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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-(3-chlorophenyl)-2,2-difluoro-1-hydroxy-1,3,6,7,9,10-hexahydro-2H-8-azacyclohepta[e]indene-8-carboxylic acid ethyl ester 1616480-18-2 C22H22ClF2NO3
1-(3-chlorophenyl)-2,2-difluoro-1-hydroxy-1,3,6,7,9,10-hexahydro-2H-8-azacyclohepta[e]indene-8-carboxylic acid ethyl ester
—— benzyl 8-fluoro-10-methoxy-2,4,5,8,9,10-hexahydro-1H-cyclopenta[i][3]benzazepine-3-carboxylate —— C22H24FNO3
benzyl 8-fluoro-10-methoxy-2,4,5,8,9,10-hexahydro-1H-cyclopenta[i][3]benzazepine-3-carboxylate
—— Benzyl 10-fluoro-10-methoxy-1,2,4,5,8,9-hexahydrocyclopenta[i][3]benzazepine-3-carboxylate —— C22H24FNO3
Benzyl 10-fluoro-10-methoxy-1,2,4,5,8,9-hexahydrocyclopenta[i][3]benzazepine-3-carboxylate
—— 1,3,6,7,9,10-hexahydro-2H-8-azacyclohepta[e]indene-8-carboxylic acid ethyl ester 1616480-03-5 C16H21NO2
1,3,6,7,9,10-hexahydro-2H-8-azacyclohepta[e]indene-8-carboxylic acid ethyl ester
—— ethyl (10E)-10-ethylidene-9,9-difluoro-2,4,5,8-tetrahydro-1H-cyclopenta[i][3]benzazepine-3-carboxylate —— C18H21F2NO2
ethyl (10E)-10-ethylidene-9,9-difluoro-2,4,5,8-tetrahydro-1H-cyclopenta[i][3]benzazepine-3-carboxylate
—— 7-methoxy-N-methyl-2-(1,2,4,5-tetrahydro-3-benzazepin-3-ylmethyl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine —— C22H24N6O
7-methoxy-N-methyl-2-(1,2,4,5-tetrahydro-3-benzazepin-3-ylmethyl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine
—— 3-(3-Hydroxypropyl)-7,8-dimethoxy-1,3-dihydro-2h-benzo[d]azepin-2-one —— C15H19NO4
3-(3-Hydroxypropyl)-7,8-dimethoxy-1,3-dihydro-2h-benzo[d]azepin-2-one
—— 8-[3-[(3,4-dimethoxy-7-bicyclo[4.2.0]octa-1,3,5-trienyl)methylamino]propyl]-3,6,9,10-tetrahydro-2H-[1,4]dioxino[2,3-h][3]benzazepin-7-one —— C26H32N2O5
8-[3-[(3,4-dimethoxy-7-bicyclo[4.2.0]octa-1,3,5-trienyl)methylamino]propyl]-3,6,9,10-tetrahydro-2H-[1,4]dioxino[2,3-h][3]benzazepin-7-one
—— 3-(3-aminopropyl)-7,8-dimethoxy-1H-3-benzazepin-2-one —— C15H20N2O3
3-(3-aminopropyl)-7,8-dimethoxy-1H-3-benzazepin-2-one
—— N-[(1R)-2-hydroxy-1-phenylethyl]-4-methyl-1,2,3,5-tetrahydro-1-benzazepine-4-carboxamide —— C20H24N2O2
N-[(1R)-2-hydroxy-1-phenylethyl]-4-methyl-1,2,3,5-tetrahydro-1-benzazepine-4-carboxamide
—— 1-[(4R)-7-bromo-8-hydroxy-4-propan-2-yl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C15H17BrF3NO2
1-[(4R)-7-bromo-8-hydroxy-4-propan-2-yl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— 1-[(4R)-4-tert-butyl-6-methylsulfonyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C17H22F3NO3S
1-[(4R)-4-tert-butyl-6-methylsulfonyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— (4R)-8-hydroxy-4-propan-2-yl-3-(2,2,2-trifluoroacetyl)-1,2,4,5-tetrahydro-3-benzazepine-7-carbonitrile —— C16H17F3N2O2
(4R)-8-hydroxy-4-propan-2-yl-3-(2,2,2-trifluoroacetyl)-1,2,4,5-tetrahydro-3-benzazepine-7-carbonitrile
—— 1-[(4R)-6-bromo-4-tert-butyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C16H19BrF3NO
1-[(4R)-6-bromo-4-tert-butyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— 1-[(4R)-7,8-diamino-4-tert-butyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C16H22F3N3O
1-[(4R)-7,8-diamino-4-tert-butyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— (7R)-7-tert-butyl-7,8,9,10-tetrahydro-6H-pyrazino[2,3-h][3]benzazepine —— C16H21N3
(7R)-7-tert-butyl-7,8,9,10-tetrahydro-6H-pyrazino[2,3-h][3]benzazepine
—— (4R)-4-propan-2-yl-2,3,4,5-tetrahydro-1H-3-benzazepine-7-carbonitrile —— C14H18N2
(4R)-4-propan-2-yl-2,3,4,5-tetrahydro-1H-3-benzazepine-7-carbonitrile
—— 1-[(4R)-8-bromo-4-tert-butyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C16H19BrF3NO
1-[(4R)-8-bromo-4-tert-butyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— 1-[(4R)-4-tert-butyl-8-methylsulfonyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone —— C17H22F3NO3S
1-[(4R)-4-tert-butyl-8-methylsulfonyl-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone
—— 2-(5-amino-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-2-yl)-1-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)ethanone 1616707-94-8 C22H22N6O2
2-(5-amino-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-2-yl)-1-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)ethanone
—— 2-(5-Amino-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-2-yl)-1-(5,7-dihydropyrrolo[3,4-b]pyridin-6-yl)ethanone;2-(5-amino-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-2-yl)-1-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethanone —— C41H39N13O4
2-(5-Amino-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-2-yl)-1-(5,7-dihydropyrrolo[3,4-b]pyridin-6-yl)ethanone;2-(5-amino-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-2-yl)-1-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethanone
—— 3-(3-Chloropropyl)-7,8-dimethoxy-1,3-dihydro-1-benzazepin-2-one —— C15H18ClNO3
3-(3-Chloropropyl)-7,8-dimethoxy-1,3-dihydro-1-benzazepin-2-one
—— 3-[3-[[1-(3,4-dimethoxyphenyl)cyclobutyl]methyl-methylamino]propyl]-7,8-dimethoxy-1H-3-benzazepin-2-one —— C29H38N2O5
3-[3-[[1-(3,4-dimethoxyphenyl)cyclobutyl]methyl-methylamino]propyl]-7,8-dimethoxy-1H-3-benzazepin-2-one
—— 7-methoxy-2-((7-methoxy-4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)methyl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine 1616708-49-6 C22H24N6O2
7-methoxy-2-((7-methoxy-4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)methyl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine
—— heptan-4-yl N-(6,11-dihydro-5H-benzo[b][1]benzazepin-2-yl)carbamate —— C22H28N2O2
heptan-4-yl N-(6,11-dihydro-5H-benzo[b][1]benzazepin-2-yl)carbamate
—— (15S)-7-cyclohexyl-10-methoxy-15-(3-methyl-3,8-diazabicyclo[3.2.1]octane-8-carbonyl)-1-azoniapentacyclo[10.7.0.02,4.06,11.014,19]nonadeca-3,5,7,9,11,14(19),17-heptaene-1-carboxylic acid —— C34H40N3O4+
(15S)-7-cyclohexyl-10-methoxy-15-(3-methyl-3,8-diazabicyclo[3.2.1]octane-8-carbonyl)-1-azoniapentacyclo[10.7.0.02,4.06,11.014,19]nonadeca-3,5,7,9,11,14(19),17-heptaene-1-carboxylic acid
—— (15S)-7-cyclohexyl-10-methoxy-15-(3-methyl-3,8-diazabicyclo[3.2.1]octane-8-carbonyl)-1-azoniapentacyclo[10.7.0.02,4.06,11.014,19]nonadeca-3,5,7,9,11,14(19),17-heptaene-1-carboxylic acid;2,2,2-trifluoroacetic acid —— C36H41F3N3O6+
(15S)-7-cyclohexyl-10-methoxy-15-(3-methyl-3,8-diazabicyclo[3.2.1]octane-8-carbonyl)-1-azoniapentacyclo[10.7.0.02,4.06,11.014,19]nonadeca-3,5,7,9,11,14(19),17-heptaene-1-carboxylic acid;2,2,2-trifluoroacetic acid
—— 10-(Propan-2-ylamino)-1,3-diazatricyclo[6.4.1.04,13]trideca-4,6,8(13)-triene-2,9-dione —— C14H17N3O2
10-(Propan-2-ylamino)-1,3-diazatricyclo[6.4.1.04,13]trideca-4,6,8(13)-triene-2,9-dione
—— [3-[2-(Ethoxycarbonylamino)-5,6-dihydrobenzo[b][1]benzazepin-11-yl]-3-oxopropyl]-(2-hydroxyethyl)azanium —— C22H28N3O4+
[3-[2-(Ethoxycarbonylamino)-5,6-dihydrobenzo[b][1]benzazepin-11-yl]-3-oxopropyl]-(2-hydroxyethyl)azanium
—— ethyl N-[11-[3-(2-hydroxyethylamino)propanoyl]-5,6-dihydrobenzo[b][1]benzazepin-2-yl]carbamate —— C22H27N3O4
ethyl N-[11-[3-(2-hydroxyethylamino)propanoyl]-5,6-dihydrobenzo[b][1]benzazepin-2-yl]carbamate
—— (5Z)-5-(aminomethylidene)-1-phenyl-3H-2-benzazepin-4-one —— C17H14N2O
(5Z)-5-(aminomethylidene)-1-phenyl-3H-2-benzazepin-4-one
—— 9-chloro-2-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-8-methyl-4,5-dihydro-3H-2-benzazepin-1-one —— C19H21ClN2O2
9-chloro-2-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-8-methyl-4,5-dihydro-3H-2-benzazepin-1-one
—— 7-chloro-2-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-8-methyl-4,5-dihydro-3H-2-benzazepin-1-one —— C19H21ClN2O2
7-chloro-2-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-8-methyl-4,5-dihydro-3H-2-benzazepin-1-one
—— 9-fluoro-9,10-dimethyl-2,3,4,5,8,10-hexahydro-1H-cyclopenta[i][3]benzazepine —— C15H20FN
9-fluoro-9,10-dimethyl-2,3,4,5,8,10-hexahydro-1H-cyclopenta[i][3]benzazepine
—— 9-fluoro-10-methoxy-9-methyl-2,3,4,5,8,10-hexahydro-1H-cyclopenta[i][3]benzazepine —— C15H20FNO
9-fluoro-10-methoxy-9-methyl-2,3,4,5,8,10-hexahydro-1H-cyclopenta[i][3]benzazepine
—— 9-chloro-7-[(2E,4Z)-hexa-2,4-dien-2-yl]-2-methyl-2,5-dihydro-1H-pyrimido[5,4-d][2]benzazepine —— C19H20ClN3
9-chloro-7-[(2E,4Z)-hexa-2,4-dien-2-yl]-2-methyl-2,5-dihydro-1H-pyrimido[5,4-d][2]benzazepine
—— 1-methanimidoyl-7-methyl-4,5-dihydro-3H-1-benzazepin-2-one —— C12H14N2O
1-methanimidoyl-7-methyl-4,5-dihydro-3H-1-benzazepin-2-one
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-2-[2-(3-methoxypropylamino)-2-oxoethyl]-6-methylheptanoate —— C33H50N2O9
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-2-[2-(3-methoxypropylamino)-2-oxoethyl]-6-methylheptanoate
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2-[2-[4-(dimethylamino)piperidin-1-yl]-2-oxoethyl]-2,6-dihydroxy-6-methylheptanoate —— C36H55N3O8
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2-[2-[4-(dimethylamino)piperidin-1-yl]-2-oxoethyl]-2,6-dihydroxy-6-methylheptanoate
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2-[2-(furan-2-ylmethylamino)-2-oxoethyl]-2,6-dihydroxy-6-methylheptanoate —— C34H46N2O9
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2-[2-(furan-2-ylmethylamino)-2-oxoethyl]-2,6-dihydroxy-6-methylheptanoate
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-6-methyl-2-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]heptanoate —— C34H51N3O8
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-6-methyl-2-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]heptanoate
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-6-methyl-2-[2-(2-methylpiperidin-1-yl)-2-oxoethyl]heptanoate —— C35H52N2O8
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-6-methyl-2-[2-(2-methylpiperidin-1-yl)-2-oxoethyl]heptanoate
—— 1-O-[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] 4-O-methyl (2R)-2-hydroxy-2-(4-hydroxy-4-methylpentyl)butanedioate —— C30H43NO9
1-O-[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] 4-O-methyl (2R)-2-hydroxy-2-(4-hydroxy-4-methylpentyl)butanedioate
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-2-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-6-methylheptanoate —— C34H50N2O9
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-2-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-6-methylheptanoate
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2-[2-(cyclohexylamino)-2-oxoethyl]-2,6-dihydroxy-6-methylheptanoate —— C35H52N2O8
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2-[2-(cyclohexylamino)-2-oxoethyl]-2,6-dihydroxy-6-methylheptanoate
—— 2-[[9-chloro-7-(2-fluoro-6-methylphenyl)-4,5-dihydro-1H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-1,3-oxazole-5-carboxylic acid —— C23H17ClFN5O3
2-[[9-chloro-7-(2-fluoro-6-methylphenyl)-4,5-dihydro-1H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-1,3-oxazole-5-carboxylic acid
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2-[2-(4-cyanopiperidin-1-yl)-2-oxoethyl]-2,6-dihydroxy-6-methylheptanoate —— C35H49N3O8
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2-[2-(4-cyanopiperidin-1-yl)-2-oxoethyl]-2,6-dihydroxy-6-methylheptanoate
—— 2-(4-aminophenyl)-5-(methoxymethyl)-8-(4-methylidenepiperidin-1-yl)-10H-furo[2,3-c][1]benzazepin-4-one —— C26H27N3O3
2-(4-aminophenyl)-5-(methoxymethyl)-8-(4-methylidenepiperidin-1-yl)-10H-furo[2,3-c][1]benzazepin-4-one
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-6-methyl-2-[2-oxo-2-(thiophen-2-ylmethylamino)ethyl]heptanoate —— C34H46N2O8S
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-6-methyl-2-[2-oxo-2-(thiophen-2-ylmethylamino)ethyl]heptanoate
—— [(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-6-methyl-2-(2-oxo-2-pyrrolidin-1-ylethyl)heptanoate —— C33H48N2O8
[(1S,18E,20S)-19-methoxy-5,7-dioxa-13-azatetracyclo[11.7.1.02,10.04,8]henicosa-2,4(8),9,18-tetraen-20-yl] (2R)-2,6-dihydroxy-6-methyl-2-(2-oxo-2-pyrrolidin-1-ylethyl)heptanoate