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—— (5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-fluorophenyl)-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione —— C30H25F2N3O4S2
(5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-fluorophenyl)-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione
—— (5S)-5-(4-butoxy-3-ethoxyphenyl)-1-(6-chloro-1,3-benzothiazol-2-yl)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]pyrrolidine-2,3-dione —— C32H29ClN2O7S
(5S)-5-(4-butoxy-3-ethoxyphenyl)-1-(6-chloro-1,3-benzothiazol-2-yl)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]pyrrolidine-2,3-dione
—— (5S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(3-fluorophenyl)pyrrolidine-2,3-dione —— C30H26FN3O4S2
(5S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(3-fluorophenyl)pyrrolidine-2,3-dione
—— (5S)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione —— C34H28FN3O7S2
(5S)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-1-[5-(naphthalen-1-ylmethylsulfanyl)-1,3,4-thiadiazol-2-yl]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C37H38N2O5
(5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-1-[3-(diethylamino)propyl]-4-[(4-ethoxyphenyl)-hydroxymethylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione —— C32H44N2O6
(5S)-1-[3-(diethylamino)propyl]-4-[(4-ethoxyphenyl)-hydroxymethylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione
—— (5S)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2,3-dione —— C31H32N2O7
(5S)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2,3-dione
—— (5S)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione —— C30H25F2N3O4S2
(5S)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(2-fluorophenyl)-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione
—— (5S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(3,4-dichlorophenyl)pyrrolidine-2,3-dione —— C30H25Cl2N3O4S2
(5S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(3,4-dichlorophenyl)pyrrolidine-2,3-dione
—— (5R)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,3-dione —— C31H32N2O7
(5R)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)methylidene]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,3-dione
—— (5S)-5-(4-butoxy-3-methoxyphenyl)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]pyrrolidine-2,3-dione —— C36H44N2O6
(5S)-5-(4-butoxy-3-methoxyphenyl)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]pyrrolidine-2,3-dione
—— (5S)-1-[3-(diethylamino)propyl]-5-(3-ethoxy-4-hydroxyphenyl)-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]pyrrolidine-2,3-dione —— C34H40N2O6
(5S)-1-[3-(diethylamino)propyl]-5-(3-ethoxy-4-hydroxyphenyl)-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]pyrrolidine-2,3-dione
—— (5S)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[5-[(2-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-5-(3,4-dichlorophenyl)pyrrolidine-2,3-dione —— C30H24Cl3N3O4S2
(5S)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[5-[(2-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-5-(3,4-dichlorophenyl)pyrrolidine-2,3-dione
—— [5-(3,4-Dimethylphenyl)-3-methoxypentyl] acetate —— C16H24O3
[5-(3,4-Dimethylphenyl)-3-methoxypentyl] acetate
—— (5R)-1-[3-(diethylamino)propyl]-4-[[4-[(4-fluorophenyl)methoxy]phenyl]-hydroxymethylidene]-5-(4-phenylmethoxyphenyl)pyrrolidine-2,3-dione —— C38H39FN2O5
(5R)-1-[3-(diethylamino)propyl]-4-[[4-[(4-fluorophenyl)methoxy]phenyl]-hydroxymethylidene]-5-(4-phenylmethoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dione —— C33H33N3O4S2
(5S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dione
—— (5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-propoxyphenyl)methylidene]-5-(3-methoxy-4-phenylmethoxyphenyl)pyrrolidine-2,3-dione —— C35H42N2O6
(5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-propoxyphenyl)methylidene]-5-(3-methoxy-4-phenylmethoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-5-(3-methoxy-4-phenylmethoxyphenyl)pyrrolidine-2,3-dione —— C35H28FN3O6S2
(5R)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-5-(3-methoxy-4-phenylmethoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[3-(diethylamino)propyl]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione —— C34H48N2O6
(5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[3-(diethylamino)propyl]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione
—— (5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C38H40N2O5
(5S)-1-[3-(diethylamino)propyl]-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-5-(4-bromophenyl)-4-[hydroxy-[4-[(3-methylphenyl)methoxy]phenyl]methylidene]-1-(3-imidazol-1-ylpropyl)pyrrolidine-2,3-dione —— C31H28BrN3O4
(5S)-5-(4-bromophenyl)-4-[hydroxy-[4-[(3-methylphenyl)methoxy]phenyl]methylidene]-1-(3-imidazol-1-ylpropyl)pyrrolidine-2,3-dione
—— 5-fluoro-2-(pyridin-2-ylmethyl)isoindoline-1,3-dione —— C14H9FN2O2
5-fluoro-2-(pyridin-2-ylmethyl)isoindoline-1,3-dione
—— 5-Anilino-2-methyl-6-propoxypyridazin-3-one —— C14H17N3O2
5-Anilino-2-methyl-6-propoxypyridazin-3-one
—— (5R)-5-(4-butoxy-3-methoxyphenyl)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]pyrrolidine-2,3-dione —— C36H44N2O6
(5R)-5-(4-butoxy-3-methoxyphenyl)-1-[3-(diethylamino)propyl]-4-[hydroxy-(4-phenylmethoxyphenyl)methylidene]pyrrolidine-2,3-dione
—— (5R)-1-[3-(diethylamino)propyl]-5-(3-ethoxy-4-hydroxyphenyl)-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]pyrrolidine-2,3-dione —— C34H40N2O6
(5R)-1-[3-(diethylamino)propyl]-5-(3-ethoxy-4-hydroxyphenyl)-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]pyrrolidine-2,3-dione
—— (5R)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-fluorophenyl)pyrrolidine-2,3-dione —— C30H26FN3O4S2
(5R)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-fluorophenyl)pyrrolidine-2,3-dione
—— [(5S,7R)-2-bromo-1-adamantyl]methanol —— C11H17BrO
[(5S,7R)-2-bromo-1-adamantyl]methanol
—— (5S)-1-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-4-[hydroxy-(4-methoxyphenyl)methylidene]-5-(4-phenylmethoxyphenyl)pyrrolidine-2,3-dione —— C31H26N2O6S
(5S)-1-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-4-[hydroxy-(4-methoxyphenyl)methylidene]-5-(4-phenylmethoxyphenyl)pyrrolidine-2,3-dione
—— 5-Cyclohexyl-2-[3-(3H-imidazol-4-yl)-propyl]-1H-imidazole —— C15H22N4
5-Cyclohexyl-2-[3-(3H-imidazol-4-yl)-propyl]-1H-imidazole
—— 5-Methanesulfonylamino-[1,3,4]thiadiazole-2-sulfonic acid amide —— C3H6N4O4S3
5-Methanesulfonylamino-[1,3,4]thiadiazole-2-sulfonic acid amide
—— 5-Hydrazinyl-4-(naphthalen-2-ylmethyl)-1,2-dihydropyrazol-3-one —— C14H14N4O
5-Hydrazinyl-4-(naphthalen-2-ylmethyl)-1,2-dihydropyrazol-3-one
—— 5-(2-Phenoxypropyl)-1,3-thiazolidine-2,4-dione —— C12H13NO3S
5-(2-Phenoxypropyl)-1,3-thiazolidine-2,4-dione
—— (5S,8aR)-5-Naphthalen-1-yl-octahydro-indolizine —— C18H21N
(5S,8aR)-5-Naphthalen-1-yl-octahydro-indolizine
—— 5-Bromo-1,2,3,4-tetrahydro-2-ethylisoquinolin-8-amine —— C11H15BrN2
5-Bromo-1,2,3,4-tetrahydro-2-ethylisoquinolin-8-amine
—— 5-Azido-4-chloro-2-(4-hydroxybutyl)pyridazin-3-one —— C8H10ClN5O2
5-Azido-4-chloro-2-(4-hydroxybutyl)pyridazin-3-one
—— (5S)-1-[3-(diethylamino)propyl]-5-(4-ethoxy-3-methoxyphenyl)-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]pyrrolidine-2,3-dione —— C35H42N2O6
(5S)-1-[3-(diethylamino)propyl]-5-(4-ethoxy-3-methoxyphenyl)-4-[hydroxy-[4-[(4-methylphenyl)methoxy]phenyl]methylidene]pyrrolidine-2,3-dione
—— (5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[3-(diethylamino)propyl]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C34H40N2O5
(5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[3-(diethylamino)propyl]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(3,4-dichlorophenyl)-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione —— C30H24Cl2FN3O4S2
(5S)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(3,4-dichlorophenyl)-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione
—— (5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-chlorophenyl)-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione —— C30H25ClFN3O4S2
(5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-chlorophenyl)-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]pyrrolidine-2,3-dione
—— (5R,7R)-N-[(6S)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H30F3N5O2S
(5R,7R)-N-[(6S)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[3-(diethylamino)propyl]-5-(4-pentoxyphenyl)pyrrolidine-2,3-dione —— C33H46N2O5
(5R)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[3-(diethylamino)propyl]-5-(4-pentoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-5-[3-[(4-chlorophenoxy)methyl]-4-methoxyphenyl]-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-pyridin-2-ylpyrrolidine-2,3-dione —— C31H25ClN2O6
(5S)-5-[3-[(4-chlorophenoxy)methyl]-4-methoxyphenyl]-4-[hydroxy-(4-methoxyphenyl)methylidene]-1-pyridin-2-ylpyrrolidine-2,3-dione
—— (5E)-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione —— C13H8N2O2S
(5E)-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione
—— (5,7-Dimethyl-6-oxo-9-thia-1,3,5-triaza-7-azoniatricyclo[6.3.1.04,12]dodeca-2,4(12),7-trien-10-yl)methanolate —— C10H12N4O2S
(5,7-Dimethyl-6-oxo-9-thia-1,3,5-triaza-7-azoniatricyclo[6.3.1.04,12]dodeca-2,4(12),7-trien-10-yl)methanolate
—— (5R)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C33H23F2N3O5S2
(5R)-4-[(3-fluoro-4-methoxyphenyl)-hydroxymethylidene]-1-[5-[(4-fluorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[3-(diethylamino)propyl]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione —— C34H48N2O6
(5S)-4-[(4-butoxyphenyl)-hydroxymethylidene]-1-[3-(diethylamino)propyl]-5-[3-methoxy-4-(3-methylbutoxy)phenyl]pyrrolidine-2,3-dione
—— (5S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-fluorophenyl)pyrrolidine-2,3-dione —— C30H26FN3O4S2
(5S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-4-[(4-butoxyphenyl)-hydroxymethylidene]-5-(4-fluorophenyl)pyrrolidine-2,3-dione
—— [(5S)-3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methanone —— C14H10F8N2O3
[(5S)-3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]methanone
—— (5R,10bS)-1'-benzyl-9-bromo-2-(4-methylphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one —— C31H24BrN3O2
(5R,10bS)-1'-benzyl-9-bromo-2-(4-methylphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one
—— (5R,7S)-N-[(6R)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C28H30F3N5O2S
(5R,7S)-N-[(6R)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide