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—— (E)-3-(4-methylphenyl)-1-[4-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]prop-2-en-1-one —— C18H21N3O4S
(E)-3-(4-methylphenyl)-1-[4-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]prop-2-en-1-one
—— (E)-3-(4-fluorophenyl)-N-[3-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide —— C15H16FN3O4S
(E)-3-(4-fluorophenyl)-N-[3-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide
—— (E)-3-(4-methylphenyl)-N-[5-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)pentyl]prop-2-enamide —— C18H23N3O4S
(E)-3-(4-methylphenyl)-N-[5-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)pentyl]prop-2-enamide
—— (E)-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methylpropyl]-2-phenylethenesulfonamide —— C20H23NO4S
(E)-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methylpropyl]-2-phenylethenesulfonamide
—— (E)-3-(4-methoxyphenyl)-N-[3-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide —— C16H19N3O5S
(E)-3-(4-methoxyphenyl)-N-[3-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide
—— (E)-3-(2,5-dimethoxyphenyl)-N-[3-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide —— C17H21N3O6S
(E)-3-(2,5-dimethoxyphenyl)-N-[3-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide
—— (E)-3-(2,4-dichlorophenyl)-N-[3-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide —— C15H15Cl2N3O4S
(E)-3-(2,4-dichlorophenyl)-N-[3-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide
—— Ethyl 4-[[2-(tert-butylamino)-2-oxoethyl]-methylsulfamoyl]benzoate —— C16H24N2O5S
Ethyl 4-[[2-(tert-butylamino)-2-oxoethyl]-methylsulfamoyl]benzoate
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]prop-2-enamide —— C20H27N3O2
(E)-3-[4-(cyanomethoxy)phenyl]-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]prop-2-enamide
—— ethyl N-[3-[[4-(propan-2-ylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate —— C19H23N3O5S
ethyl N-[3-[[4-(propan-2-ylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate
—— ethyl N-[4-[[4-(methylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate —— C17H19N3O5S
ethyl N-[4-[[4-(methylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate
—— (E)-3-(4-chlorophenyl)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]prop-2-enamide —— C14H14ClN3O4S
(E)-3-(4-chlorophenyl)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]prop-2-enamide
—— (E)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]-3-(2-propoxyphenyl)prop-2-enamide —— C17H21N3O5S
(E)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]-3-(2-propoxyphenyl)prop-2-enamide
—— (E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-propoxyphenyl)prop-2-enamide —— C16H19N3O5S
(E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-propoxyphenyl)prop-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]prop-2-enamide —— C13H12FN3O4S
(E)-3-(4-fluorophenyl)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]-3-phenylprop-2-enamide —— C14H15N3O4S
(E)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]-3-phenylprop-2-enamide
—— (E)-3-(3,4-dichlorophenyl)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]prop-2-enamide —— C13H11Cl2N3O4S
(E)-3-(3,4-dichlorophenyl)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]prop-2-enamide
—— (E)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]-3-(4-propoxyphenyl)prop-2-enamide —— C17H21N3O5S
(E)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]-3-(4-propoxyphenyl)prop-2-enamide
—— (E)-3-(2-methoxy-5-methylphenyl)-N-[4-(methylsulfamoyl)phenyl]prop-2-enamide —— C18H20N2O4S
(E)-3-(2-methoxy-5-methylphenyl)-N-[4-(methylsulfamoyl)phenyl]prop-2-enamide
—— ethyl 2-[[(2R)-2-(furan-3-carbonylamino)propanoyl]amino]-1,3-thiazole-4-carboxylate —— C14H15N3O5S
ethyl 2-[[(2R)-2-(furan-3-carbonylamino)propanoyl]amino]-1,3-thiazole-4-carboxylate
—— (E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-phenylmethoxyphenyl)prop-2-enamide —— C20H19N3O5S
(E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-phenylmethoxyphenyl)prop-2-enamide
—— (E)-3-(2,5-dimethoxyphenyl)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]prop-2-enamide —— C15H17N3O6S
(E)-3-(2,5-dimethoxyphenyl)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]prop-2-enamide
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]prop-2-enamide —— C20H27N3O2
(E)-3-[4-(cyanomethoxy)phenyl]-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]prop-2-enamide
—— (E)-3-(6-methoxynaphthalen-2-yl)-N-[4-(methylsulfamoyl)phenyl]prop-2-enamide —— C21H20N2O4S
(E)-3-(6-methoxynaphthalen-2-yl)-N-[4-(methylsulfamoyl)phenyl]prop-2-enamide
—— (E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylprop-2-enamide —— C13H13N3O4S
(E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylprop-2-enamide
—— (E)-3-(4-fluorophenyl)-1-[(2S)-2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)pyrrolidin-1-yl]prop-2-en-1-one —— C16H16FN3O4S
(E)-3-(4-fluorophenyl)-1-[(2S)-2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)pyrrolidin-1-yl]prop-2-en-1-one
—— ethyl N-[3-[(pentylcarbamothioylamino)carbamoyl]phenyl]carbamate —— C16H24N4O3S
ethyl N-[3-[(pentylcarbamothioylamino)carbamoyl]phenyl]carbamate
—— (E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(2,6-dichlorophenyl)prop-2-enamide —— C16H9Cl3N2O3
(E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(2,6-dichlorophenyl)prop-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]prop-2-enamide —— C14H14FN3O4S
(E)-3-(4-fluorophenyl)-N-[2-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)ethyl]prop-2-enamide
—— (E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-propoxyphenyl)prop-2-enamide —— C16H19N3O5S
(E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-propoxyphenyl)prop-2-enamide
—— (E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-propan-2-ylphenyl)prop-2-enamide —— C16H19N3O4S
(E)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-propan-2-ylphenyl)prop-2-enamide
—— (E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(2,3-dimethylphenyl)prop-2-enamide —— C18H15ClN2O3
(E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(2,3-dimethylphenyl)prop-2-enamide
—— (E)-N-[(1S,2R)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)butyl]-3-phenylprop-2-enamide —— C17H21N3O4S
(E)-N-[(1S,2R)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)butyl]-3-phenylprop-2-enamide
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-cyano-N-(2,6-dichlorophenyl)prop-2-enamide —— C18H11Cl3N2O3
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-cyano-N-(2,6-dichlorophenyl)prop-2-enamide
—— (E)-2-cyano-3-[5-(2-fluorophenyl)furan-2-yl]-N-(4-sulfamoylphenyl)prop-2-enamide —— C20H14FN3O4S
(E)-2-cyano-3-[5-(2-fluorophenyl)furan-2-yl]-N-(4-sulfamoylphenyl)prop-2-enamide
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-(4-sulfamoylphenyl)prop-2-enamide —— C17H12ClN3O5S
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-(4-sulfamoylphenyl)prop-2-enamide
—— (E)-2-cyano-3-[1-[(3R)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]-N-(2-methoxyphenyl)prop-2-enamide —— C20H22N4O4S
(E)-2-cyano-3-[1-[(3R)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]-N-(2-methoxyphenyl)prop-2-enamide
—— (E)-N-[(2S)-2-(dimethylamino)-2-(2-methoxyphenyl)ethyl]-3-(6-methoxynaphthalen-2-yl)prop-2-enamide —— C25H28N2O3
(E)-N-[(2S)-2-(dimethylamino)-2-(2-methoxyphenyl)ethyl]-3-(6-methoxynaphthalen-2-yl)prop-2-enamide
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-cyano-N-(3,4-dimethoxyphenyl)prop-2-enamide —— C20H17ClN2O5
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-cyano-N-(3,4-dimethoxyphenyl)prop-2-enamide
—— ethyl 2-[[(2S)-2-(furan-3-carbonylamino)propanoyl]amino]-1,3-thiazole-4-carboxylate —— C14H15N3O5S
ethyl 2-[[(2S)-2-(furan-3-carbonylamino)propanoyl]amino]-1,3-thiazole-4-carboxylate
—— (E)-N-(3-chloro-4-methoxyphenyl)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)prop-2-enamide —— C20H22ClN3O2
(E)-N-(3-chloro-4-methoxyphenyl)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)prop-2-enamide
—— (E)-4-(1,3-benzothiazol-2-yl)-5-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]pent-4-enoic acid —— C22H21N3O3S
(E)-4-(1,3-benzothiazol-2-yl)-5-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]pent-4-enoic acid
—— (E)-3-(4-ethylphenyl)-N-[4-(propan-2-ylsulfamoyl)phenyl]prop-2-enamide —— C20H24N2O3S
(E)-3-(4-ethylphenyl)-N-[4-(propan-2-ylsulfamoyl)phenyl]prop-2-enamide
—— (E)-4-(1,3-benzothiazol-2-yl)-5-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)pent-4-enoic acid —— C20H16ClNO4S
(E)-4-(1,3-benzothiazol-2-yl)-5-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)pent-4-enoic acid
—— (E)-2-cyano-N-(2,6-dichlorophenyl)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide —— C20H16Cl2N4O2
(E)-2-cyano-N-(2,6-dichlorophenyl)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide
—— (E)-3-[1-benzyl-3-(3-methoxyphenyl)pyrazol-4-yl]-N-butyl-2-cyanoprop-2-enamide —— C25H26N4O2
(E)-3-[1-benzyl-3-(3-methoxyphenyl)pyrazol-4-yl]-N-butyl-2-cyanoprop-2-enamide
—— (E)-N-[(1S,2R)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)butyl]-3-(2-propoxyphenyl)prop-2-enamide —— C20H27N3O5S
(E)-N-[(1S,2R)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)butyl]-3-(2-propoxyphenyl)prop-2-enamide
—— (E)-4-(1,3-benzothiazol-2-yl)-5-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)pent-4-enoate —— C20H15ClNO4S-
(E)-4-(1,3-benzothiazol-2-yl)-5-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)pent-4-enoate
—— (E)-3-(4-methylphenyl)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]prop-2-enamide —— C14H15N3O4S
(E)-3-(4-methylphenyl)-N-[(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)methyl]prop-2-enamide
—— (E)-2-cyano-N-(3,4-dimethoxyphenyl)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide —— C22H22N4O4
(E)-2-cyano-N-(3,4-dimethoxyphenyl)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide