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—— ethyl 2,4-dimethyl-5-[(2S)-2-[4-(5-methylthiophen-2-yl)-4-oxobutanoyl]oxypropanoyl]-1H-pyrrole-3-carboxylate —— C21H25NO6S
ethyl 2,4-dimethyl-5-[(2S)-2-[4-(5-methylthiophen-2-yl)-4-oxobutanoyl]oxypropanoyl]-1H-pyrrole-3-carboxylate
—— ethyl (4S)-4-ethyl-6-[[4-(5-methylthiophen-2-yl)-4-oxobutanoyl]oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O6S
ethyl (4S)-4-ethyl-6-[[4-(5-methylthiophen-2-yl)-4-oxobutanoyl]oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2E,5S)-2-[[3-bromo-4-[(2-chlorophenyl)methoxy]-5-methoxyphenyl]methylidene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31BrClN3O5S
ethyl (2E,5S)-2-[[3-bromo-4-[(2-chlorophenyl)methoxy]-5-methoxyphenyl]methylidene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-4-[[(3S)-1-(4-bromophenyl)-2,5-dioxopyrrolidin-3-yl]-[2-(3,4-dimethoxyphenyl)ethyl]amino]-4-oxobut-2-enoate —— C24H22BrN2O7-
(E)-4-[[(3S)-1-(4-bromophenyl)-2,5-dioxopyrrolidin-3-yl]-[2-(3,4-dimethoxyphenyl)ethyl]amino]-4-oxobut-2-enoate
—— ethyl (4S)-6-[3-(1,3-benzoxazol-2-yl)propanoyloxymethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H23N3O6
ethyl (4S)-6-[3-(1,3-benzoxazol-2-yl)propanoyloxymethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2E,5R)-2-[[3-bromo-4-[(2-chlorophenyl)methoxy]-5-methoxyphenyl]methylidene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31BrClN3O5S
ethyl (2E,5R)-2-[[3-bromo-4-[(2-chlorophenyl)methoxy]-5-methoxyphenyl]methylidene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 5-[(2R)-2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C22H24N2O6
ethyl 5-[(2R)-2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— Ethyl 4-[(4-ethylbenzoyl)hydrazinylidene]piperidine-1-carboxylate —— C17H23N3O3
Ethyl 4-[(4-ethylbenzoyl)hydrazinylidene]piperidine-1-carboxylate
—— Ethyl 5-amino-3-[3-(1,3-benzoxazol-2-yl)propanoyloxymethyl]-4-cyanothiophene-2-carboxylate —— C19H17N3O5S
Ethyl 5-amino-3-[3-(1,3-benzoxazol-2-yl)propanoyloxymethyl]-4-cyanothiophene-2-carboxylate
—— ethyl (2E,5R)-2-[(2-bromo-4,5-dimethoxyphenyl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H27BrN2O7S
ethyl (2E,5R)-2-[(2-bromo-4,5-dimethoxyphenyl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[(2,5-dimethyl-1-pyridin-3-ylpyrrol-3-yl)methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H34N4O4S
ethyl (2E,5S)-2-[(2,5-dimethyl-1-pyridin-3-ylpyrrol-3-yl)methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[(2-bromo-4,5-dimethoxyphenyl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H25BrN2O6S
ethyl (2E,5R)-2-[(2-bromo-4,5-dimethoxyphenyl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[4-(diethylamino)-2-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H39N3O5S
ethyl (2Z,5R)-2-[[4-(diethylamino)-2-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-5-[4-(dimethylamino)phenyl]-2-[[2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32FN3O5S
ethyl (2Z,5R)-5-[4-(dimethylamino)phenyl]-2-[[2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H30N2O7S
ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[(2,5-dimethyl-1-pyridin-3-ylpyrrol-3-yl)methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H34N4O4S
ethyl (2E,5R)-2-[(2,5-dimethyl-1-pyridin-3-ylpyrrol-3-yl)methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[(2-bromo-4,5-dimethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H23BrN2O7S
ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[(2-bromo-4,5-dimethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-5-[4-(dimethylamino)phenyl]-2-[[2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32FN3O5S
ethyl (2Z,5S)-5-[4-(dimethylamino)phenyl]-2-[[2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[(3-bromo-5-methoxy-4-prop-2-enoxyphenyl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H24BrClN2O5S
ethyl (2E,5S)-2-[(3-bromo-5-methoxy-4-prop-2-enoxyphenyl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H22BrClN2O5S
ethyl (2E,5S)-2-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-5-(3-bromo-4-methoxyphenyl)-7-methyl-3-oxo-2-[[5-[3-(trifluoromethyl)phenyl]furan-2-yl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H22BrF3N2O5S
ethyl (2Z,5S)-5-(3-bromo-4-methoxyphenyl)-7-methyl-3-oxo-2-[[5-[3-(trifluoromethyl)phenyl]furan-2-yl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[(4R)-2-amino-3-cyano-7,7-dimethyl-4-(3-nitrophenyl)-5-oxo-6,8-dihydro-4H-quinolin-1-yl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C30H32N4O5S
ethyl 2-[(4R)-2-amino-3-cyano-7,7-dimethyl-4-(3-nitrophenyl)-5-oxo-6,8-dihydro-4H-quinolin-1-yl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— ethyl (5S)-4-(4-bromophenyl)-2',4'-diphenylspiro[1,3,4-thiadiazole-5,1'-phthalazine]-2-carboxylate —— C30H23BrN4O2S
ethyl (5S)-4-(4-bromophenyl)-2',4'-diphenylspiro[1,3,4-thiadiazole-5,1'-phthalazine]-2-carboxylate
—— ethyl (2E,5S)-2-[[5-(2-chloro-4-nitrophenyl)furan-2-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H22ClN3O7S
ethyl (2E,5S)-2-[[5-(2-chloro-4-nitrophenyl)furan-2-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[3-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31FN2O6S
ethyl (2Z,5S)-2-[[3-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-(adamantane-1-carbonyloxy)-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H38N2O7S
ethyl (2Z,5S)-2-[[4-(adamantane-1-carbonyloxy)-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-(3-bromobenzoyl)oxy-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H27BrN2O7S
ethyl (2Z,5S)-2-[[4-(3-bromobenzoyl)oxy-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31FN2O6S
ethyl (2Z,5S)-2-[[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-[(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)oxy]-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H39N7O8S
ethyl (2Z,5S)-2-[[4-[(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)oxy]-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[(E)-3-(4-bromophenyl)prop-2-enylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H23BrN2O4S
ethyl (2Z,5S)-2-[(E)-3-(4-bromophenyl)prop-2-enylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[3-ethoxy-4-[(2-nitrophenyl)methoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31N3O8S
ethyl (2Z,5R)-2-[[3-ethoxy-4-[(2-nitrophenyl)methoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (4S)-2-amino-1-(4-bromophenyl)-4-(4-chlorophenyl)-5-oxo-4,6,7,8-tetrahydroquinoline-3-carboxylate —— C24H22BrClN2O3
ethyl (4S)-2-amino-1-(4-bromophenyl)-4-(4-chlorophenyl)-5-oxo-4,6,7,8-tetrahydroquinoline-3-carboxylate
—— ethyl N-dibenzofuran-2-ylcarbamate —— C15H13NO3
ethyl N-dibenzofuran-2-ylcarbamate
—— ethyl N-[3-(butylsulfamoyl)phenyl]carbamate —— C13H20N2O4S
ethyl N-[3-(butylsulfamoyl)phenyl]carbamate
—— Ethyl [4-[(3-methylbenzoyl)amino]phenyl] carbonate —— C17H17NO4
Ethyl [4-[(3-methylbenzoyl)amino]phenyl] carbonate
—— ethyl N-methyl-N-[(1S)-1-(4-sulfamoylphenyl)ethyl]carbamate —— C12H18N2O4S
ethyl N-methyl-N-[(1S)-1-(4-sulfamoylphenyl)ethyl]carbamate
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C23H29N2O3+
(E)-3-(3,4-dimethoxyphenyl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— ethyl N-(6-methyl-4-oxo-5-phenylthieno[2,3-d]pyrimidin-3-yl)carbamate —— C16H15N3O3S
ethyl N-(6-methyl-4-oxo-5-phenylthieno[2,3-d]pyrimidin-3-yl)carbamate
—— ethyl (4S)-2-amino-4-(4-chlorophenyl)-7,7-dimethyl-1-(4-nitrophenyl)-5-oxo-6,8-dihydro-4H-quinoline-3-carboxylate —— C26H26ClN3O5
ethyl (4S)-2-amino-4-(4-chlorophenyl)-7,7-dimethyl-1-(4-nitrophenyl)-5-oxo-6,8-dihydro-4H-quinoline-3-carboxylate
—— (E)-3-(furan-2-yl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C19H23N2O2+
(E)-3-(furan-2-yl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— (E)-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)-N-[2-oxo-2-(propylamino)ethyl]prop-2-enamide —— C20H25N3O2
(E)-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)-N-[2-oxo-2-(propylamino)ethyl]prop-2-enamide
—— ethyl (4R)-4-(4-bromophenyl)-5-cyano-2-methyl-6-(thiophen-2-ylmethylsulfanyl)-3,4-dihydropyridine-3-carboxylate —— C21H19BrN2O2S2
ethyl (4R)-4-(4-bromophenyl)-5-cyano-2-methyl-6-(thiophen-2-ylmethylsulfanyl)-3,4-dihydropyridine-3-carboxylate
—— ethyl N-(2,5-diethoxyphenyl)carbamate —— C13H19NO4
ethyl N-(2,5-diethoxyphenyl)carbamate
—— (E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[3-(3,5-dimethylpyrazol-1-yl)propyl]prop-2-enamide —— C19H24N4O3
(E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[3-(3,5-dimethylpyrazol-1-yl)propyl]prop-2-enamide
—— ethyl (4R)-6-amino-5-cyano-2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)sulfanylmethyl]-4-(4-methylsulfanylphenyl)-4H-pyran-3-carboxylate —— C26H24N4O3S2
ethyl (4R)-6-amino-5-cyano-2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)sulfanylmethyl]-4-(4-methylsulfanylphenyl)-4H-pyran-3-carboxylate
—— (E)-3-(4-methoxyphenyl)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C22H26N2O2
(E)-3-(4-methoxyphenyl)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— (E)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]-3-[3-(trifluoromethyl)phenyl]prop-2-enamide —— C22H23F3N2O
(E)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]-3-[3-(trifluoromethyl)phenyl]prop-2-enamide
—— ethyl N-[3-[3-(2,4-dimethylphenyl)propylcarbamoyl]phenyl]carbamate —— C21H26N2O3
ethyl N-[3-[3-(2,4-dimethylphenyl)propylcarbamoyl]phenyl]carbamate
—— (E)-3-(6-chloro-2H-chromen-3-yl)-N-[2-oxo-2-(propylamino)ethyl]prop-2-enamide —— C17H19ClN2O3
(E)-3-(6-chloro-2H-chromen-3-yl)-N-[2-oxo-2-(propylamino)ethyl]prop-2-enamide
—— ethyl N-methyl-N-[(1R)-1-(4-sulfamoylphenyl)ethyl]carbamate —— C12H18N2O4S
ethyl N-methyl-N-[(1R)-1-(4-sulfamoylphenyl)ethyl]carbamate