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—— (E)-N-[(2R)-2-(2,4-difluorophenyl)-2-hydroxypropyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C16H16F2N2O2S
(E)-N-[(2R)-2-(2,4-difluorophenyl)-2-hydroxypropyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (E)-N-[(2R)-2-hydroxy-2-thiophen-3-ylpropyl]-3-(4-nitrophenyl)prop-2-enamide —— C16H16N2O4S
(E)-N-[(2R)-2-hydroxy-2-thiophen-3-ylpropyl]-3-(4-nitrophenyl)prop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[(2R)-2-hydroxy-2-thiophen-3-ylpropyl]prop-2-enamide —— C18H20N2O3S
(E)-3-(4-acetamidophenyl)-N-[(2R)-2-hydroxy-2-thiophen-3-ylpropyl]prop-2-enamide
—— (E)-N-[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]-3-(4-nitrophenyl)prop-2-enamide —— C16H16N2O4S
(E)-N-[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]-3-(4-nitrophenyl)prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(2S)-2-methyl-3-pyrrolidin-1-ylpropyl]prop-2-enamide —— C22H28N4O
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(2S)-2-methyl-3-pyrrolidin-1-ylpropyl]prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(2R)-2-methyl-3-pyrrolidin-1-ylpropyl]prop-2-enamide —— C22H28N4O
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(2R)-2-methyl-3-pyrrolidin-1-ylpropyl]prop-2-enamide
—— (E)-3-(3-fluorophenyl)-N-[(2S)-2-hydroxy-2-methyl-3-morpholin-4-ylpropyl]prop-2-enamide —— C17H23FN2O3
(E)-3-(3-fluorophenyl)-N-[(2S)-2-hydroxy-2-methyl-3-morpholin-4-ylpropyl]prop-2-enamide
—— (E)-3-(3-fluorophenyl)-N-[(2S)-2-hydroxy-2-(5-methylfuran-2-yl)propyl]prop-2-enamide —— C17H18FNO3
(E)-3-(3-fluorophenyl)-N-[(2S)-2-hydroxy-2-(5-methylfuran-2-yl)propyl]prop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[(2S)-2-hydroxy-2-thiophen-2-ylpropyl]prop-2-enamide —— C18H20N2O3S
(E)-3-(4-acetamidophenyl)-N-[(2S)-2-hydroxy-2-thiophen-2-ylpropyl]prop-2-enamide
—— (E)-3-(3-fluorophenyl)-N-[(2R)-2-hydroxy-2-methyl-3-morpholin-4-ylpropyl]prop-2-enamide —— C17H23FN2O3
(E)-3-(3-fluorophenyl)-N-[(2R)-2-hydroxy-2-methyl-3-morpholin-4-ylpropyl]prop-2-enamide
—— (E)-N-[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-3-(2-methoxyphenyl)prop-2-enamide —— C17H21N3O3
(E)-N-[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-3-(2-methoxyphenyl)prop-2-enamide
—— ethyl 1-ethyl-4-[(E)-3-[[(2R)-2-hydroxy-2-methyl-3-morpholin-4-ylpropyl]amino]-3-oxoprop-1-enyl]-2,5-dimethylpyrrole-3-carboxylate —— C22H35N3O5
ethyl 1-ethyl-4-[(E)-3-[[(2R)-2-hydroxy-2-methyl-3-morpholin-4-ylpropyl]amino]-3-oxoprop-1-enyl]-2,5-dimethylpyrrole-3-carboxylate
—— (E)-N-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-3-thiophen-3-ylprop-2-enamide —— C14H17N3O2S
(E)-N-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-3-thiophen-3-ylprop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[(2R)-2-hydroxy-2-thiophen-2-ylpropyl]prop-2-enamide —— C18H20N2O3S
(E)-3-(4-acetamidophenyl)-N-[(2R)-2-hydroxy-2-thiophen-2-ylpropyl]prop-2-enamide
—— ethyl N-[(2R)-1-[4-[(4-benzylpiperazin-1-yl)methyl]anilino]-3-methyl-1-oxobutan-2-yl]carbamate —— C26H36N4O3
ethyl N-[(2R)-1-[4-[(4-benzylpiperazin-1-yl)methyl]anilino]-3-methyl-1-oxobutan-2-yl]carbamate
—— ethyl N-[(2S)-1-[4-[(4-benzylpiperazin-1-yl)methyl]anilino]-3-methyl-1-oxobutan-2-yl]carbamate —— C26H36N4O3
ethyl N-[(2S)-1-[4-[(4-benzylpiperazin-1-yl)methyl]anilino]-3-methyl-1-oxobutan-2-yl]carbamate
—— ethyl (2S)-1-[2-(4-cyanobenzoyl)oxyacetyl]piperidine-2-carboxylate —— C18H20N2O5
ethyl (2S)-1-[2-(4-cyanobenzoyl)oxyacetyl]piperidine-2-carboxylate
—— ethyl (2R)-1-[2-(8-chloro-1,3-dimethyl-2,6-dioxopurin-7-yl)acetyl]piperidine-2-carboxylate —— C17H22ClN5O5
ethyl (2R)-1-[2-(8-chloro-1,3-dimethyl-2,6-dioxopurin-7-yl)acetyl]piperidine-2-carboxylate
—— Ethyl 4-carbamoyl-5-[[2-[2-(4-methoxyphenyl)acetyl]oxyacetyl]amino]-2-methylfuran-3-carboxylate —— C20H22N2O8
Ethyl 4-carbamoyl-5-[[2-[2-(4-methoxyphenyl)acetyl]oxyacetyl]amino]-2-methylfuran-3-carboxylate
—— ethyl 1-[2-oxo-2-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]ethyl]piperidine-4-carboxylate —— C18H26N2O3S
ethyl 1-[2-oxo-2-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]ethyl]piperidine-4-carboxylate
—— ethyl 1-[2-oxo-2-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]ethyl]piperidine-4-carboxylate —— C18H26N2O3S
ethyl 1-[2-oxo-2-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]ethyl]piperidine-4-carboxylate
—— ethyl 4-[2-[(2S)-2-methylpiperidin-1-yl]ethylcarbamoylamino]-1H-pyrrole-2-carboxylate —— C16H26N4O3
ethyl 4-[2-[(2S)-2-methylpiperidin-1-yl]ethylcarbamoylamino]-1H-pyrrole-2-carboxylate
—— ethyl (3S)-1-[2-(2,3-dihydro-1,4-benzothiazin-4-yl)-2-oxoethyl]piperidine-3-carboxylate —— C18H24N2O3S
ethyl (3S)-1-[2-(2,3-dihydro-1,4-benzothiazin-4-yl)-2-oxoethyl]piperidine-3-carboxylate
—— ethyl 4-[2-[(2R)-2-methylpiperidin-1-yl]ethylcarbamoylamino]-1H-pyrrole-2-carboxylate —— C16H26N4O3
ethyl 4-[2-[(2R)-2-methylpiperidin-1-yl]ethylcarbamoylamino]-1H-pyrrole-2-carboxylate
—— ethyl (3R)-1-[2-(2,3-dihydro-1,4-benzothiazin-4-yl)-2-oxoethyl]piperidine-3-carboxylate —— C18H24N2O3S
ethyl (3R)-1-[2-(2,3-dihydro-1,4-benzothiazin-4-yl)-2-oxoethyl]piperidine-3-carboxylate
—— ethyl 5-[[(3S,5R)-3,5-dimethylmorpholin-4-yl]methyl]-2-phenyl-1,3-oxazole-4-carboxylate —— C19H24N2O4
ethyl 5-[[(3S,5R)-3,5-dimethylmorpholin-4-yl]methyl]-2-phenyl-1,3-oxazole-4-carboxylate
—— ethyl 5-[[(3R,5R)-3,5-dimethylmorpholin-4-yl]methyl]-2-phenyl-1,3-oxazole-4-carboxylate —— C19H24N2O4
ethyl 5-[[(3R,5R)-3,5-dimethylmorpholin-4-yl]methyl]-2-phenyl-1,3-oxazole-4-carboxylate
—— ethyl 5-[[(3S,5S)-3,5-dimethylmorpholin-4-yl]methyl]-2-phenyl-1,3-oxazole-4-carboxylate —— C19H24N2O4
ethyl 5-[[(3S,5S)-3,5-dimethylmorpholin-4-yl]methyl]-2-phenyl-1,3-oxazole-4-carboxylate
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide —— C21H23N3O3
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide
—— ethyl (2S)-1-[2-(3-methoxynaphthalene-2-carbonyl)oxyacetyl]piperidine-2-carboxylate —— C22H25NO6
ethyl (2S)-1-[2-(3-methoxynaphthalene-2-carbonyl)oxyacetyl]piperidine-2-carboxylate
—— (E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-(1,3-benzoxazol-2-yl)prop-2-enamide —— C19H16N4O2
(E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-(1,3-benzoxazol-2-yl)prop-2-enamide
—— ethyl (2R)-1-[2-[2-(1,3-dioxoisoindol-2-yl)acetyl]oxyacetyl]piperidine-2-carboxylate —— C20H22N2O7
ethyl (2R)-1-[2-[2-(1,3-dioxoisoindol-2-yl)acetyl]oxyacetyl]piperidine-2-carboxylate
—— (E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide —— C21H23N3O3
(E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(1,3-benzoxazol-2-yl)prop-2-enamide —— C19H16N4O2
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(1,3-benzoxazol-2-yl)prop-2-enamide
—— (E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C20H21N3O3
(E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(4-nitrophenyl)prop-2-enamide —— C18H16N4O3
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(4-nitrophenyl)prop-2-enamide
—— Ethyl 4-carbamoyl-5-[[2-(3,3-dimethylbutanoyloxy)acetyl]amino]-2-methylfuran-3-carboxylate —— C17H24N2O7
Ethyl 4-carbamoyl-5-[[2-(3,3-dimethylbutanoyloxy)acetyl]amino]-2-methylfuran-3-carboxylate
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C20H21N3O3
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— Ethyl 4-carbamoyl-5-[[2-(2,4-difluorobenzoyl)oxyacetyl]amino]-2-methylfuran-3-carboxylate —— C18H16F2N2O7
Ethyl 4-carbamoyl-5-[[2-(2,4-difluorobenzoyl)oxyacetyl]amino]-2-methylfuran-3-carboxylate
—— ethyl (2S)-1-[2-[2-(1,3-dioxoisoindol-2-yl)acetyl]oxyacetyl]piperidine-2-carboxylate —— C20H22N2O7
ethyl (2S)-1-[2-[2-(1,3-dioxoisoindol-2-yl)acetyl]oxyacetyl]piperidine-2-carboxylate
—— ethyl (4R)-4-(furan-2-yl)-6-[[4-(1,2-oxazol-3-ylmethyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H25N5O5
ethyl (4R)-4-(furan-2-yl)-6-[[4-(1,2-oxazol-3-ylmethyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(furan-2-yl)-6-[[4-(1,2-oxazol-3-ylmethyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H25N5O5
ethyl (4S)-4-(furan-2-yl)-6-[[4-(1,2-oxazol-3-ylmethyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2S)-1-[2-(3-methyl-4-nitrobenzoyl)oxyacetyl]piperidine-2-carboxylate —— C18H22N2O7
ethyl (2S)-1-[2-(3-methyl-4-nitrobenzoyl)oxyacetyl]piperidine-2-carboxylate
—— ethyl (2R)-1-[2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]piperidine-2-carboxylate —— C12H18N4O3S2
ethyl (2R)-1-[2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]piperidine-2-carboxylate
—— Ethyl 2-[[2-[methyl-[(4-methylsulfanylphenyl)methyl]amino]acetyl]amino]benzoate —— C20H24N2O3S
Ethyl 2-[[2-[methyl-[(4-methylsulfanylphenyl)methyl]amino]acetyl]amino]benzoate
—— Ethyl 4-carbamoyl-5-[[2-[2-(4-fluorophenyl)acetyl]oxyacetyl]amino]-2-methylfuran-3-carboxylate —— C19H19FN2O7
Ethyl 4-carbamoyl-5-[[2-[2-(4-fluorophenyl)acetyl]oxyacetyl]amino]-2-methylfuran-3-carboxylate
—— ethyl (4S)-4-ethyl-6-[[methyl-[(4-methylsulfanylphenyl)methyl]amino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H27N3O3S
ethyl (4S)-4-ethyl-6-[[methyl-[(4-methylsulfanylphenyl)methyl]amino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2,5-dimethyl-4-[2-(4-oxopentanoyloxy)acetyl]-1H-pyrrole-3-carboxylate —— C16H21NO6
ethyl 2,5-dimethyl-4-[2-(4-oxopentanoyloxy)acetyl]-1H-pyrrole-3-carboxylate
—— Ethyl 3-[[2-(4-oxopentanoyloxy)acetyl]amino]-5-phenylthiophene-2-carboxylate —— C20H21NO6S
Ethyl 3-[[2-(4-oxopentanoyloxy)acetyl]amino]-5-phenylthiophene-2-carboxylate
—— (E)-3-(2-tert-butyl-1,3-thiazol-5-yl)-1-[(4S)-4-hydroxy-5,8-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]prop-2-en-1-one —— C21H26N2O4S
(E)-3-(2-tert-butyl-1,3-thiazol-5-yl)-1-[(4S)-4-hydroxy-5,8-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]prop-2-en-1-one