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苯氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-amino-8-[4-(dipropylcarbamoyl)phenyl]-7-methyl-N,N-dipropyl-3H-1-benzazepine-4-carboxamide —— C31H42N4O2
2-amino-8-[4-(dipropylcarbamoyl)phenyl]-7-methyl-N,N-dipropyl-3H-1-benzazepine-4-carboxamide
—— N-butyl-2-methylimino-N-propyl-8-[4-(pyrrolidine-1-carbonyl)phenyl]-1,3-dihydro-1-benzazepine-4-carboxamide —— C30H38N4O2
N-butyl-2-methylimino-N-propyl-8-[4-(pyrrolidine-1-carbonyl)phenyl]-1,3-dihydro-1-benzazepine-4-carboxamide
—— N-butyl-2-[2-(dimethylamino)ethylimino]-N-propyl-8-[4-(pyrrolidine-1-carbonyl)phenyl]-1,3-dihydro-1-benzazepine-4-carboxamide —— C33H45N5O2
N-butyl-2-[2-(dimethylamino)ethylimino]-N-propyl-8-[4-(pyrrolidine-1-carbonyl)phenyl]-1,3-dihydro-1-benzazepine-4-carboxamide
—— 2-amino-N-(3-hydroxypropyl)-7-methyl-N-propyl-8-[4-(pyrrolidine-1-carbonyl)phenyl]-3H-1-benzazepine-4-carboxamide —— C29H36N4O3
2-amino-N-(3-hydroxypropyl)-7-methyl-N-propyl-8-[4-(pyrrolidine-1-carbonyl)phenyl]-3H-1-benzazepine-4-carboxamide
—— 2-(cyclopropylmethyl)-N'-(9-fluoro-4-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-3-(3,3,3-trifluoropropyl)butanediamide —— C26H27F4N3O3
2-(cyclopropylmethyl)-N'-(9-fluoro-4-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-3-(3,3,3-trifluoropropyl)butanediamide
—— 6,6,6-trifluoro-3-[[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]carbamoyl]-2-(3,3,3-trifluoropropyl)hexanoic acid —— C24H22F6N2O4
6,6,6-trifluoro-3-[[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]carbamoyl]-2-(3,3,3-trifluoropropyl)hexanoic acid
—— 4-Fluoro-5,7-dihydrobenzo[d][1]benzazepin-6-one —— C14H10FNO
4-Fluoro-5,7-dihydrobenzo[d][1]benzazepin-6-one
—— (2R,3S)-N'-[(7S)-9-fluoro-4-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide —— C25H24F7N3O3
(2R,3S)-N'-[(7S)-9-fluoro-4-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-3-(cyclopropylmethyl)-N'-[(7S)-4-fluoro-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-(3,3,3-trifluoropropyl)butanediamide —— C25H25F4N3O3
(2R,3S)-3-(cyclopropylmethyl)-N'-[(7S)-4-fluoro-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-(3,3,3-trifluoropropyl)butanediamide
—— 7-Amino-9-fluoro-4-methyl-5,7-dihydrobenzo[d][1]benzazepin-6-one —— C15H13FN2O
7-Amino-9-fluoro-4-methyl-5,7-dihydrobenzo[d][1]benzazepin-6-one
—— 4-fluoro-5-[(4-methoxyphenyl)methyl]-7H-benzo[d][1]benzazepin-6-one —— C22H18FNO2
4-fluoro-5-[(4-methoxyphenyl)methyl]-7H-benzo[d][1]benzazepin-6-one
—— 4-Chloro-5,7-dihydrobenzo[d][1]benzazepin-6-one —— C14H10ClNO
4-Chloro-5,7-dihydrobenzo[d][1]benzazepin-6-one
—— N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide —— C24H23F6N3O3
N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-3-[(3,3-difluorocyclobutyl)methyl]-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-(3,3,3-trifluoropropyl)butanediamide —— C26H26F5N3O3
(2R,3S)-3-[(3,3-difluorocyclobutyl)methyl]-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-3-propyl-2-(3,3,3-trifluoropropyl)butanediamide —— C24H26F3N3O3
(2R,3S)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-3-propyl-2-(3,3,3-trifluoropropyl)butanediamide
—— (2S)-2-(cyclopropylmethyl)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-N'-(3,3,3-trifluoropropyl)butanediamide —— C25H26F3N3O3
(2S)-2-(cyclopropylmethyl)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-N'-(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide —— C24H23F6N3O3
(2R,3S)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2,3-bis(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-N'-(4-chloro-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-2,3-bis(3,3,3-trifluoropropyl)butanediamide —— C24H22ClF6N3O3
(2R,3S)-N'-(4-chloro-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-2,3-bis(3,3,3-trifluoropropyl)butanediamide
—— (2R,3R)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-3-phenyl-2-(3,3,3-trifluoropropyl)butanediamide —— C27H24F3N3O3
(2R,3R)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-3-phenyl-2-(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-3-(cyclopropylmethyl)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-(3,3,3-trifluoropropyl)butanediamide —— C25H26F3N3O3
(2R,3S)-3-(cyclopropylmethyl)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-(3,3,3-trifluoropropyl)butanediamide
—— 9-Fluoro-4-methyl-5,7-dihydrobenzo[d][1]benzazepin-6-one —— C15H12FNO
9-Fluoro-4-methyl-5,7-dihydrobenzo[d][1]benzazepin-6-one
—— N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-propyl-3-(3,3,3-trifluoropropyl)butanediamide —— C24H26F3N3O3
N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-propyl-3-(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-3-(cyclopropylmethyl)-N'-[(7S)-9-fluoro-4-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-(3,3,3-trifluoropropyl)butanediamide —— C26H27F4N3O3
(2R,3S)-3-(cyclopropylmethyl)-N'-[(7S)-9-fluoro-4-methyl-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-(3,3,3-trifluoropropyl)butanediamide
—— N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-3-propyl-2-(3,3,3-trifluoropropyl)butanediamide —— C24H26F3N3O3
N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-3-propyl-2-(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-N'-(4-fluoro-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-3-propyl-2-(3,3,3-trifluoropropyl)butanediamide —— C24H25F4N3O3
(2R,3S)-N'-(4-fluoro-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl)-3-propyl-2-(3,3,3-trifluoropropyl)butanediamide
—— (2R,3S)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-propyl-3-(3,3,3-trifluoropropyl)butanediamide —— C24H26F3N3O3
(2R,3S)-N'-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-2-propyl-3-(3,3,3-trifluoropropyl)butanediamide
—— 7-bromo-5-methylphosphanyl-3,4-dihydro-1-benzazepin-2-one —— C11H11BrNOP
7-bromo-5-methylphosphanyl-3,4-dihydro-1-benzazepin-2-one
—— (7-Bromo-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-(2-chloro-6-fluorophenyl)methanone 1532517-52-4 C17H14BrClFNO
(7-Bromo-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-(2-chloro-6-fluorophenyl)methanone
—— [4-(dipropylcarbamoyl)-8-[4-(pyrrolidine-1-carbonyl)phenyl]-3H-1-benzazepin-2-yl]carbamic acid —— C29H34N4O4
[4-(dipropylcarbamoyl)-8-[4-(pyrrolidine-1-carbonyl)phenyl]-3H-1-benzazepin-2-yl]carbamic acid
—— 2-amino-7-(pyridin-2-ylmethoxy)-3H-1-benzazepine-4-carboxylic acid —— C17H15N3O3
2-amino-7-(pyridin-2-ylmethoxy)-3H-1-benzazepine-4-carboxylic acid
—— N-hydroxybenzo[b][1]benzazepine-11-carboxamide —— C15H12N2O2
N-hydroxybenzo[b][1]benzazepine-11-carboxamide
—— (8S,12R,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,22-pentazahexacyclo[17.2.1.05,21.06,13.08,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine 1581683-01-3 C23H23FN8O
(8S,12R,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,22-pentazahexacyclo[17.2.1.05,21.06,13.08,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine
—— (1R,16S,17S,18R)-13-fluoro-11-N-methyl-5-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[15.2.1.17,10.02,16.03,8.09,14]henicosa-3,5,7,9,11,13-hexaene-11,18-diamine 1581682-84-9 C23H23FN8O
(1R,16S,17S,18R)-13-fluoro-11-N-methyl-5-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[15.2.1.17,10.02,16.03,8.09,14]henicosa-3,5,7,9,11,13-hexaene-11,18-diamine
—— 12-fluoro-14-N-methyl-3-(2-methylpyrimidin-5-yl)oxyspiro[2,4,6,18-tetrazapentacyclo[13.2.1.05,17.06,9.011,16]octadeca-1(17),2,4,11,13,15-hexaene-8,2'-cyclobutane]-1',14-diamine 1581683-07-9 C23H23FN8O
12-fluoro-14-N-methyl-3-(2-methylpyrimidin-5-yl)oxyspiro[2,4,6,18-tetrazapentacyclo[13.2.1.05,17.06,9.011,16]octadeca-1(17),2,4,11,13,15-hexaene-8,2'-cyclobutane]-1',14-diamine
—— (7R,11R,13R)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,22-pentazahexacyclo[17.2.1.05,21.06,13.07,11.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine 1581683-11-5 C23H23FN8O
(7R,11R,13R)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,22-pentazahexacyclo[17.2.1.05,21.06,13.07,11.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine
—— (9R,11S,12R)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.08,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-9,17-diamine —— C23H23FN8O
(9R,11S,12R)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.08,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-9,17-diamine
—— (8R,10R)-13-fluoro-15-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,19-tetrazapentacyclo[14.2.1.05,18.06,10.012,17]nonadeca-1(18),2,4,12,14,16-hexaene-8,15-diamine 1581683-05-7 C21H21FN8O
(8R,10R)-13-fluoro-15-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,19-tetrazapentacyclo[14.2.1.05,18.06,10.012,17]nonadeca-1(18),2,4,12,14,16-hexaene-8,15-diamine
—— (1R)-1-[5-[[(1R,16S,17S,18R)-18-amino-13-fluoro-11-(methylamino)-2,4,6,21-tetrazahexacyclo[15.2.1.17,10.02,16.03,8.09,14]henicosa-3,5,7,9,11,13-hexaen-5-yl]oxy]pyrimidin-2-yl]ethanol 1581683-03-5 C24H25FN8O2
(1R)-1-[5-[[(1R,16S,17S,18R)-18-amino-13-fluoro-11-(methylamino)-2,4,6,21-tetrazahexacyclo[15.2.1.17,10.02,16.03,8.09,14]henicosa-3,5,7,9,11,13-hexaen-5-yl]oxy]pyrimidin-2-yl]ethanol
—— (9R,10S,11S)-14-fluoro-16-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,20-tetrazahexacyclo[15.2.1.05,19.06,11.07,10.013,18]icosa-1(19),2,4,13,15,17-hexaene-9,16-diamine —— C22H21FN8O
(9R,10S,11S)-14-fluoro-16-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,20-tetrazahexacyclo[15.2.1.05,19.06,11.07,10.013,18]icosa-1(19),2,4,13,15,17-hexaene-9,16-diamine
—— (9R,11S)-14-fluoro-16-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,20-tetrazahexacyclo[15.2.1.05,19.06,11.08,10.013,18]icosa-1(19),2,4,13,15,17-hexaene-9,16-diamine 1581683-08-0 C22H21FN8O
(9R,11S)-14-fluoro-16-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,20-tetrazahexacyclo[15.2.1.05,19.06,11.08,10.013,18]icosa-1(19),2,4,13,15,17-hexaene-9,16-diamine
—— (1R,16S,17R)-13-fluoro-N-methyl-5-(2-methylpyrimidin-5-yl)oxy-2,4,6,18,21-pentazahexacyclo[15.2.1.17,10.02,16.03,8.09,14]henicosa-3,5,7,9,11,13-hexaen-11-amine 1581683-12-6 C22H21FN8O
(1R,16S,17R)-13-fluoro-N-methyl-5-(2-methylpyrimidin-5-yl)oxy-2,4,6,18,21-pentazahexacyclo[15.2.1.17,10.02,16.03,8.09,14]henicosa-3,5,7,9,11,13-hexaen-11-amine
—— (9R,10S)-13-fluoro-15-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,19-tetrazapentacyclo[14.2.1.05,18.06,10.012,17]nonadeca-1(18),2,4,12,14,16-hexaene-9,15-diamine 1581683-04-6 C21H21FN8O
(9R,10S)-13-fluoro-15-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,19-tetrazapentacyclo[14.2.1.05,18.06,10.012,17]nonadeca-1(18),2,4,12,14,16-hexaene-9,15-diamine
—— (8R,9S)-12-fluoro-14-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,18-tetrazapentacyclo[13.2.1.05,17.06,9.011,16]octadeca-1(17),2,4,11,13,15-hexaene-8,14-diamine 1581683-06-8 C20H19FN8O
(8R,9S)-12-fluoro-14-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,18-tetrazapentacyclo[13.2.1.05,17.06,9.011,16]octadeca-1(17),2,4,11,13,15-hexaene-8,14-diamine
—— (8R,12R,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,11,22-pentazahexacyclo[17.2.1.05,21.06,13.08,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine 1581683-00-2 C23H23FN8O
(8R,12R,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,11,22-pentazahexacyclo[17.2.1.05,21.06,13.08,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine
—— (8S,10R,11S,12S)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.08,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-10,17-diamine 1581683-09-1 C23H23FN8O
(8S,10R,11S,12S)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.08,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-10,17-diamine
—— (1R,16R,17S,18R)-13-fluoro-11-N-methyl-5-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[15.2.1.17,10.02,16.03,8.09,14]henicosa-3,5,7,9,11,13-hexaene-11,18-diamine 1581683-02-4 C23H23FN8O
(1R,16R,17S,18R)-13-fluoro-11-N-methyl-5-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[15.2.1.17,10.02,16.03,8.09,14]henicosa-3,5,7,9,11,13-hexaene-11,18-diamine
—— (7S,9S,11S,12S)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-9,17-diamine —— C23H23FN8O
(7S,9S,11S,12S)-15-fluoro-17-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,21-tetrazahexacyclo[16.2.1.05,20.06,12.07,11.014,19]henicosa-1(20),2,4,14,16,18-hexaene-9,17-diamine
—— (7R,12S,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,22-pentazahexacyclo[17.2.1.05,21.06,13.07,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine —— C23H23FN8O
(7R,12S,13S)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,22-pentazahexacyclo[17.2.1.05,21.06,13.07,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine
—— (8R,12S,13R)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,22-pentazahexacyclo[17.2.1.05,21.06,13.08,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine 1581682-99-6 C23H23FN8O
(8R,12S,13R)-16-fluoro-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,9,22-pentazahexacyclo[17.2.1.05,21.06,13.08,12.015,20]docosa-1(21),2,4,15,17,19-hexaen-18-amine
—— (7S,9S,11S,13R)-16-fluoro-18-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,22-tetrazahexacyclo[17.2.1.05,21.06,13.07,11.015,20]docosa-1(21),2,4,15,17,19-hexaene-9,18-diamine —— C24H25FN8O
(7S,9S,11S,13R)-16-fluoro-18-N-methyl-3-(2-methylpyrimidin-5-yl)oxy-2,4,6,22-tetrazahexacyclo[17.2.1.05,21.06,13.07,11.015,20]docosa-1(21),2,4,15,17,19-hexaene-9,18-diamine