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—— (E)-2-cyano-3-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]-N-(4-fluoro-2-methylphenyl)prop-2-enamide —— C22H24FN3O2
(E)-2-cyano-3-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]-N-(4-fluoro-2-methylphenyl)prop-2-enamide
—— (E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-2-cyano-N-(2,4,6-trimethylphenyl)prop-2-enamide —— C24H23ClN4O
(E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-2-cyano-N-(2,4,6-trimethylphenyl)prop-2-enamide
—— ethyl (6R)-6-[3-(difluoromethoxy)-4-methoxyphenyl]-4-methyl-3-prop-2-enyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H22F2N2O4S
ethyl (6R)-6-[3-(difluoromethoxy)-4-methoxyphenyl]-4-methyl-3-prop-2-enyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3,4-difluorophenyl)-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C15H16F2N2O2S
ethyl (6S)-6-(3,4-difluorophenyl)-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-N-(3-chloro-2-methylphenyl)-2-cyanoprop-2-enamide —— C16H10Cl2N4OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-N-(3-chloro-2-methylphenyl)-2-cyanoprop-2-enamide
—— (E)-2-cyano-3-[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]-N-(4-fluoro-2-methylphenyl)prop-2-enamide —— C21H24FN3O
(E)-2-cyano-3-[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]-N-(4-fluoro-2-methylphenyl)prop-2-enamide
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(2,4,6-trimethylphenyl)prop-2-enamide —— C18H15ClN4OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(2,4,6-trimethylphenyl)prop-2-enamide
—— ethyl 2-[(2S)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-2-yl]acetate —— C13H19N3O4
ethyl 2-[(2S)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-2-yl]acetate
—— ethyl (6R)-6-(3,4-difluorophenyl)-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C15H16F2N2O2S
ethyl (6R)-6-(3,4-difluorophenyl)-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]-N-(2-ethoxyphenyl)prop-2-enamide —— C24H21N5O2
(E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]-N-(2-ethoxyphenyl)prop-2-enamide
—— (E)-2-cyano-3-(2,3,4-trimethoxyphenyl)-N-(2,4,6-trimethylphenyl)prop-2-enamide —— C22H24N2O4
(E)-2-cyano-3-(2,3,4-trimethoxyphenyl)-N-(2,4,6-trimethylphenyl)prop-2-enamide
—— (E)-3-(5-bromo-2-methoxyphenyl)-N-(4-fluoro-2-methylphenyl)prop-2-enamide —— C17H15BrFNO2
(E)-3-(5-bromo-2-methoxyphenyl)-N-(4-fluoro-2-methylphenyl)prop-2-enamide
—— ethyl (6S)-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H22F2N2O4S
ethyl (6S)-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3,4-dimethyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H22N2O3S
ethyl (6R)-3,4-dimethyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(5-bromothiophen-2-yl)-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C13H15BrN2O2S2
ethyl (6R)-6-(5-bromothiophen-2-yl)-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-[4-(cyanomethoxy)phenyl]-4-methyl-3-prop-2-enyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H21N3O3S
ethyl (6R)-6-[4-(cyanomethoxy)phenyl]-4-methyl-3-prop-2-enyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 2-[[(2R)-2-[4-(dimethylamino)pyridin-1-ium-1-yl]propanoyl]amino]-5-phenylthiophene-3-carboxylate —— C23H26N3O3S+
ethyl 2-[[(2R)-2-[4-(dimethylamino)pyridin-1-ium-1-yl]propanoyl]amino]-5-phenylthiophene-3-carboxylate
—— ethyl (6R)-6-[4-(cyanomethoxy)phenyl]-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C21H28N4O3S
ethyl (6R)-6-[4-(cyanomethoxy)phenyl]-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-2-cyano-N-(2-ethoxyphenyl)prop-2-enamide —— C23H21ClN4O2
(E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-2-cyano-N-(2-ethoxyphenyl)prop-2-enamide
—— (E)-2-cyano-N-(2,5-dichlorophenyl)-3-(4-methylsulfanylphenyl)prop-2-enamide —— C17H12Cl2N2OS
(E)-2-cyano-N-(2,5-dichlorophenyl)-3-(4-methylsulfanylphenyl)prop-2-enamide
—— ethyl (6S)-6-[3-(difluoromethoxy)-4-methoxyphenyl]-4-methyl-3-prop-2-enyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H22F2N2O4S
ethyl (6S)-6-[3-(difluoromethoxy)-4-methoxyphenyl]-4-methyl-3-prop-2-enyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl N-[2-[(2,2-dimethyl-3H-1-benzofuran-7-yl)oxy]acetyl]carbamate —— C15H19NO5
ethyl N-[2-[(2,2-dimethyl-3H-1-benzofuran-7-yl)oxy]acetyl]carbamate
—— (E)-3-(4-hydroxy-3-methoxyphenyl)-N-[2-[2-[(2R)-1-methylpiperidin-2-yl]ethyl]phenyl]prop-2-enamide —— C24H30N2O3
(E)-3-(4-hydroxy-3-methoxyphenyl)-N-[2-[2-[(2R)-1-methylpiperidin-2-yl]ethyl]phenyl]prop-2-enamide
—— ethyl (6R)-3-[3-(dimethylamino)propyl]-6-(3-fluorophenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H26FN3O2S
ethyl (6R)-3-[3-(dimethylamino)propyl]-6-(3-fluorophenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(3,4-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H25F2N3O2S
ethyl (6R)-6-(3,4-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-2-cyano-3-(3,5-ditert-butyl-4-hydroxyphenyl)-N-prop-2-enylprop-2-enamide —— C21H28N2O2
(E)-2-cyano-3-(3,5-ditert-butyl-4-hydroxyphenyl)-N-prop-2-enylprop-2-enamide
—— ethyl (4S)-4-ethyl-2-oxo-6-[[[(S)-phenyl(thiophen-2-yl)methyl]amino]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H25N3O3S
ethyl (4S)-4-ethyl-2-oxo-6-[[[(S)-phenyl(thiophen-2-yl)methyl]amino]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-(4-fluoro-2-methylphenyl)prop-2-enamide —— C19H19ClFNO3
(E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-(4-fluoro-2-methylphenyl)prop-2-enamide
—— ethyl (6S)-6-(3,4-difluorophenyl)-3-[(2S)-1-methoxypropan-2-yl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H22F2N2O3S
ethyl (6S)-6-(3,4-difluorophenyl)-3-[(2S)-1-methoxypropan-2-yl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(4-hydroxy-3-methoxyphenyl)-N-[2-[2-[(2S)-1-methylpiperidin-2-yl]ethyl]phenyl]prop-2-enamide —— C24H30N2O3
(E)-3-(4-hydroxy-3-methoxyphenyl)-N-[2-[2-[(2S)-1-methylpiperidin-2-yl]ethyl]phenyl]prop-2-enamide
—— (E)-2-cyano-N-prop-2-enyl-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C16H18N2O4
(E)-2-cyano-N-prop-2-enyl-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(4-hydroxyphenyl)-N-[2-[2-[(2R)-1-methylpiperidin-2-yl]ethyl]phenyl]prop-2-enamide —— C23H28N2O2
(E)-3-(4-hydroxyphenyl)-N-[2-[2-[(2R)-1-methylpiperidin-2-yl]ethyl]phenyl]prop-2-enamide
—— (E)-2-cyano-3-(2-morpholin-4-yl-4-phenyl-1,3-thiazol-5-yl)-N-prop-2-enylprop-2-enamide —— C20H20N4O2S
(E)-2-cyano-3-(2-morpholin-4-yl-4-phenyl-1,3-thiazol-5-yl)-N-prop-2-enylprop-2-enamide
—— (E)-3-(4-hydroxyphenyl)-N-[2-[2-[(2S)-1-methylpiperidin-2-yl]ethyl]phenyl]prop-2-enamide —— C23H28N2O2
(E)-3-(4-hydroxyphenyl)-N-[2-[2-[(2S)-1-methylpiperidin-2-yl]ethyl]phenyl]prop-2-enamide
—— (E)-N-(4-fluoro-2-methylphenyl)-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enamide —— C20H20FNO3
(E)-N-(4-fluoro-2-methylphenyl)-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enamide
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-[2-(3,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C19H17ClN4O3S
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-[2-(3,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-2-cyano-3-(3,4-difluorophenyl)-N-prop-2-enylprop-2-enamide —— C13H10F2N2O
(E)-2-cyano-3-(3,4-difluorophenyl)-N-prop-2-enylprop-2-enamide
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-naphthalen-1-ylprop-2-enamide —— C19H11ClN4OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-naphthalen-1-ylprop-2-enamide
—— (E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-2-cyano-N-(3-ethoxypropyl)prop-2-enamide —— C19H21ClN4O2
(E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-2-cyano-N-(3-ethoxypropyl)prop-2-enamide
—— (E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide —— C15H17ClN4O3S
(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide
—— ethyl (6S)-6-(3,4-difluorophenyl)-3-(4-methoxyphenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C21H20F2N2O3S
ethyl (6S)-6-(3,4-difluorophenyl)-3-(4-methoxyphenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-2-cyano-3-[1-[(2,6-dichlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-prop-2-enylprop-2-enamide —— C19H18Cl2N4O
(E)-2-cyano-3-[1-[(2,6-dichlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-prop-2-enylprop-2-enamide
—— (E)-3-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]-2-cyano-N-(3-ethoxypropyl)prop-2-enamide —— C19H20Cl2N4O2
(E)-3-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]-2-cyano-N-(3-ethoxypropyl)prop-2-enamide
—— (E)-3-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide —— C17H14Cl2N4O
(E)-3-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide
—— (E)-3-[5-chloro-1-(3-chlorophenyl)-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C20H18Cl2N6
(E)-3-[5-chloro-1-(3-chlorophenyl)-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide —— C19H19ClN4O
(E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(3-bromo-4-methoxyphenyl)but-3-enoate —— C18H13BrNO3S-
(E)-3-(1,3-benzothiazol-2-yl)-4-(3-bromo-4-methoxyphenyl)but-3-enoate
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-prop-2-enylprop-2-enamide —— C12H9ClN4OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-prop-2-enylprop-2-enamide
—— (E)-N-(2-chlorophenyl)-2-cyano-3-(3,4-difluorophenyl)prop-2-enamide —— C16H9ClF2N2O
(E)-N-(2-chlorophenyl)-2-cyano-3-(3,4-difluorophenyl)prop-2-enamide
—— (E)-2-cyano-3-(3,4-difluorophenyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C20H18F2N2O3
(E)-2-cyano-3-(3,4-difluorophenyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]prop-2-enamide