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—— (E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C18H21ClN6O2S
(E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(3-methylphenyl)prop-2-enamide —— C16H11ClN4OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(3-methylphenyl)prop-2-enamide
—— ethyl (6S)-6-(3,4-difluorophenyl)-3-(4-methoxyphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C21H20F2N2O4
ethyl (6S)-6-(3,4-difluorophenyl)-3-(4-methoxyphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-2-cyano-N-(4-ethylphenyl)-3-(2,3,4-trimethoxyphenyl)prop-2-enamide —— C21H22N2O4
(E)-2-cyano-N-(4-ethylphenyl)-3-(2,3,4-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(2-prop-2-enoxyphenyl)but-3-enoate —— C20H16NO3S-
(E)-3-(1,3-benzothiazol-2-yl)-4-(2-prop-2-enoxyphenyl)but-3-enoate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(3-methoxy-4-propoxyphenyl)but-3-enoic acid —— C21H21NO4S
(E)-3-(1,3-benzothiazol-2-yl)-4-(3-methoxy-4-propoxyphenyl)but-3-enoic acid
—— ethyl (6S)-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C18H22F2N2O5
ethyl (6S)-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-N-(4-butylphenyl)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyanoprop-2-enamide —— C19H17ClN4OS
(E)-N-(4-butylphenyl)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyanoprop-2-enamide
—— (E)-1-[1-(difluoromethoxy)naphthalen-2-yl]-3-(3-hydroxy-4-methoxyphenyl)prop-2-en-1-one —— C21H16F2O4
(E)-1-[1-(difluoromethoxy)naphthalen-2-yl]-3-(3-hydroxy-4-methoxyphenyl)prop-2-en-1-one
—— (E)-3-(4-methylsulfanylphenyl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C17H18N4S
(E)-3-(4-methylsulfanylphenyl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— ethyl (6S)-6-[4-(cyanomethoxy)phenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C17H19N3O4
ethyl (6S)-6-[4-(cyanomethoxy)phenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-cyano-N-(3-methylphenyl)prop-2-enamide —— C19H19ClN4O3S
(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-cyano-N-(3-methylphenyl)prop-2-enamide
—— ethyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-(4-methoxyphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H23N3O5
ethyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-(4-methoxyphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(7-methoxy-1,3-benzodioxol-5-yl)but-3-enoate —— C19H14NO5S-
(E)-3-(1,3-benzothiazol-2-yl)-4-(7-methoxy-1,3-benzodioxol-5-yl)but-3-enoate
—— (E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-N-(2-chlorophenyl)-2-cyanoprop-2-enamide —— C21H16Cl2N4O
(E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-N-(2-chlorophenyl)-2-cyanoprop-2-enamide
—— ethyl (6R)-6-(3,4-difluorophenyl)-3-(4-methoxyphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C21H20F2N2O4
ethyl (6R)-6-(3,4-difluorophenyl)-3-(4-methoxyphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(1,3-benzothiazol-2-yl)-N-(4-bromo-2-chlorophenyl)prop-2-enamide —— C16H10BrClN2OS
(E)-3-(1,3-benzothiazol-2-yl)-N-(4-bromo-2-chlorophenyl)prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-[4-(difluoromethoxy)-3-ethoxyphenyl]but-3-enoic acid —— C20H17F2NO4S
(E)-3-(1,3-benzothiazol-2-yl)-4-[4-(difluoromethoxy)-3-ethoxyphenyl]but-3-enoic acid
—— (E)-N-(4-chloro-2-methoxy-5-methylphenyl)-2-cyano-3-(3,4-difluorophenyl)prop-2-enamide —— C18H13ClF2N2O2
(E)-N-(4-chloro-2-methoxy-5-methylphenyl)-2-cyano-3-(3,4-difluorophenyl)prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(3-chloro-5-ethoxy-4-methoxyphenyl)but-3-enoic acid —— C20H18ClNO4S
(E)-3-(1,3-benzothiazol-2-yl)-4-(3-chloro-5-ethoxy-4-methoxyphenyl)but-3-enoic acid
—— (E)-3-[2,4-bis(difluoromethoxy)phenyl]-2-cyano-N-(2-phenylethyl)prop-2-enamide —— C20H16F4N2O3
(E)-3-[2,4-bis(difluoromethoxy)phenyl]-2-cyano-N-(2-phenylethyl)prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)but-3-enoic acid —— C20H17NO5S
(E)-3-(1,3-benzothiazol-2-yl)-4-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)but-3-enoic acid
—— (E)-2-cyano-3-(3,4-difluorophenyl)-N-naphthalen-1-ylprop-2-enamide —— C20H12F2N2O
(E)-2-cyano-3-(3,4-difluorophenyl)-N-naphthalen-1-ylprop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-[5-(3-nitrophenyl)furan-2-yl]but-3-enoic acid —— C21H14N2O5S
(E)-3-(1,3-benzothiazol-2-yl)-4-[5-(3-nitrophenyl)furan-2-yl]but-3-enoic acid
—— ethyl 4-[2-[[(S)-phenyl(thiophen-2-yl)methyl]amino]acetyl]piperazine-1-carboxylate —— C20H25N3O3S
ethyl 4-[2-[[(S)-phenyl(thiophen-2-yl)methyl]amino]acetyl]piperazine-1-carboxylate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]but-3-enoate —— C19H19ClN3O2S-
(E)-3-(1,3-benzothiazol-2-yl)-4-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]but-3-enoate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)but-3-enoate —— C16H9ClN3O2S2-
(E)-3-(1,3-benzothiazol-2-yl)-4-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)but-3-enoate
—— (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]-N-naphthalen-1-ylprop-2-enamide —— C26H19N5O
(E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]-N-naphthalen-1-ylprop-2-enamide
—— ethyl (6R)-6-[4-(difluoromethoxy)-3,5-dimethylphenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C18H22F2N2O4
ethyl (6R)-6-[4-(difluoromethoxy)-3,5-dimethylphenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(3-methoxy-4-propoxyphenyl)but-3-enoate —— C21H20NO4S-
(E)-3-(1,3-benzothiazol-2-yl)-4-(3-methoxy-4-propoxyphenyl)but-3-enoate
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(2-phenylethyl)prop-2-enamide —— C17H13ClN4OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(2-phenylethyl)prop-2-enamide
—— ethyl (6R)-3,4-dimethyl-2-oxo-6-(3-prop-2-enoxyphenyl)-1,6-dihydropyrimidine-5-carboxylate —— C18H22N2O4
ethyl (6R)-3,4-dimethyl-2-oxo-6-(3-prop-2-enoxyphenyl)-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(5-methylthiophen-2-yl)-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)prop-2-enoate —— C17H18NO4S3-
(E)-3-(5-methylthiophen-2-yl)-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)prop-2-enoate
—— ethyl (6R)-6-(5-bromothiophen-2-yl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C13H15BrN2O3S
ethyl (6R)-6-(5-bromothiophen-2-yl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[2-[[(R)-phenyl(thiophen-2-yl)methyl]amino]acetyl]piperazine-1-carboxylate —— C20H25N3O3S
ethyl 4-[2-[[(R)-phenyl(thiophen-2-yl)methyl]amino]acetyl]piperazine-1-carboxylate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]but-3-enoic acid —— C20H13ClN2O2S2
(E)-3-(1,3-benzothiazol-2-yl)-4-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]but-3-enoic acid
—— (E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-2-cyano-N-(2-phenylethyl)prop-2-enamide —— C23H21ClN4O
(E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-2-cyano-N-(2-phenylethyl)prop-2-enamide
—— ethyl (6R)-6-[4-(cyanomethoxy)phenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C17H19N3O4
ethyl (6R)-6-[4-(cyanomethoxy)phenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide —— C16H17ClN4OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(4-chloro-3-nitrophenyl)but-3-enoic acid —— C17H11ClN2O4S
(E)-3-(1,3-benzothiazol-2-yl)-4-(4-chloro-3-nitrophenyl)but-3-enoic acid
—— (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-2-cyano-N-(3-methylphenyl)prop-2-enamide —— C21H16ClFN4O
(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-2-cyano-N-(3-methylphenyl)prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(1-butyl-5-chloro-3-methylpyrazol-4-yl)but-3-enoate —— C19H19ClN3O2S-
(E)-3-(1,3-benzothiazol-2-yl)-4-(1-butyl-5-chloro-3-methylpyrazol-4-yl)but-3-enoate
—— (E)-1-[2,4-bis(difluoromethoxy)phenyl]-3-(3-hydroxyphenyl)prop-2-en-1-one —— C17H12F4O4
(E)-1-[2,4-bis(difluoromethoxy)phenyl]-3-(3-hydroxyphenyl)prop-2-en-1-one
—— ethyl (4R)-4-(methoxycarbonylamino)hex-5-enoate —— C10H17NO4
ethyl (4R)-4-(methoxycarbonylamino)hex-5-enoate
—— Ethyl 2-[[2-(5-ethyl-2-methylpyridin-1-ium-1-yl)acetyl]amino]-4-phenylthiophene-3-carboxylate —— C23H25N2O3S+
Ethyl 2-[[2-(5-ethyl-2-methylpyridin-1-ium-1-yl)acetyl]amino]-4-phenylthiophene-3-carboxylate
—— (E)-2-cyano-N-[(1R,2R)-2-methylcyclohexyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C20H26N2O4
(E)-2-cyano-N-[(1R,2R)-2-methylcyclohexyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-2-cyano-N-[(1R,2S)-2-methylcyclohexyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C20H26N2O4
(E)-2-cyano-N-[(1R,2S)-2-methylcyclohexyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— ethyl (6R)-6-(3,4-difluorophenyl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C15H16F2N2O3
ethyl (6R)-6-(3,4-difluorophenyl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(2,4-dimethylphenyl)but-3-enoic acid —— C19H17NO2S
(E)-3-(1,3-benzothiazol-2-yl)-4-(2,4-dimethylphenyl)but-3-enoic acid
—— (E)-3-(3-hydroxyphenyl)-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)prop-2-enoic acid —— C18H19NO5S2
(E)-3-(3-hydroxyphenyl)-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)prop-2-enoic acid