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—— (E)-3-[2,5-dimethyl-1-(2-propan-2-ylpyrazol-3-yl)pyrrol-3-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C22H27N7
(E)-3-[2,5-dimethyl-1-(2-propan-2-ylpyrazol-3-yl)pyrrol-3-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-[1-(1,3-benzodioxol-5-yl)-2,5-dimethylpyrrol-3-yl]-2-cyano-N-prop-2-enylprop-2-enamide —— C20H19N3O3
(E)-3-[1-(1,3-benzodioxol-5-yl)-2,5-dimethylpyrrol-3-yl]-2-cyano-N-prop-2-enylprop-2-enamide
—— (E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide —— C17H19ClN2O3
(E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)-N-(3-methylphenyl)prop-2-enamide —— C20H23N3O
(E)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)-N-(3-methylphenyl)prop-2-enamide
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-cyano-N-(2,4,6-trimethylphenyl)prop-2-enamide —— C21H19ClN2O3
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-cyano-N-(2,4,6-trimethylphenyl)prop-2-enamide
—— (E)-3-(4-methoxyphenyl)-N-[(1S)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide —— C17H21N3O5S
(E)-3-(4-methoxyphenyl)-N-[(1S)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide
—— (E)-2-cyano-N-cyclohexyl-3-[5-(2-fluorophenyl)furan-2-yl]prop-2-enamide —— C20H19FN2O2
(E)-2-cyano-N-cyclohexyl-3-[5-(2-fluorophenyl)furan-2-yl]prop-2-enamide
—— (E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-[(1S,2R)-2-methylcyclohexyl]prop-2-enamide —— C17H19ClN2O3
(E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-[(1S,2R)-2-methylcyclohexyl]prop-2-enamide
—— (E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(2,4,6-trimethylphenyl)prop-2-enamide —— C19H17ClN2O3
(E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(2,4,6-trimethylphenyl)prop-2-enamide
—— ethyl N-[3-[methyl-[2-oxo-2-(2,4,6-trimethylanilino)ethyl]carbamoyl]phenyl]carbamate —— C22H27N3O4
ethyl N-[3-[methyl-[2-oxo-2-(2,4,6-trimethylanilino)ethyl]carbamoyl]phenyl]carbamate
—— (E)-1-(4-tert-butylphenyl)-3-[1-[(3R)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]prop-2-en-1-one —— C22H28N2O3S
(E)-1-(4-tert-butylphenyl)-3-[1-[(3R)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]prop-2-en-1-one
—— (E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(3-methylphenyl)prop-2-enamide —— C17H13ClN2O3
(E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(3-methylphenyl)prop-2-enamide
—— (E)-2-cyano-3-[1-[(3R)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]-N-(3-methylphenyl)prop-2-enamide —— C20H22N4O3S
(E)-2-cyano-3-[1-[(3R)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]-N-(3-methylphenyl)prop-2-enamide
—— (E)-2-cyano-N-(3-ethoxypropyl)-3-[5-(2-fluorophenyl)furan-2-yl]prop-2-enamide —— C19H19FN2O3
(E)-2-cyano-N-(3-ethoxypropyl)-3-[5-(2-fluorophenyl)furan-2-yl]prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]but-3-enoate —— C21H18N3O3S-
(E)-3-(1,3-benzothiazol-2-yl)-4-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]but-3-enoate
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(2-chlorophenyl)-2-cyanoprop-2-enamide —— C18H12Cl2N2O3
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(2-chlorophenyl)-2-cyanoprop-2-enamide
—— (E)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)-N-prop-2-enylprop-2-enamide —— C16H21N3O
(E)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)-N-prop-2-enylprop-2-enamide
—— (E)-3-[1-(1,3-benzodioxol-5-yl)-2,5-dimethylpyrrol-3-yl]-2-cyano-N-(3-ethoxypropyl)prop-2-enamide —— C22H25N3O4
(E)-3-[1-(1,3-benzodioxol-5-yl)-2,5-dimethylpyrrol-3-yl]-2-cyano-N-(3-ethoxypropyl)prop-2-enamide
—— (E)-2-cyano-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-[5-(2-fluorophenyl)furan-2-yl]prop-2-enamide —— C24H21FN2O4
(E)-2-cyano-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-[5-(2-fluorophenyl)furan-2-yl]prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-[2,5-dimethyl-1-(2-propan-2-ylpyrazol-3-yl)pyrrol-3-yl]but-3-enoate —— C23H23N4O2S-
(E)-3-(1,3-benzothiazol-2-yl)-4-[2,5-dimethyl-1-(2-propan-2-ylpyrazol-3-yl)pyrrol-3-yl]but-3-enoate
—— (E)-N-(2-chlorophenyl)-2-cyano-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide —— C20H17ClN4O2
(E)-N-(2-chlorophenyl)-2-cyano-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide
—— (E)-3-[5-(2-fluorophenyl)furan-2-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C20H17FN4O
(E)-3-[5-(2-fluorophenyl)furan-2-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(3-chloro-2-methylphenyl)-2-cyanoprop-2-enamide —— C19H14Cl2N2O3
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(3-chloro-2-methylphenyl)-2-cyanoprop-2-enamide
—— (E)-3-(2,5-dimethoxyphenyl)-N-[(1S)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide —— C18H23N3O6S
(E)-3-(2,5-dimethoxyphenyl)-N-[(1S)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide
—— (E)-2-cyano-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[(1S,2R)-2-methylcyclohexyl]prop-2-enamide —— C21H26N4O2
(E)-2-cyano-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[(1S,2R)-2-methylcyclohexyl]prop-2-enamide
—— (E)-2-cyano-N-(2,6-dimethylphenyl)-3-[1-[(3S)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]prop-2-enamide —— C21H24N4O3S
(E)-2-cyano-N-(2,6-dimethylphenyl)-3-[1-[(3S)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]prop-2-enamide
—— (E)-2-cyano-N-[(2R)-1-methoxypropan-2-yl]-3-(3-methylfuran-2-yl)prop-2-enamide —— C13H16N2O3
(E)-2-cyano-N-[(2R)-1-methoxypropan-2-yl]-3-(3-methylfuran-2-yl)prop-2-enamide
—— (E)-2-cyano-3-[1-[(3S)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]-N-(2-phenylethyl)prop-2-enamide —— C21H24N4O3S
(E)-2-cyano-3-[1-[(3S)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]-N-(2-phenylethyl)prop-2-enamide
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-prop-2-enylprop-2-enamide —— C14H11ClN2O3
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-prop-2-enylprop-2-enamide
—— (E)-2-cyano-N-(2,4-dimethylphenyl)-3-[1-[(3R)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]prop-2-enamide —— C21H24N4O3S
(E)-2-cyano-N-(2,4-dimethylphenyl)-3-[1-[(3R)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]prop-2-enamide
—— (E)-2-cyano-N-[(2S)-1-methoxypropan-2-yl]-3-(3-methylfuran-2-yl)prop-2-enamide —— C13H16N2O3
(E)-2-cyano-N-[(2S)-1-methoxypropan-2-yl]-3-(3-methylfuran-2-yl)prop-2-enamide
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C17H15ClN4O2
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-cyano-N-(2,5-dichlorophenyl)prop-2-enamide —— C18H11Cl3N2O3
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-cyano-N-(2,5-dichlorophenyl)prop-2-enamide
—— (E)-3-(4-chlorophenyl)-N-[(1S)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide —— C16H18ClN3O4S
(E)-3-(4-chlorophenyl)-N-[(1S)-2-methyl-1-(5-methylsulfonyl-1,3,4-oxadiazol-2-yl)propyl]prop-2-enamide
—— ethyl 4-[[(2R)-3-methoxy-3-oxo-2-phenylpropyl]amino]-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate —— C21H23N3O4S
ethyl 4-[[(2R)-3-methoxy-3-oxo-2-phenylpropyl]amino]-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl N-[(3R)-1-[2-(6-chloro-2,3-dihydro-1,4-benzoxazin-4-yl)acetyl]piperidin-3-yl]carbamate —— C18H24ClN3O4
ethyl N-[(3R)-1-[2-(6-chloro-2,3-dihydro-1,4-benzoxazin-4-yl)acetyl]piperidin-3-yl]carbamate
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-(2-phenylethyl)prop-2-enamide —— C19H15ClN2O3
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-(2-phenylethyl)prop-2-enamide
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-[(1S,2R)-2-methylcyclohexyl]prop-2-enamide —— C18H19ClN2O3
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-[(1S,2R)-2-methylcyclohexyl]prop-2-enamide
—— (E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(4-ethylphenyl)prop-2-enamide —— C18H15ClN2O3
(E)-3-(3-chloro-4,5-dihydroxyphenyl)-2-cyano-N-(4-ethylphenyl)prop-2-enamide
—— (E)-N-(2-chlorophenyl)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)prop-2-enamide —— C19H20ClN3O
(E)-N-(2-chlorophenyl)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)prop-2-enamide
—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-1-(4-nitrophenyl)prop-2-en-1-one —— C19H17N3O4
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-1-(4-nitrophenyl)prop-2-en-1-one
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C18H17ClN4O2
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-(2,5-dichlorophenyl)prop-2-enamide —— C17H9Cl3N2O3
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-2-cyano-N-(2,5-dichlorophenyl)prop-2-enamide
—— (E)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)-N-[(1S,2R)-2-methylcyclohexyl]prop-2-enamide —— C20H29N3O
(E)-2-cyano-3-(2,5-dimethyl-1-propan-2-ylpyrrol-3-yl)-N-[(1S,2R)-2-methylcyclohexyl]prop-2-enamide
—— ethyl N-[4-[[(1R)-1-(2,4-dichloro-5-fluorophenyl)ethyl]carbamoyl]phenyl]carbamate —— C18H17Cl2FN2O3
ethyl N-[4-[[(1R)-1-(2,4-dichloro-5-fluorophenyl)ethyl]carbamoyl]phenyl]carbamate
—— ethyl N-[(3S)-1-[2-(6-chloro-2,3-dihydro-1,4-benzoxazin-4-yl)acetyl]piperidin-3-yl]carbamate —— C18H24ClN3O4
ethyl N-[(3S)-1-[2-(6-chloro-2,3-dihydro-1,4-benzoxazin-4-yl)acetyl]piperidin-3-yl]carbamate
—— ethyl N-[3-[[(1R)-1-(4-chlorophenyl)ethyl]carbamoyl]phenyl]carbamate —— C18H19ClN2O3
ethyl N-[3-[[(1R)-1-(4-chlorophenyl)ethyl]carbamoyl]phenyl]carbamate
—— (E)-N-[(1R)-1-(4-chlorophenyl)ethyl]-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide —— C18H15ClN2O5
(E)-N-[(1R)-1-(4-chlorophenyl)ethyl]-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide
—— (E)-3-[1-(1,3-benzodioxol-5-yl)-2,5-dimethylpyrrol-3-yl]-2-cyano-N-(2,6-dimethylphenyl)prop-2-enamide —— C25H23N3O3
(E)-3-[1-(1,3-benzodioxol-5-yl)-2,5-dimethylpyrrol-3-yl]-2-cyano-N-(2,6-dimethylphenyl)prop-2-enamide
—— (E)-2-cyano-N-(2,6-dimethylphenyl)-3-[5-(2-fluorophenyl)furan-2-yl]prop-2-enamide —— C22H17FN2O2
(E)-2-cyano-N-(2,6-dimethylphenyl)-3-[5-(2-fluorophenyl)furan-2-yl]prop-2-enamide