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—— (E)-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-[1-(furan-2-ylmethyl)-2,5-dimethylpyrrol-3-yl]-N-methylprop-2-enamide —— C24H26N2O4
(E)-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-[1-(furan-2-ylmethyl)-2,5-dimethylpyrrol-3-yl]-N-methylprop-2-enamide
—— (E)-N-butyl-3-(6-methoxynaphthalen-2-yl)prop-2-enamide —— C18H21NO2
(E)-N-butyl-3-(6-methoxynaphthalen-2-yl)prop-2-enamide
—— Ethyl 1-[6-(4-fluorophenyl)thieno[3,2-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C20H20FN3O2S
Ethyl 1-[6-(4-fluorophenyl)thieno[3,2-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-(2-fluorophenyl)prop-2-enamide —— C16H13F2NO2
(E)-3-(3-fluoro-4-methoxyphenyl)-N-(2-fluorophenyl)prop-2-enamide
—— ethyl (3R)-1-[2-(benzenesulfonamido)ethyl]piperidine-3-carboxylate —— C16H24N2O4S
ethyl (3R)-1-[2-(benzenesulfonamido)ethyl]piperidine-3-carboxylate
—— (E)-N-[3-(3-ethyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-3-(4-propan-2-ylphenyl)prop-2-enamide —— C23H23N5OS
(E)-N-[3-(3-ethyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-3-(4-propan-2-ylphenyl)prop-2-enamide
—— ethyl 4-[[(2S)-1-cyanopropan-2-yl]-methylamino]-5-methyl-2-(phenylsulfanylmethyl)thieno[2,3-d]pyrimidine-6-carboxylate —— C22H24N4O2S2
ethyl 4-[[(2S)-1-cyanopropan-2-yl]-methylamino]-5-methyl-2-(phenylsulfanylmethyl)thieno[2,3-d]pyrimidine-6-carboxylate
—— (E)-N-(3-chloro-2-methylphenyl)-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide —— C17H13ClN2O5
(E)-N-(3-chloro-2-methylphenyl)-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide
—— (E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-N-(2-fluorophenyl)prop-2-enamide —— C17H19ClFN3O
(E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-N-(2-fluorophenyl)prop-2-enamide
—— (E)-3-(4-chlorophenyl)-N-[3-(3-ethyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]prop-2-enamide —— C20H16ClN5OS
(E)-3-(4-chlorophenyl)-N-[3-(3-ethyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]prop-2-enamide
—— ethyl 2-[[(1R,2S,4S)-bicyclo[2.2.1]heptane-2-carbonyl]-ethylamino]-4-methyl-1,3-thiazole-5-carboxylate —— C17H24N2O3S
ethyl 2-[[(1R,2S,4S)-bicyclo[2.2.1]heptane-2-carbonyl]-ethylamino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (3S)-1-[2-(benzenesulfonamido)ethyl]piperidine-3-carboxylate —— C16H24N2O4S
ethyl (3S)-1-[2-(benzenesulfonamido)ethyl]piperidine-3-carboxylate
—— (E)-N-[3-(3-ethyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-3-(furan-2-yl)prop-2-enamide —— C18H15N5O2S
(E)-N-[3-(3-ethyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl N-[3-[[4-(diethylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate —— C20H25N3O5S
ethyl N-[3-[[4-(diethylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate
—— (E)-1-[(2S)-2-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C24H22N4OS
(E)-1-[(2S)-2-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (E)-1-(4-acetylpiperazin-1-yl)-3-(3-ethoxy-4-phenylmethoxyphenyl)prop-2-en-1-one —— C24H28N2O4
(E)-1-(4-acetylpiperazin-1-yl)-3-(3-ethoxy-4-phenylmethoxyphenyl)prop-2-en-1-one
—— ethyl N-[4-[[4-(diethylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate —— C20H25N3O5S
ethyl N-[4-[[4-(diethylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate
—— Ethyl 4-carbamoyl-5-[[2-(2,6-difluorobenzoyl)oxyacetyl]amino]-2-methylfuran-3-carboxylate —— C18H16F2N2O7
Ethyl 4-carbamoyl-5-[[2-(2,6-difluorobenzoyl)oxyacetyl]amino]-2-methylfuran-3-carboxylate
—— ethyl 4-[[(2R)-1-cyanopropan-2-yl]-methylamino]-5-methyl-2-(phenylsulfanylmethyl)thieno[2,3-d]pyrimidine-6-carboxylate —— C22H24N4O2S2
ethyl 4-[[(2R)-1-cyanopropan-2-yl]-methylamino]-5-methyl-2-(phenylsulfanylmethyl)thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl 2-[[(1R,2R,4S)-bicyclo[2.2.1]heptane-2-carbonyl]-ethylamino]-4-methyl-1,3-thiazole-5-carboxylate —— C17H24N2O3S
ethyl 2-[[(1R,2R,4S)-bicyclo[2.2.1]heptane-2-carbonyl]-ethylamino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (1S)-1-[2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-oxocyclopentane-1-carboxylate —— C19H22F2N4O4S
ethyl (1S)-1-[2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-oxocyclopentane-1-carboxylate
—— Ethyl 4-carbamoyl-2-methyl-5-[[2-(2-methylbenzoyl)oxyacetyl]amino]furan-3-carboxylate —— C19H20N2O7
Ethyl 4-carbamoyl-2-methyl-5-[[2-(2-methylbenzoyl)oxyacetyl]amino]furan-3-carboxylate
—— ethyl (1R)-1-[2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-oxocyclopentane-1-carboxylate —— C19H22F2N4O4S
ethyl (1R)-1-[2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-oxocyclopentane-1-carboxylate
—— ethyl (1S)-1-[2-[3-cyano-6-methyl-4-(trifluoromethyl)pyridin-2-yl]sulfanylethyl]-2-oxocyclopentane-1-carboxylate —— C18H19F3N2O3S
ethyl (1S)-1-[2-[3-cyano-6-methyl-4-(trifluoromethyl)pyridin-2-yl]sulfanylethyl]-2-oxocyclopentane-1-carboxylate
—— ethyl (1R)-1-[2-[3-cyano-6-methyl-4-(trifluoromethyl)pyridin-2-yl]sulfanylethyl]-2-oxocyclopentane-1-carboxylate —— C18H19F3N2O3S
ethyl (1R)-1-[2-[3-cyano-6-methyl-4-(trifluoromethyl)pyridin-2-yl]sulfanylethyl]-2-oxocyclopentane-1-carboxylate
—— ethyl (1R)-2-oxo-1-[2-[[4-(2-thiophen-2-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]cyclopentane-1-carboxylate —— C18H23N3O3S2
ethyl (1R)-2-oxo-1-[2-[[4-(2-thiophen-2-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]cyclopentane-1-carboxylate
—— (E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2R)-2-methyl-3-pyrrolidin-1-ylpropyl]prop-2-enamide —— C16H25ClN4O
(E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2R)-2-methyl-3-pyrrolidin-1-ylpropyl]prop-2-enamide
—— ethyl 1-[[(1R)-4-fluoro-2,3-dihydro-1H-inden-1-yl]carbamoyl]cyclopropane-1-carboxylate —— C16H18FNO3
ethyl 1-[[(1R)-4-fluoro-2,3-dihydro-1H-inden-1-yl]carbamoyl]cyclopropane-1-carboxylate
—— ethyl 1-[[(1S)-4-fluoro-2,3-dihydro-1H-inden-1-yl]carbamoyl]cyclopropane-1-carboxylate —— C16H18FNO3
ethyl 1-[[(1S)-4-fluoro-2,3-dihydro-1H-inden-1-yl]carbamoyl]cyclopropane-1-carboxylate
—— ethyl (1S)-1-[2-[1-(2,3-dimethylphenyl)tetrazol-5-yl]sulfanylethyl]-2-oxocyclopentane-1-carboxylate —— C19H24N4O3S
ethyl (1S)-1-[2-[1-(2,3-dimethylphenyl)tetrazol-5-yl]sulfanylethyl]-2-oxocyclopentane-1-carboxylate
—— (E)-N-[(2S)-2-methyl-3-pyrrolidin-1-ylpropyl]-3-pyridin-3-ylprop-2-enamide —— C16H23N3O
(E)-N-[(2S)-2-methyl-3-pyrrolidin-1-ylpropyl]-3-pyridin-3-ylprop-2-enamide
—— (E)-N-[(2R)-2-methyl-3-pyrrolidin-1-ylpropyl]-3-pyridin-3-ylprop-2-enamide —— C16H23N3O
(E)-N-[(2R)-2-methyl-3-pyrrolidin-1-ylpropyl]-3-pyridin-3-ylprop-2-enamide
—— ethyl (1S)-2-oxo-1-[2-[[4-(2-thiophen-2-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]cyclopentane-1-carboxylate —— C18H23N3O3S2
ethyl (1S)-2-oxo-1-[2-[[4-(2-thiophen-2-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]cyclopentane-1-carboxylate
—— ethyl (1R)-1-[2-[1-(2,3-dimethylphenyl)tetrazol-5-yl]sulfanylethyl]-2-oxocyclopentane-1-carboxylate —— C19H24N4O3S
ethyl (1R)-1-[2-[1-(2,3-dimethylphenyl)tetrazol-5-yl]sulfanylethyl]-2-oxocyclopentane-1-carboxylate
—— (E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2S)-2-methyl-3-pyrrolidin-1-ylpropyl]prop-2-enamide —— C16H25ClN4O
(E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2S)-2-methyl-3-pyrrolidin-1-ylpropyl]prop-2-enamide
—— (E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2R)-2-hydroxy-2-thiophen-2-ylpropyl]prop-2-enamide —— C15H18ClN3O2S
(E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2R)-2-hydroxy-2-thiophen-2-ylpropyl]prop-2-enamide
—— ethyl (1S,2R)-2-cyano-1,2,3,4-tetrahydronaphthalene-1-carboxylate —— C14H15NO2
ethyl (1S,2R)-2-cyano-1,2,3,4-tetrahydronaphthalene-1-carboxylate
—— (E)-N-[(2S)-2-(2,4-difluorophenyl)-2-hydroxypropyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C16H16F2N2O2S
(E)-N-[(2S)-2-(2,4-difluorophenyl)-2-hydroxypropyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (E)-3-(4-chlorophenyl)-N-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]prop-2-enamide —— C16H18ClN3O2
(E)-3-(4-chlorophenyl)-N-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-N-[(2R)-2-hydroxy-2-(5-methylfuran-2-yl)propyl]prop-2-enamide —— C18H18N2O3S
(E)-3-(1,3-benzothiazol-2-yl)-N-[(2R)-2-hydroxy-2-(5-methylfuran-2-yl)propyl]prop-2-enamide
—— ethyl 1-ethyl-4-[(E)-3-[[(2S)-2-hydroxy-2-methyl-3-morpholin-4-ylpropyl]amino]-3-oxoprop-1-enyl]-2,5-dimethylpyrrole-3-carboxylate —— C22H35N3O5
ethyl 1-ethyl-4-[(E)-3-[[(2S)-2-hydroxy-2-methyl-3-morpholin-4-ylpropyl]amino]-3-oxoprop-1-enyl]-2,5-dimethylpyrrole-3-carboxylate
—— (E)-3-(3-fluorophenyl)-N-[(2R)-2-hydroxy-2-(5-methylfuran-2-yl)propyl]prop-2-enamide —— C17H18FNO3
(E)-3-(3-fluorophenyl)-N-[(2R)-2-hydroxy-2-(5-methylfuran-2-yl)propyl]prop-2-enamide
—— (E)-N-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-3-(2-methoxyphenyl)prop-2-enamide —— C17H21N3O3
(E)-N-[(2R)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-3-(2-methoxyphenyl)prop-2-enamide
—— Ethyl 4-carbamoyl-2-methyl-5-[(2-pyrimidin-2-ylsulfanylacetyl)amino]furan-3-carboxylate —— C15H16N4O5S
Ethyl 4-carbamoyl-2-methyl-5-[(2-pyrimidin-2-ylsulfanylacetyl)amino]furan-3-carboxylate
—— (E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2S)-2-hydroxy-2-thiophen-2-ylpropyl]prop-2-enamide —— C15H18ClN3O2S
(E)-3-(5-chloro-1,3-dimethylpyrazol-4-yl)-N-[(2S)-2-hydroxy-2-thiophen-2-ylpropyl]prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-N-[(2S)-2-hydroxy-2-(5-methylfuran-2-yl)propyl]prop-2-enamide —— C18H18N2O3S
(E)-3-(1,3-benzothiazol-2-yl)-N-[(2S)-2-hydroxy-2-(5-methylfuran-2-yl)propyl]prop-2-enamide
—— (E)-N-[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-3-thiophen-3-ylprop-2-enamide —— C14H17N3O2S
(E)-N-[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]-3-thiophen-3-ylprop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]prop-2-enamide —— C18H20N2O3S
(E)-3-(4-acetamidophenyl)-N-[(2S)-2-hydroxy-2-thiophen-3-ylpropyl]prop-2-enamide
—— (E)-3-(4-chlorophenyl)-N-[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]prop-2-enamide —— C16H18ClN3O2
(E)-3-(4-chlorophenyl)-N-[(2S)-2-hydroxy-2-(1-methylpyrazol-4-yl)propyl]prop-2-enamide
—— ethyl (1S,2S)-2-cyano-1,2,3,4-tetrahydronaphthalene-1-carboxylate —— C14H15NO2
ethyl (1S,2S)-2-cyano-1,2,3,4-tetrahydronaphthalene-1-carboxylate