-2-cyclopropylpurin-6-yl)-2-(difluoromethyl)-4,5-dihydro-1-benzazepine
—— [(1R,3S,12R,16R)-9-bromo-3-(hydroxymethyl)-8-methoxy-16-methyl-14-[2-(4-nitrophenyl)hydrazinyl]-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-4-yl]-phenylmethanone —— C31H31BrN4O6
[(1R,3S,12R,16R)-9-bromo-3-(hydroxymethyl)-8-methoxy-16-methyl-14-[2-(4-nitrophenyl)hydrazinyl]-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-4-yl]-phenylmethanone
—— 4-Ethyl-3-methyl-1,2,4,5-tetrahydro-3-benzazepine —— C13H19N
4-Ethyl-3-methyl-1,2,4,5-tetrahydro-3-benzazepine
—— 2-[[(1R,3S,12R,16R)-9-bromo-4-(ethylcarbamoyl)-3-(hydroxymethyl)-8-methoxy-16-methyl-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-14-yl]amino]acetic acid —— C23H30BrN3O6
2-[[(1R,3S,12R,16R)-9-bromo-4-(ethylcarbamoyl)-3-(hydroxymethyl)-8-methoxy-16-methyl-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-14-yl]amino]acetic acid
—— [3-(3-Pyrimidin-2-ylsulfanylpropyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]methanesulfonic acid —— C18H23N3O3S2
[3-(3-Pyrimidin-2-ylsulfanylpropyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]methanesulfonic acid
—— (2S)-2-[[(2R)-2-hydroxyoctyl]amino]-N-(7-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-1-yl)propanamide —— C26H35N3O3
(2S)-2-[[(2R)-2-hydroxyoctyl]amino]-N-(7-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-1-yl)propanamide
—— 9-Ethyl-1,6,7,8-tetramethyl-2,3,4,5-tetrahydro-1-benzazepine —— C16H25N
9-Ethyl-1,6,7,8-tetramethyl-2,3,4,5-tetrahydro-1-benzazepine
—— 2-[3-(4-fluorophenyl)propyl]-N-[(3-methyl-2,1-benzoxazol-5-yl)methyl]-3H-1-benzazepin-6-amine —— C28H26FN3O
2-[3-(4-fluorophenyl)propyl]-N-[(3-methyl-2,1-benzoxazol-5-yl)methyl]-3H-1-benzazepin-6-amine
—— [(1S)-2-(16-fluoro-3,5,11,13-tetrazatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),2(6),4,7(12),8,10,15,17-octaen-4-yl)cyclopropyl]methyl 2,2,2-trifluoroacetate —— C20H14F4N4O2
[(1S)-2-(16-fluoro-3,5,11,13-tetrazatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),2(6),4,7(12),8,10,15,17-octaen-4-yl)cyclopropyl]methyl 2,2,2-trifluoroacetate
—— 1,10,10,11,14,15,19,20-Octamethyl-16,17-bis(prop-1-enyl)-20-azatetracyclo[9.8.1.02,9.013,18]icosa-2(9),3,5,7,13(18),14,16-heptaene —— C33H43N
1,10,10,11,14,15,19,20-Octamethyl-16,17-bis(prop-1-enyl)-20-azatetracyclo[9.8.1.02,9.013,18]icosa-2(9),3,5,7,13(18),14,16-heptaene
—— 10-bromo-7-[4-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]butyl]-2-(trifluoromethyl)-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine —— C29H28BrF3N6OS
10-bromo-7-[4-[[4-methyl-5-(2-methylquinolin-5-yl)-1,2,4-triazol-3-yl]sulfanyl]butyl]-2-(trifluoromethyl)-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine
—— (2,5-Dihydroxypyrrol-1-yl) 4-[2-[3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)propyl-methylamino]ethylcarbamoyl]benzoate —— C32H34N4O5
(2,5-Dihydroxypyrrol-1-yl) 4-[2-[3-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)propyl-methylamino]ethylcarbamoyl]benzoate
—— ethane;1-ethyl-3-(methylamino)-4,5-dihydro-3H-1-benzazepin-2-one —— C15H24N2O
ethane;1-ethyl-3-(methylamino)-4,5-dihydro-3H-1-benzazepin-2-one
—— 9-bromo-N-(2-methylpyridin-3-yl)-7,12-dihydroindolo[3,2-d][1]benzazepin-6-amine —— C22H17BrN4
9-bromo-N-(2-methylpyridin-3-yl)-7,12-dihydroindolo[3,2-d][1]benzazepin-6-amine
—— 5-[3-[4-[(2S)-2-aminopropanoyl]-3-methyl-1,2,4,5-tetrahydro-3-benzazepin-8-yl]-1,2,4-oxadiazol-5-yl]-2-propan-2-yloxybenzonitrile —— C26H29N5O3
5-[3-[4-[(2S)-2-aminopropanoyl]-3-methyl-1,2,4,5-tetrahydro-3-benzazepin-8-yl]-1,2,4-oxadiazol-5-yl]-2-propan-2-yloxybenzonitrile
—— 1,4-dichloro-N,N-dimethyl-3H-2-benzazepin-6-amine —— C12H12Cl2N2
1,4-dichloro-N,N-dimethyl-3H-2-benzazepin-6-amine
—— 3-[2-(4-Chlorophenoxy)ethyl]-1,2,4,5-tetrahydro-3-benzazepine-7-carboxamide —— C19H21ClN2O2
3-[2-(4-Chlorophenoxy)ethyl]-1,2,4,5-tetrahydro-3-benzazepine-7-carboxamide
—— Methyl 5-[2-[2-(cyclohexylmethyl)-5-(dimethylsulfamoylcarbamoyl)phenyl]-7-methoxy-1,3-dihydro-2-benzazepin-4-yl]-1-propan-2-yltriazole-4-carboxylate —— C34H44N6O6S
Methyl 5-[2-[2-(cyclohexylmethyl)-5-(dimethylsulfamoylcarbamoyl)phenyl]-7-methoxy-1,3-dihydro-2-benzazepin-4-yl]-1-propan-2-yltriazole-4-carboxylate
—— [(2,2,6,6-Tetramethyl-1,3-dihydropyridin-4-yl)amino] 5,6-dihydrobenzo[b][1]benzazepine-11-carboxylate —— C24H29N3O2
[(2,2,6,6-Tetramethyl-1,3-dihydropyridin-4-yl)amino] 5,6-dihydrobenzo[b][1]benzazepine-11-carboxylate
—— Pyrrolo[2,3-c][1]benzazepine —— C12H8N2
Pyrrolo[2,3-c][1]benzazepine
—— 19-cyclohexyl-15-N-dimethylsulfinamoyl-5-ethyl-18-methyl-10-N-[(3,5,8,8-tetramethyl-2-bicyclo[3.2.1]octanyl)methyl]-12-azapentacyclo[10.7.0.02,7.08,10.013,18]nonadeca-1(19),2(7),3,5,13,15-hexaene-10,15-dicarboxamide —— C44H62N4O3S
19-cyclohexyl-15-N-dimethylsulfinamoyl-5-ethyl-18-methyl-10-N-[(3,5,8,8-tetramethyl-2-bicyclo[3.2.1]octanyl)methyl]-12-azapentacyclo[10.7.0.02,7.08,10.013,18]nonadeca-1(19),2(7),3,5,13,15-hexaene-10,15-dicarboxamide
—— N'-[(1R,3S,12R,16R)-9-bromo-3-(hydroxymethyl)-8-methoxy-16-methyl-4-(thiophene-2-carbonyl)-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-14-yl]-4-methoxybenzenesulfonohydrazide —— C30H32BrN3O7S2
N'-[(1R,3S,12R,16R)-9-bromo-3-(hydroxymethyl)-8-methoxy-16-methyl-4-(thiophene-2-carbonyl)-11-oxa-4-azatetracyclo[8.6.1.01,12.06,17]heptadeca-6,8,10(17),13-tetraen-14-yl]-4-methoxybenzenesulfonohydrazide
—— (2S)-2-methoxy-N-(6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-N'-(2,2,3,3,3-pentafluoropropyl)propanediamide —— C21H18F5N3O4
(2S)-2-methoxy-N-(6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-N'-(2,2,3,3,3-pentafluoropropyl)propanediamide
—— tert-butyl N-(1-sulfanyl-2,3-dihydro-1-benzazepin-4-yl)carbamate —— C15H20N2O2S
tert-butyl N-(1-sulfanyl-2,3-dihydro-1-benzazepin-4-yl)carbamate
—— 2H-2-benzazepin-1-yl 2,2,2-trifluoroacetate —— C12H8F3NO2
2H-2-benzazepin-1-yl 2,2,2-trifluoroacetate
—— 4-[(9-chloro-6-hydroxy-7H-pyrimido[5,4-i][1]benzazepin-2-yl)amino]-N-[(5-pyridin-2-ylthiophen-2-yl)methyl]benzamide —— C29H21ClN6O2S
4-[(9-chloro-6-hydroxy-7H-pyrimido[5,4-i][1]benzazepin-2-yl)amino]-N-[(5-pyridin-2-ylthiophen-2-yl)methyl]benzamide
—— 3-[7-[5-(3-Cyano-4-propan-2-yloxyphenyl)-1,2,4-oxadiazol-3-yl]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2-methylpropanoic acid —— C26H28N4O4
3-[7-[5-(3-Cyano-4-propan-2-yloxyphenyl)-1,2,4-oxadiazol-3-yl]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2-methylpropanoic acid
—— 15-Butyl-2,4-diethyl-12-thia-1-azoniapentacyclo[9.7.0.02,4.05,10.013,18]octadeca-1(11),5,7,9,13(18),14,16-heptaene —— C24H28NS+
15-Butyl-2,4-diethyl-12-thia-1-azoniapentacyclo[9.7.0.02,4.05,10.013,18]octadeca-1(11),5,7,9,13(18),14,16-heptaene
—— 5,6-dihydro-4aH-benzo[d][1]benzazepine —— C14H13N
5,6-dihydro-4aH-benzo[d][1]benzazepine
—— 6',6'-diethyl-2'-hexylidene-1'-(2-methylprop-2-enylidene)spiro[6H-benzo[a]quinolizin-5-ium-7,8'-7H-pyrido[2,1-a][2]benzazepin-5-ium] —— C40H46N2+2
6',6'-diethyl-2'-hexylidene-1'-(2-methylprop-2-enylidene)spiro[6H-benzo[a]quinolizin-5-ium-7,8'-7H-pyrido[2,1-a][2]benzazepin-5-ium]
—— 13-Benzhydryl-3,6,10-trioxa-13-azapentacyclo[10.8.1.02,7.09,20.014,19]henicosa-1(20),2(7),8,12(21),14,16,18-heptaene —— C30H23NO3
13-Benzhydryl-3,6,10-trioxa-13-azapentacyclo[10.8.1.02,7.09,20.014,19]henicosa-1(20),2(7),8,12(21),14,16,18-heptaene
—— 14-Ethyl-9,11-difluoro-19,20-dimethyl-5-(2-methylpentyl)-17-oxo-14-propyl-16-oxa-19-aza-2,22-diazoniapentacyclo[13.8.0.02,7.08,13.018,22]tricosa-1(15),2(7),3,5,8,10,12,18(22),20-nonaene-10-carbonitrile —— C33H38F2N4O2+2
14-Ethyl-9,11-difluoro-19,20-dimethyl-5-(2-methylpentyl)-17-oxo-14-propyl-16-oxa-19-aza-2,22-diazoniapentacyclo[13.8.0.02,7.08,13.018,22]tricosa-1(15),2(7),3,5,8,10,12,18(22),20-nonaene-10-carbonitrile
—— 9-Chloro-2-[(3-methyl-2,4,5,6-tetrahydropyrido[3,2-g][1,3]oxazocin-8-yl)amino]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione —— C22H21ClN6OS
9-Chloro-2-[(3-methyl-2,4,5,6-tetrahydropyrido[3,2-g][1,3]oxazocin-8-yl)amino]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione
—— 1,7-dimethyl-4,5-dihydro-3H-2-benzazepine;ethane —— C16H27N
1,7-dimethyl-4,5-dihydro-3H-2-benzazepine;ethane
—— methyl 2-[2-[3-(1H-imidazo[4,5-b]pyridin-2-yl)propylcarbamoyl]-2-benzazepin-5-yl]acetate —— C23H23N5O3
methyl 2-[2-[3-(1H-imidazo[4,5-b]pyridin-2-yl)propylcarbamoyl]-2-benzazepin-5-yl]acetate
—— (5S)-7-benzyl-9-hydroxy-5,16-dimethyl-3,6,9,14-tetraza-7-azoniapentacyclo[11.9.0.02,10.07,14.017,22]docosa-1(13),2(10),11,17,19,21-hexaene-4,8,15-trione —— C26H24N5O4+
(5S)-7-benzyl-9-hydroxy-5,16-dimethyl-3,6,9,14-tetraza-7-azoniapentacyclo[11.9.0.02,10.07,14.017,22]docosa-1(13),2(10),11,17,19,21-hexaene-4,8,15-trione
—— 2-tert-butyl-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine —— C15H20N2O
2-tert-butyl-6,7,8,9-tetrahydro-5H-[1,3]oxazolo[4,5-h][1]benzazepine
—— (1-tert-butyl-2-oxo-4,5-dihydro-3H-1-benzazepin-3-yl) carbamate —— C15H20N2O3
(1-tert-butyl-2-oxo-4,5-dihydro-3H-1-benzazepin-3-yl) carbamate
—— 3-[1-(1H-imidazol-2-yl)ethyl]-1,2,4,5-tetrahydro-3-benzazepine —— C15H19N3
3-[1-(1H-imidazol-2-yl)ethyl]-1,2,4,5-tetrahydro-3-benzazepine
—— N-[(4-carbamimidoylphenyl)methyl]acetamide;2-(3-oxo-1,2,4,5-tetrahydro-1-benzazepin-2-yl)acetic acid —— C22H26N4O4
N-[(4-carbamimidoylphenyl)methyl]acetamide;2-(3-oxo-1,2,4,5-tetrahydro-1-benzazepin-2-yl)acetic acid
—— 7-[6-(diazonioamino)pyrimidin-4-yl]oxy-1-[[3-(trifluoromethyl)phenyl]carbamoyl]-2,3,4,5-tetrahydro-1-benzazepine —— C22H19F3N7O2+
7-[6-(diazonioamino)pyrimidin-4-yl]oxy-1-[[3-(trifluoromethyl)phenyl]carbamoyl]-2,3,4,5-tetrahydro-1-benzazepine
—— 2-[4-(16-Fluoro-3,5,11,13-tetrazatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),2(6),4,7(12),8,10,15,17-octaen-4-yl)cyclohexyl]acetaldehyde —— C22H21FN4O
2-[4-(16-Fluoro-3,5,11,13-tetrazatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),2(6),4,7(12),8,10,15,17-octaen-4-yl)cyclohexyl]acetaldehyde
—— 8-butan-2-yl-3,4-dihydro-1H-1-benzazepine-2,5-dione —— C14H17NO2
8-butan-2-yl-3,4-dihydro-1H-1-benzazepine-2,5-dione
—— N'-[1-[2-(dimethylamino)ethyl]-2,3,4,5-tetrahydro-1-benzazepin-7-yl]thiophene-2-carboximidamide;N'-[1-[2-(methylamino)ethyl]-3,4-dihydro-2H-quinolin-6-yl]thiophene-2-carboximidamide;N'-[2-methylidene-3-(1-methylpiperidin-4-yl)-1,3-dihydroindol-5-yl]thiophene-2-carboximidamide;N'-[2-methylidene-1-(2-pyrrolidin-1-ylethyl)-4,5-dihydro-3H-1-benzazepin-7-yl]thiophene-2-carboximidamide;N'-(1-pyrrolidin-3-yl-3,4-dihydro-2H-quinolin-6-yl)thiophene-2-carboximidamide;N'-[1-(2-pyrrolidin-1-ylethyl)-2,3,4,5-tetrahydro-1-benzazepin-7-yl]thiophene-2-carboximidamide —— C117H150N24S6
N'-[1-[2-(dimethylamino)ethyl]-2,3,4,5-tetrahydro-1-benzazepin-7-yl]thiophene-2-carboximidamide;N'-[1-[2-(methylamino)ethyl]-3,4-dihydro-2H-quinolin-6-yl]thiophene-2-carboximidamide;N'-[2-methylidene-3-(1-methylpiperidin-4-yl)-1,3-dihydroindol-5-yl]thiophene-2-carboximidamide;N'-[2-methylidene-1-(2-pyrrolidin-1-ylethyl)-4,5-dihydro-3H-1-benzazepin-7-yl]thiophene-2-carboximidamide;N'-(1-pyrrolidin-3-yl-3,4-dihydro-2H-quinolin-6-yl)thiophene-2-carboximidamide;N'-[1-(2-pyrrolidin-1-ylethyl)-2,3,4,5-tetrahydro-1-benzazepin-7-yl]thiophene-2-carboximidamide